Carbamates and crop protection agents containing them

ABSTRACT

Carbamates of the formula I ##STR1## where the substituents have the following meanings: Z is methoxy, NH 2 , NHCH 3 , N(CH 3 ) 2 , CH 3 , C 2  H 5 , CF 3  or CCl 3 , 
     X and Y are identical or different and each is hydrogen, F, Cl, Br, CF 3 , CN, NO 2 , alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may be condensed together to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, 
     R 1  may also be substituted or unsubstituted and is O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O--CO 2  -alkyl, 
     A is --O--, --S--, --CR 2  ═CR 3  --, CHR 2  --O--, --CHR 2  --S--, --CHR 2  --O--N═C(R 4 )--, --CR 2  ═N--O--, --O--N═C(R 4 )--, --C.tbd.C--, --CHR 2  --CHR 3  --, --CHR 2  --O--CO--, --O--CHR 2  -- or a single bond, 
     B is substituted or unsubstituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, substituted or unsubstituted alkylaryl, substituted or unsubstituted alkylhetaryl, substituted or unsubstituted alkylcycloalkyl, substituted or unsubstituted alkylcycloalkenyl, 
     R 2  and R 3  are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, 
     R 4  is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl, 
     R 5  is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl and plant-tolerated acid and base adducts thereof, and fungicides containing them.

DESCRIPTION

The present invention relates to carbamates and crop protection agents, in particular for controlling fungi, insects, nematodes and spider mites.

It is known that aniline derivatives, for example isopropyl N-phenylcarbamate or the corresponding 3-chlorophenyl ester (GB 574 995) or methyl N-3,4-dichloro-phenylcarbamate (BE 612 550) can be used as crop protection agents. However, their fungicidal action is unsatisfactory.

It has now been found, surprisingly, that carbamates of the formula I ##STR2## where the substituents have the following meanings: Z is methoxy, NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂ H₅, CF₃ or CCl₃,

X and Y independently of one another are each hydrogen,

F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R¹ is unsubstituted or substituted alkyl, alkenyl, cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH₂ --CN, --CH₂ OCH₃, --CO₂ CH₃ or --S--R⁵, O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O--CO₂ -alkyl,

A is --O--, --S--, --CR² ═CR³ --, CHR² --O, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O--, --O--N═C(R⁴)--, --C.tbd.--C--, --CHR² --CHR³ --, --CHR² --O--CO--, --O--CHR² -- or a single bond,

B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, unsubstituted or substituted alkylaryl, unsubstituted or substituted alkylhetaryl, unsubstituted or substituted alkylcycloalkyl or unsubstituted or substituted alkylcycloalkenyl,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl,

R⁴ is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl,

R⁵ is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products have a good fungicidal, acaricidal, insecticidal and nematocidal action.

Acids for addition products are, for example, mineral acids, such as hydrochloric acid, hydrobromic acid, phosphoric acid, sulfuric acid or nitric acid, or carboxylic acids, such as formic acid, acetic acid, oxalic acid, malonic acid, lactic acid, malic acid, succinic acid, tartaric acid, citric acid, salicylic acid, p-toluenesulfonic acid or dodecylbenzenesulfonic acid, as well as proton-acidic compounds generally, for example saccharin.

Bases for base addition products are, for example, potassium hydroxide, sodium hydroxide, potassium carbonate, sodium carbonate and ammonium hydroxide.

The novel compounds of the formula I may be obtained in the preparation as mixtures of stereoisomers (E/Z isomers, diastereomers, enantiomers), which can be separated into the individual components in a conventional manner, for example by crystallization or chromatography. Both the individual isomers and mixtures thereof may be used as fungicides, acaricides, nematocides or insecticides, and form the subject of the present invention.

The abovementioned alkyl radicals may be substituted and are of 1 to 6 carbon atoms.

The abovementioned alkenyl and alkynyl radicals may be substituted and are of 2 to 6 carbon atoms.

The abovementioned cycloalkyl radicals are of 3 to 10 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The abovementioned aryl radicals are of 6, 10 or 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The abovementioned hetaryl radicals have 5 to 14 ring atoms, including from 1 to 4 hetero atoms selected from the group consisting of N, O and S, are unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The above mentioned heterocyclyl radicals have 5 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S, are saturated or partially unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substitutents R⁶.

The abovementioned cycloalkenyl radicals are of 5 to 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

Two adjacent substituents R⁶, together with the carbon atoms of which they are substituents, may form a carbocyclic hydrogenated, partially unsaturated or aromatic ring having 3 to 14 carbon atoms or a heterocyclic hydrogenated, partially unsaturated or heteroaromatic ring having 3 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S.

R⁶ may be unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁷, and R⁶ is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoxyimino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl, alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsuifonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

R⁷ is is any substituent and is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoximino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl; alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

The abovementioned alkyl radicals may be substituted, are preferably of 1 to 6 carbon atoms and are, in particular, methyl, ethyl, propyl, such as n-propyl or isopropyl, butyl, such as n-butyl, isobutyl, tert-butyl or sec-butyl, pentyl or hexyl.

The abovementioned alkenyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethenyl, propenyl, such as prop-1-enyl, prop-2-enyl or prop-1-en-2-yl, butenyl, such as but-1-enyl, but-2-enyl, but-3-enyl, but-1-en-3-yl, but-2-en-2-yl, but-1-en-2-yl, 2-methyl-1-propenyl or 2-methyl-2-propenyl, pentenyl or hexenyl.

The abovementioned alkynyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethynyl, propynyl, such as prop-1-ynyl or prop-3-ynyl, butynyl, such as but-1-ynyl, but-2-ynyl, but-3-ynyl or 1-methylprop-2-ynyl, pentynyl or hexynyl.

The abovementioned halogens are fluorine, chlorine, bromine or iodine.

The abovementioned cycloalkyl radicals are preferably cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclooctyl, cyclononyl, cyclodecyl, bornanyl, norbornanyl, dicyclohexyl, bicyclo 3.3.0!octyl, bicyclo 3.2.1!octyl, bicyclo 2.2.2!octyl or bicyclo 3.3.1!nonyl.

The abovementioned cycloalkenyl radicals are preferably cyclopropenyl, cyclobutenyl, cyclopentenyl, cyclohexenyl, cycloheptenyl, cyclooctenyl, cyclononenyl, cyclodecenyl, bornenyl, norbornenyl, bicyclo 3.3.0!octenyl, bicyclo 3.2.1!octenyl, bicyclo 2.2.2!octenyl or bicyclo 3.3.1!nonenyl.

The abovementioned haloalkyl radicals are preferably C₁ -C₄ -haloalkyl, in particular C₁ - or C₂ -haloalkyl, such as chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorof luoromethyl, chlorodifluoromethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl or pentafluoroethyl.

The abovementioned haloalkoxy radicals are preferably C₁ -C₄ -haloalkoxy, in particular C₁ - or C₂ -haloalkoxy, such as chloromethoxy, dichloromethoxy, trichloromethoxy, fluoromethoxy, difluoromethoxy, trifluoromethoxy, chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 1-fluoroethoxy, 2-fluoroethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy or pentafluoroethoxy.

The abovementioned aryl radicals are preferably phenyl, 1-naphthyl, 2-naphtyl, 1-anthracenyl, 2-anthracenyl or 9-anthracenyl.

The abovementioned hetaryl radicals are preferably furyl, such as 2-furyl or 3-furyl, thienyl, such as 2-thienyl or 3-thienyl, pyrrolyl, such as 1-pyrrolyl, 2-pyrrolyl or 3-pyrrolyl, isoxazolyl, such as 3-isoxazolyl, 4-isoxazolyl or 5-isoxazolyl, isothiazolyl, such as 3-isothiazolyl, 4-isothiazolyl or 5-isothiazolyl, pyrazolyl, such as 1-pyrazolyl, 3-pyrazolyl, 4-pyrazolyl or 5-pyrazolyl, oxazolyl, such as 2-oxazolyl, 4-oxazolyl or 5-oxazolyl, thiazolyl, such as 2-thiazolyl, 4-thiazolyl or 5-thiazolyl, imidazolyl, such as 1-imidazolyl, 2-imidazolyl, 4-imidazolyl or 5-imidazolyl, 1,2,3-thiadiazolyl, 1,2,4-thiadiazolyl, 1,2,5-thiadiazolyl, 1,3,4-thiadiazolyl, tetrazolyl, 1,2,3,4-thiatriazolyl, 1,2,3,4-oxatriazolyl, pyridyl, such as 2-pyridyl or 4-pyridyl, pyridazinyl, such as 3-pyridazinyl or 4-pyridazinyl, pyrimidinyl, such as 2-pyrimidinyl, 4-pyrimidinyl or 5-pyrimidinyl, pyrazinyl, such as 2-pyrazinyl or 3-pyrazinyl, 1,2,4-triazinyl, 1,3,5-triazinyl or 1,2,4,5-tetrazinyl.

Adjacent substituents of the hetero atoms may be condensed to form an aromatic or heteroaromatic ring, so that hetaryl also comprises fused ring systems, eg. benzofuranyl, isobenzofuranyl, 1-benzothienyl, 2-benzothienyl, indolyl, isoindolyl, benzisoxazolyl, benzoxazolyl, benzisothiazolyl, benzothiazolyl, such as 2-benzothiazolyl, 4-benzothiazolyl, 5-benzothiazolyl, 6-benzothiazolyl or 7-benzothiazolyl, indazolyl, benzimidazolyl, benzofurazanyl, dibenzofuranyl, dibenzothienyl, acridinyl, phenanthridinyl, carbazolyl, quinolyl, isoquinolyl, phthalazinyl, quinazolinyl, quinoxalinyl, cinnolinyl, 1,5-naphthyridinyl, 1,6-naphthyridinyl, 1,7-naphthyridinyl, 1,8-naphthyridinyl, pteridinyl, pyrrolopyridinyl, pyrrolopyridazinyl, pyrrolopyrimidinyl, pyrrolopyrazinyl, pyrrolotriazinyl, furopyridyl, furopyridazinyl, furopyrimidinyl, furopyrazinyl, furotriazinyl, thienopyridyl, thienopyridazinyl, thienopyrimidinyl, thienopyrazinyl, thienotriazinyl, imidazopyridazinyl, imidazopyrimidinyl, imidazopyrazinyl, pyrazolopyridyl, pyrazolopyridazinyl, pyrazolopyrimidinyl, pyrazopyrazinyl, isoxazolopyrazinyl, oxazolopyridyl, oxazolopyridazinyl, oxazolopyrimidinyl, oxazolopyrazinyl, thiazolopyridyl, thiazolopyridazinyl, isothiazolopyrazinyl, triazolopyridyl, triazolopyridazinyl, triazolopyrimidinyl or triazolopyrazinyl.

The abovementioned heterocycyl radicals are preferably 2-tetrahydrofuranyl, oxiranyl, 3-tetrahydrofuranyl, 2-tetrahydrothienyl, 3-tetrahydrothienyl, 2-pyrrolidinyl, 3-pyrrolidinyl, 3-isoxazolidinyl, 4-isoxazolidinyl, 5-isoxazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl, 5-isothiazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4-oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl, 4-thiazolidinyl, 5-thiazolidinyl, 2-imidazolidinyl, 4-imidazolidinyl, 1,2,4-oxadiazolidin-3-yl, 1,2,4-oxadiazolidin-5-yl, 1,2,4-thiadiazolidin-3-yl, 1,2,4-thiadiazolidin-5-yl, 1,2,5-triazolidin-3-yl, 1,3,4-oxadiazolidin-2-yl, 1,3,4-thiadiazolidin-2-yl, 1,3,4-triazolidin-2-yl, 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,5-dihydrofur-2-yl, 2,5-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,3-dihydrothieno-2-yl, 2,3-dihydrothien-3-yl, 2,5-dihydrothien-2-yl, 2,4-pyrrolin-2-yl, 2,3-pyrrolin-3-yl, 2,5-pyrrolin-2-yl, 2,5-pyrrolin-3-yl, 2,3-isoxazolidin-3-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-2-yl, 2,3-isoxazolin-4-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-4-yl, 2,3-isoxazolin-5-yl, 3,4-isoxazolin-5-yl, 4,5-isoxazolin-5-yl, 2,3-isothiazolin-3-yl, 3,4-isothiazolin-3-yl, 4,5-isothiazolin-3-yl, 2,3-isothiazolin-4-yl, 3,4-isothiazolin-4-yl, 4,5-isothiazolin-4-yl, 2,3-isothiazolin-5-yl, 3,4-isothiazolin-5-yl, 4,5-isothiazolin-5-yl, 2,3-dihydropyrazol-1-yl, 2,3-dihydro-pyrazol-2-yl, 2,3-dihydropyrazol-3-yl, 2,3-dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol-1-yl, 3,4-dihydropyrazol-2-yl, 3,4-dihydropyrazol-4-yl, 3,4-dihydropyrazol-5-yl, 4,5-dihydropyrazol-1-yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol-4-yl, 4,5-dihydropyrazol-5-yl, 3,4-dihydrooxazol-2-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 3,4-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 2-piperidinyl, 3-piperidinyl, 4-piperidinyl, 3-tetrahydropyridazinyl, 4-tetrahydropyridazinyl, 2-tetrahydropyrimidinyl, 4-tetrahydropyrimidinyl, 5-tetrahydropyrimidinyl, 2-tetrahydropyrazinyl, 1,3,5-tetrahydrotriazin-2-yl, 1,2,4-tetrahydrotriazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, oxazol-2-in-2-yl, 2-tetrahydropyranyl, 1,3-dioxolan-2-yl, thiazol-2-in-2-yl, 3,4,5,6-tetrahydropyridin-2-yl, 4H-1,3-thiazin-2-yl, 4H-3,1-benzothiazin-2-yl, 1,1-dioxo-2,3,4,5-tetrahydrothien-2-yl, 2H-1,4-benzothiazin-3-yl, 2H-1,4-benzoxazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, N-morpholinyl or dihydroquinazolinyl.

The invention furthermore relates to carbamates of the formula I ##STR3## where the substituents have the following meanings: Z is methoxy, NH₂, NHCH₃ or CH₃,

X and Y independently of one another are each hydrogen,

F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form a phenyl ring,

R¹ is hydrogen, alkyl, alkenyl alkynyl cyclopropyl, cyclopropylmethyl, cyclobutyl, --CH₂ --CN, --CH₂ --O--CH₃, --CO₂ CH₃ or --S--R⁵,

A is --O--, --CR² ═CR³ --, --C.tbd.C--, --CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O-- or --O--N═C(R⁴)--,

a) B is substituted phenyl when A is --CR² .tbd.--CR³ --, --C═C--, --CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O-- or --O--N═C(R⁴),

b) or B is unsubstituted or substituted cyclolalkyl, unsubstituted or substituted cycloalkenyl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted hetaryl, unsubstituted or substituted naphthyl, unsubstituted or substituted arylalkyl, unsubstituted or substituted hetarylalkyl, unsubstituted or substituted cycloalkylalkyl, unsubstituted or substituted cycloalkenylalkyl or unsubstituted or substituted anthracenyl,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl,

R⁴ is CN, alkyl, alkenyl, alkynyl or cycloalkyl and

R⁵ is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula II ##STR4## where X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula III ##STR5## where X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula I as claimed in claim 2, where A is --CH═CH-- and X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula VII ##STR6## where the substituents have the following meanings: X and Y independently of one another are each hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R¹ can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or --CO₂ -alkyl,

A is --O--, --S--, --CR² ═CR³ --, CHR² --O--, --CHR² --S--, --CHR² --O--N═C(R⁴)--, --CR² ═N--O--, --O--N═C(R⁴)--, --C--.tbd.C--, --CHR² --CHR³ --, --CER² --O--CO--, --O--CHR² -- or a single bond,

B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl or hydrogen,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula VIII ##STR7## where A, B and R¹ have the meanings stated in claim 9.

The invention furthermore relates to carbamates of the formula IX ##STR8## where R¹ and B have the meanings stated in claim 1.

The invention furthermore relates to carbamates of the formula X ##STR9## where R¹ and B have the meanings stated in claim 1.

The novel compounds can be prepared, for example, by the following processes:

The nitrobenzenes 1 obtainable by standard processes are reduced to the anilines 2, for example with hydrogen or hydrogen transfer agents, such as ammonium formate, in the presence of suitable catalysts, such as Pd, Pt or Ni, with complex reducing agents, eg. Collman's reagent (Na₂ Fe(CO)₄) or by other methods known from the literature (J. March, Advanced Organic Chemistry, 3rd Edition, 1985, page 1103 et seq.). The anilines 2 are reacted under alkaline conditions with methyl chloroformate to give the carbamates 3. The reaction of the carbamates 3 under alkaline conditions with the corresponding alkylating agents, acylating agents or R⁵ --S--S(═O)₂ --R⁵ gives the derivatives 4 (Scheme 1). ##STR10##

The nitrobenzenes 5 can be converted into the carbamates 6 similarly to Scheme 1. The halogen derivatives 7 (Z=Cl or Br) are obtainable by acidic cleavage 5 of the methyl ether of 6 (Scheme 2). ##STR11##

Alternatively, the halogen derivatives 7 (Z=Cl or Br) are obtainable from the derivatives 9 by free radical halogenation. The carbamates 9 are in turn prepared from the corresponding starting materials 8, similarly to Scheme 1 (Scheme 3). ##STR12##

The halogen derivatives 7 (Z=Cl or Br) can be converted into the active ingredients 10 under alkaline conditions. Alternatively, the compounds 7 are converted into the phosphorus compounds 11a and 11b by reaction with P(C₆ H₅)₃ or P(O-Alkyl)₃, or into the carbonyl compounds 12 by oxidation (for example with N-methylmorpholine N-oxide) (Scheme 4). ##STR13##

The corresponding stilbenes 13 are obtainable from the phosphonium salts 11a or phosphonates 11b or carbonyl compounds 12 by a Wittig reaction (Scheme 5). ##STR14##

Partial reduction of the nitroaromatics 21 (for example with zinc (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278) or with hydrogen in the presence of suitable catalysts such as platinum (similarly to European Patent 85,890)) gives the hydroxylamines 22, which can be reacted under alkaline conditions with an acylating agent (eg. propionyl chloride) or a carbamoylating agent (eg. methyl isocyanate) to give the compound 23 and then with an electrophile, for example with an alkylating agent, to give the active ingredients 24 (scheme 11). ##STR15##

In addition, the hydroxylamine 25 can be acylated or aminoacylated (for example with methyl isocyanate) (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278; European Patent 85,890) to give the compound 26, which can then be alkylated or alkoxyacylated (for example with chloroformates) to give the hydroxylamine derivative 27. The free radical halogenation of 27, for example with N-bromosuccinamide, bromine, chlorine or So₂ Cl₂ in the presence of free radical initiator, eg. azobisisobutyronitrile, or with exposure to UV light, then gives the halide 28 (Hal=Cl or Br; Scheme 12). ##STR16##

The halides 28 can then be converted into the compounds 29 with the corresponding nucelphiles (Scheme 13). ##STR17##

In addition, the halides 28 can be converted by free radical reaction to the dihalide 30 and then converted with H₂ O/MeOH in the presence of AgNO₃ into the carbonyl compound 31 or reacted directly with N-methylmorpholine N-oxide to give the carbonyl compound 11. Furthermore, the phosphonates, phosphonium salts or phosphine oxides 32 (P is the particular organophosphorus radical) are obtainable from the halides 8 (Scheme 14). ##STR18##

The carbonyl compounds 31 can then be reacted with the corresponding hydroxylamines to give the oximes 33 or can be subjected to a Wittig reaction to give the olefins 34, The olefins 34 are also obtainable by a Wittig reaction starting from the phosphonates, phosphonium salts or phosphine oxides 32 (Scheme 15). ##STR19##

The saturated compounds 35 can be prepared from the olefins 34 by reduction or, where R² and R³ are each H, the acetylenes 36 can be prepared from said olef ins by halogen addition (Hal=Cl, Br or I) and subsequent two-fold elimination of hydrogen halide (Scheme 16). ##STR20##

Alternatively, the ureas 39 can be synthesized by acylation of the hydroxylamines 22 to the compounds 37, subsequent alkylation or acylation to the compounds 38 and substitution of the nucleofugic leaving group V (V is, for example, OCH₃, OCCl₃, CCl₃, O-phenyl or O-p-nitrophenyl) by NH₃, H₂ N--CH₃ or HN(CH₃)₂ (Scheme 17). ##STR21##

Alternatively, ureas of the formula 39 can also be obtained by alkylating ureas of the formula 41, which in turn are obtainable from 17 by reacting 17 with the corresponding amines, or directly from 22 by aminocarbonylation (for example with dimethylcarbamoyl chloride or methyl isocyanate) (cf. for example Houben-Weyl, volume E16a, page 208).

Furthermore, ureas of the formula 39 can also be obtained from the N-aryl-O-alkylhydroxylamines of the formula 42 in a similar manner by aminocarbonylation.

The compounds of the formula 42 are in turn obtainable by methods known from the literature, from hydroxylamines of the formula 2 (cf. for example Houben-Weyl, volume E16a, pages 271 and 282-289).

In addition, the hydroxylamines 22 are obtainable from the anilines 43 by formation of the imines 44, oxidation of the compounds 44 with the m-chloroperbenzoic acid and reaction of the oxaziridines 45 with hydroxylamine (Scheme 18; similarly to G. Grundke et al., Synthesis 1987, 1115). ##STR22##

The Examples which follow illustrate the preparation of the novel compounds.

EXAMPLES Example 1

Methyl N-ethyl-N-(2-(2'-methylphenoxymethyl)-phenyl)-carbamate (Table 7, No. 2)

a) Methyl N-(o-methylphenyl)-carbamate 50 g (0.53 mol) of methyl chloroformate are added dropwise to 53 g (0.5 mol) of o-toluidene in 500 ml of methylene chloride. During this procedure, the reaction solution heats up to the boiling point and a colorless solid is precipitated.

Stirring is carried out for one hour, after which 200 ml of 10% strength sodium hydroxide solution are added dropwise, the colorless solid going into solution. The organic phase is dried over MgSO₄ and evaporated down under reduced pressure. The remaining solid is stirred with n-hexane and filtered off under suction. 84 g (0.5 mol, quantitative yield) of the title compound are obtained as a colorless solid.

mp.=61°-62° C.; ¹ H-NMR (DMSO-d₆ ; δ (PPm)): 8.85 (s, 1H, NH); 7.35 (d, broad, 1H, aromatic); 7.1 (m, 3H, aromatic); 3.6 (s, 3H, OCH₃); 2.2 (s, 3H, CH₃)

b) Methyl N-ethyl-N-(o-methylphenyl)-carbamate

5.1 g (0.2 mol) of sodium hydride are added a little at a time to 30 g (0.18 mol) of methyl N-(o-methylphenyl)-carbamate (Example 1a) in 200 ml of dimethylformamide. After the evolution of gas has ceased, 30 g (0.2 mol) of ethyl iodide are added drop-wise, the reaction mixture being lightly cooled in a water bath. A white solid is precipitated. After about 4 hours, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is dried over MgSO₄ and evaporated down. The residue is distilled. 32.5 g (0.17 mol=93%) of the title compound are obtained as a colorless oil. bp.⁰.5 =74° C.; ¹ H-NMR (CDCl₃ ; δ (ppm): 7.2 (m, 3H, aromatic); 7.1 (m, 1H, aromatic); 3.8 (m, 1H, N--CH_(A)); 3.6 (s, 3H, OCH₃); 3.5 (m, 1H, N--CH_(B)); 2.2 (s, 3H, CH₃); 1.1 (t, 3H, CH₃)

c) Methyl N-ethyl-N-(o-bromomethylphenyl)-carbamate

A mixture of 30 g (0.155 mol) of methyl N-ethyl-N-(o-methylphenyl)-carbamate (Example 1b), 33 g (0.185 mol) of N-bromosuccinimide and 0.1 g of azoisobutyronitrile in 300 ml of carbon tetrachloride is exposed to a 300 W UV lamp for 6 hours. During this procedure, the contents of the flask heat up to about 70° C. Thereafter, the reaction mixture is washed four times with water, dried and evaporated down. The residue obtained comprises 41 g of a brown oil which contains the title compound in about 50% purity and is used without further purification in the next reaction.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.2 (m, 4H, aromatic); 4.45 (s, 2H, CH₂ --Br); 3.8 (m, 1H, N--CH_(A)); 3.6 (s, 3H, OCH₃); 3.5 (m, 1H, N--CH_(B)); 1.15 (t, 3H, J=8 Hz, CH₃)

d) Methyl N-ethyl-N-(2-(2'-methylphenoxymethyl)-phenyl)-carbamate (Table 7, No. 2)

2.4 g (17 mmol) of sodium hydride are added a little at a time to 8.6 g (80 mmol) of o-cresol in 100 ml of dimethylformamide. Stirring is carried out for 30 minutes at room temperature (20° C.), after which 20.5 g of methylN-ethyl-N-(o-bromomethylphenyl)-carbamate (Example 1c, about 50% purity, about 37 mmol) are added. Stirring is carried out overnight at room temperature, after which the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The combined ether phases are dried over MgSO₄ and evaporated down. The residue is distilled in a kugelrohr (bulb tube) apparatus. 10 g of a yellow oil are obtained at 220° C. and 0.2 mbar, and the oil is then purified by chromatography with cyclohexane/ethyl acetate mixtures over silica gel and then over alumina. The product thus obtained is purified again by kugelrohr distillation. 3.6 g (12 mmol=32%) of the title compound are obtained as a colorless oil.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.6 (m, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (dd, broad, 2H, O--CH₂); 3.8 (m, 1H, N--CH_(A)); 3.6 (s, 3H, O--CH₃); 3.5 (m, 1H, N--CH_(B)); 2.3 (s, 3H, CH₃); 1.15 (t, 3H, J=8 Hz, CH₃)

Example 2

Methyl N- 2-(2'-methylphenoxymethyl)-phenyl!-N-methyl-thiocarbamate (Table 7, No. 89)

a) 2-(2'-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide are stirred for 5 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and filtered off under suction. 73 g (0.300 mol=88%) of the title compound are obtained as a colorless solid.

mp.=83° C.; ¹ H-NMR (CDCl₃ ; δ (ppm)): 8.15 (d, 1H, J=8 Hz, aromatic); 7.95 (d, 1H, J=8 Hz, aromatic); 7.7 (t, 1H, J=8 Hz, aromatic); 7.45 (t, 1H, J=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O--CH₂); 2.35 (s, 3H, CH₃)

b) 2-(2'-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2'-methylphenoxymethyl)-nitrobenzene (Example 2a) and 10 g of 5% strength Pt/C (platinum adsorbed onto active carbon) in 50 ml of methanol are stirred vigorously for two hours under an H₂ atmosphere. Thereafter, a further 2 g of 5% strength Pt/C are added and stirring is continued overnight. The catalyst is then filtered off under suction and is replaced with 10 g of fresh catalyst. Stirring is continued overnight, the mixture is filtered under suction and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography using hexane/ethyl acetate mixtures. 61 g (0.286 mol=93%) of the title compound are obtained as a colorless solid.

mp.=56° C.; ¹ H-NMR (CDCl₃ ; δ (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, J=8 Hz, aromatic); 6.9 (t, 1H, J=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O--CH₂); 4.05 (s, broad, 2H, NH₂); 2.2 (s, 3H, CH₃)

c) Methyl N- 2-(2'-methylphenoxymethyl)-phenyl!-carbamate (Table 7, No. 3)

6 g (63 mmol) of methyl chloroformate are added dropwise to 10 g (47 mmol) of 2-(2'-methylphenoxymethyl)-aniline in 500 of methylene chloride at 20°-30° C. Stirring is carried out for 3 hours at room temperature, a white solid being precipitated, and the reaction mixture is then stirred with 20 ml of 10% strength sodium hydroxide solution. The organic phase is filtered off under suction over silica gel, the filtrate is evaporated down and the remaining residue is stirred thoroughly with methanol and filtered under suction. 10.5 g (39 mmol=82%) of the title compound are obtained as a colorless solid.

mp.=111° C.; ¹ H-NMR (CDCl₃ ; δ (ppm)): 8.0 (d, broad, 1H, aromatic); 7.7 (s, broad, 1H, aromatic); 7.7 (s, broad, 1H, NH); 6.8-7.5 (m, 6H, aromatic); 5.0 (s, 2H, O--CH₂); 3.75 (s, 3H, O--CH₃); 2.25 (s, 3H, CH₃)

d) Methyl N- 2-(2'-methylphenoxymethyl)-phenyl!-N-methylthiocarbamate (Table 7, No. 89)

0.5 g (20.8 mmol) of sodium hydride is added a little at a time to 4.9 g (17.3 mmol) of methyl N- 2-(2'-methylphenoxymethyl)!-phenylcarbamate (Example 2c) in 80 ml of toluene. After the end of gas evolution, 2.4 g (19 mmol) of methyl methanethiosulfonate are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is extracted with water, dried over MgSO₄ and evaporated down under reduced pressure. The residue is purified by column chromatography with hexane/ethyl acetate mixtures over silica gel. 3 g (9.1 mmol=53%) of the title compound are obtained as a yellow oil.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.65 (d, broad, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (m, 2H, O--CH₂); 3.75 (s, 3H, O--CH₃); 2.55 (s, 3H, S--CH₃); 2.3 (s, 3H, CH₃)

Example 3

Methyl N-allyl-N- 2-(3"-bromophenylmethyliminoxymethyl)-phenyl!-carbamate (Table 7, No. 91)

a) o-Methoxymethylnitrobenzene

125 g of 30% strength sodium methylate solution (0.69 mol) in methanol are added dropwise to 130 g (0.6 mol) of o-nitrobenzyl bromide in 200 ml of methanol. During this procedure, the reaction mixture heats up to about 50° C. Stirring is continued for a further 3 hours, the reaction mixture being cooled to room temperature, after which ice water is added to the reaction vessel and the reaction mixture is neutralized by adding dilute hydrochloric acid. The aqueous phase is extracted with three times with ether, and the organic phase is dried over MgSO₄ and evaporated down. 101 g (0.6 mol, quantitative yield) of the title compound are obtained as a residue in the form of a brownish oil. ¹ H-NMR (CDCl₃ ; δ (ppm)): 8.1 (d, broad, 1H, aromatic); 7.8 (d, broad, 1H, aromatic); 7.5 (t, broad, 1H, aromatic); 7.45 (t, broad, 1H, aromatic); 4.85 (s, 2H, O--CH₂); 3.5 (s, 3H, OCH₃)

b) Methyl N-(2-methoxymethylphenyl)-carbamate

528 g of 21.8% strength Na₂ Fe(CO)₄ ! solution (0.6 mol; 1 kg of the solution contains 633 g of water, 218 g of Na₂ Fe(CO)₄ !, 108 g of Na₂ CO₃ and 41 g of NaOH) are added dropwise to 101 g (0.6 mol) of o-methoxymethylnitrobenzene (Example 3a) in 1 l of methanol at 20°-30° C. Stirring is carried out for 1 hour at room temperature, after which the reaction mixture is diluted with ether. A brown oil separates out in the reaction vessel. The total reaction mixture is poured onto a silica gel column and is eluted with ether. Thereafter, the ether phase is evaporated, the residue is taken up in methylene chloride and the solution is dried over MgSO₄. It is filtered under suction over silica gel and the solvent is then evaporated off under reduced pressure. The residue is purified by column chromatography with hexane and methylene chloride. 83.8 g of o-methoxymethylaniline are obtained as a brown oil, which is directly reacted further.

The resulting crude product is dissolved in 700 ml of methylene chloride, 62.4 g (0.66 mol) of methyl chloroformate are added and 52.2 g (0.66 mol) of pyridine are then added dropwise. Stirring is carried out overnight at room temperature and the reaction mixture is then extracted with dilute hydrochloric acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with hexane/ethyl acetate mixtures. 89.4 g (0.41 mol=69%, based on 2-methoxymethylnitrobenzene) of the title compound are obtained as a yellow oil in a purity of about 90%.

¹ H-NMR (CDCl₃ ; δ (ppm)): 8.0 (m, 2H, 1× aromatic, NH); 7.35 (t, broad, 1H, aromatic); 7.15 (d, broad, 1H, aromatic); 7.0 (t, broad, 1H, aromatic); 4.5 (s, 2H, OCH₂); 3.8 (s, broad, 3H, OCH₃); 3.4 (s, broad, 3H, OCH₃)

c) Methyl N-(2-bromomethylphenyl)-carbamate

38.6 g (150 mmol) of boron tribromide are added dropwise to 10 g (51 mmol) of methyl N-(2-methoxymethylphenyl)-carbamate (Example 2b) in 100 ml of methylene chloride. Stirring is carried out for 2 hours, after which the vigorously stirred reaction mixture is added dropwise to a solution of 11.8 g (0.17 mol) of NaHCO₃ in water. The organic phase is separated off and the aqueous phase is extracted once with methylene chloride and once with ethyl acetate. The combined organic phases are dried over MgSO₄ and evaporated down. 9.5 g (39 mmol=76%) of the title compound are obtained as a colorless solid.

mp.=132° C.; ¹ H-NMR (CDCl₃ ; δ (ppm)): 7.85 (d, broad, 1H, aromatic); 7.3 (m, 2H, aromatic); 7.1 (t, broad, 1H, aromatic); 6.9 (s, broad, 1H, NH); 4.5 (s, 2H, CH₂ --Br); 3.8 (s, 3H, OCH₃)

d) Methyl N- 2-(3"-bromophenylmethyliminoxymethyl)-phenyl!-carbamate (Table 7, No. 88)

0.95 g (39 mmol) of sodium hydride is added a little at a time to 7 g (33 mmol) of m-bromoacetophenone oxime in 100 ml of dimethylformamide. When the evolution of gas has ended, 8 g (33 mmol) of methyl N-(2-bromomethylphenyl)-carbamate (Example 3c), dissolved in 10 ml of dimethylformamide, are added dropwise. Stirring is carried out for 3 hours at room temperature, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is washed three times with water, dried and evaporated down. The residue crystallizes and is stirred thoroughly with methanol. 5.1 g (13.5 mmol=41%) of the title compound are obtained as a colorless solid.

mp.=124°-125° C.; ¹ H-NMR (CDCl₃ ; δ (ppm)): 8.6 (s, broad, 1H, NH); 7.8-8.1 (m, 2H, aromatic); 7-7.6 (m, 6H, aromatic); 5.2 (s, 2H, O--CH₂); 3.8 (s, 3H, O--CH₃); 2.2 (s, 3H, CH₃)

e) Methyl N-allyl-N- 2-(3"-bromophenylmethyliminoxy-methyl)-phenyl!-carbamate (Table 7, No. 91)

0.1 g (4.1 mmol) of sodium hydride is added a little at a time to 1.3 g (3.5 mmol) of methyl N- 2-(3"-bromophenylmethyliminoxymethyl)-phenyl!-carbamate (Example 3d) in 20 ml of dimethylformamide. After gas evolution has ended, 0.5 g (3.8 mmol) of allyl bromide are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is diluted with water and extracted three times with ether. The combined ether phases are washed three times with water, dried over MgSO₄ and evaporated down. 1.5 g (quantitative yield) of the title compound are obtained as a residue in the form of a yellow oil.

¹ H-NMR (CDCl₃ ; δ (ppm)): 7.8 (s, broad, 1H, aromatic); 7.1-7.6 (m, 7H, aromatic); 6.0 (m, 1H, C--CH═C); 5.1 (m, 4H, O--CH2 and C═CH2); 4.4 (m, 1H, N--CH_(A)); 4.0 (m, 1H, N--CH_(B)) 3.6-3.8 (2s, broad, O--CH₃); 2.2 (S, 3H, CH₃)

The compounds described in the Tables below can be prepared in a similar manner.

                  TABLE 1                                                          ______________________________________                                          ##STR23##                                                                     I: R.sup.1 = H                                                                 II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = SCH.sub.3                                                         VI: R.sup.1 = CH.sub.2 CN                                                      VII: R.sup.1 = CH.sub.2 OCH.sub.3                                              VIII: R.sup.1 = COOCH.sub.3                                                    No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-C-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    181     3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    182     4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-CH.sub.3 CH.sub.2 CO                                            304     2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                   305     2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                         306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-CH.sub.3 CO                                            308     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   309     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          310     2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                311     2-Cl-4-CHO                                                             312     2-Cl-4-CH.sub.3 CO                                                     313     2-Cl-4-CH.sub.3 CH.sub.2 CO                                            314     2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                         315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-CH.sub.3 CO                                            317     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   318     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          319     2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                   369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2, 5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                        375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                        381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)              9                                                                      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CN-C-Allyl)                           649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-C-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 2                                                          ______________________________________                                          ##STR24##                                                                     I: R.sup.1 = H                                                                 II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = SCH.sub.3                                                         VI: R.sup.1 = CH.sub.2 CN                                                      VII: R.sup.1 = CH.sub.2 CCH.sub.3                                              VIII: R.sup.1 = COOCH.sub.3                                                    No.        B                                                                   ______________________________________                                          1         Pyrrolyl-3                                                           2         NCH.sub.3 -Pyrrolyl-3                                                3         NC.sub.6 H.sub.5 -Pyrrolyl-3                                         4         N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           5         N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           6         N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           7         N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          8         N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          9         N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          10        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           11        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           12        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           13        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  14        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  15        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  16        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  17        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  18        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  19        Pyrrolyl-2                                                           20        NCH.sub.3 -Pyrrolyl-2                                                21        NC.sub.6 H.sub.5 -Pyrrolyl-2                                         22        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           23        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           24        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           25        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          26        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          27        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          28        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           29        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           30        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           31        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  32        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  33        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  34        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  35        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  36        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  37        Furyl-2                                                              38        5-CH.sub.3 -Furyl-2                                                  39        5-C.sub.6 H.sub.5 -Furyl-2                                           40        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              41        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              42        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              43        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             44        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             45        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             46        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              47        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              48        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              49        5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     50        5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     51        5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     52        5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     53        5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     54        5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     55        4-CH.sub.3 -Furyl-2                                                  56        4-C.sub.6 H.sub.5 -Furyl-2                                           57        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              58        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              59        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              60        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             61        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             62        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             63        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              64        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              65        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              66        4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     67        4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     68        4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     69        4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     70        4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     71        4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     72        Thienyl-2                                                            73        5-CH.sub.3 -Thienyl-2                                                74        5-C.sub.6 H.sub.5 -Thienyl-2                                         75        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            76        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            77        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            78        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           79        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           80        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           81        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            82        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            83        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            84        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   85        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   86        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   87        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   88        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   89        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   90        4-CH.sub.3 -Thienyl-2                                                91        4-C.sub.6 H.sub.5 -Thienyl-2                                         92        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            93        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            94        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            95        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           96        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           97        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           98        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            99        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                           100        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                           101        4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                  102        4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                  103        4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                  104        4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                  105        4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                  106        4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                  107        Thienyl-3                                                           108        5-CH.sub.3 -Thienyl-3                                               109        5-C.sub.6 H.sub.5 -Thienyl-3                                        110        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           111        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           112        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           113        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          114        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          115        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          116        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           117        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           118        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           119        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                  120        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                  121        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                  122        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                  i23        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                  i24        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                  125        Pyrazolyl-4                                                         126        NCH.sub.3 -Pyrazolyl-4                                              127        NC.sub.6 H.sub.5 -Pyrazolyl-4                                       128        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         129        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         130        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         131        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        132        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        133        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        134        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         135        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         136        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         137        N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                138        N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                139        N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                140        N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                141        N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                142        N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                143        3-CH.sub.3 N-Methylpyrazolyl-4                                      144        3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                               145        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 146        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 147        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 148        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                149        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                150        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                151        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 152        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 153        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 154        3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                        155        3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                        156        3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                        157        3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                        158        3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                        159        3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                        160        Isoxazolyl-5                                                        161        3-CH.sub.3 -Isoxazolyl-5                                            162        3-C.sub.6 H.sub.5 -Isoxazolyl-5                                     163        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        164        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        165        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        166        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       167        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       168        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       169        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        170        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        171        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        172        3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               173        3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               174        3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               175        3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               176        3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               177        3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               178        4-Chloroisoxazolyl-5                                                179        3-CH.sub.3 -4-Chloroisoxazolyl-5                                    180        3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                             181        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                182        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                183        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                184        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               185        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               186        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               187        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                188        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                189        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                190        3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       191        3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       192        3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       193        3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       194        3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       195        3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       196        Isoxazolyl-3                                                        197        5-CH.sub.3 -Isoxazolyl-3                                            198        5-C.sub.6 H.sub.5 -Isoxazolyl-3                                     199        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        200        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        201        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        202        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       203        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       204        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       205        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        206        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        207        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        208        5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               209        5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               210        5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               211        5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               212        5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               213        5 (2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               214        Isothiazolyl-5                                                      215        3-CH.sub.3 -Isothiazolyl-5                                          216        3-C.sub.6 H.sub.5 -Isothiazolyl-5                                   217        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      218        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      219        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      220        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     221        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     222        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     223        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      224        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      225        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      226        3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             227        3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             228        3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             229        3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             230        3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             231        3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             232        Oxazolyl-4                                                          233        3-CH.sub.3 -Oxazolyl-4                                              234        3-C.sub.6 H.sub.5 -Oxazolyl-4                                       235        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          236        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          237        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          238        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         239        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         240        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         241        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          242        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          243        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          244        3-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 245        3-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 246        3-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 247        3-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 248        3-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 249        3-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 250        Thiazolyl-4                                                         251        2-CH.sub.3 -Thiazolyl-4                                             252        2-C.sub.6 H.sub.5 -Thiazolyl-4                                      253        2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         254        2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         255        2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         256        2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         267        2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                        258        2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                        259        2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         260        2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         261        2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         262        2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                263        2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                264        2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                265        2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 66        2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                267        2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                268        NCH.sub.3 -1,2,4-Triazolyl-5                                        269        3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                             270        3-C.sub.6 H.sub.5 -NCH.sub.3 -1,2,4-Triazolyl-5                     271        3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         272        3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         273        3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         274        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        275        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        276        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        277        3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         278        3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         279        3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         280        3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                281        3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                282        3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                283        3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                284        3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                285        3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                286        1,3,4-Oxadiazolyl-2                                                 287        5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                     288        5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                              289        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 290        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 291        S-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 292        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                293        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                294        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                295        S-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 296        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 297        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 298        5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        299        5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        300        5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        301        5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        302        5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        303        5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        304        1,2,4-Oxadiazolyl-3                                                 305        5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                     306        5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                              307        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 308        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 309        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 310        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                311        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                312        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                313        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 314        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 315        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 316        5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        317        5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        318        5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        319        5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        320        5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        321        5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        322        1,2,4-Oxadiazolyl-5                                                 323        3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                     324        3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                              325        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 326        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 327        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 328        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                329        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                330        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-cxadiazolyl-5                331        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 332        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 333        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 334        3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        335        3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        336        3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        337        3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        338        3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        339        3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        340        1,2,4-Thiadiazolyl-3                                                341        5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                    342        5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                             343        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                344        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                345        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                346        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               347        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               348        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               349        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                350        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                351        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                352        5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       353        5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       354        5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       355        5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       356        5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       357        5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       358        1,3,4-Thiadiazolyl-2                                                359        5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                    360        5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                             361        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                362        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                363        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                364        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               365        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               366        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               367        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazollyl-2               368        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                369        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                370        5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       371        5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       372        5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       373        5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       374        5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       375        5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       376        Pyridinyl-2                                                         377        Pyridinyl-4                                                         378        Pyridazinyl-3                                                       379        Pyridazinyl-4                                                       380        Pyridazinyl-2                                                       381        Pyrimidinyl-4                                                       382        Pyrimidinyl-5                                                       383        Pyrimidinyl-2                                                       384        1-Naphthyl                                                          385        2-Naphthyl                                                          ______________________________________                                    

                  TABLE 3                                                          ______________________________________                                          ##STR25##                                                                     I: R.sup.1 = H                                                                 II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = SCH.sub.3                                                         VI: R.sup.1 = CH.sub.2 CN                                                      VII: R.sup.1 = CH.sub.2 OCH.sub.3                                              VIII: R.sup.1 = COOCH.sub.3                                                    No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   181     3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   182     4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 C(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-CH.sub.3 CH.sub.2 CO                                            304     2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                   305     2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                         306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-CH.sub.3 CO                                            308     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   309     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          310     2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                311     2-Cl-4-CHO                                                             312     2-Cl-4-CH.sub.3 CO                                                     313     2-Cl-4-CH.sub.3 CH.sub.2 CO                                            314     2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                         315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-CH.sub.3 CO                                            317     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   318     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          319     2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NCC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NCC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NC-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NC-CH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                  369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3)2-4-(CH.sub.3 CNOCH.sub.3)                               375     2,5-(CH.sub.3)2-4-(CH.sub.3 CNOC.sub.2 H.sub.5)                        376     2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                     377     2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                     378     2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-Allyl)                                 379     2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-trans-Chloroallyl)                     380     2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-Proparyl)                              381     2,5-(CH.sub.3)2-4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                     382     2,5-(CH.sub.3)2-4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)               383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAl1yl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-C-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-C-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazo1yl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)              1                                                                      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-C-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-C-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 4                                                          ______________________________________                                          ##STR26##                                                                     I: R.sup.1 = H                                                                 II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = SCH.sub.3                                                         VI: R.sup.1 = CH.sub.2 CN                                                      VII: R.sup.1 = CH.sub.2 OCH.sub.3                                              VIII: R.sup.1 = COOCH.sub.3                                                    No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                            2        N-CH.sub.3 -Pyrrolyl-3                                                3        N-C.sub.6 H.sub.5 -Pyrrolyl-3                                         4        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            5        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            6        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            7        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           8        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           9        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           10       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            11       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            12       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            13       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   14       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   15       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   16       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   17       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   18       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   19       Pyrrolyl-2                                                            20       N-CH.sub.3 -Pyrrolyl-2                                                21       N-C.sub.6 H.sub.5 -Pyrrolyl-2                                         22       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            23       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            24       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            25       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           26       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           27       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           28       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            29       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            30       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            31       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   32       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   33       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   34       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   35       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   36       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   37       Furyl-2                                                               38       5-CH.sub.3 -Furyl-2                                                   39       5-C.sub.6 H.sub.5 -Furyl-2                                            40       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               41       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               42       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               43       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              44       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              45       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              46       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               47       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               48       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               49       5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      50       5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      51       5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      52       5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      53       5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      54       5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      55       4-CH.sub.3 -Furyl-2                                                   56       4-C.sub.6 H.sub.5 -Furyl-2                                            57       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               58       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               59       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               60       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              61       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              62       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              63       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               64       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               65       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               66       4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      67       4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      68       4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      69       4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      70       4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      71       4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      72       Thienyl-2                                                             73       5-CH.sub.3 -Thienyl-2                                                 74       5-C.sub.6 H.sub.5 -Thienyl-2                                          75       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             76       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             77       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             78       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            79       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            80       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            81       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             82       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             83       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             84       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    85       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    86       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    87       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    88       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    89       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    90       4-CH.sub.3 -Thienyl-2                                                 91       4-C.sub.6 H.sub.5 -Thienyl-2                                          92       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             93       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             94       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             95       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            96       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            97       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            98       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             99       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thieny1-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       NCH.sub.3 -Pyrazolyl-4                                               127       NC.sub.6 H.sub.5 -Pyrazolyl-4                                        128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-PyrazOlyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyraz6lyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 143       3-CH.sub.3 -N-Methylpyrazolyl-4                                      144       3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4                               145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   154       3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          155       3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          156       3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          157       3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          158       3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          159       3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          160       Isoxazolyl-5                                                         161       3-CH.sub.3 -Isoxazolyl-5                                             162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 -Isoxazolyl-3                                             198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 -Isothiazolyl-5                                           216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isbthiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       2-CH.sub.3 -Oxazolyl-4                                               234       2-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           236       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           237       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           238       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          239       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          241       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           242       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           243       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           244       2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  245       2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  246       2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  247       2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  248       2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  249       2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       NCH.sub.3 -1,2,4-Triazolyl-5                                         269       3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                              270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          280       3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 281       3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 282       3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 283       3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 284       3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 285       3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-Cl-C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-3                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-3                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-3                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        384       1-Naphthyl                                                           385       2-Naphthyl                                                           ______________________________________                                    

                  TABLE 5                                                          ______________________________________                                          ##STR27##                                                                     I: R.sup.1 = H                                                                 II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = SCH.sub.3                                                         VI: R.sup.1 = CH.sub.2 CN                                                      VII: R.sup.1 = CH.sub.2 OCH.sub.3                                              VIII: R.sup.1 = COOCH.sub.3                                                    No.       X.sub.m                                                              ______________________________________                                          1        H                                                                     2        2-F                                                                   3        3-F                                                                   4        4-F                                                                   5        2,4-F.sub.2                                                           6        2,4,6-F.sub.3                                                         7        2,3,4,5,6-F.sub.5                                                     8        2,3-F.sub.2                                                           9        2-Cl                                                                  10       3-Cl                                                                  11       4-Cl                                                                  12       2,3-Cl.sub.2                                                          13       2,4-Cl.sub.2                                                          14       2,5-Cl.sub.2                                                          15       2,6-Cl.sub.2                                                          16       3,4-Cl.sub.2                                                          17       3,5-Cl.sub.2                                                          18       2,3,4-Cl.sub.3                                                        19       2,3,5-Cl.sub.3                                                        20       2,3,6-Cl.sub.3                                                        21       2,4,5-Cl.sub.3                                                        22       2,4,6-Cl.sub.3                                                        23       3,4,5-Cl.sub.3                                                        24       2,3,4,6-Cl.sub.4                                                      25       2,3,5,6-Cl.sub.4                                                      26       2,3,4,5,6-Cl.sub.5                                                    27       2-Br                                                                  28       3-Br                                                                  29       4-Br                                                                  30       2,4-Br.sub.2                                                          31       2,5-Br.sub.2                                                          32       2,6-Br.sub.2                                                          33       2,4,6-Br.sub.3                                                        34       2,3,4,5,6-Br.sub.5                                                    35       2-I                                                                   36       3-I                                                                   37       4-I                                                                   38       2,4-I.sub.2                                                           39       2-Cl, 3-F                                                             40       2-Cl, 4-F                                                             41       2-Cl, 5-F                                                             42       2-Cl, 6-F                                                             43       2-Cl, 3-Br                                                            44       2-Cl, 4-Br                                                            45       2-Cl, 5-Br                                                            46       2-Cl, 6-Br                                                            47       2-Br, 3-Cl                                                            48       2-Br, 4-Cl                                                            49       2-Br, 5-Cl                                                            50       2-Br, 3-F                                                             51       2-Br, 4-F                                                             52       2-Br, 5-F                                                             53       2-Br, 6-F                                                             54       2-F, 3-Cl                                                             55       2-F, 4-Cl                                                             56       2-F, 5-Cl                                                             57       3-Cl, 4-F                                                             58       3-Cl, 5-F                                                             59       3-Cl, 4-Br                                                            60       3-Cl, 5-Br                                                            61       3-F, 4-Cl                                                             62       3-F, 4-Br                                                             63       3-Br, 4-Cl                                                            64       3-Br, 4-F                                                             65       2,6-Cl.sub.2, 4-Br                                                    66       2-CH.sub.3                                                            67       3-CH.sub.3                                                            68       4-CH.sub.3                                                            69       2,3-(CH.sub.3).sub.2                                                  70       2,4-(CH.sub.3).sub.2                                                  71       2,5-(CH.sub.3).sub.2                                                  72       2,6-(CH.sub.3).sub.2                                                  73       3,4-(CH.sub.3).sub.2                                                  74       3,5-(CH.sub.3).sub.2                                                  75       2,3,5-(CH.sub.3).sub.3                                                76       2,3,4-(CH.sub.3).sub.3                                                77       2,3,6-(CH.sub.3).sub.3                                                78       2,4,5-(CH.sub.3).sub.3                                                79       2,4,6-(CH.sub.3).sub.3                                                80       3,4,5-(CH.sub.3).sub.3                                                81       2,3,4,6-(CH.sub.3).sub.4                                              82       2,3,5,6-(CH.sub.3).sub.4                                              83       2,3,4,5,6-(CH.sub.3).sub.5                                            84       2-C.sub.2 H.sub.5                                                     85       3-C.sub.2 H.sub.5                                                     86       4-C.sub.2 H.sub.5                                                     87       2,4-(C.sub.2 H.sub.5).sub.2                                           88       2,6-(C.sub.2 H.sub.5).sub.2                                           89       3,5-(C.sub.2 H.sub.5).sub.2                                           90       2,4,6-(C.sub.2 H.sub.5).sub.3                                         91       2-n-C.sub.3 H.sub.7                                                   92       3-n-C.sub.3 H.sub.7                                                   93       4-n-C.sub.3 H.sub.7                                                   94       2-i-C.sub.3 H.sub.7                                                   95       3-i-C.sub.3 H.sub.7                                                   96       4-i-C.sub.3 H.sub.7                                                   97       2,4-(i-C.sub.3 H.sub.7).sub.2                                         98       2,6-(i-C.sub.3 H.sub.7).sub.2                                         99       3,5-(i-C.sub.3 H.sub.7).sub.2                                        100       2,4,6-(i-C.sub.3 H.sub.7).sub.3                                      101       2-s-C.sub.4 H.sub.9                                                  102       3-s-C.sub.4 H.sub.9                                                  103       4-s-C.sub.4 H.sub.9                                                  104       2-t-C.sub.4 H.sub.9                                                  105       3-t-C.sub.4 H.sub.9                                                  106       4-t-C.sub.4 H.sub.9                                                  107       2,3-(t-C.sub.4 H.sub.9).sub.2                                        108       2,4-(t-C.sub.4 H.sub.9).sub.2                                        109       2,5-(t-C.sub.4 H.sub.9).sub.2                                        110       2,6-(t-C.sub.4 H.sub.9).sub.2                                        111       3,4-(t-C.sub.4 H.sub.9).sub.2                                        112       2,4,6-(t-C.sub.4 H.sub.9).sub.3                                      113       4-n-C.sub.9 H.sub.19                                                 114       4-n-C.sub.12 H.sub.25                                                115       4-n-C.sub.15 H.sub.31                                                116       4-(1,1,3,3-Tetramethylbutyl)                                         117       4-(2,4,4-Trimethylpropyl)                                            118       2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                      119       2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                      120       2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                            121       2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                      122       2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                      123       2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                      124       2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                      125       3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                      126       2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                      127       2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                   128       2-Allyl                                                              129       3-Allyl                                                              130       4-Allyl                                                              131       2-Allyl, 6-CH.sub.3                                                  132       2-cyclo-C.sub.6 H.sub.11                                             133       3-cyclo-C.sub.6 H.sub.11                                             134       4-cyclo-C.sub.6 H.sub.11                                             135       2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                       136       2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                 137       2-CH.sub.2 C.sub.6 H.sub.5                                           138       3-CH.sub.2 C.sub.6 H.sub.5                                           139       4-CH.sub.2 C.sub.6 H.sub.5                                           140       2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                               141       2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                               142       2-C.sub.6 H.sub.5                                                    143       3-C.sub.6 H.sub.5                                                    144       4-C.sub.6 H.sub.5                                                    145       4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                              146       4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                              147       2-Cl, 4-C.sub.6 H.sub.5                                              148       2-Br, 4-C.sub.6 H.sub.5                                              149       2-C.sub.6 H.sub.5, 4-Cl                                              150       2-C.sub.6 H.sub.5, 4-Br                                              151       2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                     152       2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                     153       2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                     154       2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                     155       2-cyclo-C.sub.6 H.sub.11, 4-Cl                                       156       2-cyclo-C.sub.6 H.sub.11, 4-Br                                       157       2-Cl, 4-cyclo-C.sub.6 H.sub.11                                       158       2-Br, 4-cyclo-C.sub.6 H.sub.11                                       159       2-OCH.sub.3                                                          160       3-OCH.sub.3                                                          161       4-OCH.sub.3                                                          162       2-OC.sub.2 H.sub.5                                                   163       3-OC.sub.2 H.sub.5                                                   164       4-OC.sub.2 H.sub.5                                                   165       2-O-n-C.sub.3 H.sub.7                                                166       3-O-n-C.sub.3 H.sub.7                                                167       4-O-n-C.sub.3 H.sub.7                                                168       2-O-i-C.sub.3 H.sub.7                                                169       3-O-i-C.sub.3 H.sub.7                                                170       4-O-i-C.sub.3 H.sub.7                                                171       2-O-n-C.sub.6 H.sub.13                                               172       3-O-n-C.sub.6 H.sub.13                                               173       4-O-n-C.sub.6 H.sub.13                                               174       2-O-n-C.sub.8 H.sub.17                                               175       3-O-n-C.sub.8 H.sub.17                                               176       4-O-n-C.sub.8 H.sub.17                                               177       2-OCH.sub.2 C.sub.6 H.sub.5                                          178       3-OCH.sub.2 C.sub.6 H.sub.5                                          179       4-OCH.sub.2 C.sub.6 H.sub.5                                          180       2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                 181       3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                 182       4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                 183       2,4-(OCH.sub.3).sub.2                                                184       2-CF.sub.3                                                           185       3-CF.sub.3                                                           186       4-CF.sub.3                                                           187       2-OCF.sub.3                                                          188       3-OCF.sub.3                                                          189       4-OCF.sub.3                                                          190       3-OCH.sub.2 CHF.sub.2                                                191       2-NO.sub.2                                                           192       3-NO.sub.2                                                           193       4-NO.sub.2                                                           194       2-CN                                                                 195       3-CN                                                                 196       4-CN                                                                 197       2-CH.sub.3, 3-Cl                                                     198       2-CH.sub.3, 4-Cl                                                     199       2-CH.sub.3, 5-Cl                                                     200       2-CH.sub.3, 6-Cl                                                     201       2-CH.sub.3, 3-F                                                      202       2-CH.sub.3, 4-F                                                      203       2-CH.sub.3, 5-F                                                      204       2-CH.sub.3, 6-F                                                      205       2-CH.sub.3, 3-Br                                                     206       2-CH.sub.3, 4-Br                                                     207       2-CH.sub.3, 5-Br                                                     208       2-CH.sub.3, 6-Br                                                     209       2-Cl, 3-CH.sub.3                                                     210       2-Cl, 4-CH.sub.3                                                     211       2-Cl, 5-CH.sub.3                                                     212       2-F, 3-CH.sub.3                                                      213       2-F, 4-CH.sub.3                                                      214       2-F, 5-CH.sub.3                                                      215       2-Br, 3-CH.sub.3                                                     216       2-Br, 4-CH.sub.3                                                     217       2-Br, 5-CH.sub.3                                                     218       3-CH.sub.3, 4-Cl                                                     219       3-CH.sub.3, 5-Cl                                                     220       3-CH.sub.3, 4-F                                                      221       3-CH.sub.3, 5-F                                                      222       3-CH.sub.3, 4-Br                                                     223       3-CH.sub.3, 5-Br                                                     224       3-F, 4-CH.sub.3                                                      225       3-Cl, 4-CH.sub.3                                                     226       3-Br, 4-CH.sub.3                                                     227       2-Cl, 4,5-(CH.sub.3).sub.2                                           228       2-Br, 4,5-(CH.sub.3).sub.2                                           229       2-Cl, 3,5-(CH.sub.3).sub.2                                           230       2-Br, 3,5-(CH.sub.3).sub.2                                           231       2,6-Cl.sub.2, 4-CH.sub.3                                             232       2,6-F.sub.2, 4-CH.sub.3                                              233       2,6-Br.sub.2, 4-CH.sub.3                                             234       2,4-Br.sub.2, 6-CH.sub.3                                             235       2,4-F.sub.2, 6-CH.sub.3                                              236       2,4-Br.sub.2, 6-CH.sub.3                                             237       2,6-(CH.sub.3).sub.2, 4-F                                            238       2,6-(CH.sub.3).sub.2, 4-Cl                                           239       2,6-(CH.sub.3).sub.2, 4-Br                                           240       3,5-(CH.sub.3).sub.2, 4-F                                            241       3,5-(CH.sub.3).sub.2, 4-Cl                                           242       3,5-(CH.sub.3).sub.2, 4-Br                                           243       2,3,6-(CH.sub.3).sub.3, 4-F                                          244       2,3,6-(CH.sub.3).sub.3, 4-Cl                                         245       2,3,6-(CH.sub.3).sub.3, 4-Br                                         246       2,4-(CH.sub.3).sub.2, 6-F                                            247       2,4-(CH.sub.3).sub.2, 6-Cl                                           248       2,4-(CH.sub.3).sub.2, 6-Br                                           249       2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                250       2-Cl, 4-NO.sub.2                                                     251       2-NO.sub.2, 4-Cl                                                     252       2-OCH.sub.3, 5-NO.sub.2                                              253       2,4-Cl.sub.2, 5-NO.sub.2                                             254       2,4-Cl.sub.2, 5-NO.sub.2                                             255       2,6-Cl.sub.2, 4-NO.sub.2                                             256       2,6-Br.sub.2, 4-NO.sub.2                                             257       2,6-I.sub.2, 4-NO.sub.2                                              258       2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                259       2-CO.sub.2 CH.sub.3                                                  260       3-CO.sub.2 CH.sub.3                                                  261       4-CO.sub.2 CH.sub.3                                                  262       2-CO.sub.2 (C.sub.2 H.sub.5)                                         263       3-CO.sub.2 (C.sub.2 H.sub.5)                                         264       4-CO.sub.2 (C.sub.2 H.sub.5)                                         265       2-CO.sub.2 (n-C.sub.3 H.sub.7)                                       266       3-CO.sub.2 (n-C.sub.3 H.sub.7)                                       267       4-CO.sub.2 (n-C.sub.3 H.sub.7)                                       268       2-CO.sub.2 (i-C.sub.3 H.sub.7)                                       269       3-CO.sub.2 (i-C.sub.3 H.sub.7)                                       270       4-CO.sub.2 (i-C.sub.3 H.sub.7)                                       271       2-CO.sub.2 (n-C.sub.6 H.sub.13)                                      272       3-CO.sub.2 (n-C.sub.6 H.sub.13)                                      273       4-CO.sub.2 (n-C.sub.6 H.sub.13)                                      274       2-CH.sub.2 OCH.sub.3                                                 275       3-CH.sub.2 OCH.sub.3                                                 276       4-CH.sub.2 OCH.sub.3                                                 277       2-CH.sub.2 O(C.sub.2 H.sub.5)                                        278       3-CH.sub.2 C(C.sub.2 H.sub.5)                                        279       4-CH.sub.2 O(C.sub.2 H.sub.5)                                        280       2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      281       3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      282       4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      283       2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      284       3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      285       4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      286       2-CHO                                                                287       3-CHO                                                                288       4-CHO                                                                289       2-COCH.sub.3                                                         290       3-COCH.sub.3                                                         291       4-COCH.sub.3                                                         292       2-COCH.sub.2 CH.sub.3                                                293       3-COCH.sub.2 CH.sub.3                                                294       4-COCH.sub.2 CH.sub.3                                                295       2-COCH.sub.2 CH.sub.2 CH.sub.3                                       296       3-COCH.sub.2 CH.sub.2 CH.sub.3                                       297       4-COCH.sub.2 CH.sub.2 CH.sub.3                                       298       2-COCH(CH.sub.3)CH.sub.3                                             299       3-COCH(CH.sub.3)CH.sub.3                                             300       4-COCH(CH.sub.3)CH.sub.3                                             301       2-Me-4-CHO                                                           302       2-Me-4-CH.sub.3 CO                                                   303       2-Me-4-CH.sub.3 CH.sub.2 CO                                          304       2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                 305       2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                       306       2,5-Me.sub.2 -4-CHO                                                  307       2,5-Me.sub.2 -4-CH.sub.3 CO                                          308       2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                 309       2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                        310       2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                              311       2-Cl-4-CHO                                                           312       2-Cl-4-CH.sub.3 CO                                                   313       2-Cl-4-CH.sub.3 CH.sub.2 CO                                          314       2-Cl-4-CH.sub.3 CH(CH.sub.3)OC                                       315       2,5-Cl.sub.2 -4-CHO                                                  316       2,5-Cl.sub.2 -4-CH.sub.3 CO                                          317       2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                 318       2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                        319       2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                              320       2-C(NOCH.sub.3)CH.sub.3                                              321       3-C(NOCH.sub.3)CH.sub.3                                              322       4-C(NOCH.sub.3)CH.sub.3                                              323       2-C(NOC.sub.2 H.sub.5)CH.sub.3                                       324       3-C(NOC.sub.2 H.sub.5)CH.sub.3                                       325       4-C(NOC.sub.2 H.sub.5)CH.sub.3                                       326       2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    327       3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    328       4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    329       2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    330       3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    331       4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    332       2-C(NO-Allyl)-CH.sub.3                                               333       3-C(NO-Allyl)-CH.sub.3                                               334       4-C(NO-Allyl)-CH.sub.3                                               335       2-C(NO-trans-Chloroallyl)-CH.sub.3                                   336       3-C(NO-trans-Chloroallyl)-CH.sub.3                                   337       4-C(NO-trans-Chloroallyl)-CH.sub.3                                   338       2-C(NO-Propargyl)-CH.sub.3                                           339       3-C(NO-Propargyl)-CH.sub.3                                           340       4-C(NO-Propargyl)-CH.sub.3                                           341       2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    342       3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    343       4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    344       2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              345       3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              346       4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              347       2-CH.sub.3 -4-CHNOCH.sub.3                                           348       2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                    349       2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                 350       2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                 351       2-CH.sub.3 -4-CHNO-Allyl                                             352       2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                               353       2-CH.sub.3 -4-CHNO-Propargyl                                         354       2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                 355       2-CH.sub.3 -4-CHNO-CH.sub.2 C.sub.6 H.sub.5                          356       2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                 357       2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                          358       2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                       359       2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                       360       2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                   361       2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                       362       2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                               363       2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                       364       2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                 365       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                          366       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                   367       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                368       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                 369       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                            370       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                371       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                        372       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                373       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-CH.sub.2 C.sub.6 H.sub.5)         374       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                       375       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                376       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)             377       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)             378       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                         379       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)             380       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                      381       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)             382       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-CH.sub.2 C.sub.6 H.sub.5)                6                                                                    383       2-C.sub.6 H.sub.5                                                    384       3-C.sub.6 H.sub.5                                                    385       4-C.sub.6 H.sub.5                                                    386       2-(2'-FC.sub.6 H.sub.4)                                              387       2-(3'-FC.sub.6 H.sub.4)                                              388       2-(4'-FC.sub.6 H.sub.4)                                              389       3-(2'-FC.sub.6 H.sub.4)                                              390       3-(3'-FC.sub.6 H.sub.4)                                              391       3-(4'-FC.sub.6 H.sub.4)                                              392       4-(2'-FC.sub.6 H.sub.4)                                              393       4-(3'-FC.sub.6 H.sub.4)                                              394       4-(4'-FC.sub.6 H.sub.4)                                              395       2-(2'-ClC.sub.6 H.sub.4)                                             396       2-(3'-ClC.sub.6 H.sub.4)                                             397       2-(4'-ClC.sub.6 H.sub.4)                                             398       3-(2'-ClC.sub.6 H.sub.4)                                             399       3-(3'-ClC.sub.6 H.sub.4)                                             400       3-(4'-ClC.sub.6 H.sub.4)                                             401       4-(2'-ClC.sub.6 H.sub.4)                                             402       4-(3'-ClC.sub.6 H.sub.4)                                             403       4-(4'-ClC.sub.6 H.sub.4)                                             405       2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      406       2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      407       2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      408       3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      409       3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      410       3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      411       4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      412       4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      413       4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      414       2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    415       2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    416       2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    417       3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    418       3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    419       3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    420       4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    421       4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    422       4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    423       2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         424       2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         425       2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         426       3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         427       3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         428       3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         429       4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         430       4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         431       4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         432       2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             433       2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             434       2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             435       3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             436       3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             437       3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             438       4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             439       4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             440       4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             441       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     442       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     443       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     444       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     445       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     446       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     447       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     448       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     449       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     450       2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      451       2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      452       2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      453       3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      454       3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      455       3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      456       4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      457       4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      458       4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      459       2-(2'-NCC.sub.6 H.sub.4)                                             460       2-(3'-NCC.sub.6 H.sub.4)                                             461       2-(4'-NCC.sub.6 H.sub.4)                                             462       3-(2'-NCC.sub.6 H.sub.4)                                             463       3-(3'-NCC.sub.6 H.sub.4)                                             464       3-(4'-NCC.sub.6 H.sub.4)                                             465       4-(2'-NCC.sub.6 H.sub.4)                                             466       4-(3'-NCC.sub.6 H.sub.4)                                             467       4-(4'-NCC.sub.6 H.sub.4)                                             468       2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      469       2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      470       2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      471       3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      472       3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      473       3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      474       4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      475       4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      476       4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      477       2-OC.sub.6 H.sub.5                                                   475       3-OC.sub.6 H.sub.5                                                   476       4-OC.sub.6 H.sub.5                                                   478       2-O-(2'-FC.sub.6 H.sub.4)                                            479       2-O-(3'-FC.sub.6 H.sub.4)                                            480       2-O-(4'-FC.sub.6 H.sub.4)                                            481       3-O-(2'-FC.sub.6 H.sub.4)                                            482       3-O-(3'-FC.sub.6 H.sub.4)                                            483       3-O-(4'-FC.sub.6 H.sub.4)                                            484       4-O-(2'-FC.sub.6 H.sub.4)                                            485       4-O-(3'-FC.sub.6 H.sub.4)                                            486       4-O-(4'-FC.sub.6 H.sub.4)                                            487       2-O-(2'-ClC.sub.6 H.sub.4)                                           488       2-O-(3'-ClC.sub.6 H.sub.4)                                           489       2-O-(4'-ClC.sub.6 H.sub.4)                                           490       3-O-(2'-ClC.sub.6 H.sub.4)                                           491       3-O-(3'-ClC.sub.6 H.sub.4)                                           492       3-O-(4'-ClC.sub.6 H.sub.4)                                           493       3-O-(4'-ClC.sub.6 H.sub.4)                                           494       4-O-(2'-ClC.sub.6 H.sub.4)                                           495       4-O-(3'-ClC.sub.6 H.sub.4)                                           496       4-O-(4'-ClC.sub.6 H.sub.4)                                           497       2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    498       2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    499       2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    500       3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    501       3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    502       3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    503       4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    504       4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    505       4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    506       2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  507       2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  508       2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  509       3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  510       3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  511       3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  512       4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  513       4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  514       4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  515       2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       516       2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       517       2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       518       3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       519       3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       520       3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       521       4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       522       4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       523       4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       524       2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           525       2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           526       2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           527       3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           528       3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           529       3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           530       4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           531       4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           532       4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           533       2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   534       2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   535       2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   536       3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   537       3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   538       3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   539       4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   540       4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   541       4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   542       2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    543       2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    544       2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    545       3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    546       3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    547       3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    548       4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    549       4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    550       4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    551       2-O-(2'-NCC.sub.6 H.sub.4)                                           552       2-O-(3'-NCC.sub.6 H.sub.4)                                           553       2-O-(4'-NCC.sub.6 H.sub.4)                                           554       3-O-(2'-NCC.sub.6 H.sub.4)                                           555       3-O-(3'-NCC.sub.6 H.sub.4)                                           556       3-O-(4'-NCC.sub.6 H.sub.4)                                           557       4-O-(2'-NCC.sub.6 H.sub.4)                                           558       4-O-(3'-NCC.sub.6 H.sub.4)                                           559       4-O-(4'-NCC.sub.6 H.sub.4)                                           560       2-O-(2'-CF.sub.3 C.sub.6 H.sub.5)                                    561       2-O-(3'-CF.sub.3 C.sub.6 H.sub.5)                                    562       2-O-(4'-CF.sub.3 C.sub.6 H.sub.5)                                    563       3-O-(2'-CF.sub.3 C.sub.6 H.sub.5)                                    564       3-O-(3'-CF.sub.3 C.sub.6 H.sub.5)                                    565       3-O-(4'-CF.sub.3 C.sub.6 H.sub.5)                                    566       4-O-(2'-CF.sub.3 C.sub.6 H.sub.5)                                    567       4-O-(3'-CF.sub.3 C.sub.6 H.sub.5)                                    568       4-O-(4'-CF.sub.3 C.sub.6 H.sub.5)                                    569       2-Pyridinyl-2'                                                       570       2-Pyridinyl-3'                                                       571       2-Pyridinyl-4'                                                       572       3-Pyridinyl-2'                                                       573       3-Pyridinyl-3'                                                       574       3-Pyridinyl-4'                                                       575       4-Pyridinyl-2'                                                       576       4-Pyridinyl-3'                                                       577       4-Pyridinyl-4'                                                       578       2-Pyrimidinyl-2'                                                     579       2-Pyrimidinyl-3'                                                     580       2-Pyrimidinyl-4'                                                     581       3-Pyrimidinyl-2'                                                     582       3-Pyrimidinyl-3'                                                     583       3-Pyrimidinyl-4'                                                     584       4-Pyrimidinyl-2'                                                     585       4-Pyrimidinyl-3'                                                     586       4-Pyrimidinyl-4'                                                     587       2-Pyrazolyl-1'                                                       588       2-Pyrazolyl-3'                                                       589       2-Pyrazolyl-4'                                                       590       3-Pyrazolyl-1'                                                       591       3-Pyrazolyl-3'                                                       592       3-Pyrazolyl-4'                                                       593       4-Pyrazolyl-1'                                                       594       4-Pyrazolyl-3'                                                       595       4-Pyrazolyl-4'                                                       596       2-Isoxazolyl-3'                                                      597       2-Isoxazolyl-4'                                                      598       2-Isoxazolyl-5'                                                      599       3-Isoxazolyl-3'                                                      600       3-Isoxazolyl-4'                                                      601       3-Isoxazolyl-5'                                                      602       4-Isoxazolyl-3'                                                      603       4-Isoxazolyl-4'                                                      604       4-Isoxazolyl-5'                                                      605       2-Isothiazolyl-3'                                                    606       2-Isothiazolyl-4'                                                    607       2-Isothiazolyl-5'                                                    608       3-Isothiazolyl-3'                                                    609       3-Isothiazolyl-4'                                                    610       3-Isothiazolyl-5'                                                    611       4-Isothiazolyl-3'                                                    612       4-Isothiazolyl-4'                                                    613       4-Isothiazolyl-5'                                                    614       2-Imidazolyl-1'                                                      615       2-Imidazolyl-2'                                                      616       2-Imidazolyl-4'                                                      617       3-Imidazolyl-1'                                                      618       3-Imidazolyl-2'                                                      619       3-Imidazolyl-4'                                                      620       4-Imidazolyl-1'                                                      621       4-Imidazolyl-2'                                                      622       4-Imidazolyl-4'                                                      623       2-Oxazolyl-2'                                                        624       2-Oxazolyl-4'                                                        625       2-Oxazolyl-5'                                                        626       3-Oxazolyl-2'                                                        627       3-Oxazolyl-4'                                                        628       3-Oxazolyl-5'                                                        629       4-Oxazolyl-2'                                                        630       4-Oxazolyl-4'                                                        631       4-Oxazolyl-5'                                                        632       2-Thiazolyl-2'                                                       633       2-Thiazolyl-4'                                                       634       2-Thiazolyl-5'                                                       635       3-Thiazolyl-2'                                                       636       3-Thiazolyl-4'                                                       637       3-Thiazolyl-5'                                                       638       4-Thiazolyl-2'                                                       639       4-Thiazolyl-4'                                                       640       4-Thiazolyl-5'                                                       ______________________________________                                    

                  TABLE 6                                                          ______________________________________                                          ##STR28##                                                                     I: R.sup.1 = H                                                                 II: R.sup.1 = CH.sub.3                                                         III: R.sup.1 = Allyl                                                           IV: R.sup.1 = Propargyl                                                        V: R.sup.1 = SCH.sub.3                                                         VI: R.sup.1 = CH.sub.2 CN                                                      VII: R.sup.1 = CH.sub.2 OCH.sub.3                                              VIII: R.sup.1 = COOCH.sub.3                                                    No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                            2        N-CH.sub.3 -Pyrrolyl-3                                                3        N-C.sub.6 H.sub.5 -Pyrrolyl-3                                         4        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            5        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            6        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            7        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           8        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           9        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           10       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            11       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            12       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            13       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   14       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   15       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   16       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   17       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   18       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   19       Pyrrolyl-2                                                            20       N-CH.sub.3 -Pyrrolyl-2                                                21       N-C.sub.6 H.sub.5 -Pyrrolyl-2                                         22       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            23       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            24       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            25       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           26       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           27       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           28       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            29       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            30       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            31       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   32       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   33       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   34       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   35       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   36       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   37       Furyl-2                                                               38       5-CH.sub.3 -Furyl-2                                                   39       5-C.sub.6 H.sub.5 -Furyl-2                                            40       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               41       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               42       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               43       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              44       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              45       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              46       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               47       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               48       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               49       5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      50       5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      51       5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      52       5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      53       5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      54       5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      55       4-CH.sub.3 -Furyl-2                                                   56       4-C.sub.6 H.sub.5 -Furyl-2                                            57       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               58       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               59       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               60       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              61       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              62       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              63       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               64       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               65       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               66       4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      67       4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      68       4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      69       4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      70       4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      71       4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      72       Thienyl-2                                                             73       5-CH.sub.3 -Thienyl-2                                                 74       5-C.sub.6 H.sub.5 -Thienyl-2                                          75       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             76       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             77       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             78       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            79       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            80       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            81       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             82       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             83       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             84       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    85       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    86       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    87       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    88       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    89       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    90       4-CH.sub.3 -Thienyl-2                                                 91       4-C.sub.6 H.sub.5 -Thienyl-2                                          92       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             93       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             94       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             95       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            96       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            97       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            98       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             99       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       N-CH.sub.3 -Pyrazolyl-4                                              127       N-C.sub.6 H.sub.5 -Pyrazolyl-4                                       128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 143       3-CH.sub.3 -N-Methylpyrazolyl-4                                      144       3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4                               145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  154       3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         155       3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         156       3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         157       3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         158       3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         159       3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         160       Isoxazolyl-5                                                         161       3-CH.sub.3 -Isoxazolyl-5                                             162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 -Isoxazolyl-3                                             198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-I5oxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 -Isothiazolyl-5                                           216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       2-CH.sub.3 -Oxazolyl-4                                               234       2-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           236       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           237       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           238       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          239       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          241       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           242       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           243       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           244       2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  245       2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  246       2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  247       2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  248       2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  249       2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       N-CH.sub.3 -1,2,4-Triazolyl-5                                        269       3-CH.sub.3NCH.sub.3 -1,2,4-Triazolyl-5                               270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          280       3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 281       3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 282       3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 283       3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 284       3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 285       3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        ______________________________________                                    

                                      TABLE 7                                      __________________________________________________________________________     Selected physical data of some compounds                                       No.                                                                               Compound                mp/°C. IR/cm.sup.-1                          __________________________________________________________________________      1                                                                                 ##STR29##              --            1707, 1484, 1457, 1447, 1303,                                                  1277                                   2                                                                                 ##STR30##              --            1708, 1495, 1457, 1449, 1304,                                                  1241                                   3                                                                                 ##STR31##              111                                                  4                                                                                 ##STR32##               73                                                  5                                                                                 ##STR33##               54                                                  6                                                                                 ##STR34##              --            1706, 1496, 1456, 1447, 1294,                                                  1243                                   7                                                                                 ##STR35##               73                                                  8                                                                                 ##STR36##               57                                                  9                                                                                 ##STR37##               86                                                  10                                                                                ##STR38##              --            1709, 1599, 1497, 1453, 1346,                                                  1241                                   11                                                                                ##STR39##              --            1708, 1599, 1497, 1455, 1447,                                                  1397, 1238                             12                                                                                ##STR40##              --            1740, 1593, 1527, 1489, 1456,                                                  1252, 1225                             13                                                                                ##STR41##              --            1710, 1603, 1584, 1490, 1451,                                                  1364, 1254                             14                                                                                ##STR42##              --            1709, 1490, 1456, 1447, 1379,                                                  1300, 1258                             15                                                                                ##STR43##              --            1712, 1490, 1456, 1447, 1378,                                                  1298, 1259                             16                                                                                ##STR44##               88                                                  17                                                                                ##STR45##              --            1710, 1511, 1451, 1364, 1302,                                                  1238                                   18                                                                                ##STR46##              --            1709, 1511, 1456, 1447, 1379,                                                  1301, 1236                             19                                                                                ##STR47##              --            1712, 1511, 1447, 1378, 1298,                                                  1233                                   20                                                                                ##STR48##              --            1738, 1723, 1582, 1522, 1452,                                                  1223                                   21                                                                                ##STR49##              --            1711, 1492, 1480, 1447, 1362,                                                  1303, 1192, 1159                       22                                                                                ##STR50##              --            1708, 1491, 1479, 1446, 1376,                                                  1300, 1277, 1150                       23                                                                                ##STR51##              --            1712, 1511, 1447, 1378, 1298,                                                  1233                                   24                                                                                ##STR52##              --            1736, 1582, 1523, 1453, 1221           25                                                                                ##STR53##              --            1706, 1495, 1485, 1363, 1303,                                                  1193, 1160                             26                                                                                ##STR54##              --            1706, 1484, 1447, 1377, 1301,                                                  1280, 1150                             27                                                                                ##STR55##              --            1710, 1495, 1483, 1446, 1376,                                                  1299, 1233                             28                                                                                ##STR56##               92                                                  29                                                                                ##STR57##              --            1709, 1489, 1447, 1362, 1303,                                                  1192, 1159                             30                                                                                ##STR58##              --            1706, 1484, 1447, 1377, 1301,                                                  1280, 1150                             31                                                                                ##STR59##              --            1711, 1488, 1446, 1375, 1299,                                                  1232                                   32                                                                                ##STR60##              132                                                  33                                                                                ##STR61##              --            1709, 1495, 1486, 1451, 1366,                                                  1161, 1008                             34                                                                                ##STR62##              --            1708, 1487, 1455, 1447, 1379,                                                  1300, 1009                             35                                                                                ##STR63##              --            1711, 1488, 1447, 1378, 1297,                                                  1232, 1023, 1008                       36                                                                                ##STR64##              --            1696, 1532, 1515, 1453, 1267,                                                  1245, 1069                             37                                                                                ##STR65##              --            1712, 1486, 1447, 1361, 1303,                                                  1191, 1160                             38                                                                                ##STR66##              --            1708, 1485, 1446, 1376, 1300,                                                  1274                                   39                                                                                ##STR67##              --            1709, 1484, 1446, 1374, 1297,                                                  1277, 1232                             40                                                                                ##STR68##              --            1712, 1495, 1457, 1447, 1378,                                                  1298, 1237                             41                                                                                ##STR69##              110                                                  42                                                                                ##STR70##              --            1739, 1593, 1528, 1511, 1457,                                                  1226, 1035                             43                                                                                ##STR71##              102                                                  44                                                                                ##STR72##              --            1708, 1513, 1457, 1447, 1378,                                                  1302, 1246, 1035                       45                                                                                ##STR73##              102                                                  46                                                                                ##STR74##               74                                                  47                                                                                ##STR75##              --            1709, 1606, 1512, 1364, 1245,                                                  1228, 1171, 1162, 1033, 1005           48                                                                                ##STR76##               59           1709, 1447, 1364, 1261, 1157,                                                  1034, 1007                             49                                                                                ##STR77##              --            1709, 1576, 1446, 1379, 1300,                                                  1260, 1239, 1156, 1037                 50                                                                                ##STR78##              --                                                   51                                                                                ##STR79##               89                                                  52                                                                                ##STR80##              --            1740, 1593, 1575, 1527, 1457,                                                  1316, 1300, 1224, 1067, 1029           53                                                                                ##STR81##               81                                                  54                                                                                ##STR82##              --            1711, 1574, 1447, 1365, 1322,                                                  1303, 1213, 1160, 1033, 1008           55                                                                                ##STR83##              --            1709, 1574, 1446, 1378, 1321,                                                  1301, 1284, 1213, 1034                 56                                                                                ##STR84##              --            1711, 1505, 1451, 1365, 1304,                                                  1245, 1160, 1143, 1035, 1007           57                                                                                ##STR85##               63                                                  58                                                                                ##STR86##              --            1710, 1487, 1450, 1364, 1301,                                                  1246, 1160, 1030, 1006                 59                                                                                ##STR87##              --            1708, 1487, 1449, 1378, 1300,                                                  1247, 1030, 1009                       60                                                                                ##STR88##              --            1743, 1593, 1528, 1502, 1457,                                                  1301, 1255, 1190, 1066, 1006           61                                                                                ##STR89##               77                                                  62                                                                                ##STR90##              --            1712, 1503, 1453, 1363, 1303,                                                  1259, 1244, 1160, 1136, 1006           63                                                                                ##STR91##              --            1711, 1503, 1457, 1447, 1380,                                                  1301, 1258, 1239, 1136, 1015           64                                                                                ##STR92##               92           1743, 1593, 1528, 1502, 1457,                                                  1301, 1255, 1190, 1066, 1006           65                                                                                ##STR93##               90                                                  66                                                                                ##STR94##               70                                                  67                                                                                ##STR95##               75                                                  68                                                                                ##STR96##              108                                                  69                                                                                ##STR97##               93                                                  70                                                                                ##STR98##               74                                                  71                                                                                ##STR99##              --            1712, 1504, 1450, 1363, 1303,                                                  1255, 1222, 1159, 1134                 72                                                                                ##STR100##             --            1712, 1510, 1498, 1450, 1365,                                                  1327, 1246, 1150, 1035, 1005           73                                                                                ##STR101##              60                                                  74                                                                                ##STR102##             --            1711, 1509, 1497, 1451, 1363,                                                  1302, 1264, 1193, 1156, 1129           75                                                                                ##STR103##             --            1710, 1496, 1475, 1149, 1365,                                                  1301, 1263, 1195, 1159                 76                                                                                ##STR104##              66                                                  77                                                                                ##STR105##              86                                                  78                                                                                ##STR106##              91                                                  79                                                                                ##STR107##             100                                                  80                                                                                ##STR108##             --            1710, 1593, 1497, 1452, 1364,                                                  1323, 1297, 1193, 1165, 1153           81                                                                                ##STR109##             --            1715, 1510, 1447, 1367, 1324,                                                  1299, 1243, 1149, 1027, 996            82                                                                                ##STR110##             --            1710, 1509, 1456, 1446, 1377,                                                  1326, 1300, 1241, 1149, 1306           83                                                                                ##STR111##             --            1723, 1509, 1453, 1437, 1316,                                                  1292, 1241, 1149, 1064, 1036           84                                                                                ##STR112##             --            1738, 1611, 1581, 1539, 1446,                                                  1312, 1301, 1231, 1201, 1067           85                                                                                ##STR113##             --            1713, 1504, 1447, 1375, 1313,                                                  1300, 1233, 1143, 1027                 86                                                                                ##STR114##             --            1711, 1486, 1447, 1376, 1300,                                                  1281, 1150, 1034, 1013                 87                                                                                ##STR115##             --            1714, 1487, 1447, 1376, 1300,                                                  1231, 1023, 999                        88                                                                                ##STR116##             --            1733, 1594, 1533, 1457, 1306,                                                  1231, 1013, 984                        89                                                                                ##STR117##             --            1721, 1495, 1453, 1437, 1313,                                                  1290, 1239, 1123                       90                                                                                ##STR118##             --            1709, 1453, 1366, 1303, 1228,                                                  1160, 1014                             91                                                                                ##STR119##             --            1708, 1455, 1447, 1378, 1299,                                                  1282, 1015, 996                        92                                                                                ##STR120##             --            1710, 1447, 1378, 1296, 1232,                                                  1045, 1023, 995                        93                                                                                ##STR121##             108                                                  94                                                                                ##STR122##             --            1717, 1495, 1457, 1444, 1376,                                                  1298, 1241, 1228, 1193                 95                                                                                ##STR123##             --            1739, 1614, 1603, 1542, 1450,                                                  1262, 129, 1179                        96                                                                                ##STR124##             170                                                  97                                                                                ##STR125##             180                                                  98                                                                                ##STR126##             173                                                  99                                                                                ##STR127##             150                                                 100                                                                                ##STR128##             129                                                 101                                                                                ##STR129##             112                                                 102                                                                                ##STR130##             116                                                 103                                                                                ##STR131##             127                                                 104                                                                                ##STR132##             108                                                 105                                                                                ##STR133##             --            1710, 1486, 1447, 1363, 1307,                                                  1193, 1159, 1031, 1006, 919           106                                                                                ##STR134##             --            1706, 1484, 1447, 1376, 1302,                                                  1279, 1150, 1031, 1011, 923           107                                                                                ##STR135##             --            1711, 1484, 1446, 1376, 1298,                                                  1232, 1144, 1024, 995, 922            108                                                                                ##STR136##             147                                                 109                                                                                ##STR137##                           1716, 1455, 1445, 1376, 1297,                                                  1279, 1097, 1069, 1017, 1008          110                                                                                ##STR138##                           1718, 1487, 1447, 1394, 1374,                                                  1306, 1232, 1025, 1008                111                                                                                ##STR139##             109                                                 112                                                                                ##STR140##                           1706, 1487, 1450, 1387, 1304,                                                  1276, 1155, 1022, 1009, 769           113                                                                                ##STR141##                           1706, 1487, 1453, 1383, 1312,                                                  1301, 1274, 1155, 1033, 1008          114                                                                                ##STR142##             115                                                 115                                                                                ##STR143##             167                                                 116                                                                                ##STR144##                           1729, 1575, 1565, 1545, 1523,                                                  1445, 1434, 1224, 1060                117                                                                                ##STR145##             110                                                 118                                                                                ##STR146##              77                                                 119                                                                                ##STR147##                           1712, 1494, 1447, 1378, 1298,                                                  1232, 1045, 1024, 818, 771            120                                                                                ##STR148##             115                                                 121                                                                                ##STR149##                           1717, 1455, 1445, 1376, 1298,                                                  1278, 1097, 1068, 1016, 999           122                                                                                ##STR150##              81                                                 123                                                                                ##STR151##                           1712, 1493, 1447, 1378, 1297,                                                  1232, 1047, 1024, 998, 772            124                                                                                ##STR152##             107                                                 125                                                                                ##STR153##                           1717, 1455, 1445, 1376, 1298,                                                  1279, 1096, 1068, 1017, 999           126                                                                                ##STR154##             128                                                 127                                                                                ##STR155##                           1712, 1492, 1447, 1378, 1298,                                                  1232, 1096, 1044, 1023                128                                                                                ##STR156##             119                                                 129                                                                                ##STR157##                           1717, 1492, 1455, 1445, 1376,                                                  1298, 1096, 1068, 1012, 1000          130                                                                                ##STR158##             133                                                 131                                                                                ##STR159##                           1712, 1511, 1494, 1447, 1378,                                                  1298, 1232, 1045, 1024, 837           132                                                                                ##STR160##             113                                                 133                                                                                ##STR161##                           1716, 1511, 1455, 1445, 1376,                                                  1298, 1228, 1097, 1068, 999           134                                                                                ##STR162##                           1737, 1592, 1529, 1509, 1489,                                                  1455, 1303, 1231, 1067, 1014          135                                                                                ##STR163##                           1712, 1586, 1507, 1489, 1454,                                                  1378, 1297, 1239, 1023                136                                                                                ##STR164##             148                                                 137                                                                                ##STR165##                           1716, 1587, 1507, 1490, 1455,                                                  1375, 1298, 1240, 1068                138                                                                                ##STR166##              90                                                 139                                                                                ##STR167##                           1719, 1495, 1464, 1446, 1375,                                                  1295, 1239, 1104, 1075, 1014          140                                                                                ##STR168##                           1715, 1495, 1463, 1448, 1376,                                                  1298, 1239                            141                                                                                ##STR169##             134                                                 142                                                                                ##STR170##                           1744, 1583, 1522, 1503, 1458,                                                  1442, 1223, 1304, 1035, 1004          143                                                                                ##STR171##                           1720, 1465, 1446, 1372, 1296,                                                  1280, 1243, 1144, 1035, 1014          144                                                                                ##STR172##                           1716, 1505, 1465, 1448, 1374,                                                  1298, 1279, 1241, 1141, 999           145                                                                                ##STR173##             109                                                 146                                                                                ##STR174##             158                                                 147                                                                                ##STR175##                           1718, 1463, 1445, 1376, 1294,                                                  1104, 1073, 1024, 1010                148                                                                                ##STR176##                           1714, 1462, 1447, 1377, 1297,                                                  1238, 1025, 1009                      149                                                                                ##STR177##             140                                                 __________________________________________________________________________

Example 4

Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

a) Methyl N-(2-methylphenyl)-N-hydroxy-carbamate

At 25°-30° C., 14.0 g (0.148 mol) of methyl Chloroocarbonate is added dropwise to 16.4 g of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.9 g (0.163 mol) of pyridine in 100 ml of methylene Chloroide. The mixture is stirred overnight at room temperature (20° C.) and is then extracted with dilute hydroChloroic acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 7 g (39 mmol) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 8.6 (s, broad, OH); 7.3 (m, 4H, phenyl); 3.75 (s, 3H, OCH₃); 2.3 (s, 3H, CH₃)

b) Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

At 20°-30° C., 1.1 g (44.1 mmol) of sodium hydride is added in portions to 6.6 g (36.5 mmol) of the hydroxyl compound from Example 4a in 50 ml of dimethylformamide. Upon conclusion of gas evolution 5.7 g (40.1 mmol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 5.2 g (27 mmol=73%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.25 (m, 4H, phenyl); 3.8; 3.75 (s, 3H, OCH₃ ; 3.75 (s, 3H, OCH₃); 2.3 (s, 3H, CH₃)

Example 5

Methyl N-(2-bromomethylphenyl)-N-methoxy-carbamate (Table 14, No. 2)

2.5 g (12.8 mmol) of the N-methoxycarbamate from Example 4b, 2.5 g (14.1 mmol) of N-bromosuccinimide and a spatula-tip (1 g) of azoisobutyrodinitrile in 20 ml of carbon tetrachloroide were irradiated with a 300 W UV lamp; the reaction mixture heated up to 30°-40° C. After three hours the reaction mixture is extracted twice with water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.4 g (5.1 mmol=40%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.55 (s, 2H, CH₂ --Br); 3.8 (2s, 6H, 2× OCH₃)

Example 6

Methyl N- 2-(2'-methylphenoxymethyl)-phenyl!-N-methoxy-carbamate (Table 14, No. 3)

1.2 g (4.4 mmol) of the methyl bromide from Example 5, 0.45 g (4.2 mmol) o-cresol and 0.7 g (4.8 mmol) of K₂ CO₃ in 30 ml of dimethylformamide are stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.2 g of the title compound containing o-cresol as impurity. The mixture is heated in a furnace at about 1 mbar for about 1 hour at 125° C. The residue obtained is 0.9 g (3 mmol=68%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 7.15 (m, 2H, phenyl); 6.9 (t, broad, 2H, phenyl); 5.15 (s, 2H, O--CH₂); 3.8 (s, 3H, OCH₃), 3.75 (s, 3H, OCH₃); 2.3 (s, 3H, CH₃)

                  TABLE 8                                                          ______________________________________                                          ##STR178##                                                                    I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 CH.sub.3                                                No.      Xm                                                                    ______________________________________                                         1        H                                                                     2        2-F                                                                   3        3-F                                                                   4        4-F                                                                   5        2,4-F.sub.2                                                           6        2,4,6-F.sub.3                                                         7        2,3,4,5,6-F.sub.5                                                     8        2,3-F.sub.2                                                           9        2-Cl                                                                  10       3-Cl                                                                  11       4-Cl                                                                  12       2,3-Cl.sub.2                                                          13       2,4-Cl.sub.2                                                          14       2,5-Cl.sub.2                                                          15       2,6-Cl.sub.2                                                          16       3,4-Cl.sub.2                                                          17       3,5-Cl.sub.2                                                          18       2,3,4-Cl.sub.3                                                        19       2,3,5-Cl.sub.3                                                        20       2,3,6-Cl.sub.3                                                        21       2,4,5-Cl.sub.3                                                        22       2,4,6-Cl.sub.3                                                        23       3,4,5-Cl.sub.3                                                        24       2,3,4,6-Cl.sub.4                                                      25       2,3,5,6-Cl.sub.4                                                      26       2,3,4,5,6-Cl.sub.5                                                    27       2-Br                                                                  28       3-Br                                                                  29       4-Br                                                                  30       2,4-Br.sub.2                                                          31       2,5-Br.sub.2                                                          32       2,6-Br.sub.2                                                          33       2,4,6-Br.sub.3                                                        34       2,3,4,5,6-Br.sub.5                                                    35       2-I                                                                   36       3-I                                                                   37       4-I                                                                   38       2,4-I.sub.2                                                           39       2-Cl, 3-F                                                             40       2-Cl, 4-F                                                             41       2-Cl, 5-F                                                             42       2-Cl, 6-F                                                             43       2-Cl, 3-Br                                                            44       2-Cl, 4-Br                                                            45       2-Cl, 5-Br                                                            46       2-Cl, 6-Br                                                            47       2-Br, 3-Cl                                                            48       2-Br, 4-Cl                                                            49       2-Br, 5-Cl                                                            50       2-Br, 3-F                                                             51       2-Br, 4-F                                                             52       2-Br, 5-F                                                             53       2-Br, 6-F                                                             54       2-F, 3-Cl                                                             55       2-F, 4-Cl                                                             56       2-F, 5-Cl                                                             57       3-Cl, 4-F                                                             58       3-Cl, 5-F                                                             59       3-Cl, 4-Br                                                            60       3-Cl, 5-Br                                                            61       3-F, 4-Cl                                                             62       3-F, 4-Br                                                             63       3-Br, 4-Cl                                                            64       3-Br, 4-F                                                             65       2,6-Cl.sub.2, 4-Br                                                    66       2-CH.sub.3                                                            67       3-CH.sub.3                                                            68       4-CH.sub.3                                                            69       2,3-(CH.sub.3).sub.2                                                  70       2,4-(CH.sub.3).sub.2                                                  71       2,5-(CH.sub.3).sub.2                                                  72       2,6-(CH.sub.3).sub.2                                                  73       3,4-(CH.sub.3).sub.2                                                  74       3,5-(CH.sub.3).sub.2                                                  75       2,3,5-(CH.sub.3).sub.3                                                76       2,3,4-(CH.sub.3).sub.3                                                77       2,3,6-(CH.sub.3).sub.3                                                78       2,4,5-(CH.sub.3).sub.3                                                79       2,4,6-(CH.sub.3).sub.3                                                80       3,4,5-(CH.sub.3).sub.3                                                81       2,3,4,6-(CH.sub.3).sub.4                                              82       2,3,5,6-(CH.sub.3).sub.4                                              83       2,3,4,5,6-(CH.sub.3).sub.5                                            84       2-C.sub.2 H.sub.5                                                     85       3-C.sub.2 H.sub.5                                                     86       4-C.sub.2 H.sub.5                                                     87       2,4-(C.sub.2 H.sub.5).sub.2                                           88       2,6-(C.sub.2 H.sub.5).sub.2                                           89       3,5-(C.sub.2 H.sub.5).sub.2                                           90       2,4,6-(C.sub.2 H.sub.5).sub.3                                         91       2-n-C.sub.3 H.sub.7                                                   92       3-n-C.sub.3 H.sub.7                                                   93       4-n-C.sub.3 H.sub.7                                                   94       2-i-C.sub.3 H.sub.7                                                   95       3-i-C.sub.3 H.sub.7                                                   96       4-i-C.sub.3 H.sub.7                                                   97       2,4-(i-C.sub.3 H.sub.7).sub.2                                         98       2,6-(i-C.sub.3 H.sub.7).sub.2                                         99       3,5-(i-C.sub.3 H.sub.7).sub.2                                         100      2,4,6-(i-C.sub.3 H.sub.7).sub.3                                       101      2-s-C.sub.4 H.sub.9                                                   102      3-s-C.sub.4 H.sub.9                                                   103      4-s-C.sub.4 H.sub.9                                                   104      2-t-C.sub.4 H.sub.9                                                   105      3-t-C.sub.4 H.sub.9                                                   106      4-t-C.sub.4 H.sub.9                                                   107      2,3-(t-C.sub.4 H.sub.9).sub.2                                         108      2,4-(t-C.sub.4 H.sub.9).sub.2                                         109      2,5-(t-C.sub.4 H.sub.9).sub.2                                         110      2,6-(t-C.sub.4 H.sub.9).sub.2                                         111      3,4-(t-C.sub.4 H.sub.9).sub.2                                         112      2,4,6-(t-C.sub.4 H.sub.9).sub.3                                       113      4-n-C.sub.9 H.sub.19                                                  114      4-n-C.sub.12 H.sub.25                                                 115      4-n-C.sub.15 H.sub.31                                                 116      4-(1,1,3,3-Tetramethylbutyl)                                          117      4-(2,4,4-Trimethylpropyl)                                             118      2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                       119      2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                       120      2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                             121      2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                       122      2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                       123      2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                       124      2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                       125      3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                       126      2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                       127      2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                    128      2-Allyl                                                               129      3-Allyl                                                               130      4-Allyl                                                               131      2-Allyl, 6-CH.sub.3                                                   132      2-cyclo-C.sub.6 H.sub.11                                              133      3-cyclo-C.sub.6 H.sub.11                                              134      4-cyclo-C.sub.6 H.sub.11                                              135      2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                        136      2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                  137      2-CH.sub.2 C.sub.6 H.sub.5                                            138      3-CH.sub.2 C.sub.6 H.sub.5                                            139      4-CH.sub.2 C.sub.6 H.sub.5                                            140      2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                141      2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                142      2-C.sub.6 H.sub.5                                                     143      3-C.sub.6 H.sub.5                                                     144      4-C.sub.6 H.sub.5                                                     145      4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                               146      4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                               147      2-Cl, 4-C.sub.6 H.sub.5                                               148      2-Br, 4-C.sub.6 H.sub.5                                               149      2-C.sub.6 H.sub.5, 4-Cl                                               150      2-C.sub.6 H.sub.5, 4-Br                                               151      2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                      152      2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                      153      2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                      154      2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                      155      2-cyclo-C.sub.6 H.sub.11, 4-Cl                                        156      2-cyclo-C.sub.6 H.sub.11, 4-Br                                        157      2-Cl, 4-cyclo-C.sub.6 H.sub.11                                        158      2-Br, 4-cyclo-C.sub.6 H.sub.11                                        159      2-OCH.sub.3                                                           160      3-OCH.sub.3                                                           161      4-OCH.sub.3                                                           162      2-OC.sub.2 H.sub.5                                                    163      3-OC.sub.2 H.sub.5                                                    164      4-OC.sub.2 H.sub.5                                                    165      2-O-n-C.sub.3 H.sub.7                                                 166      3-O-n-C.sub.3 H.sub.7                                                 167      4-O-n-C.sub.3 H.sub.7                                                 168      2-O-i-C.sub.3 H.sub.7                                                 169      3-O-i-C.sub.3 H.sub.7                                                 170      4-O-i-C.sub.3 H.sub.7                                                 171      2-O-n-C.sub.6 H.sub.13                                                172      3-O-n-C.sub.6 H.sub.13                                                173      4-O-n-C.sub.6 H.sub.13                                                174      2-O-n-C.sub.8 H.sub.17                                                175      3-O-n-C.sub.8 H.sub.17                                                176      4-O-n-C.sub.8 H.sub.17                                                177      2-OCH.sub.2 C.sub.6 H.sub.5                                           178      3-OCH.sub.2 C.sub.6 H.sub.5                                           179      4-OCH.sub.2 C.sub.6 H.sub.5                                           180      2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   181      3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   182      4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183      2,4-(OCH.sub.3).sub.2                                                 184      2-CF.sub.3                                                            185      3-CF.sub.3                                                            186      4-CF.sub.3                                                            187      2-OCF.sub.3                                                           188      3-OCF.sub.3                                                           189      4-OCF.sub.3                                                           190      3-OCH.sub.2 CHF.sub.2                                                 191      2-NO.sub.2                                                            192      3-NO.sub.2                                                            193      4-NO.sub.2                                                            194      2-CN                                                                  195      3-CN                                                                  196      4-CN                                                                  197      2-CH.sub.3, 3-Cl                                                      198      2-CH.sub.3, 4-Cl                                                      199      2-CH.sub.3, 5-Cl                                                      200      2-CH.sub.3, 6-Cl                                                      201      2-CH.sub.3, 3-F                                                       202      2-CH.sub.3, 4-F                                                       203      2-CH.sub.3, 5-F                                                       204      2-CH.sub.3, 6-F                                                       205      2-CH.sub.3, 3-Br                                                      206      2-CH.sub.3, 4-Br                                                      207      2-CH.sub.3, 5-Br                                                      208      2-CH.sub.3, 6-Br                                                      209      2-Cl, 3-CH.sub.3                                                      210      2-Cl, 4-CH.sub.3                                                      211      2-Cl, 5-CH.sub.3                                                      212      2-F, 3-CH.sub.3                                                       213      2-F, 4-CH.sub.3                                                       214      2-F, 5-CH.sub.3                                                       215      2-Br, 3-CH.sub.3                                                      216      2-Br, 4-CH.sub.3                                                      217      2-Br, 5-CH.sub.3                                                      218      3-CH.sub.3, 4-Cl                                                      219      3-CH.sub.3, 5-Cl                                                      220      3-CH.sub.3, 4-F                                                       221      3-CH.sub.3, 5-F                                                       222      3-CH.sub.3, 4-Br                                                      223      3-CH.sub.3, 5-Br                                                      224      3-F, 4-CH.sub.3                                                       225      3-Cl, 4-CH.sub.3                                                      226      3-Br, 4-CH.sub.3                                                      227      2-Cl, 4,5-(CH.sub.3).sub.2                                            228      2-Br, 4,5-(CH.sub.3).sub.2                                            229      2-Cl, 3,5-(CH.sub.3).sub.2                                            230      2-Br, 3,5-(CH.sub.3).sub.2                                            231      2,6-Cl.sub.2, 4-CH.sub.3                                              232      2,6-F.sub.2, 4-CH.sub.3                                               233      2,6-Br.sub.2, 4-CH.sub.3                                              234      2,4-Br.sub.2, 6-CH.sub.3                                              235      2,4-F.sub.2, 6-CH.sub.3                                               236      2,4-Br.sub.2, 6-CH.sub.3                                              237      2,6-(CH.sub.3).sub.2, 4-F                                             238      2,6-(CH.sub.3).sub.2, 4-Cl                                            239      2,6-(CH.sub.3).sub.2, 4-Br                                            240      3,5-(CH.sub.3).sub.2, 4-F                                             241      3,5-(CH.sub.3).sub.2, 4-Cl                                            242      3,5-(CH.sub.3).sub.2, 4-Br                                            243      2,3,6-(CH.sub.3).sub.3, 4-F                                           244      2,3,6-(CH.sub.3).sub.3, 4-Cl                                          245      2,3,6-(CH.sub.3).sub.3, 4-Br                                          246      2,4-(CH.sub.3).sub.2, 6-F                                             247      2,4-(CH.sub.3).sub.2, 6-Cl                                            248      2,4-(CH.sub.3).sub.2, 6-Br                                            249      2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                 250      2-Cl, 4-NO.sub.2                                                      251      2-NO.sub.2, 4-Cl                                                      252      2-OCH.sub.3, 5-NO.sub.2                                               253      2,4-Cl.sub.2, 5-NO.sub.2                                              254      2,4-Cl.sub.2, 6-NO.sub.2                                              255      2,6-Cl.sub.2, 4-NO.sub.2                                              256      2,6-Br.sub.2, 4-NO.sub.2                                              257      2,6-I.sub.2, 4-NO.sub.2                                               258      2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                 259      2-CO.sub.2 CH.sub.3                                                   260      3-CO.sub.2 CH.sub.3                                                   261      4-CO.sub.2 CH.sub.3                                                   262      2-CO.sub.2 (C.sub.2 H.sub.5)                                          263      3-CO.sub.2 (C.sub.2 H.sub.5)                                          264      4-CO.sub.2 (C.sub.2 H.sub.5)                                          265      2-CO.sub.2 (n-C.sub.3 H.sub.7)                                        266      3-CO.sub.2 (n-C.sub.3 H.sub.7)                                        267      4-CO.sub.2 (n-C.sub.3 H.sub.7)                                        268      2-CO.sub.2 (i-C.sub.3 H.sub.7)                                        269      3-CO.sub.2 (i-C.sub.3 H.sub.7)                                        270      4-CO.sub.2 (i-C.sub.3 H.sub.7)                                        271      2-CO.sub.2 (n-C.sub.6 H.sub.13)                                       272      3-CO.sub.2 (n-C.sub.6 H.sub.13)                                       273      4-CO.sub.2 (n-C.sub.6 H.sub.13)                                       274      2-CH.sub.2 OCH.sub.3                                                  275      3-CH.sub.2 OCH.sub.3                                                  276      4-CH.sub.2 OCH.sub.3                                                  277      2-CH.sub.2 O (C.sub.2 H.sub.5)                                        278      3-CH.sub.2 O (C.sub.2 H.sub.5)                                        279      4-CH.sub.2 O (C.sub.2 H.sub.5)                                        280      2-CH.sub.2 O (n-C.sub.3 H.sub.7)                                      281      3-CH.sub.2 O (n-C.sub.3 H.sub.7)                                      282      4-CH.sub.2 O (n-C.sub.3 H.sub.7)                                      283      2-CH.sub.2 O (i-C.sub.3 H.sub.7)                                      284      3-CH.sub.2 O (i-C.sub.3 H.sub.7)                                      285      4-CH.sub.2 O (i-C.sub.3 H.sub.7)                                      286      2-CHO                                                                 287      3-CHO                                                                 288      4-CHO                                                                 289      2-COCH.sub.3                                                          290      3-COCH.sub.3                                                          291      4-COCH.sub.3                                                          292      2-COCH.sub.2 CH.sub.3                                                 293      3-COCH.sub.2 CH.sub.3                                                 294      4-COCH.sub.2 CH.sub.3                                                 295      2-COCH.sub.2 CH.sub.2 CH.sub.3                                        296      3-COCH.sub.2 CH.sub.2 CH.sub.3                                        297      4-COCH.sub.2 CH.sub.2 CH.sub.3                                        298      2-COCH (CH.sub.3)CH.sub.3                                             299      3-COCH (CH.sub.3)CH.sub.3                                             300      4-COCH (CH.sub.3)CH.sub.3                                             301      2-Me-4-CHO                                                            302      2-Me-4-CH.sub.3 CO                                                    303      2-Me-4-CH.sub.3 CH.sub.2 CO                                           304      2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                  305      2-Me-4-CH.sub.3 CH (CH.sub.3)CO                                       306      2,5-Me.sub.2 -4-CHO                                                   307      2,5-Me.sub.2 -4-CH.sub.3 CO                                           308      2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                  309      2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                         310      2,5-Me.sub.2 -4-CH.sub.3 CH (CH.sub.3)CO                              311      2-Cl-4-CHO                                                            312      2-Cl-4-CH.sub.3 CO                                                    313      2-Cl-4-CH.sub.3 CH.sub.2 CO                                           314      2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                        315      2,5-Cl.sub.2 -4-CHO                                                   316      2,5-Cl.sub.2 -4-CH.sub.3 CO                                           317      2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                  318      2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                         319      2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                               320      2-C(NOCH.sub.3)CH.sub.3                                               321      3-C(NOCH.sub.3)CH.sub.3                                               322      4-C(NOCH.sub.3)CH.sub.3                                               323      2-C(NOC.sub.2 H.sub.5)CH.sub.3                                        324      3-C(NOC.sub.2 H.sub.5)CH.sub.3                                        325      4-C(NOC.sub.2 H.sub.5)CH.sub.3                                        326      2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     327      3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     328      4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     329      2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     330      3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     331      4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     332      2-C(NO-Allyl)-CH.sub.3                                                333      3-C(NO-Allyl)-CH.sub.3                                                334      4-C(NO-Allyl)-CH.sub.3                                                335      2-C(NO-trans-Chloroallyl)-CH.sub.3                                    336      3-C(NO-trans-Chloroallyl)-CH.sub.3                                    337      4-C(NO-trans-Chloroallyl)-CH.sub.3                                    338      2-C(NO-Propargyl)-CH.sub.3                                            339      3-C(NO-Propargyl)-CH.sub.3                                            340      4-C(NO-Propargyl)-CH.sub.3                                            341      2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     342      3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     343      4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     344      2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               345      3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               346      4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               347      2-CH.sub.3 -4-CHNOCH.sub.3                                            348      2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                     349      2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                  350      2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                  351      2-CH.sub.3 -4-CHNO-Allyl                                              352      2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                353      2-CH.sub.3 -4-CHNO-Propargyl                                          354      2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                  355      2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                            356      2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                  357      2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                           358      2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                        359      2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                        360      2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                    361      2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                        362      2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                363      2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                        364      2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                  365      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                           366      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                    367      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                 368      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                 369      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                             370      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                 371      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                         372      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                 373      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)           374      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                        375      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                 376      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)              377      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)              378      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                          379      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)              380      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                       381      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)              382      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)        383      2-C.sub.6 H.sub.5                                                     384      3-C.sub.6 H.sub.5                                                     385      4-C.sub.6 H.sub.5                                                     386      2-(2'-FC.sub.6 H.sub.4)                                               387      2-(3'-FC.sub.6 H.sub.4)                                               388      2-(4'-FC.sub.6 H.sub.4)                                               389      3-(2'-FC.sub.6 H.sub.4)                                               390      3-(3'-FC.sub.6 H.sub.4)                                               391      3-(4'-FC.sub.6 H.sub.4)                                               392      4-(2'-FC.sub.6 H.sub.4)                                               393      4-(3'-FC.sub.6 H.sub.4)                                               394      4-(4'-FC.sub.6 H.sub.4)                                               395      2-(2'-ClC.sub.6 H.sub.4)                                              396      2-(3'-ClC.sub.6 H.sub.4)                                              397      2-(4'-ClC.sub.6 H.sub.4)                                              398      3-(2'-ClC.sub.6 H.sub.4)                                              399      3-(3'-ClC.sub.6 H.sub.4)                                              400      3-(4'-ClC.sub.6 H.sub.4)                                              401      4-(2'-ClC.sub.6 H.sub.4)                                              402      4-(3'-ClC.sub.6 H.sub.4)                                              403      4-(4'-ClC.sub.6 H.sub.4)                                              405      2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       406      2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       407      2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       408      3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       409      3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       410      3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       411      4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       412      4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       413      4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       414      2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     415      2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     416      2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     417      3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     418      3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     419      3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     420      4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     421      4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     422      4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     423      2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          424      2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          425      2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          426      3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          427      3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          428      3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          429      4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          430      4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          431      4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          432      2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              433      2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              434      2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              435      3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              436      3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              437      3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              438      4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              439      4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              440      4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              441      2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      442      2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      443      2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      444      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      445      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      446      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      447      4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      448      4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      449      4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      450      2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       451      2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       452      2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       453      3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       454      3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       455      3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       456      4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       457      4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       458      4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       459      2-(2'-NCC.sub.6 H.sub.4)                                              460      2-(3'-NCC.sub.6 H.sub.4)                                              461      2-(4'-NCC.sub.6 H.sub.4)                                              462      3-(2'-NCC.sub.6 H.sub.4)                                              463      3-(3'-NCC.sub.6 H.sub.4)                                              464      3-(4'-NCC.sub.6 H.sub.4)                                              465      4-(2'-NCC.sub.6 H.sub.4)                                              466      4-(3'-NCC.sub.6 H.sub.4)                                              467      4-(4'-NCC.sub.6 H.sub.4)                                              468      2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       469      2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       470      2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       471      3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       472      3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       473      3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       474      4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       475      4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       476      4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       477      2-OC.sub.6 H.sub.5                                                    475      3-OC.sub.6 H.sub.5                                                    476      4-OC.sub.6 H.sub.5                                                    478      2-O-(2'-FC.sub.6 H.sub.4)                                             479      2-O-(3'-FC.sub.6 H.sub.4)                                             480      2-O-(4'-FC.sub.6 H.sub.4)                                             481      3-O-(2'-FC.sub.6 H.sub.4)                                             482      3-O-(3'-FC.sub.6 H.sub.4)                                             483      3-O-(4'-FC.sub.6 H.sub.4)                                             484      4-O-(2'-FC.sub.6 H.sub.4)                                             485      4-O-(3'-FC.sub.6 H.sub.4)                                             486      4-O-(4'-FC.sub.6 H.sub.4)                                             487      2-O-(2'-ClC.sub.6 H.sub.4)                                            488      2-O-(3'-ClC.sub.6 H.sub.4)                                            489      2-O-(4'-ClC.sub.6 H.sub.4)                                            490      3-O-(2'-ClC.sub.6 H.sub.4)                                            491      3-O-(3'-ClC.sub.6 H.sub.4)                                            492      3-O-(4'-ClC.sub.6 H.sub.4)                                            493      3-O-(4'-ClC.sub.6 H.sub.4)                                            494      4-O-(2'-ClC.sub.6 H.sub.4)                                            495      4-O-(3'-ClC.sub.6 H.sub.4)                                            496      4-O-(4'-ClC.sub.6 H.sub.4)                                            497      2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     498      2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     499      2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     500      3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     501      3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     502      3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     503      4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     504      4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     505      4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     506      2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   507      2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   508      2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   509      3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   510      3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   511      3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   512      4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   513      4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   514      4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   515      2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        516      2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        517      2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        518      3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        519      3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        520      3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        521      4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        522      4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        523      4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        524      2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            525      2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            526      2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            527      3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            528      3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            529      3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            530      4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            531      4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            532      4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            533      2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    534      2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    535      2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    536      3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    537      3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    538      3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    539      4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    540      4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    541      4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    542      2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     543      2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     544      2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     545      3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     546      3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     547      3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     548      4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     549      4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     550      4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     551      2-O-(2'-NCC.sub.6 H.sub.4)                                            552      2-O-(3'-NCC.sub.6 H.sub.4)                                            553      2-O-(4'-NCC.sub.6 H.sub.4)                                            554      3-O-(2'-NCC.sub.6 H.sub.4)                                            555      3-O-(3'-NCC.sub.6 H.sub.4)                                            556      3-O-(4'-NCC.sub.6 H.sub.4)                                            557      4-O-(2'-NCC.sub.6 H.sub.4)                                            558      4-O-(3'-NCC.sub.6 H.sub.4)                                            559      4-O-(4'-NCC.sub.6 H.sub.4)                                            560      2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     561      2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     562      2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     563      3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     564      3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     565      3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     566      4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     567      4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     568      4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     569      2-Pyridinyl-2'                                                        570      2-Pyridinyl-3'                                                        571      2-Pyridinyl-4'                                                        572      3-Pyridinyl-2'                                                        573      3-Pyridinyl-3'                                                        574      3-Pyridinyl-4'                                                        575      4-Pyridinyl-2'                                                        576      4-Pyridinyl-3'                                                        577      4-Pyridinyl-4'                                                        578      2-Pyrimidinyl-2'                                                      579      2-Pyrimidinyl-3'                                                      580      2-Pyrimidinyl-4'                                                      581      3-Pyrimidinyl-2'                                                      582      3-Pyrimidinyl-3'                                                      583      3-Pyrimidinyl-4'                                                      584      4-Pyrimidinyl-2'                                                      585      4-Pyrimidinyl-3'                                                      586      4-Pyrimidinyl-4'                                                      587      2-Pyrazolyl-1'                                                        588      2-Pyrazolyl-3'                                                        589      2-Pyrazolyl-4'                                                        590      3-Pyrazolyl-1'                                                        591      3-Pyrazolyl-3'                                                        592      3-Pyrazolyl-4'                                                        593      4-Pyrazolyl-1'                                                        594      4-Pyrazolyl-3'                                                        595      4-Pyrazolyl-4'                                                        596      2-Isoxazolyl-3'                                                       597      2-Isoxazolyl-4'                                                       598      2-Isoxazolyl-5'                                                       599      3-Isoxazolyl-3'                                                       600      3-Isoxazolyl-4'                                                       601      3-Isoxazolyl-5'                                                       602      4-Isoxazolyl-3'                                                       603      4-Isoxazolyl-4'                                                       604      4-Isoxazolyl-5'                                                       605      2-Isothiazolyl-3'                                                     606      2-Isothiazolyl-4'                                                     607      2-Isothiazolyl-5'                                                     608      3-Isothiazolyl-3'                                                     609      3-Isothiazolyl-4'                                                     610      3-Isothiazolyl-5'                                                     611      4-Isothiazolyl-3'                                                     612      4-Isothiazolyl-4'                                                     613      4-Isothiazolyl-5'                                                     614      2-Imidazolyl-1'                                                       615      2-Imidazolyl-2'                                                       616      2-Imidazolyl-4'                                                       617      3-Imidazolyl-1'                                                       618      3-Imidazolyl-2'                                                       619      3-Imidazolyl-4'                                                       620      4-Imidazolyl-1'                                                       621      4-Imidazolyl-2'                                                       622      4-Imidazolyl-4'                                                       623      2-Oxazolyl-2'                                                         624      2-Oxazolyl-4'                                                         625      2-Oxazolyl-5'                                                         626      3-Oxazolyl-2'                                                         627      3-Oxazolyl-4'                                                         628      3-Oxazolyl-5'                                                         629      4-Oxazolyl-2'                                                         630      4-Oxazolyl-4'                                                         631      4-Oxazolyl-5'                                                         632      2-Thiazolyl-2'                                                        633      2-Thiazolyl-4'                                                        634      2-Thiazolyl-5'                                                        635      3-Thiazolyl-2'                                                        636      3-Thiazolyl-4'                                                        637      3-Thiazolyl-5'                                                        638      4-Thiazolyl-2'                                                        639      4-Thiazolyl-4'                                                        640      4-Thiazolyl-5'                                                        641      2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)               642      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)        643      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)              .                                                                     644      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                         645      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                  646      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)               647      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)               648      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                           649      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)               650      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                       651      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)               652      2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)         653      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                         654      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                  655      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)               656      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)               657      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                           658      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)               659      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                       660      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)               661      2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)         662      2-O-n-C.sub.4 H.sub.9                                                 663      2-O-i-C.sub.4 H.sub.9                                                 664      2-O-s-C.sub.4 H.sub.9                                                 665      2-O-t-C.sub.4 H.sub.9                                                 666      2-Neopentyloxy                                                        667      3-O-n-C.sub.4 H.sub.9                                                 668      3-O-i-C.sub.4 H.sub.9                                                 669      3-O-s-C.sub.4 H.sub.9                                                 670      3-O-t-C.sub.4 H.sub.9                                                 671      3-Neopentyloxy                                                        672      4-O-n-C.sub.4 H.sub.9                                                 673      4-O-i-C.sub.4 H.sub.9                                                 674      4-O-s-C.sub.4 H.sub.9                                                 675      4-O-t-C.sub.4 H.sub.9                                                 676      4-Neopentyloxy                                                        677      3-CH.sub.3 -4-OCH.sub.3                                               678      3-CH.sub.3 -4-OC.sub.2 H.sub.5                                        679      3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                     680      3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                     681      3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                     682      3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                     683      3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                     684      3-CH.sub.3 -4-Neopentyloxy                                            685      2-CH.sub.3 -3-OCH.sub.3                                               686      2-CH.sub.3 -4-OCH.sub.3                                               687      2-CH.sub.3 -5-OCH.sub.3                                               688      2-CH.sub.3 -6-OCH.sub.3                                               689      3-CH.sub.3 -4-OCH.sub.3                                               690      3-CH.sub.3 -5-OCH.sub.3                                               691      3-CH.sub.3 -6-OCH.sub.3                                               692      4-CH.sub.3 -5-OCH.sub.3                                               693      4-CH.sub.3 -6-OCH.sub.3                                               694      4-CH.sub.3 -6-OCH.sub.3                                               695      2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                     696      2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                     697      2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                     698      2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                     699      3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                     700      3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                     701      3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                     702      4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                     703      4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                     704      5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                     705      2-Cl-3-OCH.sub.3                                                      706      2-Cl-4-OCH.sub.3                                                      707      2-Cl-5-OCH.sub.3                                                      708      2-Cl-6-OCH.sub.3                                                      709      3-Cl-4-OCH.sub.3                                                      710      3-Cl-5-OCH.sub.3                                                      711      3-Cl-6-OCH.sub.3                                                      712      4-Cl-5-OCH.sub.3                                                      713      4-Cl-6-OCH.sub.3                                                      714      5-Cl-6-OCH.sub.3                                                      ______________________________________                                    

                  TABLE 9                                                          ______________________________________                                          ##STR179##                                                                    I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 CH.sub.3                                                No.       B                                                                    ______________________________________                                         1         Pyrrolyl-3                                                           2         NCH.sub.3 -Pyrrolyl-3                                                3         NC.sub.6 H.sub.5 -Pyrrolyl-3                                         4         N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           5         N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           6         N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           7         N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          8         N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          9         N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          10        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           11        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           12        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           13        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  14        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  15        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  16        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  17        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  18        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  19        Pyrrolyl-2                                                           20        NCH.sub.3 -Pyrrolyl-2                                                21        NC.sub.6 H.sub.5 -Pyrrolyl-2                                         22        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           23        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           24        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           25        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          26        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          27        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          28        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           29        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           30        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           31        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  32        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  33        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  34        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  35        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  36        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  37        Furyl-2                                                              38        5-CH.sub.3 -Furyl-2                                                  39        5-C.sub.6 H.sub.5 -Furyl-2                                           40        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              41        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              42        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              43        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             44        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             45        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             46        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              47        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              48        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              49        5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     50        5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     51        5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     52        5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     53        5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     54        5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     55        4-CH.sub.3 -Furyl-2                                                  56        4-C.sub.6 H.sub.5 -Furyl-2                                           57        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              58        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              59        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              60        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             61        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             62        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             63        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              64        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              65        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              66        4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     67        4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     68        4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     69        4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     70        4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     71        4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     72        Thienyl-2                                                            73        5-CH.sub.3 -Thienyl-2                                                74        5-C.sub.6 H.sub.5 -Thienyl-2                                         75        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            76        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            77        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            78        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           79        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           80        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           81        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            82        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            83        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            84        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   85        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   86        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   87        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   88        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   89        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   90        4-CH.sub.3 -Thienyl-2                                                91        4-C.sub.6 H.sub.5 -Thienyl-2                                         92        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            93        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            94        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            95        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           96        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           97        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           98        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            99        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       NCH.sub.3 -Pyrazolyl-4                                               127       NC.sub.6 H.sub.5 -Pyrazolyl-4                                        128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 143       3-CH.sub.3 N-Methylpyrazolyl-4                                       144       3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                                145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   154       3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          155       3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          156       3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          157       3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          158       3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          159       3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          160       Isoxazolyl-5                                                         161       3-CH.sub.3 -Isoxazolyl-5                                             162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 -Isoxazolyl-3                                             198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 -Isothiazolyl-5                                           216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       2-CH.sub.3 -Oxazolyl-4                                               234       2-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           236       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           237       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           238       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          239       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          241       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           242       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           243       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           244       2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  245       2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  246       2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  247       2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  248       2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  249       2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       NCH.sub.3 -1,2,4-Triazolyl-5                                         269       3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                              270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          280       3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 281       3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 282       3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 283       3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 284       3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 285       3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        384       Pyridinyl-3                                                          385       1-Naphthyl                                                           386       2-Naphthyl                                                           ______________________________________                                    

                  TABLE 10                                                         ______________________________________                                          ##STR180##                                                                    I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 CH.sub.3                                                No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-C-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    181     3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    182     4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-CH.sub.3 CH.sub.2 CO                                            304     2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                   305     2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                         306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-CH.sub.3 CO                                            308     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   309     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          310     2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                311     2-Cl-4-CHO                                                             312     2-Cl-4-CH.sub.3 CO                                                     313     2-Cl-4-CH.sub.3 CH.sub.2 CO                                            314     2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                         315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-CH.sub.3 CO                                            317     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   318     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          319     2 5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NQ-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(-NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                   369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propagyl)                           372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                        381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-C-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4                                                       607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-C-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 11                                                         ______________________________________                                          ##STR181##                                                                    I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 CH.sub.3                                                No.        B                                                                   ______________________________________                                          1         Pyrrolyl-3                                                           2         NCH.sub.3 -Pyrrolyl-3                                                3         NC.sub.6 H.sub.5 -Pyrrolyl-3                                         4         N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           5         N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           6         N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           7         N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          8         N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          9         N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          10        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           11        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           12        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           13        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  14        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  15        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  16        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  17        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  18        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  19        Pyrrolyl-2                                                           20        NCH.sub.3 -Pyrrolyl-2                                                21        NC.sub.6 H.sub.5 -Pyrrolyl-2                                         22        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           23        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           24        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           25        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          26        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          27        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          28        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           29        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           30        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           31        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  32        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  33        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  34        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  35        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  36        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  37        Furyl-2                                                              38        5-CH.sub.3 -Furyl-2                                                  39        5-C.sub.6 H.sub.5 -Furyl-2                                           40        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              41        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              42        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              43        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             44        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             45        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             46        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              47        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              48        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              49        5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     50        5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     51        5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     52        5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     53        5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     54        5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     55        4-CH.sub.3 -Furyl-2                                                  56        4-C.sub.6 H.sub.5 -Furyl-2                                           57        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              58        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              59        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              60        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             61        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             62        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             63        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              64        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              65        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              66        4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     67        4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     68        4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     69        4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     70        4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     71        4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     72        Thienyl-2                                                            73        5-CH.sub.3 -Thienyl-2                                                74        5-C.sub.6 H.sub.5 -Thienyl-2                                         75        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            76        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            77        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            78        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           79        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           80        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           81        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            82        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            83        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            84        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   85        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   86        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   87        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   88        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   89        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   90        4-CH.sub.3 -Thienyl-2                                                91        4-C.sub.6 H.sub.5 -Thienyl-2                                         92        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            93        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            94        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            95        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           96        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           97        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           98        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            99        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                           100        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                           101        4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                  102        4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                  103        4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                  104        4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                  105        4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                  106        4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                  107        Thienyl-3                                                           108        5-CH.sub.3 -Thienyl-3                                               109        5-C.sub.6 H.sub.5 -Thienyl-3                                        110        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           111        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           112        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           113        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          114        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          115        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          116        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           117        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           118        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           119        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                  120        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                  121        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                  122        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                  123        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                  124        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                  125        Pyrazolyl-4                                                         126        NCH.sub.3 -Pyrazolyl-4                                              127        NC.sub.6 H.sub.5 -Pyrazolyl-4                                       128        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         129        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         130        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         131        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        132        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        133        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        134        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         135        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         136        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         137        N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                138        N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                139        N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                140        N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                141        N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                142        N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                143        3-CH.sub.3 N-Methylpyrazolyl-4                                      144        3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                               145        3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  146        3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  147        3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  148        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                 149        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                 150        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                 151        3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  152        3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  153        3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  154        3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         155        3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         156        3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         157        3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         158        3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         159        3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         160        Isoxazolyl-5                                                        161        3-CH.sub.3 -Isoxazolyl-5                                            162        3-C.sub.6 H.sub.5 -Isoxazolyl-5                                     163        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        164        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        165        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        166        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       167        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       168        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       169        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        170        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        171        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        172        3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               173        3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               174        3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               175        3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               176        3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               177        3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               178        4-Chloroisoxazolyl-5                                                179        3-CH.sub.3 -4-Chloroisoxazolyl-5                                    180        3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                             181        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                182        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                183        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                184        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               185        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               186        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               187        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                188        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                189        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                190        3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       191        3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       192        3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       193        3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       194        3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       195        3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       196        Isoxazolyl-3                                                        197        5-CH.sub.3 -Isoxazolyl-3                                            198        5-C.sub.6 H.sub.5 -Isoxazolyl-3                                     199        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        200        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        201        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        202        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       203        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       204        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       205        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        206        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        207        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        208        5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               209        5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               210        5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               211        5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               212        5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               213        5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               214        Isothiazolyl-5                                                      215        3-CH.sub.3 -Isothiazolyl-5                                          216        3-C.sub.6 H.sub.5 -Isothiazolyl-5                                   217        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      218        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      219        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      220        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     221        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     222        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     223        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      224        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      225        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      226        3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             227        3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             228        3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             229        3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             230        3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             231        3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             232        Oxazolyl-4                                                          233        2-CH.sub.3 -Oxazolyl-4                                              234        2-C.sub.6 H.sub.5 -Oxazolyl-4                                       235        2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          236        2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          237        2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          238        2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         239        2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         240        2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         241        2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          242        2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          243        2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          244        2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 245        2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 246        2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 247        2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 248        2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 249        2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 250        Thiazolyl-4                                                         251        2-CH.sub.3 -Thiazolyl-4                                             252        2-C.sub.6 H.sub.5 -Thiazolyl-4                                      253        2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         254        2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         255        2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         256        2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                        267        2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                        258        2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                        259        2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         260        2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         261        2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         262        2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                263        2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                264        2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                265        2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                266        2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                267        2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                268        NCH.sub.3 -1,2,4-Triazolyl-5                                        269        3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                             270        3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                      271        3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         272        3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         273        3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         274        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        275        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        276        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        277        3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         278        3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         279        3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         280        3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                281        3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                282        3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                283        3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                284        3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                285        3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2 ,4-Triazolyl-5               286        1,3,4-Oxadiazolyl-2                                                 287        5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                     288        5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                              289        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 290        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 291        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 292        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                293        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                294        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                295        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 296        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 297        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 298        5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        299        5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazdlyl-2                        300        5-(2'-CNC.sub.6 H.sub.4)-1,3,4-axadiazolyl-2                        301        5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        302        5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        303        5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        304        1,2,4-Oxadiazolyl-3                                                 305        5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                     306        5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                              307        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 308        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 309        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 310        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                311        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                312        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                313        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 314        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 315        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 316        5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        317        5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        318        5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        319        5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        320        5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        321        5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        322        1,2,4-Oxadiazolyl-5                                                 323        3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                     324        3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                              325        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 326        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 327        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 328        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                329        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                330        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                331        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 332        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 333        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 334        3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        335        3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        336        3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        337        3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        338        3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        339        3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        340        1,2,4-Thiadiazolyl-3                                                341        5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                    342        5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                             343        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                344        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                345        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                346        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               347        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               348        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               349        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                350        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                351        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                352        5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       353        5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       354        5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       355        5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       356        5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       357        5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       358        1,3,4-Thiadiazolyl-2                                                359        5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                    360        5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                             361        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                362        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                363        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                364        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               365        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               366        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               367        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                368        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                369        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                370        5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       371        5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       372        5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       373        5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       374        5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       375        5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       376        Pyridinyl-2                                                         377        Pyridinyl-4                                                         378        Pyridazinyl-3                                                       379        Pyridazinyl-4                                                       380        Pyridazinyl-2                                                       381        Pyrimidinyl-4                                                       382        Pyrimidinyl-5                                                       383        Pyrimidinyl-2                                                       384        Pyridinyl-3                                                         385        1-Naphthyl                                                          386        2-Naphthyl                                                          ______________________________________                                    

                  TABLE 12                                                         ______________________________________                                          ##STR182##                                                                    I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 CH.sub.3                                                No.       X.sub.m                                                              ______________________________________                                          1        H                                                                     2        2-F                                                                   3        3-F                                                                   4        4-F                                                                   5        2,4-F.sub.2                                                           6        2,4,6-F.sub.3                                                         7        2,3,4,5,6-F.sub.5                                                     8        2,3-F.sub.2                                                           9        2-Cl                                                                  10       3-Cl                                                                  11       4-Cl                                                                  12       2,3-Cl.sub.2                                                          13       2,4-Cl.sub.2                                                          14       2,5-Cl.sub.2                                                          15       2,6-Cl.sub.2                                                          16       3,4-Cl.sub.2                                                          17       3,5-Cl.sub.2                                                          18       2,3,4-Cl.sub.3                                                        19       2,3,5-Cl.sub.3                                                        20       2,3,6-Cl.sub.3                                                        21       2,4,5-Cl.sub.3                                                        22       2,4,6-Cl.sub.3                                                        23       3,4,5-Cl.sub.3                                                        24       2,3,4,6-Cl.sub.4                                                      25       2,3,5,6-Cl.sub.4                                                      26       2,3,4,5,6-Cl.sub.5                                                    27       2-Br                                                                  28       3-Br                                                                  29       4-Br                                                                  30       2,4-Br.sub.2                                                          31       2,5-Br.sub.2                                                          32       2,6-Br.sub.2                                                          33       2,4,6-Br.sub.3                                                        34       2,3,4,5,6-Br.sub.5                                                    35       2-I                                                                   36       3-I                                                                   37       4-I                                                                   38       2,4-I.sub.2                                                           39       2-Cl, 3-F                                                             40       2-Cl, 4-F                                                             41       2-Cl, 5-F                                                             42       2-Cl, 6-F                                                             43       2-Cl, 3-Br                                                            44       2-Cl, 4-Br                                                            45       2-Cl, 5-Br                                                            46       2-Cl, 6-Br                                                            47       2-Br, 3-Cl                                                            48       2-Br, 4-Cl                                                            49       2-Br, 5-Cl                                                            50       2-Br, 3-F                                                             51       2-Br, 4-F                                                             52       2-Br, 5-F                                                             53       2-Br, 6-F                                                             54       2-F, 3-Cl                                                             55       2-F, 4-Cl                                                             56       2-F, 5-Cl                                                             57       3-Cl, 4-F                                                             58       3-Cl, 5-F                                                             59       3-Cl, 4-Br                                                            60       3-Cl, 5-Br                                                            61       3-F, 4-Cl                                                             62       3-F, 4-Br                                                             63       3-Br, 4-Cl                                                            64       3-Br, 4-F                                                             65       2,6-Cl.sub.2, 4-Br                                                    66       2-CH.sub.3                                                            67       3-CH.sub.3                                                            68       4-CH.sub.3                                                            69       2,3-(CH.sub.3).sub.2                                                  70       2,4-(CH.sub.3).sub.2                                                  71       2,5-(CH.sub.3).sub.2                                                  72       2,6-(CH.sub.3).sub.2                                                  73       3,4-(CH.sub.3).sub.2                                                  74       3,5-(CH.sub.3).sub.2                                                  75       2,3,5-(CH.sub.3).sub.3                                                76       2,3,4-(CH.sub.3).sub.3                                                77       2,3,6-(CH.sub.3).sub.3                                                78       2,4,5-(CH.sub.3).sub.3                                                79       2,4,6-(CH.sub.3).sub.3                                                80       3,4,5-(CH.sub.3).sub.3                                                81       2,3,4,6-(CH.sub.3).sub.4                                              82       2,3,5,6-(CH.sub.3).sub.4                                              83       2,3,4,5,6-(CH.sub.3).sub.5                                            84       2-C.sub.2 H.sub.5                                                     85       3-C.sub.2 H.sub.5                                                     86       4-C.sub.2 H.sub.5                                                     87       2,4-(C.sub.2 H.sub.5).sub.2                                           88       2,6-(C.sub.2 H.sub.5).sub.2                                           89       3,5-(C.sub.2 H.sub.5).sub.2                                           90       2,4,6-(C.sub.2 H.sub.5).sub.3                                         91       2-n-C.sub.3 H.sub.7                                                   92       3-n-C.sub.3 H.sub.7                                                   93       4-n-C.sub.3 H.sub.7                                                   94       2-i-C.sub.3 H.sub.7                                                   95       3-i-C.sub.3 H.sub.7                                                   96       4-i-C.sub.3 H.sub.7                                                   97       2,4-(i-C.sub.3 H.sub.7).sub.2                                         98       2,6-(i-C.sub.3 H.sub.7).sub.2                                         99       3,5-(i-C.sub.3 H.sub.7).sub.2                                        100       2,4,6-(i-C.sub.3 H.sub.7).sub.3                                      101       2-s-C.sub.4 H.sub.9                                                  102       3-s-C.sub.4 H.sub.9                                                  103       4-s-C.sub.4 H.sub.9                                                  104       2-t-C.sub.4 H.sub.9                                                  105       3-t-C.sub.4 H.sub.9                                                  106       4-t-C.sub.4 H.sub.9                                                  107       2,3-(t-C.sub.4 H.sub.9).sub.2                                        108       2,4-(t-C.sub.4 H.sub.9).sub.2                                        109       2,5-(t-C.sub.4 H.sub.9).sub.2                                        110       2,6-(t-C.sub.4 H.sub.9).sub.2                                        111       3,4-(t-C.sub.4 H.sub.9).sub.2                                        112       2,4,6-(t-C.sub.4 H.sub.9).sub.3                                      113       4-n-C.sub.9 H.sub.19                                                 114       4-n-C.sub.12 H.sub.25                                                115       4-n-C.sub.15 H.sub.31                                                116       4-(1,1,3,3-Tetramethylbutyl)                                         117       4-(2,4,4-Trimethylpropyl)                                            118       2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                      119       2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                      120       2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                            121       2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                      122       2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                      123       2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                      124       2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                      125       3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                      126       2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                      127       2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                   128       2-Allyl                                                              129       3-Allyl                                                              130       4-Allyl                                                              131       2-Allyl, 6-CH.sub.3                                                  132       2-cyclo-C.sub.6 H.sub.11                                             133       3-cyclo-C.sub.6 H.sub.11                                             134       4-cyclo-C.sub.6 H.sub.11                                             135       2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                       136       2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                 137       2-CH.sub.2 C.sub.6 H.sub.5                                           138       3-CH.sub.2 C.sub.6 H.sub.5                                           139       4-CH.sub.2 C.sub.6 H.sub.5                                           140       2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                               141       2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                               142       2-C.sub.6 H.sub.5                                                    143       3-C.sub.6 H.sub.5                                                    144       4-C.sub.6 H.sub.5                                                    145       4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                              146       4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                              147       2-Cl, 4-C.sub.6 H.sub.5                                              148       2-Br, 4-C.sub.6 H.sub.5                                              149       2-C.sub.6 H.sub.5, 4-Cl                                              150       2-C.sub.6 H.sub.5, 4-Br                                              151       2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                     152       2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                     153       2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                     154       2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                     155       2-cyclo-C.sub.6 H.sub.11, 4-Cl                                       156       2-cyclo-C.sub.6 H.sub.11, 4-Br                                       157       2-Cl, 4-cyclo-C.sub.6 H.sub.11                                       158       2-Br, 4-cyclo-C.sub.6 H.sub.11                                       159       2-OCH.sub.3                                                          160       3-OCH.sub.3                                                          161       4-OCH.sub.3                                                          162       2-OC.sub.2 H.sub.5                                                   163       3-OC.sub.2 H.sub.5                                                   164       4-OC.sub.2 H.sub.5                                                   165       2-O-n-C.sub.3 H.sub.7                                                166       3-O-n-C.sub.3 H.sub.7                                                167       4-O-n-C.sub.3 H.sub.7                                                168       2-O-i-C.sub.3 H.sub.7                                                169       3-O-i-C.sub.3 H.sub.7                                                170       4-O-i-C.sub.3 H.sub.7                                                171       2-O-n-C.sub.6 H.sub.13                                               172       3-O-n-C.sub.6 H.sub.13                                               173       4-O-n-C.sub.6 H.sub.13                                               174       2-O-n-C.sub.8 H.sub.17                                               175       3-O-n-C.sub.8 H.sub.17                                               176       4-O-n-C.sub.8 H.sub.17                                               177       2-OCH.sub.2 C.sub.6 H.sub.5                                          178       3-OCH.sub.2 C.sub.6 H.sub.5                                          179       4-OCH.sub.2 C.sub.6 H.sub.5                                          180       2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                  181       3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                  182       4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                  183       2,4-(OCH.sub.3).sub.2                                                184       2-CF.sub.3                                                           185       3-CF.sub.3                                                           186       4-CF.sub.3                                                           187       2-OCF.sub.3                                                          188       3-OCF.sub.3                                                          189       4-OCF.sub.3                                                          190       3-OCH.sub.2 CHF.sub.2                                                191       2-NO.sub.2                                                           192       3-NO.sub.2                                                           193       4-NO.sub.2                                                           194       2-CN                                                                 195       3-CN                                                                 196       4-CN                                                                 197       2-CH.sub.3, 3-Cl                                                     198       2-CH.sub.3, 4-Cl                                                     199       2-CH.sub.3, 5-Cl                                                     200       2-CH.sub.3, 6-Cl                                                     201       2-CH.sub.3, 3-F                                                      202       2-CH.sub.3, 4-F                                                      203       2-CH.sub.3, 5-F                                                      204       2-CH.sub.3, 6-F                                                      205       2-CH.sub.3, 3-Br                                                     206       2-CH.sub.3, 4-Br                                                     207       2-CH.sub.3, 5-Br                                                     208       2-CH.sub.3, 6-Br                                                     209       2-Cl, 3-CH.sub.3                                                     210       2-Cl, 4-CH.sub.3                                                     211       2-Cl, 5-CH.sub.3                                                     212       2-F, 3-CH.sub.3                                                      213       2-F, 4-CH.sub.3                                                      214       2-F, 5-CH.sub.3                                                      215       2-Br, 3-CH.sub.3                                                     216       2-Br, 4-CH.sub.3                                                     217       2-Br, 5-CH.sub.3                                                     218       3-CH.sub.3, 4-Cl                                                     219       3-CH.sub.3, 5-Cl                                                     220       3-CH.sub.3, 4-F                                                      221       3-CH.sub.3, 5-F                                                      222       3-CH.sub.3, 4-Br                                                     223       3-CH.sub.3, 5-Br                                                     224       3-F, 4-CH.sub.3                                                      225       3-Cl, 4-CH.sub.3                                                     226       3-Br, 4-CH.sub.3                                                     227       2-Cl, 4,5-(CH.sub.3).sub.2                                           228       2-Br, 4,5-(CH.sub.3).sub.2                                           229       2-Cl, 3,5-(CH.sub.3).sub.2                                           230       2-Br, 3,5-(CH.sub.3).sub.2                                           231       2,6-Cl.sub.2, 4-CH.sub.3                                             232       2,6-F.sub.2, 4-CH.sub.3                                              233       2,6-Br.sub.2, 4-CH.sub.3                                             234       2,4-Br.sub.2, 6-CH.sub.3                                             235       2,4-F.sub.2, 6-CH.sub.3                                              236       2,4-Br.sub.2, 6-CH.sub.3                                             237       2,6-(CH.sub.3).sub.2, 4-F                                            238       2,6-(CH.sub.3).sub.2, 4-Cl                                           239       2,6-(CH.sub.3).sub.2, 4-Br                                           240       3,5-(CH.sub.3).sub.2, 4-F                                            241       3,5-(CH.sub.3).sub.2, 4-Cl                                           242       3,5-(CH.sub.3).sub.2, 4-Br                                           243       2,3,6-(CH.sub.3).sub.3, 4-F                                          244       2,3,6-(CH.sub.3).sub.3, 4-Cl                                         245       2,3,6-(CH.sub.3).sub.3, 4-Br                                         246       2,4-(CH.sub.3).sub.2, 6-F                                            247       2,4-(CH.sub.3).sub.2, 6-Cl                                           248       2,4-(CH.sub.3).sub.2, 6-Br                                           249       2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                250       2-Cl, 4-NO.sub.2                                                     251       2-NO.sub.2, 4-Cl                                                     252       2-OCH.sub.3, 5-NO.sub.2                                              253       2,4-Cl.sub.2, 5-NO.sub.2                                             254       2,4-Cl.sub.2, 6-NO.sub.2                                             255       2,6-Cl.sub.2, 4-NO.sub.2                                             256       2,6-Br.sub.2, 4-NO.sub.2                                             257       2,6-I.sub.2, 4-NO.sub.2                                              258       2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                259       2-CO.sub.2 CH.sub.3                                                  260       3-CO.sub.2 CH.sub.3                                                  261       4-CO.sub.2 CH.sub.3                                                  262       2-CO.sub.2 (C.sub.2 H.sub.5)                                         263       3-CO.sub.2 (C.sub.2 H.sub.5)                                         264       4-CO.sub.2 (C.sub.2 H.sub.5)                                         265       2-CO.sub.2 (n-C.sub.3 H.sub.7)                                       266       3-CO.sub.2 (n-C.sub.3 H.sub.7)                                       267       4-CO.sub.2 (n-C.sub.3 H.sub.7)                                       268       2-CO.sub.2 (i-C.sub.3 H.sub.7)                                       269       3-CO.sub.2 (i-C.sub.3 H.sub.7)                                       270       4-CO.sub.2 (i-C.sub.3 H.sub.7)                                       271       2-CO.sub.2 (n-C.sub.6 H.sub.13)                                      272       3-CO.sub.2 (n-C.sub.6 H.sub.13)                                      273       4-CO.sub.2 (n-C.sub.6 H.sub.13)                                      274       2-CH.sub.2 OCH.sub.3                                                 275       3-CH.sub.2 OCH.sub.3                                                 276       4-CH.sub.2 OCH.sub.3                                                 277       2-CH.sub.2 O(C.sub.2 H.sub.5)                                        278       3-CH.sub.2 O(C.sub.2 H.sub.5)                                        279       4-CH.sub.2 O(C.sub.2 H.sub.5)                                        280       2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      281       3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      282       4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      283       2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      284       3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      285       4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      286       2-CHO                                                                287       3-CHO                                                                288       4-CHO                                                                289       2-COCH.sub.3                                                         290       3-COCH.sub.3                                                         291       4-COCH.sub.3                                                         292       2-COCH.sub.2 CH.sub.3                                                293       3-COCH.sub.2 CH.sub.3                                                294       4-COCH.sub.2 CH.sub.3                                                295       2-COCH.sub.2 CH.sub.2 CH.sub.3                                       296       3-COCH.sub.2 CH.sub.2 CH.sub.3                                       297       4-COCH.sub.2 CH.sub.2 CH.sub.3                                       298       2-COCH(CH.sub.3)CH.sub.3                                             299       3-COCH(CH.sub.3)CH.sub.3                                             300       4-COCH(CH.sub.3)CH.sub.3                                             301       2-Me-4-CHO                                                           302       2-Me-4-CH.sub.3 CO                                                   303       2-Me-4-CH.sub.3 CH.sub.2 CO                                          304       2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                 305       2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                       306       2,5-Me.sub.2 -4-CHO                                                  307       2, 5-Me.sub.2 -4-CH.sub.3 CO                                         308       2, 5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                309       2, 5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                       310       2, 5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                             311       2-Cl-4-CHO                                                           312       2-Cl-4-CH.sub.3 CO                                                   313       2-Cl-4-CH.sub.3 CH.sub.2 CO                                          314       2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                       315       2,5-Cl.sub.2 -4-CHO                                                  316       2,5-Cl.sub.2 -4-CH.sub.3 CO                                          317       2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                 318       2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                        319       2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                              320       2-C(NOCH.sub.3)CH.sub.3                                              321       3-C(NOCH.sub.3)CH.sub.3                                              322       4-C(NOCH.sub.3)CH.sub.3                                              323       2-C(NOC.sub.2 H.sub.5)CH.sub.3                                       324       3-C(NOC.sub.2 H.sub.5)CH.sub.3                                       325       4-C(NOC.sub.2 H.sub.5)CH.sub.3                                       326       2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    327       3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    328       4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    329       2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    330       3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    331       4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    332       2-C(NO-Allyl)-CH.sub.3                                               333       3-C(NO-Allyl)-CH.sub.3                                               334       4-C(NO-Allyl)-CH.sub.3                                               335       2-C(NO-trans-Chloroallyl)-CH.sub.3                                   336       3-C(NO-trans-Chloroallyl)-CH.sub.3                                   337       4-C(NO-trans-Chloroallyl)-CH.sub.3                                   338       2-C(NO-Propargyl)-CH.sub.3                                           339       3-C(NO-Propargyl)-CH.sub.3                                           340       4-C(NO-Propargyl)-CH.sub.3                                           341       2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    342       3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    343       4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    344       2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              345       3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              346       4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              347       2-CH.sub.3 -4-CHNOCH.sub.3                                           348       2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                    349       2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                 350       2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                 351       2-CH.sub.3 -4-CHNO-Allyl                                             352       2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                               353       2-CH.sub.3 -4-CHNO-Propargyl                                         354       2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                 355       2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                           356       2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                 357       2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                          358       2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                       359       2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                       360       2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                   361       2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                       362       2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                               363       2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                       364       2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                 365       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                          366       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                   367       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                368       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                369       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                            370       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                371       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                        372       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                373       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)          374       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                       375       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                376       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)             377       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)             378       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                         379       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)             380       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                      381       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)             382       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)       383       2-C.sub.6 H.sub.5                                                    384       3-C.sub.6 H.sub.5                                                    385       4-C.sub.6 H.sub.5                                                    386       2-(2'-FC.sub.6 H.sub.4)                                              387       2-(3'-FC.sub.6 H.sub.4)                                              388       2-(4'-FC.sub.6 H.sub.4)                                              389       3-(2'-FC.sub.6 H.sub.4)                                              390       3-(3'-FC.sub.6 H.sub.4)                                              391       3-(4'-FC.sub.6 H.sub.4)                                              392       4-(2'-FC.sub.6 H.sub.4)                                              393       4-(3'-FC.sub.6 H.sub.4)                                              394       4-(4'-FC.sub.6 H.sub.4)                                              395       2-(2'-ClC.sub.6 H.sub.4)                                             396       2-(3'-ClC.sub.6 H.sub.4)                                             397       2-(4'-ClC.sub.6 H.sub.4)                                             398       3-(2'-ClC.sub.6 H.sub.4)                                             399       3-(3'-ClC.sub.6 H.sub.4)                                             400       3-(4'-ClC.sub.6 H.sub.4)                                             401       4-(2'-ClC.sub.6 H.sub.4)                                             402       4-(3'-ClC.sub.6 H.sub.4)                                             403       4-(4'-ClC.sub.6 H.sub.4)                                             405       2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      406       2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      407       2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      408       3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      409       3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      410       3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      411       4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      412       4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      413       4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      414       2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    415       2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    416       2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    417       3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    418       3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    419       3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    420       4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    421       4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    422       4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    423       2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         424       2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         425       2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         426       3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         427       3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         428       3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         429       4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         430       4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         43i       4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         432       2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             433       2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             434       2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             435       3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             436       3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             437       3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             438       4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             439       4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             440       4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             441       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     442       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     443       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     444       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     445       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     446       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     447       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     448       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     449       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     450       2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      451       2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      452       2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      453       3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      454       3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      455       3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      456       4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      457       4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      458       4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      459       2-(2'-NCC.sub.6 H.sub.4)                                             460       2-(3'-NCC.sub.6 H.sub.4)                                             461       2-(4'-NCC.sub.6 H.sub.4)                                             462       3-(2'-NCC.sub.6 H.sub.4)                                             463       3-(3'-NCC.sub.6 H.sub.4)                                             464       3-(4'-NCC.sub.6 H.sub.4)                                             465       4-(2'-NCC.sub.6 H.sub.4)                                             466       4-(3'-NCC.sub.6 H.sub.4)                                             467       4-(4'-NCC.sub.6 H.sub.4)                                             468       2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      469       2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      470       2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      471       3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      472       3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      473       3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      474       4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      475       4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      476       4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      477       2-OC.sub.6 H.sub.5                                                   475       3-OC.sub.6 H.sub.5                                                   476       4-OC.sub.6 H.sub.5                                                   478       2-O-(2'-FC.sub.6 H.sub.4)                                            479       2-O-(3'-FC.sub.6 H.sub.4)                                            480       2-O-(4'-FC.sub.6 H.sub.4)                                            481       3-O-(2'-FC.sub.6 H.sub.4)                                            482       3-O-(3'-FC.sub.6 H.sub.4)                                            483       3-O-(4'-FC.sub.6 H.sub.4)                                            484       4-O-(2'-FC.sub.6 H.sub.4)                                            485       4-O-(3'-FC.sub.6 H.sub.4)                                            486       4-O-(4'-FC.sub.6 H.sub.4)                                            487       2-O-(2'-ClC.sub.6 H.sub.4)                                           488       2-O-(3'-ClC.sub.6 H.sub.4)                                           489       2-O-(4'-ClC.sub.6 H.sub.4)                                           490       3-O-(2'-ClC.sub.6 H.sub.4)                                           491       3-O-(3'-ClC.sub.6 H.sub.4)                                           492       3-O-(4'-ClC.sub.6 H.sub.4)                                           493       3-O-(4'-ClC.sub.6 H.sub.4)                                           494       4-O-(2'-ClC.sub.6 H.sub.4)                                           495       4-O-(3'-ClC.sub.6 H.sub.4)                                           496       4-O-(4'-ClC.sub.6 H.sub.4)                                           497       2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    498       2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    499       2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    500       3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    501       3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    502       3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    503       4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    504       4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    505       4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    506       2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  507       2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  508       2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  509       3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  510       3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  511       3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  512       4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  513       4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  514       4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  515       2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       516       2-C-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       517       2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       518       3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       519       3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       520       3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       521       4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       522       4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       523       4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       524       2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           525       2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           526       2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           527       3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           528       3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           529       3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           530       4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           531       4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           532       4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           533       2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   534       2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   535       2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   536       3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   537       3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   538       3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   539       4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   540       4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   541       4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   542       2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    543       2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    544       2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    545       3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    546       3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    547       3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    548       4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    549       4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    550       4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    551       2-O-(2'-NCC.sub.6 H.sub.4)                                           552       2-O-(3'-NCC.sub.6 H.sub.4)                                           553       2-O-(4'-NCC.sub.6 H.sub.4)                                           554       3-O-(2'-NCC.sub.6 H.sub.4)                                           555       3-O-(3'-NCC.sub.6 H.sub.4)                                           556       3-O-(4'-NCC.sub.6 H.sub.4)                                           557       4-O-(2'-NCC.sub.6 H.sub.4)                                           558       4-O-(3'-NCC.sub.6 H.sub.4)                                           559       4-O-(4'-NCC.sub.6 H.sub.4)                                           560       2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                    561       2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                    562       2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                    563       3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                    564       3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                    565       3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                    566       4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                    567       4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                    568       4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                    569       2-Pyridinyl-2'                                                       570       2-Pyridinyl-3'                                                       571       2-Pyridinyl-4'                                                       572       3-Pyridinyl-2'                                                       573       3-Pyridinyl-3'                                                       574       3-Pyridinyl-4'                                                       575       4-Pyridinyl-2'                                                       576       4-Pyridinyl-3'                                                       577       4-Pyridinyl-4'                                                       578       2-Pyrimidinyl-2'                                                     579       2-Pyrimidinyl-3'                                                     580       2-Pyrimidinyl-4'                                                     581       3-Pyrimidinyl-2'                                                     582       3-Pyrimidinyl-3'                                                     583       3-Pyrimidinyl-4'                                                     584       4-Pyrimidinyl-2'                                                     585       4-Pyrimidinyl-3'                                                     586       4-Pyrimidinyl-4'                                                     587       2-Pyrazolyl-1'                                                       588       2-Pyrazolyl-3'                                                       589       2-Pyrazolyl-4'                                                       590       3-Pyrazolyl-1'                                                       591       3-Pyrazolyl-3'                                                       592       3-Pyrazolyl-4'                                                       593       4-Pyrazolyl-1'                                                       594       4-Pyrazolyl-3'                                                       595       4-Pyrazolyl-4'                                                       596       2-Isoxazolyl-3'                                                      597       2-Isoxazolyl-4'                                                      598       2-Isoxazolyl-5'                                                      599       3-Isoxazolyl-3'                                                      600       3-Isoxazolyl-4'                                                      601       3-Isoxazolyl-5'                                                      602       4-Isoxazolyl-3'                                                      603       4-Isoxazolyl-4'                                                      604       4-Isoxazolyl-5'                                                      605       2-Isothiazolyl-3'                                                    606       2-Isothiazolyl-4'                                                    607       2-Isothiazolyl-5'                                                    608       3-Isothiazolyl-3'                                                    609       3-Isothiazolyl-4'                                                    610       3-Isothiazolyl-5'                                                    611       4-Isothiazolyl-3'                                                    612       4-Isothiazolyl-4'                                                    613       4-Isothiazolyl-5'                                                    614       2-Imidazolyl-1'                                                      615       2-Imidazolyl-2'                                                      616       2-Imidazolyl-4'                                                      617       3-Imidazolyl-1'                                                      618       3-Imidazolyl-2'                                                      619       3-Imidazolyl-4'                                                      620       4-Imidazolyl-1'                                                      621       4-Imidazolyl-2'                                                      622       4-Imidazolyl-4'                                                      623       2-Oxazolyl-2'                                                        624       2-Oxazolyl-4'                                                        625       2-Oxazolyl-5'                                                        626       3-Oxazolyl-2'                                                        627       3-Oxazolyl-4'                                                        628       3-Oxazolyl-5'                                                        629       4-Oxazolyl-2'                                                        630       4-Oxazolyl-4'                                                        631       4-Oxazolyl-5'                                                        632       2-Thiazolyl-2'                                                       633       2-Thiazolyl-4'                                                       634       2-Thiazolyl-5'                                                       635       3-Thiazolyl-2'                                                       636       3-Thiazolyl-4'                                                       637       3-Thiazolyl-5'                                                       638       4-Thiazolyl-2'                                                       639       4-Thiazolyl-4'                                                       640       4-Thiazolyl-5'                                                       ______________________________________                                    

                  TABLE 13                                                         ______________________________________                                          ##STR183##                                                                    I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = CH.sub.2 CH.sub.3                                                No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                            2        NCH.sub.3 -Pyrrolyl-3                                                 3        NC.sub.6 H.sub.5 -Pyrrolyl-3                                          4        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            5        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            6        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            7        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           8        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           9        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           10       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            11       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            12       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            13       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   14       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   15       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   16       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   17       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   18       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   19       Pyrrolyl-2                                                            20       NCH.sub.3 -Pyrrolyl-2                                                 21       NC.sub.6 H.sub.5 -Pyrrolyl-2                                          22       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            23       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            24       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            25       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           26       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           27       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           28       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            29       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            30       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            31       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   32       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   33       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   34       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   35       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   36       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   37       Furyl-2                                                               38       5-CH.sub.3 -Furyl-2                                                   39       5-C.sub.6 H.sub.5 -Furyl-2                                            40       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               41       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               42       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               43       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              44       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              45       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              46       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               47       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               48       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               49       5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      50       5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      51       5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      52       5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      53       5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      54       5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      55       4-CH.sub.3 -Furyl-2                                                   56       4-C.sub.6 H.sub.5 -Furyl-2                                            57       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               58       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               59       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               60       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              61       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              62       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              63       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               64       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               65       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               66       4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      67       4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      68       4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      69       4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      70       4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      71       4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      72       Thienyl-2                                                             73       5-CH.sub.3 -Thienyl-2                                                 74       5-C.sub.6 H.sub.5 -Thienyl-2                                          75       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             76       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             77       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             78       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            79       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            80       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            81       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             82       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             83       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             84       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    85       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    86       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    87       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    88       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    89       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    90       4-CH.sub.3 -Thienyl-2                                                 91       4-C.sub.6 H.sub.5 -Thienyl-2                                          92       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             93       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             94       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             95       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            96       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            97       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            98       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             99       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       NCH.sub.3 -Pyrazolyl-4                                               127       NC.sub.6 H.sub.5 -Pyrazolyl-4                                        128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 143       3-CH.sub.3 N-Methylpyrazolyl-4                                       144       3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                                145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   154       3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          155       3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          156       3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          157       3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          158       3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          159       3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          160       Isoxazolyl-5                                                         161       3-CH.sub.3 -Isoxazolyl-5                                             162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 -Isoxazolyl-3                                             198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 -Isothiazolyl-5                                           216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       2-CH.sub.3 -Oxazolyl-4                                               234       2-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           236       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           237       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           238       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          239       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          241       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           242       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           243       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           244       2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  245       2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  246       2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  247       2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  248       2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  249       2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       NCH.sub.3 -1,2,4-Triazolyl-5                                         269       3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                              270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          280       3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 281       3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 282       3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 283       3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 284       3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 285       3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        384       Pyridinyl-3                                                          ______________________________________                                    

                                      TABLE 14                                     __________________________________________________________________________     Selected physical data of some compounds                                       No.                                                                               Compound                        .sup.1 H-NMR (ppm)                          __________________________________________________________________________      1                                                                                 ##STR184##                     3.8 (s, 3H); 3.75 (s, 3H)                    2                                                                                 ##STR185##                     3.8 (2s, 2 × 3H)                       3                                                                                 ##STR186##                     3.8 (s, 3H); 3.75 (s, 3H)                    4                                                                                 ##STR187##                     3.95 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H)        5                                                                                 ##STR188##                     4.05 (q, 2H, I = 7.5 Hz); 3.85 (s,                                             3H)                                          6                                                                                 ##STR189##                     4.0 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H)         7                                                                                 ##STR190##                     3.8 (s, 3H); 3.75 (s, 3H)                    8                                                                                 ##STR191##                     3.8 (s, 3H); 3.75 (s, 3H)                    9                                                                                 ##STR192##                     3.85 (s, 3H); 3.8 (s, 3H)                   10                                                                                 ##STR193##                     4.0 (s, 3H); 3.8 (s, 3H), 3.75 (s,                                             3H)                                         11                                                                                 ##STR194##                     3.8 (s, 3H); 3.75 (s, 3H)                   12                                                                                 ##STR195##                     3.8 (s, 3H); 3.75 (s, 3H)                   13                                                                                 ##STR196##                     3.8 (s, 3H); 3.75 (s, 3H)                   14                                                                                 ##STR197##                     3.8 (s, 3H); 3.75 (s, 3H) 66                15                                                                                 ##STR198##                     3.8 (s, 3H); 3.75 (s, 3H)                   16                                                                                 ##STR199##                     4.0 (q, 2H, I = 7.5 Hz); 3.8 (s, 3H)        17                                                                                 ##STR200##                     3.8 (2s, each 3H)                           18                                                                                 ##STR201##                     3.8 (2s, each 3H)                           19                                                                                 ##STR202##                     3.8 (s, 3H); 3.75 (s, 3H)                   20                                                                                 ##STR203##                     3.8 (s, 3H); 3.75 (s, 3H)                   21                                                                                 ##STR204##                     3.8 (s, 3H); 3.75 (s, 3H)                   22                                                                                 ##STR205##                     3.8 (s, 3H); 3.75 (s, 3H)                   23                                                                                 ##STR206##                     3.8 (s, 3H); 3.75 (s, 3H)                   24                                                                                 ##STR207##                     3.8 (s, 6H)                                 25                                                                                 ##STR208##                     3.75 (2s, each 3H)                          26                                                                                 ##STR209##                     3.8 (s, 3H); 3.75 (s, 3H)                   27                                                                                 ##STR210##                     3.8 (s, 3H); 3.75 (s, 3H)                   28                                                                                 ##STR211##                     3.8 (s, 3H); 3.75 (s, 3H)                   29                                                                                 ##STR212##                     3.8 (s, 3H); 3.75 (s, 3H)                   30                                                                                 ##STR213##                     3.8 (s, 6H)                                 __________________________________________________________________________

                  TABLE 52                                                         ______________________________________                                         Selected physical data of some compounds                                        ##STR214##                                                                                         mp       .sup.1 H-NMR (ppm) or IR                         No.     X.sub.m      (°C.)                                                                            (cm.sup.-1)                                      ______________________________________                                          1      H                     3.75 (2s, each 3H)                                2      2-CH.sub.3            3.75 (2s, each 3H)                                3      3-CH.sub.3            3.75 (2s, each 3H)                                4      2,4-(CH.sub.3).sub.2  3.75 (2s, each 3H)                                5      4-C.sub.2 H.sub.5     3.75 (2s, each 3H)                                6      4-i-C.sub.3 H.sub.7   3.75 (2s, each 3H)                                7      4-t-C.sub.4 H.sub.9   3.75 (2s, each 3H)                                8      3,4-(CH.sub.3).sub.2  3.75 (2s, each 3H)                                9      3-Cl                  3.75 (2s, each 3H)                               10      3-Br                  3.75 (2s, each 3H)                               11      3-CF.sub.3            3.75 (2s, each 3H)                               12      4-Br                  3.75 (2s, each 3H)                               13      4-F                   3.75 (2s, each 3H)                               14      4-CF.sub.3            3.75 (2s, each 3H)                               15      4-OCH.sub.3           3.8 (s, 3H); 3.75 (2s,                                                         each 3H)                                         16      4-CN                  3.75 (2s, each 3H)                               17      3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                                                    3.75 (2s, each 3H)                               18      3,4-Cl.sub.2          3.75 (2s, each 3H)                               19      3-CH.sub.3 -4-OCH.sub.3                                                                              3.85 (s, 3H); 3.75                                                             (2s, each 3H)                                    20      4-NO.sub.2   112                                                       21      3,5-(CH.sub.3).sub.2  3.75 (2s, each 3H)                               22      3-CH.sub.3 -4-Cl      3.75 (2s, each 3H)                               23      3-Cl-4-CH.sub.3       3.75 (2s, each 3H)                               ______________________________________                                    

                                      TABLE 53                                     __________________________________________________________________________     Selected physical data of some compounds                                        ##STR215##                                                                                                     .sup.1 H-NMR (ppm) or IR                      No.                                                                               X.sub.m                  mp (°C.)                                                                     (cm.sup.-1)                                   __________________________________________________________________________      1 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                                                   3.8 (s, 3H); 3.75 (s, 3H)                      2 2-CH.sub.3 -4-C(CH.sub.3)NO-(trans-CH.sub.2 CHCHCl)                                                          3.8 (s, 3H); 3.75 (s, 3H)                      3 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NOCH.sub.3                                                                3.95 (s, 3H); 3.8 (s,                                                          3H); 3.75 (s, 3H)                              4 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                                         3.8 (s, 3H); 3.75 (s, 3H)                      5 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-(trans-CH.sub.2 CHCHCl)                                                3.85 (s, 3H: 3.75 (s, 3H)                      6 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NOCH.sub.3                                                                   3.95 (s, 3H); 3.8 (s,                                                          3H); 3.75 (s, 3H)                              7 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NOC.sub.2 H.sub.5                                                            3.8 (s, 3H); 3.75 (s, 3H)                      8 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NO-Allyl                                                                     3.8 (s, 3H); 3.75 (s, 3H)                      9 2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NO-(trans-CH.sub.2 CHCHCl)                                                   3.8 (s, 3H); 3.75 (s, 3H)                     10 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)NOCH.sub.3                                                         3.95 (s, 3H); 3.8 (s,                                                          3H); 3.75 (s, 3H)                             11 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)NOC.sub.2 H.sub.5                                                  3.8 (s, 3H); 3.75 (s, 3H)                     12 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)NO-Allyl                                                           3.8 (s, 3H); 3.75 (s, 3H)                     13 2-Cl                          3.8 (s, 3H); 3.75 (s, 3H)                     14 4-Cl                          3.8 (s, 3H); 3.75 (s, 3H)                     15 2-CH.sub.3 -4-Cl              3.8 (s, 3H); 3.75 (s, 3H)                     16 2-Cl-4-CH.sub.3               3.8 (s, 3H); 3.75 (s, 3H)                     17 2-Cl-5-CH.sub.3               3.8 (s, 3H); 3.75 (s, 3H)                     18 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl                                                                  3.8 (s, 3H); 3.75 (s, 3H)                     19 2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)NO-(trans-CH.sub.2 CHCHCl)                                         3.8 (s, 3H); 3.75 (s, 3H)                     __________________________________________________________________________

                  TABLE 54                                                         ______________________________________                                          ##STR216##                                                                    I: R.sup.1 = CH.sub.3                                                          II: R.sup.1 = C.sub.2 H.sub.5                                                  No.     B                                                                      ______________________________________                                          1      2-Pyridyl                                                               2      3-Trifluormethyl-2-pyridyl                                              3      5-Trifluormethyl-2-pyridyl                                              4      3,5-Bis-(trifluoromethyl)-2-pyridyl                                     5      3,5-Dichloro-2-pyridyl                                                  6      3-Chloro-5-trifluoromethyl-2-pyridyl                                    7      3,5-Dichloro-2-pyridyl                                                  8      2-Chloro-4-trifluoromethylphenyl                                        9      2-Benzothiazolyl                                                       10      5-Chloro-4-methyl-2-benzimidazolyl                                     11      2-Benzoxazolyl                                                         12      1-Methyl-5-trifluoromethylimidazo 5,4-a!-pyridin-2-yl                  13      5-Chloro-2-pyrimidinyl                                                 14      4-Methyl-5-phenyl-2-thiazolin-2-yl                                     15      4-Methyl-5-phenyl-2-oxazolin-2-yl                                      16      7-Trifluoromethyl-4-quinolinyl                                         ______________________________________                                    

                  TABLE 55                                                         ______________________________________                                         Selected physical data of some compounds                                        ##STR217##                                                                    No.  X.sub.m   mp (°C.)                                                                         .sup.1 H-NMR (ppm) or IR (cm.sup.-1)                   ______________________________________                                         1    H              3.75 (s, 3H); 3.65 (s, 3H)                                 2    4-OCH.sub.3    3.8 (s, 3H); 3.75 (s, 3H); 3.65 (s, 3H)                    3    4-CH.sub.3     3.75 (s, 3H); 3.65 (s, 3H)                                 4    4-Cl           3.75 (s, 3H); 3.65 (s, 3H)                                 5    4-CF.sub.3     3.75 (s, 3H); 3.65 (s, 3H)                                 6    3,5-(CF.sub.3).sub.2                                                                          3.75 (s, 3H); 3.65 (s, 3H)                                 7    2,4-Cl.sub.2   3.75 (s, 3H); 3.65 (s, 3H)                                 8    3,4-Cl.sub.2   3.75 (s, 3H); 3.65 (s, 3H)                                 ______________________________________                                    

Example 6

O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

a) N-(2-Methylphenyl)-N-propionyl-hydroxylamine

At 25° to 30° C., 12,5 g (0.135 mol) of propionyl Chloroide and then 10.7 g (0.135 mol) of pyridine are dripped into 30 g of N-(2-methylphenyl)-hydroxylamine (crude product, prepared according to Bamberger et al., Anm. Chem. 316 (1901), 278; content approx. 80% =0.2 mol) in 500 ml of methylene Chloroide. The mixture is stirred for 30 minutes at room temperature, and is then extracted with dilute hydroChloroic acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 22.7 g (0.127 mol =63%) of the title compound as a yellow oil.

¹ H-NMR (COCl₃ ; δ in ppm): 9.4 (s, broad, 1H, OH); 7.2 (m, 4H, phenyl); 2.4 (s, 3H, CH₃); 2.1 (q, broad, 2H, CH₂); 1.1 (t, 3H, I=7 Hz, CH₃)

b) O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

At 25° to 30° C., a solution of 22.7 g (0.127 mol) (Example 6a) of N-(2-methylphenyl)-N-propionyl-hydroxylamine in 50 ml of dimethylformamide is dripped into a stirred mixture of 3.4 g (0.14 mol) of NaH in 150 ml of dimethylformamide. After completion of gas evolution (15 mins) 18.4 g (0.13 mol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 18 g (0.081 mol =64%) of the title compound as a yellow oil.

¹ H-NMR (COCl₃ ; δ in ppm): 7.2 (m, 4H, phenyl); 3.7 (s, broad, 3H, OCH₃); 2.6 (s, very broad, 2H, CH₂); 2.3 (s, 3H, CH₃); 1.2 (s, broad, 3H, CH₃)

Example 7

O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 2)

A mixture of 10 g (51.8 mmol) of the hydroxylamine derivative from Example 1, 11 g (61 mmol) of N-bromosuccinimide and 0.1 g of azoisobutyrodinitrile in 100 ml of CCl₄ is refluxed. One drop of bromine is added and the mixture is refluxed for a further 2.5 hours. The reaction mixture is cooled to room temperature, washed with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained in this sequence 3.4 g (7.9 mmol =15%) of O-methyl-N-(2-bromomethylphenyl)-d-(α, α-dibromopropionyl)-hydroxylamine, 3.8 g (10.8 mmol =21%) of O-methyl-N-(2-bromomethylphenyl)-N-(α-bromopropionyl)-hydroxylamine, 2.3 g (8.5 g (8.5 mmol =16%) of the title compound and 3.5 g of starting material, each as brown oils.

a) O-Methyl-N-(2-bromomethylphenyl)-N-(α, α-dibromopropionyl)-hydroxylamine

7.55 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 4.5 (s, 2H, CH₂, Br); 3.8 (s, 3H, OCH₃); 2.75 (s, 3H, CH₃)

b) O-Methyl-N-(2-bromomethylphenyl)-N-(α-bromopropionyl)-hydroxylamine

7.5 (s, broad, 1H, phenyl); 7.4 (s, broad, 3H, phenyl); 5.15 (s, broad, 1H, CH--Br); 4.5 (dd, broad, 2H, CH₂ --Br); 3.8 (s, 3H, OCH₃); 1.85 (s, broad, 3H, CH₃)

c) O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine

7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.5 (s, broad, 2H, CH₂ --Br); 3.75 (s, 3H, OCH₃); 2.55 (s, very broad, CH₂); 1.2 (t, 3H, I=7 Hz, CH₃)

Example 8

O-Methyl-N-(2-(2'-methylphenyloxymethyl)-phenyl)-N-propionyl-hydroxylamine (Table 21, No. 3)

0.12 g (5 mmol) of sodium hydride is added to a solution of 0.4 g (3.7 mmol) of o-cresol in 5 ml of dimethylformamide. Upon completion of gas evolution, 1 g (3.6 mmol) of the benzyl bromide from Example 2c is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is diluted with water and extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MgSO₄ and evaporated down. The residue is chromatographed with mixtures of cyclohexane and ethyl acetate using Al₂ O₃ and silica gel. There is obtained 0.4 g (1.33 mmol =37%) of the title compound as a yellow oil.

¹ H-NMR (COCl₃ ; δ in ppm): 7.7 (d, broad, 1H, phenyl); 7.35 (m, 3H, phenyl); 7.1 (m, 2H, phenyl); 6.85 (t, broad, 2H, phenyl); 5.05 (s, 2H, OCH₃); 3.7 (s, 3H, OCH₃); 2.55 (s, very broad, 2H, CH₂); 2.3 (s, 3H, CH₃); 1.2 (t, broad, 3H, CH₃)

Example 9

N-Methyl-N'-methoxy-N'-2-methylphenylurea (Table 21, No. 5)

a) Phenyl N-hydroxy-N-(2-methylphenyl)-carbamate

A mixture of 2.5 g (20 mmol) of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Anm. Chem. 316 (1901), 278), 3.5 g (25 mmol) of K₂ CO₃ and 3.5 g (22 mmol) of phenyl Chlorooformate in 20 ml of CH₂ Cl₂ is stirred for 2 hours at room temperature. The reaction mixture is then extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 2.0 g (8.2 mmol =42%) of the title compound as a colorless solid (mp=98° C.).

¹ H-NMR (COCl₃ ; δ in ppm): 7-7.6 (m, 10H, phenyl, OH); 2.35 (s, 3H, CH₃)

b) Phenyl N-methoxy-N-(2-methylphenyl)-carbamate

A mixture of 2.0 g (8.2 mmol) of the phenyl carbamate from Example 4a, 2 g (15 mmol) of K₂ CO₃ and 1.3 g (10 mmol) of dimethyl sulfate in 20 ml of acetone is stirred for 3 hours at room temperature. The reaction mixture is then filtered and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.5 g (5.8 mmol =71%) of the title compound as a colorless oil, which slowly crystallizes (mp=60° C.).

¹ H-NMR (COCl₃ ; δ in ppm): 7.1-7.5 (m, 9H, phenyl); 3.8 (s, 3H, OCH₃); 2.4 (s, 3H, CH₃)

c) N-Methyl-N'-methoxy-N'-2-methylphenylurea (Table 21, No. 5)

1.5 g (5.8 mmol) of the phenyl carbamate from Example 4b in 20 ml of 40% strength aqueous methylamine solution is stirred for 1 hour at 50° C. The reaction mixture is then cooled and extracted with CH₂ Cl₂. The combined organic phases are dried over MgCO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 0.6 g (3.1 mmol =53%) of the title compound as a colorless solid (mp=99° C.).

¹ H-NMR (COCl₃ ; δ in ppm): 7.2 (m, 4H, phenyl); 5.9 (s, broad, 1H, NH); 3.6 (s, 3H, OCH₃); 2.9 (d, 3H, I=approx. 2 Hz, N--CH₃); 2.3 (s, 3H, CH₃)

Example 18

N-Methyl-N'-methoxy-N'-(2-2',5'-dimethylphenoxymethyl)-phenyl)-urea

a) Phenyl N-methoxy-N-(2-bromomethylphenyl)-carbamate

A mixture of 125 g (0.486 mol) of methyl N-methoxy-N-(2-methylphenyl)-carbamate (Example 4b), 88 g (0.494 mol) of N-bromosuccinimide and 1 g of azoisobutyrodinitrile (AIBN) in 800 ml of CCl₄ is refluxed for about 12 hours. 10 g of N-bromosuccinimide is then added and the mixture is refluxed for about 4 hours. The reaction mixture is extracted with water and sodium thiosulfate solution, and the organic phase is dried over MgSO₄ and evaporated down under reduced pressure. The residue crystallizes, is stirred with hexane/methyl tert-butyl ether and suction dried. There is obtained 107 g (63%) of the title compound as a colorless solid.

¹ H-NMR (CDCl₃ ; δ in ppm): 7.1-7.6 (m, 9H, phenyl); 4.5 (s, 2H, CH₂ Br); 3.9 (s, 3H, OCH₃)

b) Phenyl N-methoxy-N-(2-(2',5'-dimethylphenoxymethyl)-phenyl)-carbamate

A mixture of 7 g (20 mmol) of the bromide of Example 5a and 3.3 g (22 mmol) of sodium iodide in 50 ml of acetone is refluxed for 30 minutes. The precipitated solid is then filtered off and the organic phase is evaporated down under reduced pressure. The crude product obtained is the iodide corresponding to Example 5a, which is used in the next reaction without any further purification.

The crude product obtained above is dissolved in 100 ml of dimethylformamide, 3 g (21.6 mmol) of K₂ CO₃ and 7.3 g (60 mmol) of 2,5-dimethylphenol are added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography using methylene chloride/cyclohexane (1:2) over Al₂ O₃. There is obtained 7.3 g (94%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in PPM): 7.7 (d, broad, 1H, phenyl); 7-7.6 (m, 9H, phenyl); 6.7 (m, 2H, phenyl); 5.2 (s, 2H, OCH₂); 3.85 (s, 3H, OCH₃); 2.3 (s, 6H, 2×CH₃).

c) N-Methyl-N'-methoxy-N'-(2-(2', 5'-dimethylphenoxymethyl)-phenyl)-urea (Table 1, No. V. 71)

A mixture of 3.4 g (8.8 mmol) of the phenyl carbamate of Example 5b and 20 ml of 40% strength aqueous methylamine solution is stirred for 2 hours at 50° C. The mixture is allowed to cool and is then extracted with methylene chloride. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of cyclohexane/ethyl acetate. There is obtained 1 g (36%) of the title compound as a colorless solid (mp=101° C).

¹ H-NMR (CDCl₃ ; δ in PPM):

7.75 (m, 1H, phenyl); 6.6-7.4 (m, 6H, phenyl); 6.0 (s, broad, NH); 5.15 (s, 2H, OCH₂); 3.65 (s, 3H, OCH₃); 2.9 (d, 3H, N--CH₃); 2.3 (s, 3H, CH₃); 2.25 (s, 3H, CH₃).

The compounds listed in the tables below may be prepared analogously. Compound I.1 from Table 15 has for instance the following formula ##STR218##

                  TABLE 15                                                         ______________________________________                                         I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, Z = CH.sub.3                                  III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5                           V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3                                No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5)3                                                91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    181     3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    182     4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2O (C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-CH.sub.3 CH.sub.2 CO                                            304     2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                   305     2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                         306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-CH.sub.3 CO                                            308     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   309     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          310     2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                311     2-Cl-4-CHO                                                             312     2-Cl-4-CH.sub.3 CO                                                     313     2-Cl-4-CH.sub.3 CH.sub.2 CO                                            314     2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                         315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-CH.sub.3 CO                                            317     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   318     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          319     2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NO-CH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               345     3-C(NO-CH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               346     4-C(NO-CH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                  369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 -CNO-n-C.sub.4 H.sub.9)                 373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                        381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 16                                                         ______________________________________                                          ##STR219##                                                                    I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, Z = CH.sub.3                                  III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5                           V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3                                No.      B                                                                     ______________________________________                                         1        Pyrrolyl-3                                                            2        NCH.sub.3 -Pyrrolyl-3                                                 3        NC.sub.6 H.sub.5 -Pyrrolyl-3                                          4        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            5        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            6        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            7        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           8        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           9        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           10       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            11       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            12       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            13       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   14       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   15       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   16       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   17       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   18       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   19       Pyrrolyl-2                                                            20       NCH.sub.3 -Pyrrolyl-2                                                 21       NC.sub.6 H.sub.5 -Pyrrolyl-2                                          22       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            23       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            24       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            25       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           26       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           27       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           28       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            29       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            30       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            31       N-(4'-CNC.sub.6 H.sub.4 )-Pyrrolyl-2                                  32       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   33       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   34       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   35       N-(3'-ClC.sub.6 H.sub.4 )-Pyrrolyl-2                                  36       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   37       Furyl-2                                                               38       5-CH.sub.3 -Furyl-2                                                   39       5-C.sub.6 H.sub.5 -Furyl-2                                            40       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               41       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               42       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               43       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              44       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              45       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              46       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               47       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               48       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               49       5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      50       5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      51       5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      52       5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      53       5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      54       5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      55       4-CH.sub.3 -Furyl-2                                                   56       4-C.sub.6 H.sub.5 -Furyl-2                                            57       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               58       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               59       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               60       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              61       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              62       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              63       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               64       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               65       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               66       4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      67       4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      68       4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      69       4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      70       4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      71       4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      72       Thienyl-2                                                             73       5-CH.sub.3 -Thienyl-2                                                 74       5-C.sub.6 H.sub.5 -Thienyl-2                                          75       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             76       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             77       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             78       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            79       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            80       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            81       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             82       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             83       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             84       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    85       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    86       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    87       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    88       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    89       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    90       4-CH.sub.3 -Thienyl-2                                                 91       4-C.sub.6 H.sub.5 -Thienyl-2                                          92       4-(4'-,CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            93       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             94       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             95       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            96       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            97       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            98       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             99       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             100      4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             101      4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    102      4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    103      4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    104      4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    105      4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    106      4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    107      Thienyl-3                                                             108      5-CH.sub.3 -Thienyl-3                                                 109      5-C.sub.6 H.sub.5 -Thienyl-3                                          110      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                             111      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                             112      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                             113      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                            114      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                            115      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                            116      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                             117      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                             118      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                             119      5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                    120      5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                    121      5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                    122      5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                    123      5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                    124      5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                    125      Pyrazolyl-4                                                           126      NCH.sub.3 -Pyrazolyl-4                                                127      NC.sub.6 H.sub.5 -Pyrazolyl-4                                         128      N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                           129      N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                           130      N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                           131      N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                          132      N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                          133      N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                          134      N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                           135      N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                           136      N-(2'-NO.sub.2 C.sub.6 HA)-Pyrazolyl-4                                137      N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                  138      N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                  139      N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                  140      N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                  141      N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                  142      N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                  143      3-CH.sub.3 N-Methylpyrazolyl-4                                        144      3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                                 145      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   146      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   147      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   148      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  149      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  150      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  151      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   152      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   153      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   154      3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          155      3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          156      3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          157      3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          158      3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          159      3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          160      Isoxazolyl-5                                                          161      3-CH.sub.3 -Isoxazolyl-5                                              162      3-C.sub.6 H.sub.5 -Isoxazolyl-5                                       163      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                          164      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                          165      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                          166      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                         167      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                         168      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                         169      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                          170      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                          171      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                          172      3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                 173      3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                 174      3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                 175      3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                 176      3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                 177      3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                 178      4-Chloroisoxazolyl-5                                                  179      3-CH.sub.3 -4-Chloroisoxazolyl-5                                      180      3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                               181      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  182      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  183      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  184      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 185      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 186      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 187      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  188      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  189      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  190      3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         191      3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         192      3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         193      3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         194      3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         195      3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         196      Isoxazolyl-3                                                          197      5-CH.sub.3 -Isoxazolyl-3                                              198      5-C.sub.6 H.sub.5 -Isoxazolyl-3                                       199      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                          200      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                          201      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                          202      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                         203      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                         204      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                         205      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                          206      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                          207      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                          208      5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                 209      5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                 210      5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                 211      5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                 212      5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                 213      5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                 214      Isothiazolyl-5                                                        215      3-CH.sub.3 -Isothiazolyl-5                                            216      3-C.sub.6 H.sub.5 -Isothiazolyl-5                                     217      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                        218      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                        219      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                        220      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                       221      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                       222      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                       223      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                        224      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                        225      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                        226      3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                               227      3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                               228      3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                               229      3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                               230      3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                               231      3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                               232      Oxazolyl-4                                                            233      2-CH.sub.3 -Oxazolyl-4                                                234      2-C.sub.6 H.sub.5 -Oxazolyl-4                                         235      2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                            236      2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                            237      2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                            238      2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                           239      2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                           240      2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                           241      2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                            242      2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                            243      2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                            244      2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                   245      2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                   246      2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                   247      2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                   248      2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                   249      2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                   250      Thiazolyl-4                                                           251      2-CH.sub.3 -Thiazolyl-4                                               252      2-C.sub.6 H.sub.5 -Thiazolyl-4                                        253      2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                           254      2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                           255      2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                           256      2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                          267      2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                          258      2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                          259      2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                           260      2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                           261      2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                           262      2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                  263      2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                  264      2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                  265      2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                  266      2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                  267      2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                  268      NCH.sub.3 -1,2,4-Triazolyl-5                                          269      3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                               270      3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                        271      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          272      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          273      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          274      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         275      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         276      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         277      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          278      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          279      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          280      3-(4'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 281      3-(3'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 282      3-(2'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 283      3-(4'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 284      3-(3'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 285      3-(2'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 286      1,3,4-Oxadiazolyl-2                                                   287      5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                       288      5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                289      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   290      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   291      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   292      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  293      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  294      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  295      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   296      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   297      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   298      5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          299      5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          300      5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          301      5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          302      5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          303      5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          304      1,2,4-Oxadiazolyl-3                                                   305      5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                       306      5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                307      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   308      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   309      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   310      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  311      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  312      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  313      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   314      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   315      5-(2'-NO.sub.2 -C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316      5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          317      5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          318      5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          319      5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          320      5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          321      5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          322      1,2,4-Oxadiazolyl-5                                                   323      3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                       324      3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                325      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   326      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   327      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   328      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  329      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  330      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  331      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   332      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   333      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   334      3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          335      3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          336      3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          337      3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          338      3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          339      3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          340      1,2,4-Thiadiazolyl-3                                                  341      5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                      342      5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                               343      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  344      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  345      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  346      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 347      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 348      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 349      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  350      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  351      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  352      5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         353      5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         354      5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         355      5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         356      5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         357      5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         358      1,3,4-Thiadiazolyl-2                                                  359      5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                      360      5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                               361      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  362      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  363      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  364      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 365      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 366      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 367      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  368      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  369      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  370      5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         371      5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         372      5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         373      5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         374      5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         375      5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         376      Pyridinyl-2                                                           377      Pyridinyl-4                                                           378      Pyridazinyl-3                                                         379      Pyridazinyl-4                                                         380      Pyridazinyl-2                                                         381      Pyrimidinyl-4                                                         382      Pyrimidinyl-5                                                         383      Pyrimidinyl-2                                                         384      Pyridinyl-3                                                           385      1-Naphthyl                                                            386      2-Naphthyl                                                            ______________________________________                                    

                  TABLE 17                                                         ______________________________________                                          ##STR220##                                                                    I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                            II: R.sup.1 CH.sub.2 CH.sub.3, Z = CH.sub.3                                    III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5                           V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH                                      NO.       X.sub.m                                                              ______________________________________                                         1         H                                                                    2         2-F                                                                  3         3-F                                                                  4         4-F                                                                  5         2,4-F.sub.2                                                          6         2,4,6-F.sub.3                                                        7         2,3,4,5,6-F.sub.5                                                    8         2,3-F.sub.2                                                          9         2-Cl                                                                 10        3-Cl                                                                 11        4-Cl                                                                 12        2,3-Cl.sub.2                                                         13        2,4-Cl.sub.2                                                         14        2,5-Cl.sub.2                                                         15        2,6-Cl.sub.2                                                         16        3,4-Cl.sub.2                                                         17        3,5-Cl.sub.2                                                         18        2,3,4-Cl.sub.3                                                       19        2,3,5-Cl.sub.3                                                       20        2,3,6-Cl.sub.3                                                       21        2,4,5-Cl.sub.3                                                       22        2,4,6-Cl.sub.3                                                       23        3,4,5-Cl.sub.3                                                       24        2,3,4,6-Cl.sub.4                                                     25        2,3,5,6-Cl.sub.4                                                     26        2,3,4,5,6-Cl.sub.5                                                   27        2-Br                                                                 28        3-Br                                                                 29        4-Br                                                                 30        2,4-Br.sub.2                                                         31        2,5-Br.sub.2                                                         32        2,6-Br.sub.2                                                         33        2,4,6-Br.sub.3                                                       34        2,3,4,5,6-Br.sub.5                                                   35        2-I                                                                  36        3-I                                                                  37        4-I                                                                  38        2,4-I.sub.2                                                          39        2-Cl, 3-F                                                            40        2-Cl, 4-F                                                            41        2-Cl, 5-F                                                            42        2-Cl, 6-F                                                            43        2-Cl, 3-Br                                                           44        2-Cl, 4-Br                                                           45        2-Cl, 5-Br                                                           46        2-Cl, 6-Br                                                           47        2-Br, 3-Cl                                                           48        2-Br, 4-Cl                                                           49        2-Br, 5-Cl                                                           50        2-Br, 3-F                                                            51        2-Br, 4-F                                                            52        2-Br, 5-F                                                            53        2-Br, 6-F                                                            54        2-F, 3-Cl                                                            55        2-F, 4-Cl                                                            56        2-F, 5-Cl                                                            57        3-Cl, 4-F                                                            58        3-Cl, 5-F                                                            59        3-Cl, 4-Br                                                           60        3-Cl, 5-Br                                                           61        3-F, 4-Cl                                                            62        3-F, 4-Br                                                            63        3-Br, 4-Cl                                                           64        3-Br, 4-F                                                            65        2,6-Cl.sub.2, 4-Br                                                   66        2-CH.sub.3                                                           67        3-CH.sub.3                                                           68        4-CH.sub.3                                                           69        2,3-(CH.sub.3).sub.2                                                 70        2,4-(CH.sub.3).sub.2                                                 71        2,5-(CH.sub.3).sub.2                                                 72        2,6-(CH.sub.3).sub.2                                                 73        3,4-(CH.sub.3).sub.2                                                 74        3,5-(CH.sub.3).sub.2                                                 75        2,3,5-(CH.sub.3).sub.3                                               76        2,3,4-(CH.sub.3).sub.3                                               77        2,3,6-(CH.sub.3).sub.3                                               78        2,4,5-(CH.sub.3).sub.3                                               79        2,4,6-(CH.sub.3).sub.3                                               80        3,4,5-(CH.sub.3).sub.3                                               81        2,3,4,6-(CH.sub.3).sub.4                                             82        2,3,5,6-(CH.sub.3).sub.4                                             83        2,3,4,5,6-(CH.sub.3).sub.5                                           84        2-C.sub.2 H.sub.5                                                    85        3-C.sub.2 H.sub.5                                                    86        4-C.sub.2 H.sub.5                                                    87        2,4-(C.sub.2 H.sub.5).sub.2                                          88        2,6-(C.sub.2 H.sub.5).sub.2                                          89        3,5-(C.sub.2 H.sub.5).sub.2                                          90        2,4,6-(C.sub.2 H.sub.5).sub.3                                        91        2-n-C.sub.3 H.sub.7                                                  92        3-n-C.sub.3 H.sub.7                                                  93        4-n-C.sub.3 H.sub.7                                                  94        2-i-C.sub.3 H.sub.7                                                  95        3-i-C.sub.3 H.sub.7                                                  96        4-i-C.sub.3 H.sub.7                                                  97        2,4-(i-C.sub.3 H.sub.7).sub.2                                        98        2,6-(i-C.sub.3 H.sub.7).sub.2                                        99        3,5-(i-C.sub.3 H.sub.7).sub.2                                        100       2,4,6-(i-C.sub.3 H.sub.7).sub.3                                      101       2-s-C.sub.4 H.sub.9                                                  102       3-s-C.sub.4 H.sub.9                                                  103       4-s-C.sub.4 H.sub.9                                                  104       2-t-C.sub.4 H.sub.9                                                  105       3-t-C.sub.4 H.sub.9                                                  106       4-t-C.sub.4 H.sub.9                                                  107       2,3-(t-C.sub.4 H.sub.9).sub.2                                        108       2,4-(t-C.sub.4 H.sub.9).sub.2                                        109       2,5-(t-C.sub.4 H.sub.9).sub.2                                        110       2,6-(t-C.sub.4 H.sub.9).sub.2                                        111       3,4-(t-C.sub.4 H.sub.9).sub.2                                        112       2,4,6-(t-C.sub.4 H.sub.9).sub.3                                      113       4-n-C.sub.9 H.sub.19                                                 114       4-n-C.sub.12 H.sub.25                                                115       4-n-C.sub.15 H.sub.31                                                116       4-(1,1,3,3-Tetramethylbutyl)                                         117       4-(2,4,4-Trimethylpropyl)                                            118       2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                      119       2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                      120       2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                            121       2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                      122       2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                      123       2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                      124       2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                      125       3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                      126       2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                      127       2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                   128       2-Allyl                                                              129       3-Allyl                                                              130       4-Allyl                                                              131       2-Allyl, 6-CH.sub.3                                                  132       2-cyclo-C.sub.6 H.sub.11                                             133       3-cyclo-C.sub.6 H.sub.11                                             134       4-cyclo-C.sub.6 H.sub.11                                             135       2,4-(Cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                       136       2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                 137       2-CH.sub.2 C.sub.6 H.sub.5                                           138       3-CH.sub.2 C.sub.6 H.sub.5                                           139       4-CH.sub.2 C.sub.6 H.sub.5                                           140       2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                               141       2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                               142       2-C.sub.6 H.sub.5                                                    143       3-C.sub.6 H.sub.5                                                    144       4-C.sub.6 H.sub.5                                                    145       4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                              146       4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                              147       2-Cl, 4-C.sub.6 H.sub.5                                              148       2-Br, 4-C.sub.6 H.sub.5                                              149       2-C.sub.6 H.sub.5, 4-Cl                                              150       2-C.sub.6 H.sub.5, 4-Br                                              151       2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                     152       2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                     153       2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                     154       2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                     155       2-cyclo-C.sub.6 H.sub.11, 4-Cl                                       156       2-cyclo-C.sub.6 H.sub.11, 4-Br                                       157       2-Cl, 4-cyclo-C.sub.6 H.sub.11                                       158       2-Br, 4-cyclo-C.sub.6 H.sub.11                                       159       2-OCH.sub.3                                                          160       3-OCH.sub.3                                                          161       4-OCH.sub.3                                                          162       2-OC.sub.2 H.sub.5                                                   163       3-OC.sub.2 H.sub.5                                                   164       4-OC.sub.2 H.sub.5                                                   165       2-O-n-C.sub.3 H.sub.7                                                166       3-O-n-C.sub.3 H.sub.7                                                167       4-O-n-C.sub.3 H.sub.7                                                168       2-O-i-C.sub.3 H.sub.7                                                169       3-O-i-C.sub.3 H.sub.7                                                170       4-O-i-C.sub.3 H.sub.7                                                171       2-O-n-C.sub.6 H.sub.13                                               172       3-O-n-C.sub.6 H.sub.13                                               173       4-O-n-C.sub.6 H.sub.13                                               174       2-O-n-C.sub.8 H.sub.17                                               175       3-O-n-C.sub.8 H.sub.17                                               176       4-O-n-C.sub.8 H.sub.17                                               177       2-OCH.sub.2 C.sub.6 H.sub.5                                          178       3-OCH.sub.2 C.sub.6 H.sub.5                                          179       4-OCH.sub.2 C.sub.6 H.sub.5                                          180       2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                  181       3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                  182       4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                  183       2,4-(OCH.sub.3).sub.2                                                184       2-CF.sub.3                                                           185       3-CF.sub.3                                                           186       4-CF.sub.3                                                           187       2-OCF.sub.3                                                          188       3-OCF.sub.3                                                          189       4-OCF.sub.3                                                          190       3-OCH.sub.2 CHF.sub.2                                                191       2-NO.sub.2                                                           192       3-NO.sub.2                                                           193       4-NO.sub.2                                                           194       2-CN                                                                 195       3-CN                                                                 196       4-CN                                                                 197       2-CH.sub.3, 3-Cl                                                     198       2-CH.sub.3, 4-Cl                                                     199       2-CH.sub.3, 5-Cl                                                     200       2-CH.sub.3, 6-Cl                                                     201       2-CH.sub.3, 3-F                                                      202       2-CH.sub.3, 4-F                                                      203       2-CH.sub.3, 5-F                                                      204       2-CH.sub.3, 6-F                                                      205       2-CH.sub.3, 3-Br                                                     206       2-CH.sub.3, 4-Br                                                     207       2-CH.sub.3, 5-Br                                                     208       2-CH.sub.3, 6-Br                                                     209       2-Cl, 3-CH.sub.3                                                     210       2-Cl, 4-CH.sub.3                                                     211       2-Cl, 5-CH.sub.3                                                     212       2-F, 3-CH.sub.3                                                      213       2-F, 4-CH.sub.3                                                      214       2-F, 5-CH.sub.3                                                      215       2-Br, 3-CH.sub.3                                                     216       2-Br, 4-CH.sub.3                                                     217       2-Br, 5-CH.sub.3                                                     218       3-CH.sub.3, 4-Cl                                                     219       3-CH.sub.3, 5-Cl                                                     220       3-CH.sub.3, 4-F                                                      221       3-CH.sub.3, 5-F                                                      222       3-CH.sub.3, 4-Br                                                     223       3-CH.sub.3, 5-Br                                                     224       3-F, 4-CH.sub.3                                                      225       3-Cl, 4-CH.sub.3                                                     226       3-Br, 4-CH.sub.3                                                     227       2-Cl, 4,5-(CH.sub.3).sub.2                                           228       2-Br, 4,5-(CH.sub.3).sub.2                                           229       2-Cl, 3,5-(CH.sub.3).sub.2                                           230       2-Br, 3,5-(CH.sub.3).sub.2                                           231       2,6-Cl.sub.2, 4-CH.sub.3                                             232       2,6-F.sub.2, 4-CH.sub.3                                              233       2,6-Br.sub.2, 4-CH.sub.3                                             234       2,4-Br.sub.2, 6-CH.sub.3                                             235       2,4-F.sub.2, 6-CH.sub.3                                              236       2,4-Br.sub.2, 6-CH.sub.3                                             237       2,6-(CH.sub.3).sub.2, 4-F                                            238       2,6-(CH.sub.3).sub.2, 4-Cl                                           239       2,6-(CH.sub.3).sub.2, 4-Br                                           240       3,5-(CH.sub.3).sub.2, 4-F                                            241       3,5-(CH.sub.3).sub.2, 4-Cl                                           242       3,5-(CH.sub.3).sub.2, 4-Br                                           243       2,3,6-(CH.sub.3).sub.3, 4-F                                          244       2,3,6-(CH.sub.3).sub.3, 4-Cl                                         245       2,3,6-(CH.sub.3).sub.3, 4-Br                                         246       2,4-(CH.sub.3).sub.2, 6-F                                            247       2,4-(CH.sub.3).sub.2, 6-Cl                                           248       2,4-(CH.sub.3).sub.2, 6-Br                                           249       2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                250       2-Cl, 4-NO.sub.2                                                     251       2-NO.sub.2, 4-Cl                                                     252       2-OCH.sub.3, 5-NO.sub.2                                              253       2,4-Cl.sub.2, 5-NO.sub.2                                             254       2,4-Cl.sub.2, 6-NO.sub.2                                             255       2,6-Cl.sub.2, 4-NO.sub.2                                             256       2,6-Br.sub.2, 4-NO.sub.2                                             257       2,6-I.sub.2, 4-NO.sub.2                                              258       2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                259       2-CO.sub.2 CH.sub.3                                                  260       3-CO.sub.2 CH.sub.3                                                  261       4-CO.sub.2 CH.sub.3                                                  262       2-CO.sub.2 (C.sub.2 H.sub.5)                                         263       3-CO.sub.2 (C.sub.2 H.sub.5)                                         264       4-CO.sub.2 (C.sub.2 H.sub.5)                                         265       2-CO.sub.2 (n-C.sub.3 H.sub.7)                                       266       3-CO.sub.2 (n-C.sub.3 H.sub.7)                                       267       4-CO.sub.2 (n-C.sub.3 H.sub.7)                                       268       2-CO.sub.2 (i-C.sub.3 H.sub.7)                                       269       3-CO.sub.2 (i-C.sub.3 H.sub.7)                                       270       4-CO.sub.2 (i-C.sub.3 H.sub.7)                                       271       2-CO.sub.2 (n-C.sub.6 H.sub.13)                                      272       3-CO.sub.2 (n-C.sub.6 H.sub.13)                                      273       4-CO.sub.2 (n-C.sub.6 H.sub.13)                                      274       2-CH.sub.2 OCH.sub.3                                                 275       3-CH.sub.2 OCH.sub.3                                                 276       4-CH.sub.2 OCH.sub.3                                                 277       2-CH.sub.2 O(C.sub.2 H.sub.5)                                        278       3-CH.sub.2 O(C.sub.2 H.sub.5)                                        279       4-CH.sub.2 O(C.sub.2 H.sub.5)                                        280       2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      281       3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      282       4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                      283       2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      284       3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      285       4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                      286       2-CHO                                                                287       3-CHO                                                                288       4-CHO                                                                289       2-COCH.sub.3                                                         290       3-COCH.sub.3                                                         291       4-COCH.sub.3                                                         292       2-COCH.sub.2 CH.sub.3                                                293       3-COCH.sub.2 CH.sub.3                                                294       4-COCH.sub.2 CH.sub.3                                                295       2-COCH.sub.2 CH.sub.2 CH.sub.3                                       296       3-COCH.sub.2 CH.sub.2 CH.sub.3                                       297       4-COCH.sub.2 CH.sub.2 CH.sub.3                                       298       2-COCH(CH.sub.3)CH.sub.3                                             299       3-COCH(CH.sub.3)CH.sub.3                                             300       4-COCH (CH.sub.3)CH.sub.3                                            301       2-Me-4-CHO                                                           302       2-Me-4-CH.sub.3 CO                                                   303       2-Me-4-CH.sub.3 CH.sub.2 CO                                          304       2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                 305       2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                       306       2,5-Me.sub.2 -4-CHO                                                  307       2,5-Me.sub.2 -4-CH.sub.3 CO                                          308       2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                 309       2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                        310       2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                              311       2-Cl-4-CHO                                                           312       2-Cl-4-CH.sub.3 CO                                                   313       2-Cl-4-CH.sub.3 CH.sub.2 CO                                          314       2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                       315       2,5-Cl.sub.2 -4-CHO                                                  316       2,5-Cl.sub.2 -4-CH.sub.3 CO                                          317       2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                 318       2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                        319       2,5-Cl.sub.2 -4-CH.sub.3 -CH(CH.sub.3)CO                             320       2-C(NOCH.sub.3)CH.sub.3                                              321       3-C(NOCH.sub.3)CH.sub.3                                              322       4-C(NOCH.sub.3)CH.sub.3                                              323       2-C(NOC.sub.2 H.sub.5)CH.sub.3                                       324       3-C(NOC.sub.2 H.sub.5)CH.sub.3                                       325       4-C(NOC.sub.2 H.sub.5)CH.sub.3                                       326       2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    327       3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    328       4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                    329       2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    330       3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    331       4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                    332       2-C(NO-Allyl)-CH.sub.3                                               333       3-C(NO-Allyl)-CH.sub.3                                               334       4-C(NO-Allyl)-CH.sub.3                                               335       2-C(NO-trans-Chloroallyl)-CH.sub.3                                   336       3-C(NO-trans-Chloroallyl)-CH.sub.3                                   337       4-C(NO-trans-Chloroallyl)-CH.sub.3                                   338       2-C(NO-Propargyl)-CH.sub.3                                           339       3-C(NO-Propargyl)-CH.sub.3                                           340       4-C(NO-Propargyl)-CH.sub.3                                           341       2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    342       3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    343       4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                    344       2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              345       3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              346       4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                              347       2-CH.sub.3 -4-CHNOCH.sub.3                                           348       2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                    349       2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                 350       2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                 351       2-CH.sub.3 -4-CHNO-Allyl                                             352       2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                               353       2-CH.sub.3 -4-CHNO-Propargyl                                         354       2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                 355       2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                           356       2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                 357       2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                          358       2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                       359       2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                       360       2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                   361       2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                       362       2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                               363       2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                       364       2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                 365       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                          366       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                   367       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                368       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                 369       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                            370       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                371       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                        372       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                373       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-CH.sub.2 C.sub.6 H.sub.5)         374       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                       375       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                376       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)             377       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)             378       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                         379       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)             380       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)                     381       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)             382       2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)       383       2-C.sub.6 H.sub.5                                                    384       3-C.sub.6 H.sub.5                                                    385       4-C.sub.6 H.sub.5                                                    386       2-(2'-FC.sub.6 H.sub.4)                                              387       2-(3'-FC.sub.6 H.sub.4)                                              388       2-(4'-FC.sub.6 H.sub.4)                                              389       3-(2'-FC.sub.6 H.sub.4)                                              390       3-(3'-FC.sub.6 H.sub.4)                                              391       3-(4'-FC.sub.6 H.sub.4)                                              392       4-(2'-FC.sub.6 H.sub.4)                                              393       4-(3'-FC.sub.6 H.sub.4)                                              394       4-(4'-FC.sub.6 H.sub.4)                                              395       2-(2'-ClC.sub.6 H.sub.4)                                             396       2-(3'-ClC.sub.6 H.sub.4)                                             397       2-(4'-ClC.sub.6 H.sub.4)                                             398       3-(2'-ClC.sub.6 H.sub.4)                                             399       3-(3'-ClC.sub.6 H.sub.4)                                             400       3-(4'-ClC.sub.6 H.sub.4)                                             401       4-(2'-ClC.sub.6 H.sub.4)                                             402       4-(3'-ClC.sub.6 H.sub.4)                                             403       4-(4'-ClC.sub.6 H.sub.4)                                             405       2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      406       2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      407       2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      408       3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      409       3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      410       3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      411       4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      412       4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      413       4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      414       2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    415       2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    416       2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    417       3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    418       3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    419       3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    420       4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    421       4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    422       4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    423       2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         424       2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         425       2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         426       3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         427       3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         428       3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         429       4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         430       4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         431       4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         432       2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             433       2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             434       2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             435       3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             436       3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             437       3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             438       4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             439       4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             440       4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             441       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     442       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     443       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     444       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     445       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     446       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     447       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     448       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     449       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     450       2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      451       2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      452       2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      453       3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      454       3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      455       3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      456       4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      457       4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      458       4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      459       2-(2'-NCC.sub.6 H.sub.4)                                             460       2-(3'-NCC.sub.6 H.sub.4)                                             461       2-(4'-NCC.sub.6 H.sub.4)                                             462       3-(2'-NCC.sub.6 H.sub.4)                                             463       3-(3'-NCC.sub.6 H.sub.4)                                             464       3-(4'-NCC.sub.6 H.sub.4)                                             465       4-(2'-NCC.sub.6 H.sub.4)                                             466       4-(3'-NCC.sub.6 H.sub.4)                                             467       4-(4'-NCC.sub.6 H.sub.4)                                             468       2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      469       2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      470       2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      471       3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      472       3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      473       3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      474       4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      475       4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      476       4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      477       2-OC.sub.6 H.sub.5                                                   475       3-OC.sub.6 H.sub.5                                                   476       4-OC.sub.6 H.sub.5                                                   478       2-O-(2'-FC.sub.6 H.sub.4)                                            479       2-O-(3'-FC.sub.6 H.sub.4)                                            480       2-O-(4'-FC.sub.6 H.sub.4)                                            481       3-O-(2'-FC.sub.6 H.sub.4)                                            482       3-O-(3'-FC.sub.6 H.sub.4)                                            483       3-O-(4'-FC.sub.6 H.sub.4)                                            484       4-O-(2'-FC.sub.6 H.sub.4)                                            485       4-O-(3'-FC.sub.6 H.sub.4)                                            486       4-O-(4'-FC.sub.6 H.sub.4)                                            487       2-O-(2'-ClC.sub.6 H.sub.4)                                           488       2-O-(3'-ClC.sub.6 H.sub.4)                                           489       2-O-(4'-ClC.sub.6 H.sub.4)                                           490       3-O-(2'-ClC.sub.6 H.sub.4)                                           491       3-O-(3'-ClC.sub.6 H.sub.4)                                           492       3-O-(4'-ClC.sub.6 H.sub.4)                                           493       3-O-(4'-ClC.sub.6 H.sub.4)                                           494       4-O-(2'-ClC.sub.6 H.sub.4)                                           495       4-O-(3'-ClC.sub.6 H.sub.4)                                           496       4-O-(4'-ClC.sub.6 H.sub.4)                                           497       2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    498       2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    499       2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    500       3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    501       3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    502       3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    503       4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                    504       4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                    505       4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                    506       2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  507       2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  508       2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  509       3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  510       3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  511       3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  512       4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                  513       4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                  514       4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                  515       2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       516       2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       517       2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       518       3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       519       3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       520       3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       521       4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       522       4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       523       4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                       524       2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           525       2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           526       2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           527       3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           528       3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           529       3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           530       4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           531       4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           532       4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                           533       2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   534       2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   535       2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   536       3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   537       3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   538       3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   539       4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                   540       4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                   541       4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                   542       2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    543       2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    544       2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    545       3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    546       3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    547       3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    548       4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                    549       4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                    550       4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                    551       2-O-(2'-NCC.sub.6 H.sub.4)                                           552       2-O-(3'-NCC.sub.6 H.sub.4)                                           553       2-O-(4'-NCC.sub.6 H.sub.4)                                           554       3-O-(2'-NCC.sub.6 H.sub.4)                                           555       3-O-(3'-NCC.sub.6 H.sub.4)                                           556       3-O-(4'-NCC.sub.6 H.sub.4)                                           557       4-O-(2'-NCC.sub.6 H.sub.4)                                           558       4-O-(3'-NCC.sub.6 H.sub.4)                                           559       4-O-(4'-NCC.sub.6 H.sub.4)                                           560       2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                    561       2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                    562       2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                    563       3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                    564       3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                    565       3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                    566       4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                    567       4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                    568       4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                    569       2-Pyridinyl-2'                                                       570       2-Pyridinyl-3'                                                       571       2-Pyridinyl-4'                                                       572       3-Pyridinyl-2'                                                       573       3-Pyridinyl-3'                                                       574       3-Pyridinyl-4'                                                       575       4-Pyridinyl-2'                                                       576       4-Pyridinyl-3'                                                       577       4-Pyridinyl-4'                                                       578       2-Pyrimidinyl-2'                                                     579       2-Pyrimidinyl-3'                                                     580       2-Pyrimidinyl-4'                                                     581       3-Pyrimidinyl-2'                                                     582       3-Pyrimidinyl-3'                                                     583       3-Pyrimidinyl-4'                                                     584       4-Pyrimidinyl-2'                                                     585       4-Pyrimidinyl-3'                                                     586       4-Pyrimidinyl-4'                                                     587       2-Pyrazolyl-1'                                                       588       2-Pyrazolyl-3'                                                       589       2-Pyrazolyl-4'                                                       590       3-Pyrazolyl-1'                                                       591       3-Pyrazolyl-3'                                                       592       3-Pyrazolyl-4'                                                       593       4-Pyrazolyl-1'                                                       594       4-Pyrazolyl-3'                                                       595       4-Pyrazolyl-4'                                                       596       2-Isoxazolyl-3'                                                      597       2-Isoxazolyl-4'                                                      598       2-Isoxazolyl-5'                                                      599       3-Isoxazolyl-3'                                                      600       3-Isoxazolyl-4'                                                      601       3-Isoxazolyl-5'                                                      602       4-Isoxazolyl-3'                                                      603       4-Isoxazolyl-4'                                                      604       4-Isoxazolyl-5'                                                      605       2-Isothiazolyl-3'                                                    606       2-Isothiazolyl-4'                                                    607       2-Isothiazolyl-5'                                                    608       3-Isothiazolyl-3'                                                    609       3-Isothiazolyl-4'                                                    610       3-Isothiazolyl-5'                                                    611       4-Isothiazolyl-3'                                                    612       4-Isothiazolyl-4'                                                    613       4-Isothiazolyl-5'                                                    614       2-Imidazolyl-1'                                                      615       2-Imidazolyl-2'                                                      616       2-Imidazolyl-4'                                                      617       3-Imidazolyl-1'                                                      618       3-Imidazolyl-2'                                                      619       3-Imidazolyl-4'                                                      620       4-Imidazolyl-1'                                                      621       4-Imidazolyl-2'                                                      622       4-Imidazolyl-4'                                                      623       2-Oxazolyl-2'                                                        624       2-Oxazolyl-4'                                                        625       2-Oxazolyl-5'                                                        626       3-Oxazolyl-2'                                                        627       3-Oxazolyl-4'                                                        628       3-Oxazolyl-5'                                                        629       4-Oxazolyl-2'                                                        630       4-Oxazolyl-4'                                                        631       4-Oxazolyl-5'                                                        632       2-Thiazolyl-2'                                                       633       2-Thiazolyl-4'                                                       634       2-Thiazolyl-5'                                                       635       3-Thiazolyl-2'                                                       636       3-Thiazolyl-4'                                                       637       3-Thiazolyl-5'                                                       638       4-Thiazolyl-2'                                                       639       4-Thiazolyl-4'                                                       640       4-Thiazolyl-5'                                                       641       2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)              642       2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)       643       2,5-(CH.sub.3).sub.2 -4-                                                       (CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                            644       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                        645       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                 646       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)              647       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)              648       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                          649       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)              650       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                      651       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)              652       2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)        653       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                        654       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                 655       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)              656       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)              657       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                          658       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)              659       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                      660       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)              661       2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)        662       2-O-n-C.sub.4 H.sub.9                                                663       2-O-i-C.sub.4 H.sub.9                                                664       2-O-s-C.sub.4 H.sub.9                                                665       2-O-t-C.sub.4 H.sub.9                                                666       2-Neopentyloxy                                                       667       3-O-n-C.sub.4 H.sub.9                                                668       3-O-i-C.sub.4 H.sub.9                                                669       3-O-s-C.sub.4 H.sub.9                                                670       3-O-t-C.sub.4 H.sub.9                                                671       3-Neopentyloxy                                                       672       4-O-n-C.sub.4 H.sub.9                                                673       4-O-i-C.sub.4 H.sub.9                                                674       4-O-s-C.sub.4 H.sub.9                                                675       4-O-t-C.sub.4 H.sub.9                                                676       4-Neopentyloxy                                                       677       3-CH.sub.3 -4-OCH.sub.3                                              678       3-CH.sub.3 -4-OC.sub.2 H.sub.5                                       679       3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                    680       3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                    681       3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                    682       3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                    683       3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                    684       3-CH.sub.3 -4-Neopentyloxy                                           685       2-CH.sub.3 -3-OCH.sub.3                                              686       2-CH.sub.3 -4-OCH.sub.3                                              687       2-CH.sub.3 -5-OCH.sub.3                                              688       2-CH.sub.3 -6-OCH.sub.3                                              689       3-CH.sub.3 -4-CCH.sub.3                                              690       3-CH.sub.3 -5-OCH.sub.3                                              691       3-CH.sub.3 -6-OCH.sub.3                                              692       4-CH.sub.3 -5-OCH.sub.3                                              693       4-CH.sub.3 -6-OCH.sub.3                                              694       4-CH.sub.3 -6-OCH.sub.3                                              695       2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                    696       2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                    697       2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                    698       2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                    699       3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                    700       3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                    701       3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                    702       4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                    703       4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                    704       5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                    705       2-Cl-3-OCH.sub.3                                                     706       2-Cl-4-OCH.sub.3                                                     707       2-Cl-5-OCH.sub.3                                                     708       2-Cl-6-OCH.sub.3                                                     709       3-Cl-4-OCH.sub.3                                                     710       3-Cl-5-OCH.sub.3                                                     711       3-Cl-6-OCH.sub.3                                                     712       4-Cl-5-OCH.sub.3                                                     713       4-Cl-6-OCH.sub.3                                                     714       5-Cl-6-OCH.sub.3                                                     ______________________________________                                    

                  TABLE 18                                                         ______________________________________                                          ##STR221##                                                                    I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, Z = CH.sub.3                                  III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5                           V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3                                No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                            2        N-CH.sub.3 -Pyrrolyl-3                                                3        N-C.sub.6 H.sub.5 -Pyrrolyl-3                                         4        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            5        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            6        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            7        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           8        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           9        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           10       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            11       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            12       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            13       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   14       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   15       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   16       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   17       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   18       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   19       Pyrrolyl-2                                                            20       NCH.sub.3 -Pyrrolyl-2                                                 21       NC.sub.6 H.sub.5 -Pyrrolyl-2                                          22       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            23       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            24       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            25       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           26       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           27       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           28       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            29       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            30       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            31       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   32       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   33       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   34       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   35       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   36       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   37       Furyl-2                                                               38       5-CH.sub.3 -Furyl-2                                                   39       5-C.sub.6 H.sub.5 -Furyl-2                                            40       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               41       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               42       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               43       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              44       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              45       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              46       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               47       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               48       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               49       5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      50       5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      51       5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      52       5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      53       5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      54       5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      55       4-CH.sub.3 -Furyl-2                                                   56       4-C.sub.6 H.sub.5 -Furyl-2                                            57       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               58       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               59       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               60       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              61       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              62       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              63       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               64       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               65       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               66       4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      67       4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      68       4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      69       4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      70       4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      71       4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      72       Thienyl-2                                                             73       5-CH.sub.3 -Thienyl-2                                                 74       5-C.sub.6 H.sub.5 -Thienyl-2                                          75       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             76       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             77       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             78       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            79       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            80       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            81       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             82       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             83       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             84       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    85       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    86       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    87       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    88       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    89       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    90       4-CH.sub.3 -Thienyl-2                                                 91       4-C.sub.6 H.sub.5 -Thienyl-2                                          92       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             93       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             94       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             95       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            96       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            97       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            98       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             99       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       NCH.sub.3 -Pyrazolyl-4                                               127       NC.sub.6 H.sub.5 -Pyrazolyl-4                                        128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 143       3-CH.sub.3 N-Methylpyrazolyl-4                                       144       3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4                               145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   154       3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          155       3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          156       3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          157       3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          158       3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          159       3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          160       Isoxazolyl-5                                                         161       3-CH.sub.3 Isoxazolyl-5                                              162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 Isoxazolyl-3                                              198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 Isothiazolyl-5                                            216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       2-CH.sub.3 -Oxazolyl-4                                               234       2-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           236       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           237       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           238       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          239       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          241       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           242       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           243       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           244       2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  245       2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  246       2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  247       2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  248       2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  249       2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       NCH.sub.3 -1,2,4-Triazolyl-5                                         269       3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                              270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          280       3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 281       3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 282       3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 283       3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 284       3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 285       3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        384       Pyridinyl-3                                                          385       1-Naphthyl                                                           386       2-Naphthyl                                                           ______________________________________                                    

                  TABLE 19                                                         ______________________________________                                          ##STR222##                                                                    I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, Z = CH.sub.3                                  III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5                           V: R.sup.1 CH.sub.3, Z = NHCH.sub.3                                            VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3                                No.        X.sub.m                                                             ______________________________________                                          1         H                                                                    2         2-F                                                                  3         3-F                                                                  4         4-F                                                                  5         2,4-F.sub.2                                                          6         2,4,6-F.sub.3                                                        7         2,3,4,5,6-F.sub.5                                                    8         2,3-F.sub.2                                                          9         2-Cl                                                                 10        3-Cl                                                                 11        4-Cl                                                                 12        2,3-Cl.sub.2                                                         13        2,4-Cl.sub.2                                                         14        2,5-Cl.sub.2                                                         15        2,6-Cl.sub.2                                                         16        3,4-Cl.sub.2                                                         17        3,5-Cl.sub.2                                                         18        2.3,4-Cl.sub.3                                                       19        2,3,5-Cl.sub.3                                                       20        2,3,6-Cl.sub.3                                                       21        2,4,5-Cl.sub.3                                                       22        2,4,6-Cl.sub.3                                                       23        3,4,5-Cl.sub.3                                                       24        2,3,4,6-Cl.sub.4                                                     25        2,3,5,6-Cl.sub.4                                                     26        2,3,4,5,6-Cl.sub.5                                                   27        2-Br                                                                 28        3-Br                                                                 29        4-Br                                                                 30        2,4-Br.sub.2                                                         31        2,5-Br.sub.2                                                         32        2,6-Br.sub.2                                                         33        2,4,6-Br.sub.3                                                       34        2,3,4,5,6-Br.sub.5                                                   35        2-I                                                                  36        3-I                                                                  37        4-I                                                                  38        2,4-I.sub.2                                                          39        2-Cl, 3-F                                                            40        2-Cl, 4-F                                                            41        2-Cl, 5-F                                                            42        2-Cl, 6-F                                                            43        2-Cl, 3-Br                                                           44        2-Cl, 4-Br                                                           45        2-Cl, 5-Br                                                           46        2-Cl, 6-Br                                                           47        2-Br, 3-Cl                                                           48        2-Br, 4-Cl                                                           49        2-Br, 5-Cl                                                           50        2-Br, 3-F                                                            51        2-Br, 4-F                                                            52        2-Br, 5-F                                                            53        2-Br, 6-F                                                            54        2-F, 3-Cl                                                            55        2-F, 4-Cl                                                            56        2-F, 5-Cl                                                            57        3-Cl, 4-F                                                            58        3-Cl, 5-F                                                            59        3-Cl, 4-Br                                                           60        3-Cl, 5-Br                                                           61        3-F, 4-Cl                                                            62        3-F, 4-Br                                                            63        3-Br, 4-Cl                                                           64        3-Br, 4-F                                                            65        2,6-Cl.sub.2, 4-Br                                                   66        2-CH.sub.3                                                           67        3-CH.sub.3                                                           68        4-CH.sub.3                                                           69        2,3-(CH.sub.3).sub.2                                                 70        2,4-(CH.sub.3).sub.2                                                 71        2,5-(CH.sub.3).sub.2                                                 72        2,6-(CH.sub.3).sub.2                                                 73        3,4-(CH.sub.3).sub.2                                                 74        3,5-(CH.sub.3).sub.2                                                 75        2,3,5-(CH.sub.3).sub.3                                               76        2,3,4-(CH.sub.3).sub.3                                               77        2,3,6-(CH.sub.3).sub.3                                               78        2,4,5-(CH.sub.3).sub.3                                               79        2,4,6-(CH.sub.3).sub.3                                               80        3,4,5-(CH.sub.3).sub.3                                               81        2,3,4,6-(CH.sub.3).sub.4                                             82        2,3,5,6-(CH.sub.3).sub.4                                             83        2,3,4,5,6-(CH.sub.3).sub.5                                           84        2-C.sub.2 H.sub.5                                                    85        3-C.sub.2 H.sub.5                                                    86        4-C.sub.2 H.sub.5                                                    87        2,4-(C.sub.2 H.sub.5).sub.2                                          88        2,6-(C.sub.2 H.sub.5).sub.2                                          89        3,5-(C.sub.2 H.sub.5).sub.2                                          90        2,4,6-(C.sub.2 H.sub.5).sub.3                                        91        2-n-C.sub.3 H.sub.7                                                  92        3-n-C.sub.3 H.sub.7                                                  93        4-n-C.sub.3 H.sub.7                                                  94        2-i-C.sub.3 H.sub.7                                                  95        3-i-C.sub.3 H.sub.7                                                  96        4-i-C.sub.3 H.sub.7                                                  97        2,4-(i-C.sub.3 H.sub.7).sub.2                                        98        2,6-(i-C.sub.3 H.sub.7).sub.2                                        99        3,5-(i-C.sub.3 H.sub.7).sub.2                                       100        2,4,6-(i-C.sub.3 H.sub.7).sub.3                                     101        2-s-C.sub.4 H.sub.9                                                 102        3-s-C.sub.4 H.sub.9                                                 103        4-s-C.sub.4 H.sub.9                                                 104        2-t-C.sub.4 H.sub.9                                                 105        3-t-C.sub.4 H.sub.9                                                 106        4-t-C.sub.4 H.sub.9                                                 107        2,3-(t-C.sub.4 H.sub.9).sub.2                                       108        2,4-(t-C.sub.4 H.sub.9).sub.2                                       109        2,5-(t-C.sub.4 H.sub.9).sub.2                                       110        2,6-(t-C.sub.4 H.sub.9).sub.2                                       111        3,4-(t-C.sub.4 H.sub.9).sub.2                                       112        2,4,6-(t-C.sub.4 H.sub.9).sub.3                                     113        4-n-C.sub.9 H.sub.19                                                114        4-n-C.sub.12 H.sub.25                                               115        4-n-C.sub.15 H.sub.31                                               116        4-(1,1,3,3-Tetramethylbutyl)                                        117        4-(2,4,4-Trimethylpropyl)                                           118        2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                     119        2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                     120        2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                           121        2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                     122        2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                     123        2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                     124        2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                     125        3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                     126        2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                     127        2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                  128        2-Allyl                                                             129        3-Allyl                                                             130        4-Allyl                                                             131        2-Allyl, 6-CH.sub.3                                                 132        2-cyclo-C.sub.6 H.sub.11                                            133        3-cyclo-C.sub.6 H.sub.11                                            134        4-cyclo-C.sub.6 H.sub.11                                            135        2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                      136        2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                137        2-CH.sub.2 C.sub.6 H.sub.5                                          138        3-CH.sub.2 C.sub.6 H.sub.5                                          139        4-CH.sub.2 C.sub.6 H.sub.5                                          140        2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                              141        2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                              142        2-C.sub.6 H.sub.5                                                   143        3-C.sub.6 H.sub.5                                                   144        4-C.sub.6 H.sub.5                                                   145        4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                             146        4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                             147        2-Cl, 4-C.sub.6 H.sub.5                                             148        2-Br, 4-C.sub.6 H.sub.5                                             149        2-C.sub.6 H.sub.5, 4-Cl                                             150        2-C.sub.6 H.sub.5, 4-Br                                             151        2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                    152        2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                    153        2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                    154        2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                    155        2-cyclo-C.sub.6 H.sub.11, 4-Cl                                      156        2-cyclo-C.sub.6 H.sub.11, 4-Br                                      157        2-Cl, 4-cyclo-C.sub.6 H.sub.11                                      158        2-Br, 4-cyclo-C.sub.6 H.sub.11                                      159        2-OCH.sub.3                                                         160        3-OCH.sub.3                                                         161        4-OCH.sub.3                                                         162        2-OC.sub.2 H.sub.5                                                  163        3-O-C.sub.2 H.sub.5                                                 164        4-O-C.sub.2 H.sub.5                                                 165        2-O-n-C.sub.3 H.sub.7                                               166        3-O-n-C.sub.3 H.sub.7                                               167        4-O-n-C.sub.3 H.sub.7                                               168        2-O-i-C.sub.3 H.sub.7                                               169        3-O-i-C.sub.3 H.sub.7                                               170        4-O-i-C.sub.3 H.sub.7                                               171        2-O-n-C.sub.6 H.sub.13                                              172        3-O-n-C.sub.6 H.sub.13                                              173        4-O-n-C.sub.6 H.sub.13                                              174        2-O-n-C.sub.8 H.sub.17                                              175        3-O-n-C.sub.8 H.sub.17                                              176        4-O-n-C.sub.8 H.sub.17                                              177        2-O-CH.sub.2 C.sub.6 H.sub.5                                        178        3-O-CH.sub.2 C.sub.6 H.sub.5                                        179        4-O-CH.sub.2 C.sub.6 H.sub.5                                        180        2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                181        3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                182        4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                183        2,4-(OCH.sub.3).sub.2                                               184        2-CF.sub.3                                                          185        3-CF.sub.3                                                          186        4-CF.sub.3                                                          187        2-OCF.sub.3                                                         188        3-OCF.sub.3                                                         189        4-OCF.sub.3                                                         190        3-OCH.sub.2 CHF.sub.2                                               191        2-NO.sub.2                                                          192        3-NO.sub.2                                                          193        4-NO.sub.2                                                          194        2-CN                                                                195        3-CN                                                                196        4-CN                                                                197        2-CH.sub.3, 3-Cl                                                    198        2-CH.sub.3, 4-Cl                                                    199        2-CH.sub.3, 5-Cl                                                    200        2-CH.sub.3, 6-Cl                                                    201        2-CH.sub.3, 3-F                                                     202        2-CH.sub.3, 4-F                                                     203        2-CH.sub.3, 5-F                                                     204        2-CH.sub.3, 6-F                                                     205        2-CH.sub.3, 3-Br                                                    206        2-CH.sub.3, 4-Br                                                    207        2-CH.sub.3, 5-Br                                                    208        2-CH.sub.3, 6-Br                                                    209        2-Cl, 3-CH.sub.3                                                    210        2-Cl, 4-CH.sub.3                                                    211        2-Cl, 5-CH.sub.3                                                    212        2-F, 3-CH.sub.3                                                     213        2-F, 4-CH.sub.3                                                     214        2-F, 5-CH.sub.3                                                     215        2-Br, 3-CH.sub.3                                                    216        2-Br, 4-CH.sub.3                                                    217        2-Br, 5-CH.sub.3                                                    218        3-CH.sub.3, 4-Cl                                                    219        3-CH.sub.3, 5-Cl                                                    220        3-CH.sub.3, 4-F                                                     221        3-CH.sub.3, 5-F                                                     222        3-CH.sub.3, 4-Br                                                    223        3-CH.sub.3, 5-Br                                                    224        3-F, 4-CH.sub.3                                                     225        3-Cl, 4-CH.sub.3                                                    226        3-Br, 4-CH.sub.3                                                    227        2-Cl, 4,5-(CH.sub.3).sub.2                                          228        2-Br, 4,5-(CH.sub.3).sub.2                                          229        2-Cl, 3,5-(CH.sub.3).sub.2                                          230        2-Br, 3,5-(CH.sub.3).sub.2                                          231        2,6-Cl.sub.2, 4-CH.sub.3                                            232        2,6-F.sub.2, 4-CH.sub.3                                             233        2,6-Br.sub.2, 4-CH.sub.3                                            234        2,4-Br.sub.2, 6-CH.sub.3                                            235        2,4-F.sub.2, 6-CH.sub.3                                             236        2,4-Br.sub.2, 6-CH.sub.3                                            237        2,6-(CH.sub.3).sub.2, 4-F                                           238        2,6-(CH.sub.3).sub.2, 4-Cl                                          239        2,6-(CH.sub.3).sub.2, 4-Br                                          240        3,5-(CH.sub.3).sub.2, 4-F                                           241        3,5-(CH.sub.3).sub.2, 4-Cl                                          242        3,5-(CH.sub.3).sub.2, 4-Br                                          243        2,3,6-(CH.sub.3).sub.3, 4-F                                         244        2,3,6-(CH.sub.3).sub.3, 4-Cl                                        245        2,3,6-(CH.sub.3).sub.3, 4-Br                                        246        2,4-(CH.sub.3).sub.2, 6-F                                           247        2,4-(CH.sub.3).sub.2, 6-Cl                                          248        2,4-(CH.sub.3).sub.2, 6-Br                                          249        2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                               250        2-Cl, 4-NO.sub.2                                                    251        2-NO.sub.2, 4-Cl                                                    252        2-OCH.sub.3, 5-NO.sub.2                                             253        2,4-Cl.sub.2, 5-NO.sub.2                                            254        2,4-Cl.sub.2, 6-NO.sub.2                                            255        2,6-Cl.sub.2, 4-NO.sub.2                                            256        2,6-Br.sub.2, 4-NO.sub.2                                            257        2,6-I.sub.2, 4-NO.sub.2                                             258        2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                               259        2-CO.sub.2 CH.sub.3                                                 260        3-CO.sub.2 CH.sub.3                                                 261        4-CO.sub.2 CH.sub.3                                                 262        2-CO.sub.2 (C.sub.2 H.sub.5)                                        263        3-CO.sub.2 (C.sub.2 H.sub.5)                                        264        4-CO.sub.2 (C.sub.2 H.sub.5)                                        265        2-CO.sub.2 (n-C.sub.3 H.sub.7)                                      266        3-CO.sub.2 (n-C.sub.3 H.sub.7)                                      267        4-CO.sub.2 (n-C.sub.3 H.sub.7)                                      268        2-CO.sub.2 (i-C.sub.3 H.sub.7)                                      269        3-CO.sub.2 (i-C.sub.3 H.sub.7)                                      270        4-CO.sub.2 (i-C.sub.3 H.sub.7)                                      271        2-CO.sub.2 (n-C.sub.6 H.sub.13)                                     272        3-CO.sub.2 (n-C.sub.6 H.sub.13)                                     273        4-CO.sub.2 (n-C.sub.6 H.sub.13)                                     274        2-CH.sub.2 OCH.sub.3                                                275        3-CH.sub.2 OCH.sub.3                                                276        4-CH.sub.2 OCH.sub.3                                                277        2-CH.sub.2 O(C.sub.2 H.sub.5)                                       278        3-CH.sub.2 O(C.sub.2 H.sub.5)                                       279        4-CH.sub.2 O(C.sub.2 H.sub.5)                                       280        2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                     281        3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                     282        4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                     283        2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                     284        3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                     285        4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                     286        2-CHO                                                               287        3-CHO                                                               288        4-CHO                                                               289        2-COCH.sub.3                                                        290        3-COCH.sub.3                                                        291        4-COCH.sub.3                                                        292        2-COCH.sub.2 CH.sub.3                                               293        3-COCH.sub.2 CH.sub.3                                               294        4-COCH.sub.2 CH.sub.3                                               295        2-COCH.sub.2 CH.sub.2 CH.sub.3                                      296        3-COCH.sub.2 CH.sub.2 CH.sub.3                                      297        4-COCH.sub.2 CH.sub.2 CH.sub.3                                      298        2-COCH(CH.sub.3)CH.sub.3                                            299        3-COCH(CH.sub.3)CH.sub.3                                            300        4-COCH(CH.sub.3)CH.sub.3                                            301        2-Me-4-CHO                                                          302        2-Me-4-CH.sub.3 CO                                                  303        2-Me-4-CH.sub.3 CH.sub.2 CO                                         304        2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                305        2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                      306        2,5-Me.sub.2 -4-CHO                                                 307        2,5-Me.sub.2 -4-CH.sub.3 CO                                         308        2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                309        2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                       310        2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                             311        2-Cl-4-CHO                                                          312        2-Cl-4-CH.sub.3 CO                                                  313        2-Cl-4-CH.sub.3 CH.sub.2 CO                                         314        2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                      315        2,5-Cl.sub.2 -4-CHO                                                 316        2,5-Cl.sub.2 -4-CH.sub.3 CO                                         317        2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                318        2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                       319        2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                             320        2-C(NOCH.sub.3)CH.sub.3                                             321        3-C(NOCH.sub.3)CH.sub.3                                             322        4-C(NOCH.sub.3)CH.sub.3                                             323        2-C(NOC.sub.2 H.sub.5)CH.sub.3                                      324        3-C(NOC.sub.2 H.sub.5)CH.sub.3                                      325        4-C(NOC.sub.2 H.sub.5)CH.sub.3                                      326        2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                   327        3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                   328        4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                   329        2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                   330        3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                   331        4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                   332        2-C(NO-Allyl)-CH.sub.3                                              333        3-C(NO-Allyl)-CH.sub.3                                              334        4-C(NO-Allyl)-CH.sub.3                                              335        2-C(NO-trans-Chloroallyl)-CH.sub.3                                  336        3-C(NO-trans-Chloroallyl)-CH.sub.3                                  337        4-C(NO-trans-Chloroallyl)-CH.sub.3                                  338        2-C(NO-Propargyl)-CH.sub.3                                          339        3-C(NO-Propargyl)-CH.sub.3                                          340        4-C(NO-Propargyl)-CH.sub.3                                          341        2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                   342        3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                   343        4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                   344        2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                             345        3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                             346        4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                             347        2-CH.sub.3 -4-CHNOCH.sub.3                                          348        2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                   349        2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                350        2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                351        2-CH.sub.3 -4-CHNO-Allyl                                            352        2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                              353        2-CH.sub.3 -4-CHNO-Propargyl                                        354        2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                355        2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                          356        2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                357        2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                         358        2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                      359        2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                      360        2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                  361        2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                      362        2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                              363        2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                      364        2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                365        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                         366        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                  367        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)               368        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                369        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                           370        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)               371        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                       372        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)               373        2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)         374        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                      375        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)               376        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)            377        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)            378        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                        379        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)            380        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                     381        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)            382        2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)      383        2-C.sub.6 H.sub.5                                                   384        3-C.sub.6 H.sub.5                                                   385        4-C.sub.6 H.sub.5                                                   386        2-(2'-FC.sub.6 H.sub.4)                                             387        2-(3'-FC.sub.6 H.sub.4)                                             388        2-(4'-FC.sub.6 H.sub.4)                                             389        3-(2'-FC.sub.6 H.sub.4)                                             390        3-(3'-FC.sub.6 H.sub.4)                                             391        3-(4'-FC.sub.6 H.sub.4)                                             392        4-(2'-FC.sub.6 H.sub.4)                                             393        4-(3'-FC.sub.6 H.sub.4)                                             394        4-(4'-FC.sub.6 H.sub.4)                                             395        2-(2'-ClC.sub.6 H.sub.4)                                            396        2-(3'-ClC.sub.6 H.sub.4)                                            397        2-(4'-ClC.sub.6 H.sub.4)                                            398        3-(2'-ClC.sub.6 H.sub.4)                                            399        3-(3'-ClC.sub.6 H.sub.4)                                            400        3-(4'-ClC.sub.6 H.sub.4)                                            401        4-(2'-ClC.sub.6 H.sub.4)                                            402        4-(3'-ClC.sub.6 H.sub.4)                                            403        4-(4'-ClC.sub.6 H.sub.4)                                            405        2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     406        2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     407        2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     408        3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     409        3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     410        3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     411        4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     412        4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     413        4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     414        2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   415        2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   416        2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   417        3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   418        3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   419        3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   420        4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   421        4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   422        4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   423        2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        424        2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        425        2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        426        3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        427        3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        428        3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        429        4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        430        4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        431        4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        432        2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            433        2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            434        2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            435        3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            436        3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            437        3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            438        4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            439        4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            440        4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            441        2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    442        2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    443        2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    444        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    445        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    446        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    447        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    448        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    449        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    450        2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     451        2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     452        2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     453        3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     454        3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     455        3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     456        4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     457        4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     458        4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     459        2-(2'-NCC.sub.6 H.sub.4)                                            460        2-(3'-NCC.sub.6 H.sub.4)                                            461        2-(4'-NCC.sub.6 H.sub.4)                                            462        3-(2'-NCC.sub.6 H.sub.4)                                            463        3-(3'-NCC.sub.6 H.sub.4)                                            464        3-(4'-NCC.sub.6 H.sub.4)                                            465        4-(2'-NCC.sub.6 H.sub.4)                                            466        4-(3'-NCC.sub.6 H.sub.4)                                            467        4-(4'-NCC.sub.6 H.sub.4)                                            468        2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     469        2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     470        2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     471        3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     472        3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     473        3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     474        4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     475        4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     476        4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     477        2-OC.sub.6 H.sub.5                                                  475        3-OC.sub.6 H.sub.5                                                  476        4-OC.sub.6 H.sub.5                                                  478        2-O-(2'-FC.sub.6 H.sub.4)                                           479        2-O-(3'-FC.sub.6 H.sub.4)                                           480        2-O-(4'-FC.sub.6 H.sub.4)                                           481        3-O-(2'-FC.sub.6 H.sub.4)                                           482        3-O-(3'-FC.sub.6 H.sub.4)                                           483        3-O-(4'-FC.sub.6 H.sub.4)                                           484        4-O-(2'-FC.sub.6 H.sub.4)                                           485        4-O-(3'-FC.sub.6 H.sub.4)                                           486        4-O-(4'-FC.sub.6 H.sub.4)                                           487        2-O-(2'-ClC.sub.6 H.sub.4)                                          488        2-O-(3'-ClC.sub.6 H.sub.4)                                          489        2-O-(4'-ClC.sub.6 H.sub.4)                                          490        3-O-(2'-ClC.sub.6 H.sub.4)                                          491        3-O-(3'-ClC.sub.6 H.sub.4)                                          492        3-O-(4'-ClC.sub.6 H.sub.4)                                          493        3-O-(4'-ClC.sub.6 H.sub.4)                                          494        4-O-(2'-ClC.sub.6 H.sub.4)                                          495        4-O-(3'-ClC.sub.6 H.sub.4)                                          496        4-O-(4'-ClC.sub.6 H.sub.4)                                          497        2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                   498        2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                   499        2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                   500        3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                   501        3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                   502        3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                   503        4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                   504        4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                   505        4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                   506        2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                 507        2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                 508        2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                 509        3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                 510        3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                 511        3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                 512        4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                 513        4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                 514        4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                 515        2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      516        2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      517        2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      518        3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      519        3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      520        3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      521        4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      522        4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      523        4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                      524        2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          525        2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          526        2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          527        3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          528        3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          529        3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          530        4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          531        4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          532        4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                          533        2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                  534        2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                  535        2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                  536        3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                  537        3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                  538        3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                  539        4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                  540        4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                  541        4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                  542        2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                   543        2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                   544        2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                   545        3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                   546        3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                   547        3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                   548        4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                   549        4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                   550        4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                   551        2-O-(2'-NCC.sub.6 H.sub.4)                                          552        2-O-(3'-NCC.sub.6 H.sub.4)                                          553        2-O-(4'-NCC.sub.6 H.sub.4)                                          554        3-O-(2'-NCC.sub.6 H.sub.4)                                          555        3-O-(3'-NCC.sub.6 H.sub.4)                                          556        3-O-(4'-NCC.sub.6 H.sub.4)                                          557        4-O-(2'-NCC.sub.6 H.sub.4)                                          558        4-O-(3'-NCC.sub.6 H.sub.4)                                          559        4-O-(4'-NCC.sub.6 H.sub.4)                                          560        2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                   561        2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                   562        2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                   563        3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                   564        3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                   565        3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                   566        4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                   567        4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                   568        4-0-(4'-CF.sub.3 C.sub.6 H.sub.4)                                   569        2-Pyridinyl-2'                                                      570        2-Pyridinyl-3'                                                      571        2-Pyridinyl-4'                                                      572        3-Pyridinyl-2'                                                      573        3-Pyridinyl-3'                                                      574        3-Pyridinyl-4'                                                      575        4-Pyridinyl-2'                                                      576        4-Pyridinyl-3'                                                      577        4-Pyridinyl-4'                                                      578        2-Pyrimidinyl-2'                                                    579        2-Pyrimidinyl-3'                                                    580        2-Pyrimidinyl-4'                                                    581        3-Pyrimidinyl-2'                                                    582        3-Pyrimidinyl-3'                                                    583        3-Pyrimidinyl-4'                                                    584        4-Pyrimidinyl-2'                                                    585        4-Pyrimidinyl-3'                                                    586        4-Pyrimidinyl-4'                                                    587        2-Pyrazolyl-1'                                                      588        2-Pyrazolyl-3'                                                      589        2-Pyrazolyl-4'                                                      590        3-Pyrazolyl-1'                                                      591        3-Pyrazolyl-3'                                                      592        3-Pyrazolyl-4'                                                      593        4-Pyrazolyl-1'                                                      594        4-Pyrazolyl-3'                                                      595        4-Pyrazolyl-4'                                                      596        2-Isoxazolyl-3'                                                     597        2-Isoxazolyl-4'                                                     598        2-Isoxazolyl-5'                                                     599        3-Isoxazolyl-3'                                                     600        3-Isoxazolyl-4'                                                     601        3-Isoxazolyl-5'                                                     602        4-Isoxazolyl-3'                                                     603        4-Isoxazolyl-4'                                                     604        4-Isoxazolyl-5'                                                     605        2-Isothiazolyl-3'                                                   606        2-Isothiazolyl-4'                                                   607        2-Isothiazolyl-5'                                                   608        3-Isothiazolyl-3'                                                   609        3-Isothiazolyl-4'                                                   610        3-Isothiazolyl-5'                                                   611        4-Isothiazolyl-3'                                                   612        4-Isothiazolyl-4'                                                   613        4-Isothiazolyl-5'                                                   614        2-Imidazolyl-1'                                                     615        2-Imidazolyl-2'                                                     616        2-Imidazolyl-4'                                                     617        3-Imidazolyl-1'                                                     618        3-Imidazolyl-2'                                                     619        3-Imidazolyl-4'                                                     620        4-Imidazolyl-1'                                                     621        4-Imidazolyl-2'                                                     622        4-Imidazolyl-4'                                                     623        2-Oxazolyl-2'                                                       624        2-Oxazolyl-4'                                                       625        2-Oxazolyl-5'                                                       626        3-Oxazolyl-2'                                                       627        3-Oxazolyl-4'                                                       628        3-Oxazolyl-5'                                                       629        4-Oxazolyl-2'                                                       630        4-Oxazolyl-4'                                                       631        4-Oxazolyl-5'                                                       632        2-Thiazolyl-2'                                                      633        2-Thiazolyl-4'                                                      634        2-Thiazolyl-5'                                                      635        3-Thiazolyl-2'                                                      636        3-Thiazolyl-4'                                                      637        3-Thiazolyl-5'                                                      638        4-Thiazolyl-2'                                                      639        4-Thiazolyl-4'                                                      640        4-Thiazolyl-5'                                                      ______________________________________                                    

                  TABLE 20                                                         ______________________________________                                          ##STR223##                                                                    I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, Z CH.sub.3                                    III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5                           V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3                                No.        B                                                                   ______________________________________                                          1         Pyrrolyl-3                                                           2         NCH.sub.3 -Pyrrolyl-3                                                3         NC.sub.6 H.sub.5 -Pyrrolyl-3                                         4         N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           5         N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           6         N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           7         N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          8         N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          9         N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          10        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           11        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           12        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           13        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  14        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  15        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  16        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  17        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  18        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  19        Pyrrolyl-2                                                           20        NCH.sub.3 -Pyrrolyl-2                                                21        NC.sub.6 H.sub.5 -Pyrrolyl-2                                         22        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           23        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           24        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           25        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          26        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          27        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          28        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           29        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           30        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           31        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  32        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  33        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  34        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  35        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  36        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  37        Furyl-2                                                              38        5-CH.sub.3 -Furyl-2                                                  39        5-C.sub.6 H.sub.5 -Furyl-2                                           40        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              41        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              42        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              43        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             44        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             45        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             46        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              47        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              48        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              49        5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     50        5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     51        5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     52        5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     53        5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     54        5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     55        4-CH.sub.3 -Furyl-2                                                  56        4-C.sub.6 H.sub.5 -Furyl-2                                           57        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              58        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              59        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              60        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             61        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             62        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             63        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              64        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              65        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              66        4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     67        4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     68        4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     69        4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     70        4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     71        4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     72        Thienyl-2                                                            73        5-CH.sub.3 -Thienyl-2                                                74        5-C.sub.6 H.sub.5 -Thienyl-2                                         75        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            76        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            77        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            78        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           79        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           80        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           81        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            82        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            83        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            84        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   85        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   86        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   87        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   88        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   89        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   90        4-CH.sub.3 -Thienyl-2                                                91        4-C.sub.6 H.sub.5 -Thienyl-2                                         92        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            93        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            94        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            95        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           96        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           97        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           98        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            99        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                           100        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                           101        4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                  102        4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                  103        4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                  104        4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                  105        4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                  106        4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                  107        Thienyl-3                                                           108        5-CH.sub.3 -Thienyl-3                                               109        5-C.sub.6 H.sub.5 -Thienyl-3                                        110        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           111        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           112        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                           113        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          114        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          115        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                          116        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           117        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           118        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                           119        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                  120        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                  121        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                  122        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                  123        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                  124        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                  125        Pyrazolyl-4                                                         126        NCH.sub.3 -Pyrazolyl-4                                              127        NC.sub.6 H.sub.5 -Pyrazolyl-4                                       128        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         129        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         130        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                         131        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        132        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        133        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                        134        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         135        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         136        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                         137        N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                138        N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                139        N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                140        N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                141        N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                142        N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                143        3-CH.sub.3 N-Methylpyrazolyl-4                                      144        3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                               145        3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  146        3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  147        3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  148        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                 149        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                 150        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                 151        3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  152        3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  153        3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                  154        3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         155        3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         156        3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         157        3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         158        3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         159        3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                         160        Isoxazolyl-5                                                        161        3-CH.sub.3 -Isoxazolyl-5                                            162        3-C.sub.6 H.sub.5 -Isoxazolyl-5                                     163        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        164        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        165        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                        166        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       167        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       168        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                       169        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        170        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        171        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                        172        3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               173        3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               174        3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                               175        3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               176        3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               177        3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                               178        4-Chloroisoxazolyl-5                                                179        3-CH.sub.3 -4-Chloroisoxazolyl-5                                    180        3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                             181        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                182        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                183        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                184        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               185        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               186        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5               187        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                188        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                189        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                190        3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       191        3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       192        3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       193        3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       194        3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       195        3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                       196        Isoxazolyl-3                                                        197        5-CH.sub.3 -Isoxazolyl-3                                            198        5-C.sub.6 H.sub.5 -Isoxazolyl-3                                     199        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        200        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        201        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                        202        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       203        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       204        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                       205        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        206        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        207        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                        208        5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               209        5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               210        5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                               211        5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               212        5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               213        5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                               214        Isothiazolyl-5                                                      215        3-CH.sub.3 -Isothiazolyl-5                                          216        3-C.sub.6 H.sub.5 -Isothiazolyl-5                                   217        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      218        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      219        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                      220        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     221        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     222        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                     223        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      224        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      225        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                      226        3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             227        3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             228        3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                             229        3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             230        3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             231        3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                             232        Oxazolyl-4                                                          233        2-CH.sub.3 -Oxazolyl-4                                              234        2-C.sub.6 H.sub.5 -Oxazolyl-4                                       235        2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          236        2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          237        2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                          238        2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         239        2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         240        2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                         241        2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          242        2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          243        2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                          244        2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 245        2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 246        2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                 247        2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 248        2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 249        2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                 250        Thiazolyl-4                                                         251        2-CH.sub.3 -Thiazolyl-4                                             252        2-C.sub.6 H.sub.5 -Thiazolyl-4                                      253        2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         254        2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         255        2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                         256        2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                        267        2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                        258        2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                        259        2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         260        2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         261        2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                         262        2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                263        2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                264        2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                265        2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                266        2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                267        2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                268        NCH.sub.3 -1,2,4-Triazolyl-5                                        269        3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                             270        3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                      271        3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         272        3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         273        3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         274        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        275        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        276        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5        277        3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         278        3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         279        3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         280        3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                281        3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                282        3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                283        3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                284        3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                285        3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                286        1,3,4-Oxadiazolyl-2                                                 287        5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                     288        5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                              289        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 290        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 291        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 292        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                293        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                294        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                295        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 296        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 297        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 298        5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        299        5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        300        5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        301        5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        302        5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        303        5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                        304        1,2,4-Oxadiazolyl-3                                                 305        5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                     306        5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                              307        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 308        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 309        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 310        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                311        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                312        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                313        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 314        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 315        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 316        5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        317        5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        318        5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        319        5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        320        5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        321        5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                        322        1,2,4-Oxadiazolyl-5                                                 323        3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                     324        3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                              325        3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 326        3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 327        3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 328        3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                329        3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                330        3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                331        3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 332        3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 333        3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 334        3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        335        3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        336        3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        337        3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        338        3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        339        3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                        340        1,2,4-Thiadiazolyl-3                                                341        5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                    342        5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                             343        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                344        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                345        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                346        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               347        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               348        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3               349        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                350        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                351        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                352        5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       353        5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       354        5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       355        5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       356        5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       357        5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                       358        1,3,4-Thiadiazolyl-2                                                359        5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                    360        5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                             361        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                362        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                363        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                364        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               365        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               366        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2               367        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                368        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                369        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                370        5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       371        5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       372        5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       373        5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       374        5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       375        5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                       376        Pyridinyl-2                                                         377        Pyridinyl-4                                                         378        Pyridazinyl-3                                                       379        Pyridazinyl-4                                                       380        Pyridazinyl-2                                                       381        Pyrimidinyl-4                                                       382        Pyrimidinyl-5                                                       383        Pyrimidinyl-2                                                       384        Pyridinyl-3                                                         ______________________________________                                    

                                      TABLE 21                                     __________________________________________________________________________     Selected physical data of some compounds                                       No.                                                                               Compound                    .sup.1 H-NMR (ppm)                                                                      m.p.                                   __________________________________________________________________________      1                                                                                 ##STR224##                 3.7 (s, broad, 3H); 1.2 (s, broad, 3H)           2                                                                                 ##STR225##                 3.75 (s, 3H); 1.2 (t, 3H)                        3                                                                                 ##STR226##                 3.7 (s, 3H); 1.2 (t, 3H)                         4                                                                                 ##STR227##                 3.95 (s, 3H); 3.7 (s, 3H); 1,2 (t, 3H)           5                                                                                 ##STR228##                 3.6 (s, 3H); 2.9 (d, 3H)                         6                                                                                 ##STR229##                          123                                     7                                                                                 ##STR230##                          118                                     8                                                                                 ##STR231##                 3.7 (s, 3H); 2.55 (s, very                      __________________________________________________________________________                                    broad, 2H)                                 

                  TABLE 56                                                         ______________________________________                                         Selected physical data of some compounds                                        ##STR232##                                                                                             mp     .sup.1 H-NMR (ppm) or                          No.  X.sub.m             (°C.)                                                                          IR (cm.sup.-1)                                 ______________________________________                                         1    H                   90                                                    2    2-CH.sub.3          80                                                    3    2,5-(CH.sub.3).sub.2                                                                               101                                                   4    2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                                       3.95 (s, 3H); 3.65                                                             (s, 3H); 2.9 (d, 3H)                           5    2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl                                                               3.65 (s, 3H); 2.9                                                              (d, 3H)                                        ______________________________________                                    

                  TABLE 22                                                         ______________________________________                                          ##STR233##                                                                    No.     X        Z         A                                                   ______________________________________                                          1      H        CH.sub.3  CH.sub.2 O                                           2      H        CH.sub.3  CH.sub.2 ONC(CH.sub.3)                               3      H        CH.sub.3  CHCH                                                 4      H        NH.sub.2  CH.sub.2 O                                           5      H        NH.sub.2  CH.sub.2 ONC(CH.sub.3)                               6      H        NH.sub.2  CHCH                                                 7      H        N(CH.sub.3).sub.2                                                                        CH.sub.2 O                                           8      H        N(CH.sub.3).sub.2                                                                        CH.sub.2 ONC(CH.sub.3)                               9      H        N(CH.sub.3).sub.2                                                                        CHCH                                                10      H        CCl.sub.3 CH.sub.2 O                                          11      H        CCl.sub.3 CH.sub.2 ONC(CH.sub.3)                              12      H        CCl.sub.3 CHCH                                                13      H        CF.sub.3  CH.sub.2 O                                          14      H        CF.sub.3  CH.sub.2 ONC(CH.sub.3)                              15      H        CF.sub.3  CHCH                                                16      CH.sub.3 CH.sub.3  CH.sub.2 O                                          17      CH.sub.3 CH.sub.3  CH.sub.2 ONC(CH.sub.3)                              18      CH.sub.3 CH.sub.3  CHCH                                                19      CH.sub.3 NH.sub.2  CH.sub.2 O                                          20      CH.sub.3 NH.sub.2  CH.sub.2 ONC(CH.sub.3)                              21      CH.sub.3 NH.sub.2  CHCH                                                22      CH.sub.3 N(CH.sub.3).sub.2                                                                        CH.sub.2 O                                          23      CH.sub.3 N(CH.sub.3).sub.2                                                                        CH.sub.2 ONC(CH.sub.3)                              24      CH.sub.3 N(CH.sub.3).sub.2                                                                        CHCH                                                25      CH.sub.3 CCl.sub.3 CH.sub.2 O                                          26      CH.sub.3 CCl.sub.3 CH.sub.2 ONC(CH.sub.3)                              27      CH.sub.3 CCl.sub.3 CHCH                                                28      CH.sub.3 CF.sub.3  CH.sub.2 O                                          29      CH.sub.3 CF.sub.3  CH.sub.2 ONC(CH.sub.3)                              30      CH.sub.3 CF.sub.3  CHCH                                                31      Cl       CH.sub.3  CH.sub.2 O                                          32      Cl       CH.sub.3  CH.sub.2 ONC(CH.sub.3)                              33      Cl       CH.sub.3  CHCH                                                34      Cl       NH.sub.2  CH.sub.2 O                                          35      Cl       NH.sub.2  CH.sub.2 ONC(CH.sub.3)                              36      Cl       NH.sub.2  CHCH                                                37      Cl       N(CH.sub.3).sub.2                                                                        CH.sub.2 O                                          38      Cl       N(CH.sub.3).sub.2                                                                        CH.sub.2 ONC(CH.sub.3)                              39      Cl       N(CH.sub.3).sub.2                                                                        CHCH                                                40      Cl       CCl.sub.3 CH.sub.2 O                                          41      Cl       CCl.sub.3 CH.sub.2 ONC(CH.sub.3)                              42      Cl       CCl.sub.3 CHCH                                                43      Cl       CF.sub.3  CH.sub.2 O                                          44      Cl       CF.sub.3  CH.sub.2 ONC(CH.sub.3)                              45      Cl       CF.sub.3  CHCH                                                ______________________________________                                    

                  TABLE 23                                                         ______________________________________                                          ##STR234##                                                                    I: R.sup.1 = CH.sub.3, Z = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, Z =CH.sub.3                                   III: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                   IV: R.sup.1 = CH.sub.2 CH.sub.3, Z = C.sub.2 H.sub.5                           V: R.sup.1 = CH.sub.3, Z = NHCH.sub.3                                          VI: R.sup.1 = CH.sub.2 CH.sub.3, Z = NHCH.sub.3                                No.          B                                                                 ______________________________________                                          1           2-pyridyl                                                          2           3-Trifluoromethyl-2-pyridyl                                        3           5-Trifluoromethyl-2-pyridyl                                        4           3,5-Bis-(trifluoromethyl)-2-pyridyl                                5           3,5-Dichloro-2-pyridyl                                             6           3-Chloro-5-trifluoromethyl-2-pyridyl                               7           3,5-Dichloro-2-pyridyl                                             8           2-Chloro-4-trifluormethylphenyl                                    9           2-Benzothiazolyl                                                  10           5-Chloro-4-methyl-2-benzimidazolyl                                11           2-Benzoxazolyl                                                    12           1-Methyl-5-trifluoromethylimi-                                                 dazo 5,4-a!-pyridin-2-yl                                          13           5-Chloro-2-pyrimidinyl                                            14           4-Methyl-5-phenyl-2-thiazolin-2-yl                                15           4-Methyl-5-phenyl-2-Oxazolin-2-yl                                 16           7-Trifluoromethyl-4-quinolinyl                                    ______________________________________                                    

Example 10

N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methyl-hydroxylamine (Table 30, No. 1)

a) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-hydroxylamine

At 0° to 5° C., 7.0 g (70 mmol) of methyl chloroformate is added dropwise to 11.3 g (80 mmol) of N-2,6-dimethylphenyl-hydroxylamine (prepared analogously to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.5 g (90 mmol) of K₂ CO₃ in 30 ml of methylene chloride. The mixture is stirred for 30 mins at 0°-5° C., the insoluble solid is filtered off and the filtrate is evaporated down under reduced pressure. The residure is purified by column chromatography with mixtures of cyclohexand and ethyl acetate. There is obtained 1.4 g (7.2 mmol=9%) of the title compound as a dark oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 8.85 (s, broad, 1H, OH); 7.1 (m, 3H, phenyl); 3.75 (s, 3H, OCH₃); 2.3 (s, 6H, 2×CH₃)

b) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methylhydroxylamine (Table 7, No. 1)

A mixture of 1.4 g (7.2 mmol) of N-(2,6-dimethylphenyl)-N-methoxycarbonyl-hydroxylamine (Example 1a), 1.3 g (9 mmol) of K₂ CO₃ and 10 g (8 mmol) of dimethyl sulfate in 10 ml of acetone is stirred overnight at room temperature. The reaction mixture is then diluted with CH₂ Cl₂ and stirred with dilute NH₃ solution. The phases are then separated and the organic phase is extracted another twice with water. The organic phase is dried over MgSO₄ and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.2 g (6 mmol=83%) of the title compound as a colorless solid (mp=81° C.).

¹ H-NMR (CDCl₃ ; δ in ppm): 7.1 (m, 3H, phenyl); 3.75 (s, broad, 6H, 2×OCH3); 2.3 (s, 3H, CH₃)

The compounds listed in the following tables may be prepared similarly. Compound I, No. 1 from Table 24, No. 1 has for example the following formula: ##STR235##

                  TABLE 24                                                         ______________________________________                                         a I: R.sup.1 = CH.sub.3, X = CH.sub.3                                          b II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3                                c III: R.sup.1 = CH.sub.3, X = Cl                                              d IV: R.sup.1 = CH.sub.2 CH.sub.2, X = Cl                                      No.     T.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          1I1     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    181     3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    182     4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 -CO                                                    303     2-Me-4-CH.sub.3 -CH.sub.2 CO                                           304     2-Me-4-CH.sub.3 -CH.sub.2 CH.sub.2 CO                                  305     2-Me-4-CH.sub.3 -CH(CH.sub.3)CO                                        306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-CH.sub.3 -CO                                           308     2,5-Me.sub.2 -4-CH.sub.3 -CH.sub.2 CO                                  309     2,5-Me.sub.2 -4-CH.sub.3 -CH.sub.2 CH.sub.2 CO                         310     2,5-Me.sub.2 -4-CH.sub.3 -CH(CH.sub.3)CO                               311     2-Cl-4-CHO                                                             312     2-Cl-4-CH.sub.3 -CO                                                    313     2-Cl-4-CH.sub.3 -CH.sub.2 CO                                           314     2-Cl-4-CH.sub.3 -CH(CH.sub.3)CO                                        315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-CH.sub.3 -CO                                           317     2,5-Cl.sub.2 -4-CH.sub.3 -CH.sub.2 CO                                  318     2,5-Cl.sub.2 -4-CH.sub.3 -CH.sub.2 CH.sub.2 CO                         319     2,5-Cl.sub.2 -4-CH.sub.3 -CH(CH.sub.3)CO                               320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)CH.sub.3                                                  333     3-C(NO-Allyl)CH.sub.3                                                  334     4-C(NO-Allyl)CH.sub.3                                                  335     2-C(NO-trans-Chloroallyl)CH.sub.3                                      336     3-C(NO-trans-Chloroallyl)CH.sub.3                                      337     4-C(NO-trans-Chloroallyl)CH.sub.3                                      338     2-C(NO-Propargyl)CH.sub.3                                              339     3-C(NO-Propargyl)CH.sub.3                                              340     4-C(NO-Propargyl)CH.sub.3                                              341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 -CNOCH.sub.3)                                  357     2-CH.sub.3 -4-(CH.sub.3 -CNOC.sub.2 H.sub.5)                           358     2-CH.sub.3 -4-(CH.sub.3 -CNO-n-C.sub.3 H.sub.7)                        359     2-CH.sub.3 -4-(CH.sub.3 -CNO-i-C.sub.3 H.sub.7)                        360     2-CH.sub.3 -4-(CH.sub.3 -CNO-Allyl)                                    361     2-CH.sub.3 -4-(CH.sub.3 -CNO-trans-Chloroallyl)                        362     2-CH.sub.3 -4-(CH.sub.3 -CNO-Propargyl)                                363     2-CH.sub.3 -4-(CH.sub.3 -CNO-n-C.sub.4 H.sub.9)                        364     2-CH.sub.3 -4-(CH.sub.3 -CNOCH.sub.2 C.sub.6 H.sub.5)                  365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                   369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNOCH.sub.3)                        375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNOC.sub.2 H.sub.5)                 376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-n-C.sub.3 H.sub.7)              377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-i-C.sub.3 H.sub.7)              378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-Allyl)                          379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-trans-Chloroallyl)              380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-Proparyl)                       381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNO-n-C.sub.4 H.sub.9)              382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 -CNOCH.sub.2 C.sub.6 H.sub.5)        383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 25                                                         ______________________________________                                          ##STR236##                                                                    I: R.sup.1 = CH.sub.3, X = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3                                  III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = CH.sub.2 CH.sub.3, X = Cl                                        No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                            2        NCH.sub.3 -Pyrrolyl-3                                                 3        NC.sub.6 H.sub.5 -Pyrrolyl-3                                          4        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            5        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            6        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            7        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           8        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           9        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           10       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            11       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            12       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            13       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   14       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   15       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   16       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   17       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   18       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   19       Pyrrolyl-2                                                            20       NCH.sub.3 -Pyrrolyl-2                                                 21       NC.sub.6 H.sub.5 -Pyrrolyl-2                                          22       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            23       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            24       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            25       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           26       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           27       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           28       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            29       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            30       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            31       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   32       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   33       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   34       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   35       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   36       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   37       Furyl-2                                                               38       5-CH.sub.3 -Furyl-2                                                   39       5-C.sub.6 H.sub.5 -Furyl-2                                            40       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               41       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               42       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               43       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              44       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              45       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              46       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               47       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               48       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               49       5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      50       5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      51       5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      52       5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      53       5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      54       5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      55       4-CH.sub.3 -Furyl-2                                                   56       4-C.sub.6 H.sub.5 -Furyl-2                                            57       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               58       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               59       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               60       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              61       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              62       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              63       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               64       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               65       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               66       4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      67       4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      68       4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      69       4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      70       4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      71       4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      72       Thienyl-2                                                             73       5-CH.sub.3 -Thienyl-2                                                 74       5-C.sub.6 H.sub.5 -Thienyl-2                                          75       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             76       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             77       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             78       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            79       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            80       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            81       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             82       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             83       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             84       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    85       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    86       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    87       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    88       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    89       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    90       4-CH.sub.3 -Thienyl-2                                                 91       4-C.sub.6 H.sub.5 -Thienyl-2                                          92       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             93       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             94       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             95       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            96       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            97       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            98       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             99       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(41-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       NCH.sub.3 -Pyrazolyl-4                                               127       NC.sub.6 H.sub.5 -Pyrazolyl-4                                        128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 143       3-CH.sub.3 -N-Methylpyrazolyl-4                                      144       3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                                145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                 151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  154       3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         155       3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         156       3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         157       3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         158       3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         159       3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                         160       Isoxazolyl-5                                                         161       3-CH.sub.3 -Isoxazolyl-5                                             162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4 -4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 -Isoxazolyl-3                                             198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 -Isothiazolyl-5                                           216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       2-CH.sub.3 -Oxazolyl-4                                               234       2-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       2-(4'-CH.sub.3 C.sub.6 H.sub.4)Oxazolyl-4                            236       2-(3'-CH.sub.3 C.sub.6 H.sub.4)Oxazolyl-4                            237       2-(2'-CH.sub.3 C.sub.6 H.sub.4)Oxazolyl-4                            238       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)Oxazolyl-4                           239       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)Oxazolyl-4                           241       2-(4'-NO.sub.2 C.sub.6 H.sub.4)Oxazolyl-4                            242       2-(3'-NO.sub.2 C.sub.6 H.sub.4)Oxazolyl-4                            243       2-(2'-NO.sub.2 C.sub.6 H.sub.4)Oxazolyl-4                            244       2-(4'-CNC.sub.6 H.sub.4)Oxazolyl-4                                   245       2-(3'-CNC.sub.6 H.sub.4)Oxazolyl-4                                   246       2-(2'-CNC.sub.6 H.sub.4)Oxazolyl-4                                   247       2-(4'-ClC.sub.6 H.sub.4)Oxazolyl-4                                   248       2-(3'-ClC.sub.6 H.sub.4)Oxazolyl-4                                   249       2-(2'-ClC.sub.6 H.sub.4)Oxazolyl-4                                   250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       NCH.sub.3 -1,2,4-Triazolyl-5                                         269       3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                              270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5        275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5        276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5        277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         280       3-(4'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                281       3-(3'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                282       3-(2'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                283       3-(4'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                284       3-(3'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                285       3-(2'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazoiyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        384       Pyridinyl-3                                                          385       1-Naphthyl                                                           386       2-Naphthyl                                                           ______________________________________                                    

                  TABLE 26                                                         ______________________________________                                          ##STR237##                                                                    I: R.sup.1 = CH.sub.3, X = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3                                  III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = CH.sub.2 CH.sub.3, X = Cl                                        No.     T.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    181     3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    182     4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-CH.sub.3 CH.sub.2 CO                                            304     2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                   305     2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                         306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-CH.sub.3 CO                                            308     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   309     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          310     2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                311     2-Cl-4-CHO                                                             312     2-Cl-4-CH.sub.3 CO                                                     313     2-Cl-4-CH.sub.3 CH.sub.2 CO                                            314     2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                         315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-CH.sub.3 CO                                            317     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   318     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          319     2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                  369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                        381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-CH.sub.2 C.sub.6 H.sub.5)        383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyI))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 27                                                         ______________________________________                                          ##STR238##                                                                    I: R.sup.1 = CH.sub.3, X = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3                                  III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = CH.sub.2 CH.sub.3, X = Cl                                        No.     B                                                                      ______________________________________                                          1      Pyrrolyl-3                                                              2      NCH.sub.3 -Pyrrolyl-3                                                   3      NC.sub.6 H.sub.5 -Pyrrolyl-3                                            4      N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                              5      N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                              6      N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                              7      N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                             8      N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                             9      N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                             10     N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                              11     N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                              12     N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                              13     N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                     14     N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                     15     N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                     16     N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                     17     N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                     18     N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                     19     Pyrrolyl-2                                                              20     N-CH.sub.3 -Pyrrolyl-2                                                  21     N-C.sub.6 H.sub.5 -Pyrrolyl-2                                           22     N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                              23     N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                              24     N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                              25     N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                             26     N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                             27     N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                             28     N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                              29     N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                              30     N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                              31     N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                     32     N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                     33     N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                     34     N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                     35     N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                     36     N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                     37     Furyl-2                                                                 38     5-CH.sub.3 -Furyl-2                                                     39     5-C.sub.6 H.sub.5 -Furyl-2                                              40     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 41     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 42     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 43     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                44     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                45     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                46     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 47     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 48     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 49     5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                        50     5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                        51     5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                        52     5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                        53     5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                        54     5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                        55     4-CH.sub.3 -Furyl-2                                                     56     4-C.sub.6 H.sub.5 -Furyl-2                                              57     4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 58     4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 59     4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 60     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                61     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                62     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                63     4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 64     4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 65     4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 66     4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                        67     4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                        68     4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                        69     4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                        70     4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                        71     4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                        72     Thienyl-2                                                               73     5-CH.sub.3 -Thienyl-2                                                   74     5-C.sub.6 H.sub.5 -Thienyl-2                                            75     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               76     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               77     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               78     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              79     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              80     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              81     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                               82     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                               83     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                               84     5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                      85     5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                      86     5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                      87     5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                      88     5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                      89     5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                      90     4-CH.sub.3 -Thienyl-2                                                   91     4-C.sub.6 H.sub.5 -Thienyl-2                                            92     4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               93     4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               94     4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               95     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              96     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              97     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              98     4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                               99     4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                              100     4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                              101     4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                     102     4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                     103     4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                     104     4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                     105     4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                     106     4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                     107     Thienyl-3                                                              108     5-CH.sub.3 -Thienyl-3                                                  109     5-C.sub.6 H.sub.5 -Thienyl-3                                           110     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                              111     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                              112     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                              113     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                             114     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                             115     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                             116     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                              117     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                              118     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                              119     5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                     120     5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                     121     5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                     122     5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                     123     5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                     124     5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                     125     Pyrazolyl-4                                                            126     NCH.sub.3 -Pyrazolyl-4                                                 127     NC.sub.6 H.sub.5 -Pyrazolyl-4                                          128     N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                            129     N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                            130     N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                            131     N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                           132     N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                           133     N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                           134     N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                            135     N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                            136     N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                            137     N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                   138     N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                   139     N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                   140     N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                   141     N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                   142     N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                   143     3-CH.sub.3 -N-Methylpyrazolyl-4                                        144     3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4                                 145     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                    146     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                    147     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                    148     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   149     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   150     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   151     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                    152     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                    153     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                    154     3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                           155     3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                           156     3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                           157     3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                           158     3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                           159     3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                           160     Isoxazolyl-5                                                           161     3-CH.sub.3 -Isoxazolyl-5                                               162     3-C.sub.6 H.sub.5 -Isoxazolyl-5                                        163     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                           164     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                           165     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                           166     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                          167     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                          168     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                          169     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                           170     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                           171     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                           172     3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                  173     3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                  174     3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                  175     3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                  176     3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                  177     3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                  178     4-Chloroisoxazolyl-5                                                   179     3-CH.sub.3 -4-Chloroisoxazolyl-5                                       180     3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                                181     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                   182     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                   183     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                   184     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  185     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  186     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  187     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                   188     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                   189     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                   190     3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                          191     3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                          192     3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                          193     3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                          194     3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                          195     3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                          196     Isoxazolyl-3                                                           197     5-CH.sub.3 -Isoxazolyl-3                                               198     5-C.sub.6 H.sub.5 -Isoxazolyl-3                                        199     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                           200     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                           201     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                           202     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                          203     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                          204     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                          205     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                           206     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                           207     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                           208     5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                  209     5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                  210     5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                  211     5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                  212     5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                  213     5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                  214     Isothiazolyl-5                                                         215     3-CH.sub.3 -Isothiazolyl-5                                             216     3-C.sub.6 H.sub.5 -Isothiazolyl-5                                      217     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                         218     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                         219     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                         220     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                        221     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                        222     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                        223     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                         224     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                         225     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                         226     3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                                227     3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                                228     3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                                229     3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                                230     3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                                231     3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                                232     Oxazolyl-4                                                             233     2-CH.sub.3 -Oxazolyl-4                                                 234     2-C.sub.6 H.sub.5 -Oxazolyl-4                                          235     2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                             236     2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                             237     2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                             238     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                            239     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                            240     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                            241     2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                             242     2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                             243     2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                             244     2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                    245     2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                    246     2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                    247     2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                    248     2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                    249     2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                    250     Thiazolyl-4                                                            251     2-CH.sub.3 -Thiazolyl-4                                                252     2-C.sub.6 H.sub.5 -Thiazolyl-4                                         253     2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                            254     2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                            255     2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                            256     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                           267     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                           258     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                           259     2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                            260     2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                            261     2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                            262     2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                   263     2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                   264     2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                   265     2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                   266     2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                   267     2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                   268     NCH.sub.3 -1,2,4-Triazolyl-5                                           269     3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                                270     3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                         271     3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            272     3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            273     3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            274     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5           275     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5           276     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5           277     3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            278     3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            279     3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            280     3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   281     3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   282     3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   283     3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   284     3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   285     3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   286     1,3,4-Oxadiazolyl-2                                                    287     5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                        288     5-C.sub.6 H.sub.5 -1,2,3-Oxadiazolyl-2                                 289     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    290     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    291     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    292     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   293     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   294     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   295     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    296     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    297     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    298     5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           299     5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           300     5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           301     5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           302     5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           303     5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           304     1,2,4-Oxadiazolyl-3                                                    305     5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                        306     5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                 307     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    308     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    309     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    310     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   311     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   312     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   313     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    314     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    315     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    316     5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           317     5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           318     5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           319     5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           320     5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           321     5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           322     1,2,4-Oxadiazolyl-5                                                    323     3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                        324     3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                 325     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    326     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    327     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    328     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   329     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   330     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   331     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    332     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    333     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    334     3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           335     3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           336     3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           337     3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           338     3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           339     3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           340     1,2,4-Thiadiazolyl-3                                                   341     5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                       342     5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                343     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   344     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   345     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   346     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  347     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  348     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  349     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   350     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   351     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   352     5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          353     5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          354     5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          355     5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          356     5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          357     5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          358     1,3,4-Thiadiazolyl-2                                                   359     5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                       360     5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                361     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   362     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   363     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   364     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  365     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  366     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  367     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   368     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   369     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   370     5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          371     5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          372     5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          373     5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          374     5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          375     5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          376     Pyridinyl-2                                                            377     Pyridinyl-4                                                            378     Pyridazinyl-3                                                          379     Pyridazinyl-4                                                          380     Pyridazinyl-2                                                          381     Pyrimidinyl-4                                                          382     Pyrimidinyl-5                                                          383     Pyrimidinyl-2                                                          384     Pyridinyl-3                                                            385     1-Naphthyl                                                             386     2-Naphthyl                                                             ______________________________________                                    

                  TABLE 28                                                         ______________________________________                                          ##STR239##                                                                    I: R.sup.1 = CH.sub.3, X = CH.sub.3                                            II: R.sup.1 = CH.sub.2 CH.sub.3, X = CH.sub.3                                  III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = CH.sub.2 CH.sub.3, X = Cl                                        No.      T.sub.m                                                               ______________________________________                                         1        H                                                                     2        2-F                                                                   3        3-F                                                                   4        4-F                                                                   5        2,4-F.sub.2                                                           6        2,4,6-F.sub.3                                                         7        2,3,4,5,6-F.sub.5                                                     8        2,3-F.sub.2                                                           9        2-Cl                                                                  10       3-Cl                                                                  11       4-Cl                                                                  12       2,3-Cl.sub.2                                                          13       2,4-Cl.sub.2                                                          14       2,5-Cl.sub.2                                                          15       2,6-Cl.sub.2                                                          16       3,4-Cl.sub.2                                                          17       3,5-Cl.sub.2                                                          18       2,3,4-Cl.sub.3                                                        19       2,3,5-Cl.sub.3                                                        20       2,3,6-Cl.sub.3                                                        21       2,4,5-Cl.sub.3                                                        22       2,4,6-Cl.sub.3                                                        23       3,4,5-Cl.sub.3                                                        24       2,3,4,6-Cl.sub.4                                                      25       2,3,5,6-Cl.sub.4                                                      26       2,3,4,5,6-Cl.sub.5                                                    27       2-Br                                                                  28       3-Br                                                                  29       4-Br                                                                  30       2,4-Br.sub.2                                                          31       2,5-Br.sub.2                                                          32       2,6-Br.sub.2                                                          33       2,4,6-Br.sub.3                                                        34       2,3,4,5,6-Br.sub.5                                                    35       2-I                                                                   36       3-I                                                                   37       4-I                                                                   38       2,4-I.sub.2                                                           39       2-Cl, 3-F                                                             40       2-Cl, 4-F                                                             41       2-Cl, 5-F                                                             42       2-Cl, 6-F                                                             43       2-Cl, 3-Br                                                            44       2-Cl, 4-Br                                                            45       2-Cl, 5-Br                                                            46       2-Cl, 6-Br                                                            47       2-Br, 3-Cl                                                            48       2-Br, 4-Cl                                                            49       2-Br, 5-Cl                                                            50       2-Br, 3-F                                                             51       2-Br, 4-F                                                             52       2-Br, 5-F                                                             53       2-Br, 6-F                                                             54       2-F, 3-Cl                                                             55       2-F, 4-Cl                                                             56       2-F, 5-Cl                                                             57       3-Cl, 4-F                                                             58       3-Cl, 5-F                                                             59       3-Cl, 4-Br                                                            60       3-Cl, 5-Br                                                            61       3-F, 4-Cl                                                             62       3-F, 4-Br                                                             63       3-Br, 4-Cl                                                            64       3-Br, 4-F                                                             65       2,6-Cl.sub.2, 4-Br                                                    66       2-CH.sub.3                                                            67       3-CH.sub.3                                                            68       4-CH.sub.3                                                            69       2,3-(CH.sub.3).sub.2                                                  70       2,4-(CH.sub.3).sub.2                                                  71       2,5-(CH.sub.3).sub.2                                                  72       2,6-(CH.sub.3).sub.2                                                  73       3,4-(CH.sub.3).sub.2                                                  74       3,5-(CH.sub.3).sub.2                                                  75       2,3,5-(CH.sub.3).sub.3                                                76       2,3,4-(CH.sub.3).sub.3                                                77       2,3,6-(CH.sub.3).sub.3                                                78       2,4,5-(CH.sub.3).sub.3                                                79       2,4,6-(CH.sub.3).sub.3                                                80       3,4,5-(CH.sub.3).sub.3                                                81       2,3,4,6-(CH.sub.3).sub.4                                              82       2,3,5,6-(CH.sub.3).sub.4                                              83       2,3,4,5,6-(CH.sub.3).sub.5                                            84       2-C.sub.2 H.sub.5                                                     85       3-C.sub.2 H.sub.5                                                     86       4-C.sub.2 H.sub.5                                                     87       2,4-(C.sub.2 H.sub.5).sub.2                                           88       2,6-(C.sub.2 H.sub.5).sub.2                                           89       3,5-(C.sub.2 H.sub.5).sub.2                                           90       2,4,6-(C.sub.2 H.sub.5).sub.3                                         91       2-n-C.sub.3 H.sub.7                                                   92       3-n-C.sub.3 H.sub.7                                                   93       4-n-C.sub.3 H.sub.7                                                   94       2-i-C.sub.3 H.sub.7                                                   95       3-i-C.sub.3 H.sub.7                                                   96       4-i-C.sub.3 H.sub.7                                                   97       2,4-(i-C.sub.3 H.sub.7).sub.2                                         98       2,6-(i-C.sub.3 H.sub.7).sub.2                                         99       3,5-(i-C.sub.3 H.sub.7).sub.2                                         100      2,4,6-(i-C.sub.3 H.sub.7).sub.3                                       101      2-s-C.sub.4 H.sub.9                                                   102      3-s-C.sub.4 H.sub.9                                                   103      4-s-C.sub.4 H.sub.9                                                   104      2-t-C.sub.4 H.sub.9                                                   105      3-t-C.sub.4 H.sub.9                                                   106      4-t-C.sub.4 H.sub.9                                                   107      2,3-(t-C.sub.4 H.sub.9).sub.2                                         108      2,4-(t-C.sub.4 H.sub.9).sub.2                                         109      2,5-(t-C.sub.4 H.sub.9).sub.2                                         110      2,6-(t-C.sub.4 H.sub.9).sub.2                                         111      3,4-(t-C.sub.4 H.sub.9).sub.2                                         112      2,4,6-(t-C.sub.4 H.sub.9).sub.3                                       113      4-n-C.sub.9 H.sub.19                                                  114      4-n-C.sub.12 H.sub.25                                                 115      4-n-C.sub.15 H.sub.31                                                 116      4-(1,1,3,3-Tetramethylbutyl)                                          117      4-(2,4,4-Trimethylpropyl)                                             118      2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                       119      2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                       120      2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                             121      2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                       122      2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                       123      2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                       124      2-CH.sub.3,5-i-C.sub.3 H.sub.7                                        125      3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                       126      2-i-C.sub.3 H.sub.7,5-CH.sub.3                                        127      2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                    128      2-Allyl                                                               129      3-Allyl                                                               130      4-Allyl                                                               131      2-Allyl, 6-CH.sub.3                                                   132      2-cyclo-C.sub.6 H.sub.11                                              133      3-cyclo-C.sub.6 H.sub.11                                              134      4-cyclo-C.sub.6 H.sub.11                                              135      2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                        136      2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                  137      2-CH.sub.2 C.sub.6 H.sub.5                                            138      3-CH.sub.2 C.sub.6 H.sub.5                                            139      4-CH.sub.2 C.sub.6 H.sub.5                                            140      2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                141      2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                142      2-C.sub.6 H.sub.5                                                     143      3-C.sub.6 H.sub.5                                                     144      4-C.sub.6 H.sub.5                                                     145      4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                               146      4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                               147      2-Cl, 4-C.sub.6 H.sub.5                                               148      2-Br, 4-C.sub.6 H.sub.5                                               149      2-C.sub.6 H.sub.5, 4-Cl                                               150      2-C.sub.6 H.sub.5, 4-Br                                               151      2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                      152      2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                      153      2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                      154      2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                      155      2-cyclo-C.sub.6 H.sub.11, 4-Cl                                        156      2-cyclo-C.sub.6 H.sub.11, 4-Br                                        157      2-Cl, 4-cyclo-C.sub.6 H.sub.11                                        158      2-Br, 4-cyclo-C.sub.6 H.sub.11                                        159      2-OCH.sub.3                                                           160      3-OCH.sub.3                                                           161      4-OCH.sub.3                                                           162      2-OC.sub.2 H.sub.5                                                    163      3-OC.sub.2 H.sub.5                                                    164      4-OC.sub.2 H.sub.5                                                    165      2-O-n-C.sub.3 H.sub.7                                                 166      3-O-n-C.sub.3 H.sub.7                                                 167      4-O-n-C.sub.3 H.sub.7                                                 168      2-O-i-C.sub.3 H.sub.7                                                 169      3-O-i-C.sub.3 H.sub.7                                                 170      4-O-i-C.sub.3 H.sub.7                                                 171      2-O-n-C.sub.6 H.sub.13                                                172      3-O-n-C.sub.6 H.sub.13                                                173      4-O-n-C.sub.6 H.sub.13                                                174      2-O-n-C.sub.8 H.sub.17                                                175      3-O-n-C.sub.8 H.sub.17                                                176      4-O-n-C.sub.8 H.sub.17                                                177      2-OCH.sub.2 C.sub.6 H.sub.5                                           178      3-OCH.sub.2 C.sub.6 H.sub.5                                           179      4-OCH.sub.2 C.sub.6 H.sub.5                                           180      2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   181      3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   182      4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183      2,4-(OCH.sub.3).sub.2                                                 184      2-CF.sub.3                                                            185      3-CF.sub.3                                                            186      4-CF.sub.3                                                            187      2-OCF.sub.3                                                           188      3-CCF.sub.3                                                           189      4-OCF.sub.3                                                           190      3-OCH.sub.2 CHF.sub.2                                                 191      2-NO.sub.2                                                            192      3-NO.sub.2                                                            193      4-NO.sub.2                                                            194      2-CN                                                                  195      3-CN                                                                  196      4-CN                                                                  197      2-CH.sub.3, 3-Cl                                                      198      2-CH.sub.3, 4-Cl                                                      199      2-CH.sub.3, 5-Cl                                                      200      2-CH.sub.3, 6-Cl                                                      201      2-CH.sub.3, 3-F                                                       202      2-CH.sub.3, 4-F                                                       203      2-CH.sub.3, 5-F                                                       204      2-CH.sub.3, 6-F                                                       205      2-CH.sub.3, 3-Br                                                      206      2-CH.sub.3, 4-Br                                                      207      2-CH.sub.3, 5-Br                                                      208      2-CH.sub.3, 6-Br                                                      209      2-Cl, 3-CH.sub.3                                                      210      2-Cl, 4-CH.sub.3                                                      211      2-Cl, 5-CH.sub.3                                                      212      2-F, 3-CH.sub.3                                                       213      2-F, 4-CH.sub.3                                                       214      2-F, 5-CH.sub.3                                                       215      2-Br, 3-CH.sub.3                                                      216      2-Br, 4-CH.sub.3                                                      217      2-Br, 5-CH.sub.3                                                      218      3-CH.sub.3, 4-Cl                                                      219      3-CH.sub.3, 5-Cl                                                      220      3-CH.sub.3, 4-F                                                       221      3-CH.sub.3, 5-F                                                       222      3-CH.sub.3, 4-Br                                                      223      3-CH.sub.3, 5-Br                                                      224      3-F, 4-CH.sub.3                                                       225      3-Cl, 4-CH.sub.3                                                      226      3-Br, 4-CH.sub.3                                                      227      2-Cl, 4, 5-(CH.sub.3).sub.2                                           228      2-Br, 4, 5-(CH.sub.3).sub.2                                           229      2-Cl, 3, 5-(CH.sub.3).sub.2                                           230      2-Br, 3, 5-(CH.sub.3).sub.2                                           231      2,6-Cl.sub.2, 4-CH.sub.3                                              232      2,6-F.sub.2, 4-CH.sub.3                                               233      2,6-Br.sub.2, 4-CH.sub.3                                              234      2,4-Br.sub.2, 6-CH.sub.3                                              235      2,4-F.sub.2, 6-CH.sub.3                                               236      214-Br.sub.2, 6-CH.sub.3                                              237      2,6-(CH.sub.3).sub.2, 4-F                                             238      2,6-(CH.sub.3).sub.2, 4-Cl                                            239      2,6-(CH.sub.3).sub.2, 4-Br                                            240      3,5-(CH.sub.3).sub.2, 4-F                                             241      3,5-(CH.sub.3).sub.2, 4-Cl                                            242      3,5-(CH.sub.3).sub.2, 4-Br                                            243      2,3,6-(CH.sub.3).sub.3, 4-F                                           244      2,3,6-(CH.sub.3).sub.3, 4-Cl                                          245      2,3,6-(CH.sub.3).sub.3, 4-Br                                          246      2,4-(CH.sub.3).sub.2, 6-F                                             247      2,4-(CH.sub.3).sub.2, 6-Cl                                            248      2,4-(CH.sub.3).sub.2, 6-Br                                            249      2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                 250      2-Cl, 4-NO.sub.2                                                      251      2-NO.sub.2, 4-Cl                                                      252      2-OCH.sub.3, 5-NO.sub.2                                               253      2,4-Cl.sub.2, 5-NO.sub.2                                              254      2,4-Cl.sub.2, 6-NO.sub.2                                              255      2,6-Cl.sub.2, 4-NO.sub.2                                              256      2,6-Br.sub.2, 4-NO.sub.2                                              257      2,6-I.sub.2, 4-NO.sub.2                                               258      2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                 259      2-CO.sub.2 CH.sub.3                                                   260      3-CO.sub.2 CH.sub.3                                                   261      4-CO.sub.2 CH.sub.3                                                   262      2-CO.sub.2 (C.sub.2 H.sub.5)                                          263      3-CO.sub.2 (C.sub.2 H.sub.5)                                          264      4-CO.sub.2 (C.sub.2 H.sub.5)                                          265      2-CO.sub.2 (n-C.sub.3 H.sub.7)                                        266      3-CO.sub.2 (n-C.sub.3 H.sub.7)                                        267      4-CO.sub.2 (n-C.sub.3 H.sub.7)                                        268      2-CO.sub.2 (i-C.sub.3 H.sub.7)                                        269      3-CO.sub.2 (i-C.sub.3 H.sub.7)                                        270      4-CO.sub.2 (i-C.sub.3 H.sub.7)                                        271      2-CO.sub.2 (n-C.sub.6 H.sub.13)                                       272      3-CO.sub.2 (n-C.sub.6 H.sub.13)                                       273      4-CO.sub.2 (n-C.sub.6 H.sub.13)                                       274      2-CH.sub.2 OCH.sub.3                                                  275      3-CH.sub.2 OCH.sub.3                                                  276      4-CH.sub.2 OCH.sub.3                                                  277      2-CH.sub.2 O(C.sub.2 H.sub.5)                                         278      3-CH.sub.2 O(C.sub.2 H.sub.5)                                         279      4-CH.sub.2 O(C.sub.2 H.sub.5)                                         280      2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                       281      3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                       282      4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                       283      2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                       284      3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                       285      4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                       286      2-CHO                                                                 287      3-CHO                                                                 288      4-CHO                                                                 289      2-COCH.sub.3                                                          290      3-COCH.sub.3                                                          291      4-COCH.sub.3                                                          292      2-COCH.sub.2 CH.sub.3                                                 293      3-COCH.sub.2 CH.sub.3                                                 294      4-COCH.sub.2 CH.sub.3                                                 295      2-COCH.sub.2 CH.sub.2 CH.sub.3                                        296      3-COCH.sub.2 CH.sub.2 CH.sub.3                                        297      4-COCH.sub.2 CH.sub.2 CH.sub.3                                        298      2-COCH(CH.sub.3)CH.sub.3                                              299      3-COCH(CH.sub.3)CH.sub.3                                              300      4-COCH(CH.sub.3)CH.sub.3                                              301      2-Me-4-CHO                                                            302      2-Me-4-CH.sub.3 CO                                                    303      2-Me-4-CH.sub.3 CH.sub.2 CO                                           304      2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                  305      2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                        306      2,5-Me.sub.2 -4-CHO                                                   307      2,5-Me.sub.2 -4-CH.sub.3 CO                                           308      2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                  309      2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                         310      2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                               311      2-Cl-4-CHO                                                            312      2-Cl-4-CH.sub.3 CO                                                    313      2-Cl-4-CH.sub.3 CH.sub.2 CO                                           314      2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                        315      2,5-Cl.sub.2 -4-CHO                                                   316      2,5-Cl.sub.2 -4-CH.sub.3 CO                                           317      2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                  318      2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                         319      2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                               320      2-C(NOCH.sub.3)CH.sub.3                                               321      3-C(NOCH.sub.3)CH.sub.3                                               322      4-C(NOCH.sub.3)CH.sub.3                                               323      2-C(NOC.sub.2 H.sub.5)CH.sub.3                                        324      3-C(NOC.sub.2 H.sub.5)CH.sub.3                                        325      4-C(NOC.sub.2 H.sub.5)CH.sub.3                                        326      2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     327      3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     328      4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     329      2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     330      3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     331      4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     332      2-C(NO-Allyl)-CH.sub.3                                                333      3-C(NO-Allyl)-CH.sub.3                                                334      4-C(NO-Allyl)-CH.sub.3                                                335      2-C(NO-trans-Chloroallyl)-CH.sub.3                                    336      3-C(NO-trans-Chloroallyl)-CH.sub.3                                    337      4-C(NO-trans-Chloroallyl)-CH.sub.3                                    338      2-C(NO-Propargyl)-CH.sub.3                                            339      3-C(NO-Propargyl)-CH.sub.3                                            340      4-C(NO-Propargyl)-CH.sub.3                                            341      2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     342      3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     343      4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     344      2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               345      3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               346      4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               347      2-CH.sub.3 -4-CHNOCH.sub.3                                            348      2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                     349      2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                  350      2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                  351      2-CH.sub.3 -4-CHNO-Allyl                                              352      2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                353      2-CH.sub.3 -4-CHNO-Propargyl                                          354      2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                  355      2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                            356      2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                  357      2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                           358      2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                        359      2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                        360      2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                    361      2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                        362      2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                363      2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                        364      2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                  365      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                           366      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                    367      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                 368      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                 369      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                             370      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                 371      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                         372      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                 373      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)           374      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                        375      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                 376      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)              377      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)              378      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                          379      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)              380      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                       381      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)              382      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)        383      2-C.sub.6 H.sub.5                                                     384      3-C.sub.6 H.sub.5                                                     385      4-C.sub.6 H.sub.5                                                     386      2-(2'-FC.sub.6 H.sub.4)                                               387      2-(3'-FC.sub.6 H.sub.4)                                               388      2-(4'-FC.sub.6 H.sub.4)                                               389      3-(2'-FC.sub.6 H.sub.4)                                               390      3-(3'-FC.sub.6 H.sub.4)                                               391      3-(4'-FC.sub.6 H.sub.4)                                               392      4-(2'-FC.sub.6 H.sub.4)                                               393      4-(3'-FC.sub.6 H.sub.4)                                               394      4-(4'-FC.sub.6 H.sub.4)                                               395      2-(2'-ClC.sub.6 H.sub.4)                                              396      2-(3'-ClC.sub.6 H.sub.4)                                              397      2-(4'-ClC.sub.6 H.sub.4)                                              398      3-(2'-ClC.sub.6 H.sub.4)                                              399      3-(3'-ClC.sub.6 H.sub.4)                                              400      3-(4'-ClC.sub.6 H.sub.4)                                              401      4-(2'-ClC.sub.6 H.sub.4)                                              402      4-(3'-ClC.sub.6 H.sub.4)                                              403      4-(4'-ClC.sub.6 H.sub.4)                                              405      2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       406      2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       407      2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       408      3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       409      3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       410      3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       411      4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       412      4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       413      4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       414      2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     415      2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     416      2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     417      3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     418      3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     419      3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     420      4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     421      4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     422      4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     423      2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          424      2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          425      2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          426      3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          427      3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          428      3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          429      4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          430      4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          431      4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          432      2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              433      2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              434      2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              435      3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              436      3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              437      3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              438      4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              439      4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              440      4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              441      2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      442      2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      443      2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      444      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      445      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      446      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      447      4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      448      4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      449      4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      450      2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       451      2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       452      2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       453      3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       454      3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       455      3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       456      4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       457      4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       458      4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       459      2-(2'-NCC.sub.6 H.sub.4)                                              460      2-(3'-NCC.sub.6 H.sub.4)                                              461      2-(4'-NCC.sub.6 H.sub.4)                                              462      3-(2'-NCC.sub.6 H.sub.4)                                              463      3-(3'-NCC.sub.6 H.sub.4)                                              464      3-(4'-NCC.sub.6 H.sub.4)                                              465      4-(2'-NCC.sub.6 H.sub.4)                                              466      4-(3'-NCC.sub.6 H.sub.4)                                              467      4-(4'-NCC.sub.6 H.sub.4)                                              468      2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       469      2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       470      2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       471      3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       472      3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       473      3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       474      4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       475      4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       476      4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       477      2-OC.sub.6 H.sub.5                                                    475      3-OC.sub.6 H.sub.5                                                    476      4-OC.sub.6 H.sub.5                                                    478      2-O-(2'-FC.sub.6 H.sub.4)                                             479      2-O-(3'-FC.sub.6 H.sub.4)                                             480      2-O-(4'-FC.sub.6 H.sub.4)                                             481      3-O-(2'-FC.sub.6 H.sub.4)                                             482      3-O-(3'-FC.sub.6 H.sub.4)                                             483      3-O-(4'-FC.sub.6 H.sub.4)                                             484      4-O-(2'-FC.sub.6 H.sub.4)                                             485      4-O-(3'-FC.sub.6 H.sub.4)                                             486      4-O-(4'-FC.sub.6 H.sub.4)                                             487      2-O-(2'-ClC.sub.6 H.sub.4)                                            488      2-O-(3'-ClC.sub.6 H.sub.4)                                            489      2-O-(4'-ClC.sub.6 H.sub.4)                                            490      3-O-(2'-ClC.sub.6 H.sub.4)                                            491      3-O-(3'-ClC.sub.6 H.sub.4)                                            492      3-O-(4'-ClC.sub.6 H.sub.4)                                            493      3-O-(4'-ClC.sub.6 H.sub.4)                                            494      4-O-(2'-ClC.sub.6 H.sub.4)                                            495      4-O-(3'-ClC.sub.6 H.sub.4)                                            496      4-O-(4'-ClC.sub.6 H.sub.4)                                            497      2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     498      2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     499      2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     500      3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     501      3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     502      3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     503      4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     504      4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     505      4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     506      2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   507      2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   508      2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   509      3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   510      3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   511      3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   512      4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   513      4-O-(3'-CH.sub.3 CO-C.sub.6 H.sub.4)                                  514      4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   515      2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        516      2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        517      2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        518      3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        519      3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        520      3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        521      4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        522      4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        523      4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        524      2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            525      2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            526      2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            527      3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            528      3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            529      3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            530      4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            531      4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            532      4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            533      2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    534      2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    535      2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    536      3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    537      3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    538      3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    539      4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    540      4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    541      4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    542      2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     543      2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     544      2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     545      3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     546      3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     547      3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     548      4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     549      4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     550      4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     551      2-O-(2'-NCC.sub.6 H.sub.4)                                            552      2-O-(3'-NCC.sub.6 H.sub.4)                                            553      2-O-(4'-NCC.sub.6 H.sub.4)                                            554      3-O-(2'-NCC.sub.6 H.sub.4)                                            555      3-O-(3'-NCC.sub.6 H.sub.4)                                            556      3-O-(4'-NCC.sub.6 H.sub.4)                                            557      4-O-(2'-NCC.sub.6 H.sub.4)                                            558      4-O-(3'-NCC.sub.6 H.sub.4)                                            559      4-O-(4'-NCC.sub.6 H.sub.4)                                            560      2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     561      2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     562      2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     563      3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     564      3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     565      3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     566      4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                     567      4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                     568      4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                     569      2-Pyridinyl-2'                                                        570      2-Pyridinyl-3'                                                        571      2-Pyridinyl-4'                                                        572      3-Pyridinyl-2'                                                        573      3-Pyridinyl-3'                                                        574      3-Pyridinyl-4'                                                        575      4-Pyridinyl-2'                                                        576      4-Pyridinyl-3'                                                        577      4-Pyridinyl-4'                                                        578      2-Pyrimidinyl-2'                                                      579      2-Pyrimidinyl-3'                                                      580      2-Pyrimidinyl-4'                                                      581      3-Pyrimidinyl-2'                                                      582      3-Pyrimidinyl-3'                                                      583      3-Pyrimidinyl-4'                                                      584      4-Pyrimidinyl-2'                                                      585      4-Pyrimidinyl-3'                                                      586      4-Pyrimidinyl-4'                                                      587      2-Pyrazolyl-1'                                                        588      2-Pyrazolyl-3'                                                        589      2-Pyrazolyl-4'                                                        590      3-Pyrazolyl-1'                                                        591      3-Pyrazolyl-3'                                                        592      3-Pyrazolyl-4'                                                        593      4-Pyrazolyl-1'                                                        594      4-Pyrazolyl-3'                                                        595      4-Pyrazolyl-4'                                                        596      2-Isoxazolyl-3'                                                       597      2-Isoxazolyl-4'                                                       598      2-Isoxazolyl-5'                                                       599      3-Isoxazolyl-3'                                                       600      3-Isoxazolyl-4'                                                       601      3-Isoxazolyl-5'                                                       602      4-Isoxazolyl-3'                                                       603      4-Isoxazolyl-4'                                                       604      4-Isoxazolyl-5'                                                       605      2-Isothiazolyl-3'                                                     606      2-Isothiazolyl-4'                                                     607      2-Isothiazolyl-5'                                                     608      3-Isothiazolyl-3                                                      609      3-Isothiazolyl-4'                                                     610      3-Isothiazolyl-5'                                                     611      4-Isothiazolyl-3'                                                     612      4-Isothiazolyl-4'                                                     613      4-Isothiazolyl-5'                                                     614      2-Imidazolyl-1'                                                       615      2-Imidazolyl-2'                                                       616      2-Imidazolyl-4'                                                       617      3-Imidazolyl-1'                                                       618      3-Imidazolyl-2'                                                       619      3-Imidazolyl-4'                                                       620      4-Imidazolyl-1'                                                       621      4-Imidazolyl-2'                                                       622      4-Imidazolyl-4'                                                       623      2-Oxazolyl-2'                                                         624      2-Oxazolyl-4'                                                         625      2-Oxazolyl-5'                                                         626      3-Oxazolyl-2'                                                         627      3-Oxazolyl-4'                                                         628      3-Oxazolyl-5'                                                         629      4-Oxazolyl-2'                                                         630      4-Oxazolyl-4'                                                         631      4-Oxazolyl-5'                                                         632      2-Thiazolyl-2'                                                        633      2-Thiazolyl-4'                                                        634      2-Thiazolyl-5'                                                        635      3-Thiazolyl-2'                                                        636      3-Thiazolyl-4'                                                        637      3-Thiazolyl-5'                                                        638      4-Thiazolyl-2'                                                        639      4-Thiazolyl-4                                                         640      4-Thiazolyl-5'                                                        ______________________________________                                    

                  TABLE 29                                                         ______________________________________                                          ##STR240##                                                                    I: R.sup.1 = CH.sub.3, XCH.sub.3                                               II: R.sup.1 = CH.sub.2 CH.sub.3, XCH.sub.3                                     III: R.sup.1 = CH.sub.3, XCl                                                   IV: R.sup.1 = CH.sub.2 CH.sub.3, XCl                                           No.       B                                                                    ______________________________________                                         1         Pyrrolyl-3                                                           2         NCH.sub.3 -Pyrrolyl-3                                                3         NC.sub.6 H.sub.5 -Pyrrolyl-3                                         4         N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           5         N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           6         N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           7         N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          8         N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          9         N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          10        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           11        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           12        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           13        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  14        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  15        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  16        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  17        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  18        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  19        Pyrrolyl-2                                                           20        NCH.sub.3 -Pyrrolyl-2                                                21        NC.sub.6 H.sub.5 -Pyrrolyl-2                                         22        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           23        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           24        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           25        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          26        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          27        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          28        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           29        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           30        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           31        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  32        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  33        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  34        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  35        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  36        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  37        Furyl-2                                                              38        5-CH.sub.3 -Furyl-2                                                  39        5-C.sub.6 H.sub.5 -Furyl-2                                           40        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              41        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              42        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              43        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             44        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             45        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             46        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              47        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              48        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              49        5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     50        5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     51        5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     52        5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     53        5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     54        5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     55        4-CH.sub.3 -Furyl-2                                                  56        4-C.sub.6 H.sub.5 -Furyl-2                                           57        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              58        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              59        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              60        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             61        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             62        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             63        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              64        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              65        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              66        4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     67        4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     68        4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     69        4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     70        4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     71        4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     72        Thienyl-2                                                            73        5-CH.sub.3 -Thienyl-2                                                74        5-C.sub.6 H.sub.5 -Thienyl-2                                         75        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            76        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            77        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            78        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           79        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           80        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           81        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            82        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            83        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            84        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   85        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   86        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   87        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   88        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   89        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   90        4-CH.sub.3 -Thienyl-2                                                91        4-C.sub.6 H.sub.5 -Thienyl-2                                         92        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            93        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            94        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            95        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           96        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           97        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           98        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            99        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       NCH.sub.3 -Pyrazolyl-4                                               127       NC.sub.6 H.sub.5 -Pyrazolyl-4                                        128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 143       3-CH.sub.3 N-Methylpyrazolyl-4                                       144       3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                                145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   154       3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          155       3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          156       3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          157       3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          158       3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          159       3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          160       Isoxazolyl-5                                                         161       3-CH.sub.3 -Isoxazolyl-5                                             162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 -Isoxazolyl-3                                             198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 -Isothiazolyl-5                                           216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       2-CH.sub.3 -Oxazolyl-4                                               234       2-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           236       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           237       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           238       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          239       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          241       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           242       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           243       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           244       2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  245       2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  246       2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  247       2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  248       2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  249       2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       NCH.sub.3 -1,2,4-Triazolyl-5                                         269       3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                              270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          280       3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 281       3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 282       3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 283       3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 284       3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 285       3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        384       Pyridinyl-3                                                          ______________________________________                                    

                                      TABLE 30                                     __________________________________________________________________________     Selected physical data of some compounds                                                                    IR (cm.sup.-) or                                  No.                                                                               Compound                  .sup.1 H-NMR (ppm)                                                                       m.p                                     __________________________________________________________________________         ##STR241##                         81                                      2                                                                                  ##STR242##                         60                                      3                                                                                  ##STR243##               3.85 (s, broad, 3H); 3.7 (s, broad, 3H)           4                                                                                  ##STR244##               3.85 (s, broad, 3H); 3.75 (s, broad, 3H)          5                                                                                  ##STR245##               3.75 (2s, broad, each 3H)                         6                                                                                  ##STR246##                         91                                      7                                                                                  ##STR247##               3.8 (s, 3H); 3.75 (s, broad, 3H)                  8                                                                                  ##STR248##               3.85 (s, 3H); 3.8 (s, broad,                      __________________________________________________________________________                                  3H)                                          

                  TABLE 31                                                         ______________________________________                                          ##STR249##                                                                    I: R.sup.1 = CH.sub.3, X = CH.sub.3                                            II: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                    III: R.sup.1 = CH.sub.3, X = Cl                                                IV: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                          No.          B                                                                 ______________________________________                                          1           2-Pyridyl                                                          2           3-Trifluoromethyl-2-Pyridyl                                        3           5-Trifluoromethyl-2-Pyridyl                                        4           3,5-Bis-(trifluoromethyl)-2-Pyridyl                                5           3,5-Dichloro-2-Pyridyl                                             6           3-Chloro-5-trifluoromethyl-2-Pyridyl                               7           3,5-Dichloro-2-Pyridyl                                             8           2-Chloro-4-trifluoromethylphenyl                                   9           2-Benzothiazolyl                                                  10           5-Chloro-1-methyl-2-benzimidazolyl                                11           2-Benzoxazolyl                                                    12           1-Methyl-5-trifluoromethylimidazo-                                              5,4-a!-Pyridin-2-yl                                              13           5-Chloro-2-Pyrimidinyl                                            14           4-Methyl-5-Phenyl-2-thiazolin-2-yl                                15           4-Methyl-5-Phenyl-2-oxazolin-2-yl                                 16           7-Trifluoromethyl-4-quinolinyl                                    ______________________________________                                    

                  TABLE 57                                                         ______________________________________                                         Selected physical data of some compounds                                        ##STR250##                                                                                                  mp   .sup.1 H-NMR (ppm)                          No.  X      T.sub.m           (°C.)                                                                        or IR (cm.sup.-1)                           ______________________________________                                         1    Cl     2-CH.sub.3             3.8 (s, broad, 6H)                          2    Cl     2,5-(CH.sub.3).sub.2   3.8 (s, broad, 6H)                          3    Cl     2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                                   4.0 (s, 3H); 3.8                                                               (s, broad, 6H)                              4    Cl     2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-                                                                3.8 (s, broad, 6H)                                      Allyl                                                              5    CH.sub.3                                                                              2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                                   4.0 (s, 3H); 3.75                                                              (s, broad, 6H)                              6    CH.sub.3                                                                              2-CH.sub.3             3.75 (s, broad,                                                                6H)                                         7    CH.sub.3                                                                              2,5-(CH.sub.3).sub.2   3.75 (s, broad,                                                                6H)                                         8    CH.sub.3                                                                              2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-                                                                3.75 (s, broad,                                         Allyl                  6H)                                         ______________________________________                                    

Example 11

2-(2'-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

a) 2-(2'-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide is stirred for 5 hours at room temperature (20° C.). The reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and suction filtered. There is obtained 73 g (0.300 mol=88%) of the title compound as a colorless solid.

Mp=83° C. ¹ H-NMR, (CDCl₃ ; δ (ppm)): 8.15 (d, 1H, I=8 Hz, aromatic); 7.95 (d, 1H, I=8 Hz, aromatic); 7.7 (t, 1H, I=8 Hz, aromatic); 7.45 (t, 1H, I=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O--CH₂); 2.35 (s, 3H, CH₃)

b) 2-(2'-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2'-methylphenoxymethyl)-nitrobenzene (Example 11a) and 10 g of 5% Pt/C (platinum adsorbed on activated carbon) in 50 ml of methanol are stirred vigorously under a hydrogen blanket for 2 hours. A further 2 g of 5% Pt/C is added and the mixture is stirred overnight. The catalyst is filtered off and replaced by 10 g of fresh catalyst. The mixture is stirred overnight and suction filtered, and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 61 g (0.286 mol=93%) of the title compound as a colorless solid.

Mp=56° C. ¹ H-NMR (CDCl₃ ; δ (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, I=8 Hz, aromatic); 6.9 (t, 1H, I=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O--CH₂); 4.05 (s, broad, 2H, NH₂); 2.2 (s, 3H, CH₃)

c) 2-(2'-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

At 10°-15° C., a solution of 6 g of 2-(2'-methylphenoxymethyl)-aniline (Example 1b) in 20 ml of CH₂ Cl₂ is added to a mixture of 6.6 g (36 mmol) of trichloroacetyl chloride and 3 g (38 mmol) of pyridine in 50 ml of CH₂ Cl₂. The mixture is stirred for 1 hour at room temperature, and then extracted with water, dried over MgSO₄ and evaporated down. The residue is suction filtered over silica gel and the filtrate which is obtained is evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 7.9 g (22 mmol=78%) of the title compound as a crystalline solid (mp=128° C.).

¹ H-NMR (CDCl₃ ; δ (ppm)): 9.6 (s, broad, 1H, NH); 8.1 (d, 1H, I=8 Hz, phenyl); 7.5 (t, broad, 1H, phenyl); 7.4 (d, broad, 1H, phenyl); 7.2 (m, 3H, phenyl); 6.95 (m, 2H, phenyl); 5.1 (s, 2H, OCH₂); 2.2 (s, 3H, CH₃)

Example 12

N-Methyl-N'-(2-(2'-methylphenoxymethyl)-phenyl)-urea (Table 7, No. 2)

In a laboratory autoclave, about 10 ml of methylamine is added to 2 g (5.5 mmol) of the trichloroacetanilide from Example 1c. The autoclave is then closed and the reaction mixture is heated for about 6 hours at 80° C. The reaction mixture is cooled and the autoclave opened. The methylamine is allowed to evaporate off and the solid residue is stirred with methyl tert-butyl ether. The insoluble solid is filtered off and dried under reduced pressure. There is obtained 1.4 g (5.2 mmol=94%) of the title compound as a crystalline solid (mp=144° C.).

¹ H-NMR (DMSO-d₆ ; δ (ppm)): 8.05 (s, 1H, NH); 7.8 (d, 1H, I=8 Hz, phenyl); 7.4 (d, 1H, I=8 Hz, phenyl); 6.8-7.3 (m, 6H, phenyl); 6.7 (s, 1H, NH); 5.1 (s, 2H, OCH₂); 2.65 (d, 3H, I=5 Hz, N--CH₃); 2.2 (s, 3H, CH₃)

Example 13

2-(2'-Methylphenoxymethyl)-propionyl anilide (Table 38, No. 3)

A mixture of 3 g (14.1 mmol) of the aniline from Example 11b, 1.35 g (17 mmol) of pyridine and 1.4 g (15.5 mmol) of propionyl chloride in 30 ml of methylene chloride is stirred for 1 hour at room temperature. The reaction mixture is then extracted with diluted hydrochloric acid and water, dried over MgSO₄ and evaporated down. There is obtained 3.8 g (quantitative yield) of the title compound.

¹ H-NMR (COCl₃ ; δ (ppm)): 8.25 (s, broad, 1H, NH); 8.15 (d, 1H, I=8 Hz, phenyl); 6.9-7.5 (m, 7H, phenyl); 5.1 (s, 2H, OCH₂); 2.35 (q, 2H, I=8 Hz, CH₂); 2.25 (s, 3H, CH₃); 1.2 (t, 3H, I=8 Hz, CH₃)

Example 14

N-Propionyl-2-(2'-methylphenoxymethyl)-propionyl anilide (Table 38, No. 4)

0.41 g (17.1 mmol) of sodium hydride is added in portions to 3.8 g (14 mmol) of the propionyl anilide from Example 13 in 40 ml of dimethylformamide. Upon completion of gas evolution 1.4 g (15.9 mmol) of propionyl chloride is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2.6 g (8 mmol=57%) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃): δ (ppm): 7.6 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.15 (m, 3H, phenyl); 6.85 (m, 2H, phenyl); 4.85 (m, 2H, OCH₂); 2.6 (m, 4H, 2×CH₂); 2.2 (s, 3H, CH₃); 1.1 (t, 6H, I=8 Hz, 2×CH₃)

Example 15

N-Methyl-2-(2'-methylphenoxymethyl)-propionyl anilide (Table 38, No. 5)

0.45 g (19 mmol) of sodium hydride is added in portions to 4.0 g (14.8 mmol) of the propionyl anilide from Example 13 in 50 ml of dimethylformamide. Upon completion of gas evolution 3.0 g (21 mmol) of methyl iodide is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 3.7 g (11.7 mmol=90%) of the title compound as a colorless solid (mp=80° C.).

¹ H-NMR (CDCl₃ ; δ (ppm): 5 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH₂); 3.2 (s, 3H, N--CH₃); 2.2 (s, 3H, CH₃); 2.0 (m, 2H, CH₂); 1.0 (t, 3H, I=8 Hz, CH₃)

Example 19

N-Methyl-2-(2'-methylphenoxymethyl)-acetanilide

a) N-Methyl-2-(2'-methylphenoxymethyl)-aniline

A mixture of 5 g (23 mmol) of 2-(2'-methylphenoxymethyl)-aniline (Example 1b), 5 g (36 mmol) of K₂ CO₃ and 3.4 g (24 mmol) of methyl iodide in 50 ml of dimethylformamide is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified chromatographically using mixtures of hexane and methylene chloride. There is obtained 3.0 g (70% purity, about 40% yield) of the title compound as a yellow oil.

¹ H-NMR (CDCl₃ ; δ in ppm): 6.6-7.4 (m, 8H, phenyl); 5.0 (s, 2H, OCH₂); 4.6 (s, broad, 1H, NH); 2.9 (d, 3H, N--CH₃); 2.2 (s, 3H, CH₃).

b) N-Methyl-2-(2'-methylphenoxymethyl)-acetanilide (Table 7, No. 9)

3 g (approx. 9.3 mmol) of N-methyl-2-(2'-methylphenoxymethyl)-aniline (from Example 5a) is added to a mixture of 1.6 g (16 mmol) of acetoanhydride and 1.3 g (16 mmol) of pyridine in 20 ml of methylene chloride. The mixture is stirred for 1 hour at room temperature and is then extracted with dilute hydrochloric acid and water. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2 g (80%) of the title compound as a colorless solid (mp=76° C.).

¹ H-NMR (CDCl₃ ; δ in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH₂); 3.25 (s, 3H, CH₃); 2.25 (s, 3H, CH₃); 1.8 (s, 3H, CH₃).

The compounds listed in the tables below may be prepared correspondingly.

Compound I from Table 32, No. 1 has for example the following structural formula: ##STR251##

The compounds described in the following tables may be prepared analogously.

                  TABLE 32                                                         ______________________________________                                          ##STR252##                                                                    I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                            II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                    III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5                                       V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5                                    VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5                          VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                          VIII: R.sup.1 = H, Z = NH(CH.sub.3)                                            IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                                       X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)                                 XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)                                          XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)                                     XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)                           XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)                             No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   181     3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   182     4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4 -COCH.sub.2 CH.sub.2 CH.sub.3                                        298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-COCH.sub.3                                                      303     2-Me-4-CH.sub.3 CH.sub.2 CO                                            304     2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3                                    305     2-Me-4-COCH(CH.sub.3).sub.2                                            306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-COCH.sub.3                                             308     2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3                                    309     2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3                           310     2,5-Me.sub.2 -4-COCH(CH.sub.3).sub.2                                   311     2-Cl-4-CHO                                                             312     2-Cl-4-COCH.sub.3                                                      313     2-Cl-4-COCH.sub.2 CH.sub.3                                             314     2-Cl-4-COCH(CH.sub.3).sub.2                                            315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-COCH.sub.3                                             317     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3                                    318     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3                           319     2,5-Cl.sub.2 -4-COCH(CH.sub.3).sub.2                                   320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2 -CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                  351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                  369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)                       381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-C-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CN-OCH.sub.2 CH.sub.2 OCH.sub.3)               642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 33                                                         ______________________________________                                          ##STR253##                                                                    I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                            II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                    III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5                                       V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5                                    VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5                          VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                          VIII: R.sup.1 = H, Z = NH(CH.sub.3)                                            IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                                       X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)                                 XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)                                          XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)                                     XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)                           XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)                             No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C6H5, 4-CH.sub.3                                            141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   181     3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   182     4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-COCH.sub.3                                                      303     2-Me-4-COCH.sub.2 CH.sub.3                                             304     2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3                                    305     2-Me-4-COCH(CH.sub.3).sub.2                                            306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-COCH.sub.3                                             308     2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3                                    309     2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3                           310     2,5-Me.sub.2 -4-COCH(CH.sub.3).sub.2                                   311     2-Cl-4-CHO                                                             312     2-Cl-4-COCH.sub.3                                                      313     2-Cl-4-COCH.sub.2 CH.sub.3                                             314     2-Cl-4-COCH(CH.sub.3).sub.2                                            315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-COCH.sub.3                                             317     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3                                    318     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3                           319     2,5-Cl.sub.2 -4-COCH(CH.sub.3).sub.2                                   320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)CH.sub.3                                              339     3-C(NO-Propargyl)CH.sub.3                                              340     4-C(NO-Propargyl)CH.sub.3                                              341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                   369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                        381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'CH.sub.3 C.sub.6 H.sub.4)                                         406     2-(3'CH.sub.3 C.sub.6 H.sub.4)                                         407     2-(4'CH.sub.3 C.sub.6 H.sub.4)                                         408     3-(2'CH.sub.3 C.sub.6 H.sub.4)                                         409     3-(3'CH.sub.3 C.sub.6 H.sub.4)                                         410     3-(4'CH.sub.3 C.sub.6 H.sub.4)                                         411     4-(2'CH.sub.3 C.sub.6 H.sub.4)                                         412     4-(3'CH.sub.3 C.sub.6 H.sub.4)                                         413     4-(4'CH.sub.3 C.sub.6 H.sub.4)                                         414     2-(2'CH.sub.3 COC.sub.6 H.sub.4)                                       415     2-(3'CH.sub.3 COC.sub.6 H.sub.4)                                       416     2-(4'CH.sub.3 COC.sub.6 H.sub.4)                                       417     3-(2'CH.sub.3 COC.sub.6 H.sub.4)                                       418     3-(3'CH.sub.3 COC.sub.6 H.sub.4)                                       419     3-(4'CH.sub.3 COC.sub.6 H.sub.4)                                       420     4-(2'CH.sub.3 COC.sub.6 H.sub.4)                                       421     4-(3'CH.sub.3 COC.sub.6 H.sub.4)                                       422     4-(4'CH.sub.3 COC.sub.6 H.sub.4)                                       423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                433     2-(3'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                434     2-(4'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                435     3-(2'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                436     3-(3'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                437     3-(4'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                438     4-(2'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                439     4-(3'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                440     4-(4'CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                                441     2-(2'CH.sub.3 OC.sub.6 H.sub.4)                                        442     2-(3'CH.sub.3 OC.sub.6 H.sub.4)                                        443     2-(4'CH.sub.3 OC.sub.6 H.sub.4)                                        444     3-(2'CH.sub.3 OC.sub.6 H.sub.4)                                        445     3-(3'CH.sub.3 OC.sub.6 H.sub.4)                                        446     3-(4'CH.sub.3 OC.sub.6 H.sub.4)                                        447     4-(2'CH.sub.3 OC.sub.6 H.sub.4)                                        448     4-(3'CH.sub.3 OC.sub.6 H.sub.4)                                        449     4-(4'CH.sub.3 OC.sub.6 H.sub.4)                                        450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyll))-C.sub.6 H.sub.4)                        518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chlorallyl)                 650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chlorallyl)                 659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 34                                                         ______________________________________                                          ##STR254##                                                                    I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                            II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                    III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5                                       V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5                                    VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5                          VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                          VIII: R.sup.1 = H, Z, = NH(CH.sub.3)                                           IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                                       X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)                                 XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)                                          XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)                                     XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = CH.sub.3)                              XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)                             No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.3                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   181     3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   182     4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-COCH.sub.3                                                      303     2-Me-4-COCH.sub.2 CH.sub.3                                             304     2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3                                    305     2-Me-4-COCH(CH.sub.3).sub.2                                            306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-COCH.sub.3                                             308     2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3                                    309     2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3                           310     2, 5-Me.sub.2 -4-COCH(CH.sub.3)2                                       311     2-Cl-4-CHO                                                             312     2-Cl-4-COCH.sub.3                                                      313     2-Cl-4-COCH.sub.2 CH.sub.3                                             314     2-Cl-4-COCH(CH.sub.3)2                                                 315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-COCH.sub.3                                             317     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3                                    318     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3                           319     2,5-Cl.sub.2 -4-COCH(CH.sub.3)2                                        320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NCC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)CH.sub.3                                              339     3-C(NO-Propargyl)CH.sub.3                                              340     4-C(NO-Propargyl)CH.sub.3                                              341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                  369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.4)            374     2,5-(CH.sub.3).sub.2-4-(CH.sub.3 CNOCH.sub.3)                          375     2,5-(CH.sub.3).sub.2-4-(CH.sub.3 CNOC.sub.2 H.sub.5)                   376     2,5-(CH.sub.3).sub.2-4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                        381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 35                                                         ______________________________________                                          ##STR255##                                                                    I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                            II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                    III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5                                       V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5                                    VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5                          VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                          VIII: R.sup.1 = H, Z = NH(CH.sub.3)                                            IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                                       X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)                                 XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)                                          XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)                                     XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)                           XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)                             No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-Cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    181     3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    182     4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-COCH.sub.2 CH.sub.3                                             304     2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3                                    305     2-Me-4-COCH(CH.sub.3).sub.2                                            306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-COCH.sub.3                                             308     2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3                                    309     2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3                           310     2,5-Me.sub.2 -4-COCH(CH.sub.3).sub.2                                   311     2-Cl-4-CHO                                                             312     2-Cl-4-COCH.sub.3                                                      313     2-Cl-4-COCH.sub.2 CH.sub.3                                             314     2-Cl-4-COCH(CH.sub.3).sub.2                                            315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-COCH.sub.3                                             317     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3                                    318     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3                           319     2,5-Cl.sub.2 -4-COCH(CH.sub.3).sub.2                                   320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                   369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2;5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)                       381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 36                                                         ______________________________________                                          ##STR256##                                                                    I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                            II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                    III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5                                       V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5                                    VI: R.sup.1 = CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5                          VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                          VIII: R.sup.1 = H, Z = NH(CH.sub.3)                                            IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                                       X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)                                 XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)                                          XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)                                     XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)                           XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)                             No.     X.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    181     3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    182     4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-COCH.sub.2 CH.sub.3                                             304     2-Me-4-COCH.sub.2 CH.sub.2 CH.sub.3                                    305     2-Me-4-COCH(CH.sub.3).sub.2                                            306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-COCH.sub.3                                             308     2,5-Me.sub.2 -4-COCH.sub.2 CH.sub.3                                    309     2,5-Me.sub.2 -4-CH.sub.2 CH.sub.2 COCH.sub.3                           310     2,5-Me.sub.2 -4-COCH(CH.sub.3).sub.2                                   311     2-Cl-4-CHO                                                             312     2-Cl-4-COCH.sub.3                                                      313     2-Cl-4-COCH.sub.2 CH.sub.3                                             314     2-Cl-4-COCH(CH.sub.3).sub.2                                            315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-COCH.sub.3                                             317     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.3                                    318     2,5-Cl.sub.2 -4-COCH.sub.2 CH.sub.2 CH.sub.3                           319     2,5-Cl.sub.2 -4-COCH(CH.sub.3).sub.2                                   320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                  369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)                       381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FFC.sub.6 H.sub.4)                                             484     4-O-(2'-Fab,4 C.sub.6 H.sub.4)                                         485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         ______________________________________                                    

                  TABLE 37                                                         ______________________________________                                          ##STR257##                                                                    I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                            II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                    III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5                                       V: R.sup.1 Propargyl, Z = C.sub.2 H.sub.5                                      VI: R.sup.1 CH.sub.2 OCH.sub.3, Z = C.sub.2 H.sub.5                            VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                          VIII: R.sup.1 = H, Z = NH(CH.sub.3)                                            IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                                       X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)                                 XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)                                          XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)                                     XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)                           XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)                             No.      B                                                                     ______________________________________                                         1        Pyrrolyl-3                                                            2        NCH.sub.3 -Pyrrolyl-3                                                 3        NC.sub.6 H.sub.5 -Pyrrolyl-3                                          4        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            5        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            6        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            7        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           8        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           9        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           10       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            11       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            12       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            13       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   14       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   15       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   16       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   17       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   18       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   19       Pyrrolyl-2                                                            20       NCH.sub.3 -Pyrrolyl-2                                                 21       NC.sub.6 H.sub.5 -Pyrrolyl-2                                          22       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            23       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            24       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            25       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           26       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           27       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           28       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            29       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            30       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            31       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   32       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   33       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   34       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   35       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   36       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   37       Furyl-2                                                               38       5-CH.sub.3 -Furyl-2                                                   39       5-C.sub.6 H.sub.5 -Furyl-2                                            40       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               41       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               42       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               43       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              44       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              45       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              46       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               47       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               48       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               49       5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      50       5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      51       5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      52       5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      53       5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      54       5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      55       4-CH.sub.3 -Furyl-2                                                   56       4-C.sub.6 H.sub.5 -Furyl-2                                            57       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               58       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               59       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               60       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              61       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              62       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              63       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               64       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               65       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               66       4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      67       4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      68       4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      69       4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      70       4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      71       4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      72       Thienyl-2                                                             73       5-CH.sub.3 -Thienyl-2                                                 74       5-C.sub.6 H.sub.5 -Thienyl-2                                          75       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             76       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             77       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             78       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            79       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            80       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            81       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             82       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             83       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             84       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    85       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    86       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    87       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    88       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    89       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    90       4-CH.sub.3 -Thienyl-2                                                 91       4-C.sub.6 H.sub.5 -Thienyl-2                                          92       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             93       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             94       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             95       4-(4'-CH.sub.3 O-C.sub.6 H.sub.4)-Thienyl-2                           96       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            97       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            98       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             99       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             100      4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             101      4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    102      4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    103      4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    104      4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    105      4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    106      4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    107      Thienyl-3                                                             108      5-CH.sub.3 -Thienyl-3                                                 109      5-C.sub.6 H.sub.5 -Thienyl-3                                          110      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                             111      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                             112      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                             113      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                            114      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                            115      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                            116      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                             117      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                             118      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                             119      5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                    120      5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                    121      5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                    122      5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                    123      5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                    124      5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                    125      Pyrazolyl-4                                                           126      NCH.sub.3 -Pyrazolyl-4                                                127      NC.sub.6 H.sub.5 -Pyrazolyl-4                                         128      N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                           129      N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                           130      N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                           131      N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                          132      N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                          133      N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                          134      N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                           135      N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                           136      N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                           137      N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                  138      N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                  139      N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                  140      N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                  141      N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                  142      N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                  143      3-CH.sub.3 N-Methylpyrazolyl-4                                        144      3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                                 145      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   146      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   147      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   148      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  149      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  150      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                  151      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   152      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   153      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-N-Methylpyrazolyl-4                   154      3-(4'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          155      3-(3'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          156      3-(2'-CNC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          157      3-(4'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          158      3-(3'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          159      3-(2'-ClC.sub.6 H.sub.4)-N-Methylpyrazolyl-4                          160      Isoxazolyl-5                                                          161      3-CH.sub.3 -Isoxazolyl-5                                              162      3-C.sub.6 H.sub.5 -Isoxazolyl-5                                       163      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                          164      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                          165      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                          166      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                         167      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                         168      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                         169      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                          170      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                          171      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                          172      3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                 173      3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                 174      3-(2'-CNC.sub.6 H.sub.4) Isoxazolyl-5                                 175      3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                 176      3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                 177      3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                 178      4-Chloroisoxazolyl-5                                                  179      3-CH.sub.3 -4-Chloroisoxazolyl-5                                      180      3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                               181      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  182      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  183      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  184      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 185      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 186      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 187      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  188      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  189      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                  190      3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         191      3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         192      3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         193      3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         194      3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         195      3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                         196      Isoxazolyl-3                                                          197      5-CH.sub.3 -Isoxazolyl-3                                              198      5-C.sub.6 H.sub.5 -Isoxazolyl-3                                       199      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                          200      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                          201      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                          202      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                         203      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                         204      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                         205      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                          206      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                          207      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                          208      5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                 209      5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                 210      5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                 211      5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                 212      5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                 213      5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                 214      Isothiazolyl-5                                                        215      3-CH.sub.3 -Isothiazolyl-5                                            216      3-C.sub.6 H.sub.5 -Isothiazolyl-5                                     217      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                        218      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                        219      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                        220      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                       221      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Is6thiazolyl-5                       222      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                       223      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                        224      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                        225      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                        226      3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                               227      3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                               228      3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                               229      3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                               230      3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                               231      3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                               232      Oxazolyl-4                                                            233      3-CH.sub.3 -Oxazolyl-4                                                234      3-C.sub.6 H.sub.5 -Oxazolyl-4                                         235      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                            236      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                            237      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                            238      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                           239      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                           240      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                           241      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                            242      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                            243      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                            244      3-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                   245      3-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                   246      3-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                   247      3-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                   248      3-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                   249      3-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                   250      Thiazolyl-4                                                           251      2-CH.sub.3 -Thiazolyl-4                                               252      2-C.sub.6 H.sub.5 -Thiazolyl-4                                        253      2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                           254      2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                           255      2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                           256      2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                          267      2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                          258      2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                          259      2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                           260      2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                           261      2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                           262      2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                  263      2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                  264      2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                  265      2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                  266      2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                  267      2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                  268      NCH.sub.3 -1,2,4-Triazolyl-5                                          269      3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                               270      3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                        271      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          272      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          273      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          274      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         275      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         276      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5         277      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          278      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          279      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5          280      3-(4'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 281      3-(3'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 282      3-(2'-CNC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 283      3-(4'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 284      3-(3'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 285      3-(2'-ClC.sub.6 H.sub.4)-NCH.sub.3 -1,2,4-Triazolyl-5                 286      1,3,4-Oxadiazolyl-2                                                   287      5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                       288      5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                289      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   290      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   291      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   292      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  293      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  294      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  295      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   296      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   297      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   298      5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          299      5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          300      5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          301      5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          302      5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          303      5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                          304      1,2,4-Oxadiazolyl-3                                                   305      5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                       306      5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                307      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   308      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   309      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   310      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  311      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  312      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  313      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   314      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   315      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   316      5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          317      5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          318      5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          319      5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          320      5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          321      5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                          322      1,2,4-Oxadiazolyl-5                                                   323      3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                       324      3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                325      3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   326      3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   327      3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   328      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  329      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  330      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  331      3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   332      3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   333      3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   334      3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          335      3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          336      3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          337      3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          338      3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          339      3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                          340      1,2,4-Thiadiazolyl-3                                                  341      5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                      342      5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                               343      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  344      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  345      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  346      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 347      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 348      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 349      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  350      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  351      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  352      5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         353      5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         354      5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         355      5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         356      5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         357      5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                         358      1,3,4-Thiadiazolyl-2                                                  359      5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                      360      5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                               361      5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  362      5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  363      5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  364      5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 365      5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 366      5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 367      5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  368      5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  369      5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  370      5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         371      5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         372      5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         373      5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         374      5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         375      5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                         376      Pyridinyl-2                                                           377      Pyridinyl-4                                                           378      Pyridazinyl-3                                                         379      Pyridazinyl-4                                                         380      Pyridazinyl-2                                                         381      Pyrimidinyl-4                                                         382      Pyrimidinyl-5                                                         383      Pyrimidinyl-2                                                         ______________________________________                                    

                  TABLE 38                                                         ______________________________________                                         Selected physical data of some compounds                                                                    IR (cm.sup.-1)                                                                 or                                                                             .sup.1 H-NMR                                                                            mp                                       No.  Compound                (ppm)    (°C.)                             ______________________________________                                               ##STR258##                      128                                      2                                                                                    ##STR259##                      144                                      3                                                                                    ##STR260##                                                               4                                                                                    ##STR261##                                                               5                                                                                    ##STR262##                      80                                       6                                                                                    ##STR263##                      75                                       7                                                                                    ##STR264##                      188                                      8                                                                                    ##STR265##                      115                                      9                                                                                    ##STR266##                      76                                       10                                                                                   ##STR267##                      96                                       11                                                                                   ##STR268##             3.3 (s, 3H); 2.25 (s, 3H)                         ______________________________________                                    

                                      TABLE 58                                     __________________________________________________________________________     Selected physical data of some compounds                                        ##STR269##                                                                                                IR (cm.sup.-1)                                                                 or .sup.1 H-NMR                                                                      mp                                           No.                                                                               X.sub.m          R.sup.1 (ppm) (°C.)                                 __________________________________________________________________________     1  2-CH.sub.3       H             120                                          2  2-CH.sub.3       CH.sub.3      oil                                          3  2-CH.sub.3       C.sub.2 H.sub.5                                                                              oil                                          4  2-CH.sub.3       Allyl         oil                                          5  2-CH.sub.3       Propargyl     oil                                          6  2-CH.sub.3       CH.sub.2 OCH.sub.3                                                                           oil                                          7  2,5-(CH.sub.3).sub.2                                                                            H             170                                          8  2,5-(CH.sub.3).sub.2                                                                            CH.sub.3      oil                                          9  2,5-(CH.sub.3).sub.2                                                                            C.sub.2 H.sub.5                                                                              oil                                          10 2,5-(CH.sub.3).sub.2                                                                            Allyl         oil                                          11 2,5-(CH.sub.3).sub.2                                                                            Propargyl     oil                                          12 2,5-(CH.sub.3).sub.2                                                                            CH.sub.2 OCH.sub.3                                                                           oil                                          13 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                             H             125                                          14 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                             CH.sub.3      oil                                          15 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                             C.sub.2 H.sub.5                                                                              oil                                          16 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                             Allyl          87                                          17 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                             Propargyl     oil                                          18 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                             CH.sub.2 OCH.sub.3                                                                           oil                                          19 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl                                                     H              85                                          20 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl                                                     CH.sub.3      oil                                          21 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl                                                     C.sub.2 H.sub.5                                                                              oil                                          22 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl                                                     Allyl          87                                          23 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl                                                     Propargyl     oil                                          24 2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NO-Allyl                                                     CH.sub.2 OCH.sub.3                                                                           oil                                          __________________________________________________________________________

                  TABLE 59                                                         ______________________________________                                         Selected physical data of some compounds                                        ##STR270##                                                                                                 IR (cm.sup.-1)                                                                 or .sup.1 H-NMR                                                                        mp                                        No.     X.sub.m  R.sup.1     (ppm)   (°C.)                              ______________________________________                                         1       4-CH.sub.3                                                                              H                   118                                       2       4-CH.sub.3                                                                              CH.sub.3            oil                                       3       4-CH.sub.3                                                                              C.sub.2 H.sub.5     oil                                       4       4-CH.sub.3                                                                              Allyl               oil                                       5       4-CH.sub.3                                                                              Propargyl           oil                                       6       4-CH.sub.3                                                                              CH.sub.2 OCH.sub.3  oil                                       7       3,5-Cl.sub.2                                                                            H                   160                                       8       3,5-Cl.sub.2                                                                            CH.sub.3            oil                                       9       3,5-Cl.sub.2                                                                            C.sub.2 H.sub.5     oil                                       10      3,5-Cl.sub.2                                                                            Allyl                85                                       11      3,5-Cl.sub.2                                                                            Propargyl           oil                                       12      3,5-Cl.sub.2                                                                            CH.sub.2 OCH.sub.3  oil                                       ______________________________________                                    

                  TABLE 39                                                         ______________________________________                                          ##STR271##                                                                    No.   X      R.sup.1   Z      A                                                ______________________________________                                         1     H      H         CH.sub.3                                                                              CH.sub.2 O                                       2     H      H         CH.sub.3                                                                              CH.sub.2 ONC (CH.sub.3)                          3     H      H         CH.sub.3                                                                              CHCH                                             4     H      H         NH.sub.2                                                                              CH.sub.2 O                                       5     H      H         NH.sub.2                                                                              CH.sub.2 ONC(CH.sub.3)                           6     H      H         NH.sub.2                                                                              CHCH                                             7     H      H         N(CH.sub.3).sub.2                                                                     CH.sub.2 O                                       8     H      H         N(CH.sub.3).sub.2                                                                     CH.sub.2 ONC(CH.sub.3)                           9     H      H         N(CH.sub.3).sub.2                                                                     CHCH                                             10    H      H         CCl.sub.3                                                                             CH.sub.2 O                                       11    H      H         CCl.sub.3                                                                             CH.sub.2 ONC(CH.sub.3)                           12    H      H         CCl.sub.3                                                                             CHCH                                             13    H      H         CF.sub.3                                                                              CH.sub.2 O                                       14    H      H         CF.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           15    H      H         CF.sub.3                                                                              CHCH                                             16    H      Propargyl CH.sub.3                                                                              CH.sub.2 O                                       17    H      Propargyl CH.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           18    H      Propargyl CH.sub.3                                                                              CHCH                                             19    H      Propargyl NH.sub.2                                                                              CH.sub.2 O                                       20    H      Propargyl NH.sub.2                                                                              CH.sub.2 ONC(CH.sub.3)                           21    H      Propargyl NH.sub.2                                                                              CHCH                                             22    H      Propargyl N(CH.sub.3).sub.2                                                                     CH.sub.2 O                                       23    H      Propargyl N(CH.sub.3).sub.2                                                                     CH.sub.2 ONC(CH.sub.3)                           24    H      Propargyl N(CH.sub.3).sub.2                                                                     CHCH                                             25    H      Propargyl CCl.sub.3                                                                             CH.sub.2 O                                       26    H      Propargyl CCl.sub.3                                                                             CH.sub.2 ONC(CH.sub.3)                           27    H      Propargyl CCl.sub.3                                                                             CHCH                                             28    H      Propargyl CF.sub.3                                                                              CH.sub.2 O                                       29    H      Propargyl CF.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           30    H      Propargyl CF.sub.3                                                                              CHCH                                             31    CH.sub.3                                                                              H         CH.sub.3                                                                              CH.sub.2 O                                       32    CH.sub.3                                                                              H         CH.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           33    CH.sub.3                                                                              H         CH.sub.3                                                                              CHCH                                             34    CH.sub.3                                                                              H         NH.sub.2                                                                              CH.sub.2 O                                       35    CH.sub.3                                                                              H         NH.sub.2                                                                              CH.sub.2 ONC(CH.sub.3)                           36    CH.sub.3                                                                              H         NH.sub.2                                                                              CHCH                                             37    CH.sub.3                                                                              H         N(CH.sub.3).sub.2                                                                     CH.sub.2 O                                       38    CH.sub.3                                                                              H         N(CH.sub.3).sub.2                                                                     CH.sub.2 ONC(CH.sub.3)                           39    CH.sub.3                                                                              H         N(CH.sub.3).sub.2                                                                     CHCH                                             40    CH.sub.3                                                                              H         CCl.sub.3                                                                             CH.sub.2 O                                       41    CH.sub.3                                                                              H         CCl.sub.3                                                                             CH.sub.2 ONC(CH.sub.3)                           42    CH.sub.3                                                                              H         CCl.sub.3                                                                             CHCH                                             43    CH.sub.3                                                                              H         CF.sub.3                                                                              CH.sub.2 O                                       44    CH.sub.3                                                                              H         CF.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           45    CH.sub.3                                                                              H         CF.sub.3                                                                              CHCH                                             46    CH.sub.3                                                                              Propargyl CH.sub.3                                                                              CH.sub.2 O                                       47    CH.sub.3                                                                              Propargyl CH.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           48    CH.sub.3                                                                              Propargyl CH.sub.3                                                                              CHCH                                             49    CH.sub.3                                                                              Propargyl NH.sub.2                                                                              CH.sub.2 O                                       50    CH.sub.3                                                                              Propargyl NH.sub.2                                                                              CH.sub.2 ONC(CH.sub.3)                           51    CH.sub.3                                                                              Propargyl NH.sub.2                                                                              CHCH                                             52    CH.sub.3                                                                              Propargyl N(CH.sub.3).sub.2                                                                     CH.sub.2 O                                       53    CH.sub.3                                                                              Propargyl N(CH.sub.3).sub.2                                                                     CH.sub.2 ONC(CH.sub.3)                           54    CH.sub.3                                                                              Propargyl N(CH.sub.3).sub.2                                                                     CHCH                                             55    CH.sub.3                                                                              Propargyl CCl.sub.3                                                                             CH.sub.2 O                                       56    CH.sub.3                                                                              Propargyl CCl.sub.3                                                                             CH.sub.2 ONC(CH.sub.3)                           57    CH.sub.3                                                                              Propargyl CCl.sub.3                                                                             CHCH                                             58    CH.sub.3                                                                              Propargyl CF.sub.3                                                                              CH.sub.2 O                                       59    CH.sub.3                                                                              Propargyl CF.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           60    CH.sub.3                                                                              Propargyl CF.sub.3                                                                              CHCH                                             61    Cl     H         CH.sub.3                                                                              CH.sub.2 O                                       62    Cl     H         CH.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           63    Cl     H         CH.sub.3                                                                              CHCH                                             64    Cl     H         NH.sub.2                                                                              CH.sub.2 O                                       65    Cl     H         NH.sub.2                                                                              CH.sub.2 ONC(CH.sub.3)                           66    Cl     H         NH.sub.2                                                                              CHCH                                             67    Cl     H         N(CH.sub.3).sub.2                                                                     CH.sub.2 O                                       68    Cl     H         N(CH.sub.3).sub.2                                                                     CH.sub.2 ONC(CH.sub.3)                           69    Cl     H         N(CH.sub.3).sub.2                                                                     CHCH                                             70    Cl     H         CCl.sub.3                                                                             CH.sub.2 O                                       71    Cl     H         CCl.sub.3                                                                             CH.sub.2 ONC(CH.sub.3)                           72    Cl     H         CCl.sub.3                                                                             CHCH                                             73    Cl     H         CF.sub.3                                                                              CH.sub.2 O                                       74    Cl     H         CF.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           75    Cl     H         CF.sub.3                                                                              CHCH                                             76    Cl     Propargyl CH.sub.3                                                                              CH.sub.2 O                                       77    Cl     Propargyl CH.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           78    Cl     Propargyl CH.sub.3                                                                              CHCH                                             79    Cl     Propargyl NH.sub.2                                                                              CH.sub.2 O                                       80    CI     Propargyl NH.sub.2                                                                              CH.sub.2 ONC(CH.sub.3)                           81    Cl     Propargyl NH.sub.2                                                                              CHCH                                             82    Cl     Propargyl N(CH.sub.3).sub.2                                                                     CH.sub.2 O                                       83    Cl     Propargyl N(CH.sub.3).sub.2                                                                     CH.sub.2 ONC(CH.sub.3)                           84    Cl     Propargyl N(CH.sub.3).sub.2                                                                     CHCH                                             85    Cl     Propargyl CCl.sub.3                                                                             CH.sub.2 O                                       86    Cl     Propargyl CCl.sub.3                                                                             CH.sub.2 ONC(CH.sub.3)                           87    Cl     Propargyl CCl.sub.3                                                                             CHCH                                             88    Cl     Propargyl CF.sub.3                                                                              CH.sub.2 O                                       89    Cl     Propargyl CF.sub.3                                                                              CH.sub.2 ONC(CH.sub.3)                           90    Cl     Propargyl CF.sub.3                                                                              CHCH                                             ______________________________________                                    

                  TABLE 40                                                         ______________________________________                                          ##STR272##                                                                    I: R.sup.1 = H, Z = C.sub.2 H.sub.5                                            II: R.sup.1 = CH.sub.3, Z = C.sub.2 H.sub.5                                    III: R.sup.1 = C.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                            IV: R.sup.1 = Allyl, Z = C.sub.2 H.sub.5                                       V: R.sup.1 = Propargyl, Z = C.sub.2 H.sub.5                                    VI: R.sup.1 = CH.sub.2OCH.sub.3, Z = C.sub.2 H.sub.5                           VII: R.sup.1 = COC.sub.2 H.sub.5, Z = C.sub.2 H.sub.5                          VIII: R.sup.1 = H, Z = NH(CH.sub.3)                                            IX: R.sup.1 = CH.sub.3, Z = NH(CH.sub.3)                                       X: R.sup.1 = C.sub.2 H.sub.5, Z = NH(CH.sub.3)                                 XI: R.sup.1 = Allyl, Z = NH(CH.sub.3)                                          XII: R.sup.1 = Propargyl, Z = NH(CH.sub.3)                                     XIII: R.sup.1 = CH.sub.2 OCH.sub.3, Z = NH(CH.sub.3)                           XIV: R.sup.1 = COC.sub.2 H.sub.5, Z = NH(CH.sub.3)                             No.          B                                                                 ______________________________________                                         1            2-Pyridyl                                                         2            3-Trifluoromethyl-2-pyridyl                                       3            5-Trifluoromethyl-2-pyridyl                                       4            3,5-Bis-(trifluoromethyl)-2-pyridyl                               5            3,5-Dichloro-2-pyridyl                                            6            3-chloroo-5-trifluoromethyl-2-pyridyl                             7            3,5-Dichloro-2-pyridyl                                            8            2-Chloroo-4-trifluoromethylphenyl                                 9            2-Benzothiazolyl                                                  10           5-Chloroo-1-methyl-2-benzimidazolyl                               11           2-Benzoxazolyl                                                    12           1-Methyl-5-trifluoromethylimidazo-                                              5,4-a)!-pyridin-2-yl                                             13           5-Chloroo-2-pyrimidinyl                                           14           4-Methyl-5-phenyl-2-thiazolin-2-yl                                15           4-Methyl-5-phenyl-2-oxazolin-2-yl                                 16           7-Trifluoromethyl-4-quinolinyl                                    ______________________________________                                    

Example 16

Methyl N- 2-(3", 4"-dichlorophenyl-1'-methyliminooxy-methyl-4')-6-methylphenyl!-carbamate (Table 47, No. 2)

a) 2-(Methanesulfonyloxymethyl)-6-methyl-nitrobenzene

At 10°-15° C., 27 g (0.23 mol) of methanesulfonyl chloride dissolved in 20 ml of CH₂ Cl₂ is dripped into a mixture of 34 g (0.2 mol) of 3-methyl-2-nitrobenzyl alcohol and 27 g (0.27 mol) of triethylamine in 100 ml of CH₂ Cl₂. The reaction mixture is stirred for 1 hour at room temperature and is then extracted with water. The organic phase is dried over MgSO₄ and evaporated down. There is obtained as residue 48 g of the title compound as a yellow oil, containing about 10% of the corresponding benzyl chloride as impurity. The crude product is used for the next reaction without any further purification.

¹ H-NMR(COCl₃ ; δ bin ppm): 7.3-7.6 (m, 3H, phenyl); 5.3 (S, 2H, OCH₂); 3.0 (S, 3H, CH₃ -SO₃); 2.4 (S, 3H, CH₃)

b) 2-(3", 4"-Dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methyl-nitrobenzene

At room temperature, 1.8 g (75 mmol) of sodium hydride is added in portions to a solution of 13 g (64 mmol) of 3,4-dichloroacetophenonoxime in 100 ml of dimethylformamide. Upon conclusion of gas evolution, a solution of 16 g (65 mmol) of the mesylate from Example 1a in 30 ml of dimethylformamide is dripped in at 25°-30° C., and the mixture is then stirred for 1 hour at room temperature. The reaction mixture is diluted with water and the aqueous phase is then extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MGSO₄ and evaporated down. The residue crystallizes and is stirred with methanol. The mother liquor is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained a total of 20.4 g (58 mmol=90%) of the title compound as pale yellow crystals.

¹ H-NMR(CDCl₃ ; δ in ppm): 7.7 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.3 (S, 2H, OCH₂); 2.4 (S, 3H, CH₃); 2.2 (S, 3H, CH₃)

c) 2-(3", 4"-Dichlorophenyl-1-methyl-iminooxymethyl-4')-6-methyl-aniline

At 20°-30° C., 53 g of 21.8% strength Na₂ Fe(CO)₄ ! solution (1 kg of the solution contains 633 g of water, 218 g of Na₂ Fe(CO)₄ !, 108 g of Na₂ CO₃ and 41 g of NaOH) is added dropwise to 19 g (52.8 mmol) of the nitrobenzene from Example 16b in 150 ml of methanol. The brown suspension is stirred for 2 hours at room temperature, and the reaction mixture is then diluted with methylene chloride and the mixture is suction filtered using kieselguhr. The residue is again washed with CH₂ Cl₂ and the combined extracts are extracted with water, dried over MgSO₄ and evaporated down. The brown residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 14.3 g (44.3 inmol=82%) of the title compound as a beige solid.

1H-NMR(CDCl₃ ; δ in ppm): 7.7 (S, 1H, phenyl); 7.5 (m, 2H, phenyl); 7.1 (t, broad, 2H, phenyl); 6.7 (t, 1H, I=8 Hz, phenyl); 5.2 (S, 2H, OCH₂); 4.15 (S, 2H, NH₂ ; 2.2 (S, 3H, CH₃)

d) Methyl N- 2-(3", 4"-dichlorophenyl-1'-methyl-iminooxymethyl-4'-6-methylphenyl!-carbamate (Table 47, No. 2)

At 20°-30° C., 4.8 g (50 mmol) of methyl chloroformate and subsequently 4.8 g (60 mmol) of pyridine are dripped into a solution of 14.3 g (44 mmol) of the aniline from Example 1c in 150 ml of CH₂ Cl₂. The mixture is stirred overnight at room temperature and is then extracted with dilute hydrochloric acid and water. The reaction mixture is suction filtered using silica gel, dried over MgSO₄ and evaporated down. The residue crystallizes and is stirred with cyclohexane. There is obtained 13.8 g (36 mmol=82%) of the title compound as a colorless solid (mp=109° C.).

¹ H-NMR(CDCl₃ ; δ in ppm): 7.8 (S, 1H, phenyl); 7.6 (S, broad, 1H, NH); 7.4 (S, 2H, phenyl); 7.2 (m, 3H, phenyl); 5.2 (S, 2H, OCH₂); 3.8 (S, 3H, OCH₃); 2.3 (S, 3H, CH₃); 2.2 (S, 3H, CH₃)

Example 17

Methyl N- 2-(3", 4"-dichlorophenyl-1'-methyl-iminooxymethyl-4')-6-methylphenyl!-N-propargyl-carbamate (Table 47, No. 13)

At 25°-30° C., 0.15 g (6.3 mmol) of sodium hydride is added in portions to a solution of 1.9 g (5 mmol) of the carbamate from Example 16d in 20 ml of dimethylformamide. When no more gas evolves, 0.75 g (6.3 mmol) of propargyl bromide is added and the whole is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. There is obtained 1.4 g (3.3 mmol=67%) of the title compound as a yellow oil.

1H-NMR (CDCl₃ ; δ in ppm): 7.75 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.2 (dd, 2H, I=12 Hz, OCH₂); 4.4 (dd, broad, I=16 Hz, NCH₂); (S, 3H, OCH₃); 2.3 (S, 3H, CH₃); 2.25 (S, broad, 1H, C.tbd.CH); 2.2 (S, 3H, CH₃); the ¹ H-NMR spectrum also contains signals of about 20% of the amide rotamer.

The compounds described in the following tables may be prepared analogously.

                  TABLE 41                                                         ______________________________________                                          ##STR273##                                                                    I: R.sup.1 = H, X = CH.sub.3                                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3                                 VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = Cl                                     XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       Compound I from Table 41 has for instance the following                        structural formula:                                                             ##STR274##                                                                    No.     T.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.5, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-OCH.sub.2 C.sub.6 H.sub.5                                            178     3-OCH.sub.2 C.sub.6 H.sub.5                                            179     4-OCH.sub.2 C.sub.6 H.sub.5                                            180     2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    181     3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                    182     4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-Cl                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CH.sub.3).sub.2, 6-F                                              247     2,4-(CH.sub.3).sub.2, 6-Cl                                             248     2,4-(CH.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-CH.sub.3 CH.sub.2 CO                                            304     2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                   305     2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                         306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-CH.sub.3 CO                                            308     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   309     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          310     2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                311     2-Cl-4-CHO                                                             312     2-Cl-4-CH.sub.3 CO                                                     313     2-Cl-4-CH.sub.3 CH.sub.2 CO                                            314     2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                         315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-CH.sub.3 CO                                            317     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   318     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          319     2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                   369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOn-C.sub.3 H.sub.7)                377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                        381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.3)                          645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOn-C.sub.3 H.sub.7)                 647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Allyl)                            649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-Propargyl)                        651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.3)                          654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOC.sub.2 H.sub.5)                   655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.3 H.sub.7)                656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-i-C.sub.3 H.sub.7)                657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Allyl)                            658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-trans-Chloroallyl)                659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-Propargyl)                        660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNO-n-C.sub.4 H.sub.9)                661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7 CNOCH.sub.2 C.sub.6 H.sub.5)          662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     5-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 42                                                         ______________________________________                                          ##STR275##                                                                    I: R.sup.1 = H, X = CH.sub.3                                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3                                 VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = Cl                                     XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       No.       B                                                                    ______________________________________                                          1        Pyrrolyl-3                                                            2        NCH.sub.3 -Pyrrolyl-3                                                 3        NC.sub.6 H.sub.5 -Pyrrolyl-3                                          4        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            5        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            6        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                            7        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           8        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           9        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                           10       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            11       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            12       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                            13       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   14       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   15       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                   16       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   17       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   18       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                   19       Pyrrolyl-2                                                            20       NCH.sub.3 -Pyrrolyl-2                                                 21       NC.sub.6 H.sub.5 -Pyrrolyl-2                                          22       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            23       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            24       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                            25       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           26       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           27       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                           28       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            29       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            30       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                            31       N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   32       N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   33       N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                   34       N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   35       N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   36       N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                   37       Furyl-2                                                               38       5-CH.sub.3 -Furyl-2                                                   39       5-C.sub.6 H.sub.5 -Furyl-2                                            40       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               41       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               42       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               43       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              44       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              45       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              46       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               47       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               48       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               49       5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      50       5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      51       5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      52       5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      53       5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      54       5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      55       4-CH.sub.3 -Furyl-2                                                   56       4-C.sub.6 H.sub.5 -Furyl-2                                            57       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               58       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               59       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                               60       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              61       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              62       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                              63       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               64       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               65       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                               66       4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                      67       4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                      68       4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                      69       4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                      70       4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                      71       4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                      72       Thienyl-2                                                             73       5-CH.sub.3 -Thienyl-2                                                 74       5-C.sub.6 H.sub.5 -Thienyl-2                                          75       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             76       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             77       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             78       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            79       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            80       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            81       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             82       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             83       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             84       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                    85       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                    86       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                    87       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                    88       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                    89       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                    90       4-CH.sub.3 -Thienyl-2                                                 91       4-C.sub.6 H.sub.5 -Thienyl-2                                          92       4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             93       4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             94       4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                             95       4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            96       4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            97       4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                            98       4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                             99       4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       NCH.sub.3 -Pyrazolyl-4                                               127       NC.sub.6 H.sub.5 -Pyrazolyl-4                                        128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-pyrazolyl-4                                 143       3-CH.sub.3 -N-Methylpyrazolyl-4                                      144       3-C.sub.6 H.sub.5 -N-Methylpyrazolyl-4                               145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   154       3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          155       3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          156       3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          157       3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          158       3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          159       3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          160       Isoxazolyl-5                                                         161       3-CH.sub.3 -Isoxazolyl-5                                             162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C6H4 -4-Chloroisoxazolyl-5                            188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 -Isoxazolyl-3                                             198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazqlyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 -Isothiazolyl-5                                           216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       3-CH.sub.3 -Oxazolyl-4                                               234       3-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           236       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           237       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           238       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          239       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          241       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           242       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           243       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           244       3-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  245       3-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  246       3-(2'-CNC.sub.6 H.sub.4)-oxazolyl-4                                  247       3-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  248       3-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  249       3-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       NCH.sub.3 -1,2,4-Triazolyl-5                                         269       3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                              270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          280       3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 281       3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 282       3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 283       3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 284       3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 285       3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        384       1-Naphthyl                                                           385       2-Naphthyl                                                           ______________________________________                                    

                  TABLE 43                                                         ______________________________________                                          ##STR276##                                                                    I: R.sup.1 = H, X = CH.sub.3                                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3                                 VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = Cl                                     XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       No.     T.sub.m                                                                ______________________________________                                          1      H                                                                       2      2-F                                                                     3      3-F                                                                     4      4-F                                                                     5      2,4-F.sub.2                                                             6      2,4,6-F.sub.3                                                           7      2,3,4,5,6-F.sub.5                                                       8      2,3-F.sub.2                                                             9      2-Cl                                                                    10     3-Cl                                                                    11     4-Cl                                                                    12     2,3-Cl.sub.2                                                            13     2,4-Cl.sub.2                                                            14     2,5-Cl.sub.2                                                            15     2,6-Cl.sub.2                                                            16     3,4-Cl.sub.2                                                            17     3,5-Cl.sub.2                                                            18     2,3,4-Cl.sub.3                                                          19     2,3,5-Cl.sub.3                                                          20     2,3,6-Cl.sub.3                                                          21     2,4,5-Cl.sub.3                                                          22     2,4,6-Cl.sub.3                                                          23     3,4,5-Cl.sub.3                                                          24     2,3,4,6-Cl.sub.4                                                        25     2,3,5,6-Cl.sub.4                                                        26     2,3,4,5,6-Cl.sub.5                                                      27     2-Br                                                                    28     3-Br                                                                    29     4-Br                                                                    30     2,4-Br.sub.2                                                            31     2,5-Br.sub.2                                                            32     2,6-Br.sub.2                                                            33     2,4,6-Br.sub.3                                                          34     2,3,4,5,6-Br.sub.5                                                      35     2-I                                                                     36     3-I                                                                     37     4-I                                                                     38     2,4-I.sub.2                                                             39     2-Cl, 3-F                                                               40     2-Cl, 4-F                                                               41     2-Cl, 5-F                                                               42     2-Cl, 6-F                                                               43     2-Cl, 3-Br                                                              44     2-Cl, 4-Br                                                              45     2-Cl, 5-Br                                                              46     2-Cl, 6-Br                                                              47     2-Br, 3-Cl                                                              48     2-Br, 4-Cl                                                              49     2-Br, 5-Cl                                                              50     2-Br, 3-F                                                               51     2-Br, 4-F                                                               52     2-Br, 5-F                                                               53     2-Br, 6-F                                                               54     2-F, 3-Cl                                                               55     2-F, 4-Cl                                                               56     2-F, 5-Cl                                                               57     3-Cl, 4-F                                                               58     3-Cl, 5-F                                                               59     3-Cl, 4-Br                                                              60     3-Cl, 5-Br                                                              61     3-F, 4-Cl                                                               62     3-F, 4-Br                                                               63     3-Br, 4-Cl                                                              64     3-Br, 4-F                                                               65     2,6-Cl.sub.2, 4-Br                                                      66     2-CH.sub.3                                                              67     3-CH.sub.3                                                              68     4-CH.sub.3                                                              69     2,3-(CH.sub.3).sub.2                                                    70     2,4-(CH.sub.3).sub.2                                                    71     2,5-(CH.sub.3).sub.2                                                    72     2,6-(CH.sub.3).sub.2                                                    73     3,4-(CH.sub.3).sub.2                                                    74     3,5-(CH.sub.3).sub.2                                                    75     2,3,5-(CH.sub.3).sub.3                                                  76     2,3,4-(CH.sub.3).sub.3                                                  77     2,3,6-(CH.sub.3).sub.3                                                  78     2,4,5-(CH.sub.3).sub.3                                                  79     2,4,6-(CH.sub.3).sub.3                                                  80     3,4,5-(CH.sub.3).sub.3                                                  81     2,3,4,6-(CH.sub.3).sub.4                                                82     2,3,5,6-(CH.sub.3).sub.4                                                83     2,3,4,5,6-(CH.sub.3).sub.5                                              84     2-C.sub.2 H.sub.5                                                       85     3-C.sub.2 H.sub.5                                                       86     4-C.sub.2 H.sub.5                                                       87     2,4-(C.sub.2 H.sub.5).sub.2                                             88     2,6-(C.sub.2 H.sub.5).sub.2                                             89     3,5-(C.sub.2 H.sub.5).sub.2                                             90     2,4,6-(C.sub.2 H.sub.5).sub.3                                           91     2-n-C.sub.3 H.sub.7                                                     92     3-n-C.sub.3 H.sub.7                                                     93     4-n-C.sub.3 H.sub.7                                                     94     2-i-C.sub.3 H.sub.7                                                     95     3-i-C.sub.3 H.sub.7                                                     96     4-i-C.sub.3 H.sub.7                                                     97     2,4-(i-C.sub.3 H.sub.7).sub.2                                           98     2,6-(i-C.sub.3 H.sub.7).sub.2                                           99     3,5-(i-C.sub.3 H.sub.7).sub.2                                          100     2,4,6-(i-C.sub.3 H.sub.7).sub.3                                        101     2-s-C.sub.4 H.sub.9                                                    102     3-s-C.sub.4 H.sub.9                                                    103     4-s-C.sub.4 H.sub.9                                                    104     2-t-C.sub.4 H.sub.9                                                    105     3-t-C.sub.4 H.sub.9                                                    106     4-t-C.sub.4 H.sub.9                                                    107     2,3-(t-C.sub.4 H.sub.9).sub.2                                          108     2,4-(t-C.sub.4 H.sub.9).sub.2                                          109     2,5-(t-C.sub.4 H.sub.9).sub.2                                          110     2,6-(t-C.sub.4 H.sub.9).sub.2                                          111     3,4-(t-C.sub.4 H.sub.9).sub.2                                          112     2,4,6-(t-C.sub.4 H.sub.9).sub.3                                        113     4-n-C.sub.9 H.sub.19                                                   114     4-n-C.sub.12 H.sub.25                                                  115     4-n-C.sub.15 H.sub.31                                                  116     4-(1,1,3,3-Tetramethylbutyl)                                           117     4-(2,4,4-Trimethylpropyl)                                              118     2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                        119     2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                        120     2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                              121     2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                        122     2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                        123     2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        124     2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                        125     3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                        126     2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                        127     2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                     128     2-Allyl                                                                129     3-Allyl                                                                130     4-Allyl                                                                131     2-Allyl, 6-CH.sub.3                                                    132     2-cyclo-C.sub.6 H.sub.11                                               133     3-cyclo-C.sub.6 H.sub.11                                               134     4-cyclo-C.sub.6 H.sub.11                                               135     2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                         136     2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                   137     2-CH.sub.2 C.sub.6 H.sub.5                                             138     3-CH.sub.2 C.sub.6 H.sub.5                                             139     4-CH.sub.2 C.sub.6 H.sub.5                                             140     2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                 141     2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                 142     2-C.sub.6 H.sub.5                                                      143     3-C.sub.6 H.sub.5                                                      144     4-C.sub.6 H.sub.5                                                      145     4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                                146     4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                                147     2-Cl, 4-C.sub.6 H.sub.5                                                148     2-Br, 4-C.sub.6 H.sub.5                                                149     2-C.sub.6 H.sub.4, 4-Cl                                                150     2-C.sub.6 H.sub.5, 4-Br                                                151     2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                       152     2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                       153     2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                       154     2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                       155     2-cyclo-C.sub.6 H.sub.11, 4-Cl                                         156     2-cyclo-C.sub.6 H.sub.11, 4-Br                                         157     2-Cl, 4-cyclo-C.sub.6 H.sub.11                                         158     2-Br, 4-cyclo-C.sub.6 H.sub.11                                         159     2-OCH.sub.3                                                            160     3-OCH.sub.3                                                            161     4-OCH.sub.3                                                            162     2-OC.sub.2 H.sub.5                                                     163     3-OC.sub.2 H.sub.5                                                     164     4-OC.sub.2 H.sub.5                                                     165     2-O-n-C.sub.3 H.sub.7                                                  166     3-O-n-C.sub.3 H.sub.7                                                  167     4-O-n-C.sub.3 H.sub.7                                                  168     2-O-i-C.sub.3 H.sub.7                                                  169     3-O-i-C.sub.3 H.sub.7                                                  170     4-O-i-C.sub.3 H.sub.7                                                  171     2-O-n-C.sub.6 H.sub.13                                                 172     3-O-n-C.sub.6 H.sub.13                                                 173     4-O-n-C.sub.6 H.sub.13                                                 174     2-O-n-C.sub.8 H.sub.17                                                 175     3-O-n-C.sub.8 H.sub.17                                                 176     4-O-n-C.sub.8 H.sub.17                                                 177     2-O-CH.sub.2 C.sub.6 H.sub.5                                           178     3-O-CH.sub.2 C.sub.6 H.sub.5                                           179     4-O-CH.sub.2 C.sub.6 H.sub.5                                           180     2-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   181     3-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   182     4-O-(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183     2,4-(OCH.sub.3).sub.2                                                  184     2-CF.sub.3                                                             185     3-CF.sub.3                                                             186     4-CF.sub.3                                                             187     2-OCF.sub.3                                                            188     3-OCF.sub.3                                                            189     4-OCF.sub.3                                                            190     3-OCH.sub.2 CHF.sub.2                                                  191     2-NO.sub.2                                                             192     3-NO.sub.2                                                             193     4-NO.sub.2                                                             194     2-CN                                                                   195     3-CN                                                                   196     4-CN                                                                   197     2-CH.sub.3, 3-Cl                                                       198     2-CH.sub.3, 4-Cl                                                       199     2-CH.sub.3, 5-Cl                                                       200     2-CH.sub.3, 6-Cl                                                       201     2-CH.sub.3, 3-F                                                        202     2-CH.sub.3, 4-F                                                        203     2-CH.sub.3, 5-F                                                        204     2-CH.sub.3, 6-F                                                        205     2-CH.sub.3, 3-Br                                                       206     2-CH.sub.3, 4-Br                                                       207     2-CH.sub.3, 5-Br                                                       208     2-CH.sub.3, 6-Br                                                       209     2-Cl, 3-CH.sub.3                                                       210     2-Cl, 4-CH.sub.3                                                       211     2-Cl, 5-CH.sub.3                                                       212     2-F, 3-CH.sub.3                                                        213     2-F, 4-CH.sub.3                                                        214     2-F, 5-CH.sub.3                                                        215     2-Br, 3-CH.sub.3                                                       216     2-Br, 4-CH.sub.3                                                       217     2-Br, 5-CH.sub.3                                                       218     3-CH.sub.3, 4-Cl                                                       219     3-CH.sub.3, 5-Cl                                                       220     3-CH.sub.3, 4-F                                                        221     3-CH.sub.3, 5-F                                                        222     3-CH.sub.3, 4-Br                                                       223     3-CH.sub.3, 5-Br                                                       224     3-F, 4-CH.sub.3                                                        225     3-Cl, 4-CH.sub.3                                                       226     3-Br, 4-CH.sub.3                                                       227     2-Cl, 4,5-(CH.sub.3).sub.2                                             228     2-Br, 4,5-(CH.sub.3).sub.2                                             229     2-Cl, 3,5-(CH.sub.3).sub.2                                             230     2-Br, 3,5-(CH.sub.3).sub.2                                             231     2,6-Cl.sub.2, 4-CH.sub.3                                               232     2,6-F.sub.2, 4-CH.sub.3                                                233     2,6-Br.sub.2, 4-CH.sub.3                                               234     2,4-Br.sub.2, 6-CH.sub.3                                               235     2,4-F.sub.2, 6-CH.sub.3                                                236     2,4-Br.sub.2, 6-CH.sub.3                                               237     2,6-(CH.sub.3).sub.2, 4-F                                              238     2,6-(CH.sub.3).sub.2, 4-Cl                                             239     2,6-(CH.sub.3).sub.2, 4-Br                                             240     3,5-(CH.sub.3).sub.2, 4-F                                              241     3,5-(CH.sub.3).sub.2, 4-CL                                             242     3,5-(CH.sub.3).sub.2, 4-Br                                             243     2,3,6-(CH.sub.3).sub.3, 4-F                                            244     2,3,6-(CH.sub.3).sub.3, 4-Cl                                           245     2,3,6-(CH.sub.3).sub.3, 4-Br                                           246     2,4-(CB.sub.3).sub.2, 6-F                                              247     2,4-(CB.sub.3).sub.2, 6-Cl                                             248     2,4-(CB.sub.3).sub.2, 6-Br                                             249     2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                  250     2-Cl, 4-NO.sub.2                                                       251     2-NO.sub.2, 4-Cl                                                       252     2-OCH.sub.3, 5-NO.sub.2                                                253     2,4-Cl.sub.2, 5-NO.sub.2                                               254     2,4-Cl.sub.2, 6-NO.sub.2                                               255     2,6-Cl.sub.2, 4-NO.sub.2                                               256     2,6-Br.sub.2, 4-NO.sub.2                                               257     2,6-I.sub.2, 4-NO.sub.2                                                258     2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                  259     2-CO.sub.2 CH.sub.3                                                    260     3-CO.sub.2 CH.sub.3                                                    261     4-CO.sub.2 CH.sub.3                                                    262     2-CO.sub.2 (C.sub.2 H.sub.5)                                           263     3-CO.sub.2 (C.sub.2 H.sub.5)                                           264     4-CO.sub.2 (C.sub.2 H.sub.5)                                           265     2-CO.sub.2 (n-C.sub.3 H.sub.7)                                         266     3-CO.sub.2 (n-C.sub.3 H.sub.7)                                         267     4-CO.sub.2 (n-C.sub.3 H.sub.7)                                         268     2-CO.sub.2 (i-C.sub.3 H.sub.7)                                         269     3-CO.sub.2 (i-C.sub.3 H.sub.7)                                         270     4-CO.sub.2 (i-C.sub.3 H.sub.7)                                         271     2-CO.sub.2 (n-C.sub.6 H.sub.13)                                        272     3-CO.sub.2 (n-C.sub.6 H.sub.13)                                        273     4-CO.sub.2 (n-C.sub.6 H.sub.13)                                        274     2-CH.sub.2 OCH.sub.3                                                   275     3-CH.sub.2 OCH.sub.3                                                   276     4-CH.sub.2 OCH.sub.3                                                   277     2-CH.sub.2 O(C.sub.2 H.sub.5)                                          278     3-CH.sub.2 O(C.sub.2 H.sub.5)                                          279     4-CH.sub.2 O(C.sub.2 H.sub.5)                                          280     2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        281     3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        282     4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                        283     2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        284     3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        285     4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                        286     2-CHO                                                                  287     3-CHO                                                                  288     4-CHO                                                                  289     2-COCH.sub.3                                                           290     3-COCH.sub.3                                                           291     4-COCH.sub.3                                                           292     2-COCH.sub.2 CH.sub.3                                                  293     3-COCH.sub.2 CH.sub.3                                                  294     4-COCH.sub.2 CH.sub.3                                                  295     2-COCH.sub.2 CH.sub.2 CH.sub.3                                         296     3-COCH.sub.2 CH.sub.2 CH.sub.3                                         297     4-COCH.sub.2 CH.sub.2 CH.sub.3                                         298     2-COCH(CH.sub.3)CH.sub.3                                               299     3-COCH(CH.sub.3)CH.sub.3                                               300     4-COCH(CH.sub.3)CH.sub.3                                               301     2-Me-4-CHO                                                             302     2-Me-4-CH.sub.3 CO                                                     303     2-Me-4-CH.sub.3 CH.sub.2 CO                                            304     2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                   305     2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                         306     2,5-Me.sub.2 -4-CHO                                                    307     2,5-Me.sub.2 -4-CH.sub.3 CO                                            308     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   309     2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          310     2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                311     2-Cl-4-CHO                                                             312     2-Cl-4-CH.sub.3 CO                                                     313     2-Cl-4-CH.sub.3 CH.sub.2 CO                                            314     2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                         315     2,5-Cl.sub.2 -4-CHO                                                    316     2,5-Cl.sub.2 -4-CH.sub.3 CO                                            317     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                   318     2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                          319     2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                                320     2-C(NOCH.sub.3)CH.sub.3                                                321     3-C(NOCH.sub.3)CH.sub.3                                                322     4-C(NOCH.sub.3)CH.sub.3                                                323     2-C(NOC.sub.2 H.sub.5)CH.sub.3                                         324     3-C(NOC.sub.2 H.sub.5)CH.sub.3                                         325     4-C(NOC.sub.2 H.sub.5)CH.sub.3                                         326     2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      327     3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      328     4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                      329     2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      330     3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      331     4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                      332     2-C(NO-Allyl)-CH.sub.3                                                 333     3-C(NO-Allyl)-CH.sub.3                                                 334     4-C(NO-Allyl)-CH.sub.3                                                 335     2-C(NO-trans-Chloroallyl)-CH.sub.3                                     336     3-C(NO-trans-Chloroallyl)-CH.sub.3                                     337     4-C(NO-trans-Chloroallyl)-CH.sub.3                                     338     2-C(NO-Propargyl)-CH.sub.3                                             339     3-C(NO-Propargyl)-CH.sub.3                                             340     4-C(NO-Propargyl)-CH.sub.3                                             341     2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      342     3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      343     4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                      344     2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                345     3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                346     4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                                347     2-CH.sub.3 -4-CHNOCH.sub.3                                             348     2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                      349     2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                   350     2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                   351     2-CH.sub.3 -4-CHNO-Allyl                                               352     2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                 353     2-CH.sub.3 -4-CHNO-Propargyl                                           354     2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                   355     2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                             356     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                   357     2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                            358     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                         359     2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                         360     2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                     361     2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                         362     2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                 363     2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                         364     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                   365     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                            366     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                     367     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                  368     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7)                  369     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                              370     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                  371     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                          372     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                  373     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)            374     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                         375     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                  376     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)               377     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)               378     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                           379     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)               380     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Propargyl)                       381     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)               382     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)         383     2-C.sub.6 H.sub.5                                                      384     3-C.sub.6 H.sub.5                                                      385     4-C.sub.6 H.sub.5                                                      386     2-(2'-FC.sub.6 H.sub.4)                                                387     2-(3'-FC.sub.6 H.sub.4)                                                388     2-(4'-FC.sub.6 H.sub.4)                                                389     3-(2'-FC.sub.6 H.sub.4)                                                390     3-(3'-FC.sub.6 H.sub.4)                                                391     3-(4'-FC.sub.6 H.sub.4)                                                392     4-(2'-FC.sub.6 H.sub.4)                                                393     4-(3'-FC.sub.6 H.sub.4)                                                394     4-(4'-FC.sub.6 H.sub.4)                                                395     2-(2'-ClC.sub.6 H.sub.4)                                               396     2-(3'-ClC.sub.6 H.sub.4)                                               397     2-(4'-ClC.sub.6 H.sub.4)                                               398     3-(2'-ClC.sub.6 H.sub.4)                                               399     3-(3'-ClC.sub.6 H.sub.4)                                               400     3-(4'-ClC.sub.6 H.sub.4)                                               401     4-(2'-ClC.sub.6 H.sub.4)                                               402     4-(3'-ClC.sub.6 H.sub.4)                                               403     4-(4'-ClC.sub.6 H.sub.4)                                               405     2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        406     2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        407     2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        408     3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        409     3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        410     3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        411     4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                        412     4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                        413     4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                        414     2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      415     2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      416     2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      417     3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      418     3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      419     3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      420     4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                      421     4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                      422     4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                      423     2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           424     2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           425     2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           426     3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           427     3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           428     3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           429     4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           430     4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           431     4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                           432     2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               433     2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               434     2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               435     3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               436     3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               437     3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               438     4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               439     4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               440     4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                               441     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       442     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       443     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       444     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       445     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       446     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       447     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                       448     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                       449     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                       450     2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        451     2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        452     2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        453     3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        454     3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        455     3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        456     4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                        457     4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                        458     4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                        459     2-(2'-NCC.sub.6 H.sub.4)                                               460     2-(3'-NCC.sub.6 H.sub.4)                                               461     2-(4'-NCC.sub.6 H.sub.4)                                               462     3-(2'-NCC.sub.6 H.sub.4)                                               463     3-(3'-NCC.sub.6 H.sub.4)                                               464     3-(4'-NCC.sub.6 H.sub.4)                                               465     4-(2'-NCC.sub.6 H.sub.4)                                               466     4-(3'-NCC.sub.6 H.sub.4)                                               467     4-(4'-NCC.sub.6 H.sub.4)                                               468     2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        469     2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        470     2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        471     3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        472     3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        473     3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        474     4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                        475     4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                        476     4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                        477     2-OC.sub.6 H.sub.5                                                     475     3-OC.sub.6 H.sub.5                                                     476     4-OC.sub.6 H.sub.5                                                     478     2-O-(2'-FC.sub.6 H.sub.4)                                              479     2-O-(3'-FC.sub.6 H.sub.4)                                              480     2-O-(4'-FC.sub.6 H.sub.4)                                              481     3-O-(2'-FC.sub.6 H.sub.4)                                              482     3-O-(3'-FC.sub.6 H.sub.4)                                              483     3-O-(4'-FC.sub.6 H.sub.4)                                              484     4-O-(2'-FC.sub.6 H.sub.4)                                              485     4-O-(3'-FC.sub.6 H.sub.4)                                              486     4-O-(4'-FC.sub.6 H.sub.4)                                              487     2-O-(2'-ClC.sub.6 H.sub.4)                                             488     2-O-(3'-ClC.sub.6 H.sub.4)                                             489     2-O-(4'-ClC.sub.6 H.sub.4)                                             490     3-O-(2'-ClC.sub.6 H.sub.4)                                             491     3-O-(3'-ClC.sub.6 H.sub.4)                                             492     3-O-(4'-ClC.sub.6 H.sub.4)                                             493     3-O-(4'-ClC.sub.6 H.sub.4)                                             494     4-O-(2'-ClC.sub.6 H.sub.4)                                             495     4-O-(3'-ClC.sub.6 H.sub.4)                                             496     4-O-(4'-ClC.sub.6 H.sub.4)                                             497     2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      498     2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      499     2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      500     3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      501     3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      502     3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      503     4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                      504     4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                      505     4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                      506     2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    507     2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    508     2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    509     3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    510     3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    511     3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    512     4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                    513     4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                    514     4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                    515     2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         516     2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         517     2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         518     3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         519     3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         520     3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         521     4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         522     4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         523     4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                         524     2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             525     2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             526     2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             527     3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             528     3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             529     3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             530     4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             531     4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             532     4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                             533     2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     534     2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     535     2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     536     3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     537     3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     538     3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     539     4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                     540     4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                     541     4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                     542     2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      543     2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      544     2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      545     3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      546     3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      547     3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      548     4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                      549     4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                      550     4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                      551     2-O-(2'-NCC.sub.6 H.sub.4)                                             552     2-O-(3'-NCC.sub.6 H.sub.4)                                             553     2-O-(4'-NCC.sub.6 H.sub.4)                                             554     3-O-(2'-NCC.sub.6 H.sub.4)                                             555     3-O-(3'-NCC.sub.6 H.sub.4)                                             556     3-O-(4'-NCC.sub.6 H.sub.4)                                             557     4-O-(2'-NCC.sub.6 H.sub.4)                                             558     4-O-(3'-NCC.sub.6 H.sub.4)                                             559     4-O-(4'-NCC.sub.6 H.sub.4)                                             560     2-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      561     2-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      562     2-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      563     3-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      564     3-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      565     3-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      566     4-O-(2'-CF.sub.3 C.sub.6 H.sub.4)                                      567     4-O-(3'-CF.sub.3 C.sub.6 H.sub.4)                                      568     4-O-(4'-CF.sub.3 C.sub.6 H.sub.4)                                      569     2-Pyridinyl-2'                                                         570     2-Pyridinyl-3'                                                         571     2-Pyridinyl-4'                                                         572     3-Pyridinyl-2'                                                         573     3-Pyridinyl-3'                                                         574     3-Pyridinyl-4'                                                         575     4-Pyridinyl-2'                                                         576     4-Pyridinyl-3'                                                         577     4-Pyridinyl-4'                                                         578     2-Pyrimidinyl-2'                                                       579     2-Pyrimidinyl-3'                                                       580     2-Pyrimidinyl-4'                                                       581     3-Pyrimidinyl-2'                                                       582     3-Pyrimidinyl-3'                                                       583     3-Pyrimidinyl-4'                                                       584     4-Pyrimidinyl-2'                                                       585     4-Pyrimidinyl-3'                                                       586     4-Pyrimidinyl-4'                                                       587     2-Pyrazolyl-1'                                                         588     2-Pyrazolyl-3'                                                         589     2-Pyrazolyl-4'                                                         590     3-Pyrazolyl-1'                                                         591     3-Pyrazolyl-3'                                                         592     3-Pyrazolyl-4'                                                         593     4-Pyrazolyl-1'                                                         594     4-Pyrazolyl-3'                                                         595     4-Pyrazolyl-4'                                                         596     2-Isoxazolyl-3'                                                        597     2-Isoxazolyl-4'                                                        598     2-Isoxazolyl-5'                                                        599     3-Isoxazolyl-3'                                                        600     3-Isoxazolyl-4'                                                        601     3-Isoxazolyl-5'                                                        602     4-Isoxazolyl-3'                                                        603     4-Isoxazolyl-4'                                                        604     4-Isoxazolyl-5'                                                        605     2-Isothiazolyl-3'                                                      606     2-Isothiazolyl-4'                                                      607     2-Isothiazolyl-5'                                                      608     3-Isothiazolyl-3'                                                      609     3-Isothiazolyl-4'                                                      610     3-Isothiazolyl-5'                                                      611     4-Isothiazolyl-3'                                                      612     4-Isothiazolyl-4'                                                      613     4-Isothiazolyl-5'                                                      614     2-Imidazolyl-1'                                                        615     2-Imidazolyl-2'                                                        616     2-Imidazolyl-4'                                                        617     3-Imidazolyl-1'                                                        618     3-Imidazolyl-2'                                                        619     3-Imidazolyl-4'                                                        620     4-Imidazolyl-1'                                                        621     4-Imidazolyl-2'                                                        622     4-Imidazolyl-4'                                                        623     2-Oxazolyl-2'                                                          624     2-Oxazolyl-4'                                                          625     2-Oxazolyl-5'                                                          626     3-Oxazolyl-2'                                                          627     3-Oxazolyl-4'                                                          628     3-Oxazolyl-5'                                                          629     4-Oxazolyl-2'                                                          630     4-Oxazolyl-4'                                                          631     4-Oxazolyl-5'                                                          632     2-Thiazolyl-2'                                                         633     2-Thiazolyl-4'                                                         634     2-Thiazolyl-5'                                                         635     3-Thiazolyl-2'                                                         636     3-Thiazolyl-4'                                                         637     3-Thiazolyl-5'                                                         638     4-Thiazolyl-2'                                                         639     4-Thiazolyl-4'                                                         640     4-Thiazolyl-5'                                                         641     2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)                642     2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 CH.sub.2 OCH.sub.3)         643     2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 CH.sub.2 OCH.sub.3)      644     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNOCH.sub.3)                           645     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNOC.sub.2 H.sub.5)                    646     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-n-C.sub.3 H.sub.7)                 647     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-i-C.sub.3 H.sub.7)                 648     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-Allyl)                             649     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-trans-Chloroallyl)                 650     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-Propargyl)                         651     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNO-n-C.sub.4 H.sub.9)                 652     2-CH.sub.3 -4-(n-C.sub.3 H.sub.7CNOCH.sub.2 C.sub.6 H.sub.5)           653     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNOCH.sub.3)                           654     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNOC.sub.2 H.sub.5)                    655     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-n-C.sub.3 H.sub.7)                 656     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-i-C.sub.3 H.sub.7)                 657     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-Allyl)                             658     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-trans-Chloroallyl)                 659     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-Propargyl)                         660     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNO-n-C.sub.4 H.sub.9)                 661     2-CH.sub.3 -4-(i-C.sub.3 H.sub.7CNOCH.sub.2 C.sub.6 H.sub.5)           662     2-O-n-C.sub.4 H.sub.9                                                  663     2-O-i-C.sub.4 H.sub.9                                                  664     2-O-s-C.sub.4 H.sub.9                                                  665     2-O-t-C.sub.4 H.sub.9                                                  666     2-Neopentyloxy                                                         667     3-O-n-C.sub.4 H.sub.9                                                  668     3-O-i-C.sub.4 H.sub.9                                                  669     3-O-s-C.sub.4 H.sub.9                                                  670     3-O-t-C.sub.4 H.sub.9                                                  671     3-Neopentyloxy                                                         672     4-O-n-C.sub.4 H.sub.9                                                  673     4-O-i-C.sub.4 H.sub.9                                                  674     4-O-s-C.sub.4 H.sub.9                                                  675     4-O-t-C.sub.4 H.sub.9                                                  676     4-Neopentyloxy                                                         677     3-CH.sub.3 -4-OCH.sub.3                                                678     3-CH.sub.3 -4-OC.sub.2 H.sub.5                                         679     3-CH.sub.3 -4-O-n-C.sub.3 H.sub.7                                      680     3-CH.sub.3 -4-O-n-C.sub.4 H.sub.9                                      681     3-CH.sub.3 -4-O-i-C.sub.4 H.sub.9                                      682     3-CH.sub.3 -4-O-s-C.sub.4 H.sub.9                                      683     3-CH.sub.3 -4-O-t-C.sub.4 H.sub.9                                      684     3-CH.sub.3 -4-Neopentyloxy                                             685     2-CH.sub.3 -3-OCH.sub.3                                                686     2-CH.sub.3 -4-OCH.sub.3                                                687     2-CH.sub.3 -5-OCH.sub.3                                                688     2-CH.sub.3 -6-OCH.sub.3                                                689     3-CH.sub.3 -4-OCH.sub.3                                                690     3-CH.sub.3 -5-OCH.sub.3                                                691     3-CH.sub.3 -6-OCH.sub.3                                                692     4-CH.sub.3 -5-OCH.sub.3                                                693     4-CH.sub.3 -6-OCH.sub.3                                                694     4-CH.sub.3 -6-OCH.sub.3                                                695     2-CH.sub.3 -3-O-i-C.sub.3 H.sub.7                                      696     2-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      697     2-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      698     2-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      699     3-CH.sub.3 -4-O-i-C.sub.3 H.sub.7                                      700     3-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      701     3-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      702     4-CH.sub.3 -5-O-i-C.sub.3 H.sub.7                                      703     4-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      704     5-CH.sub.3 -6-O-i-C.sub.3 H.sub.7                                      705     2-Cl-3-OCH.sub.3                                                       706     2-Cl-4-OCH.sub.3                                                       707     2-Cl-5-OCH.sub.3                                                       708     2-Cl-6-OCH.sub.3                                                       709     3-Cl-4-OCH.sub.3                                                       710     3-Cl-5-OCH.sub.3                                                       711     3-Cl-6-OCH.sub.3                                                       712     4-Cl-5-OCH.sub.3                                                       713     4-Cl-6-OCH.sub.3                                                       714     4-Cl-6-OCH.sub.3                                                       ______________________________________                                    

                  TABLE 44                                                         ______________________________________                                          ##STR277##                                                                    I: R.sup.1 = H, X = CH.sub.3                                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3                                 VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2OCH.sub.3, X = Cl                                      XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       No.     B                                                                      ______________________________________                                          1      Pyrrolyl-3                                                              2      NCH.sub.3 -Pyrrolyl-3                                                   3      NC.sub.6 H.sub.5 -Pyrrolyl-3                                            4      N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                              5      N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                              6      N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                              7      N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                             8      N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                             9      N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                             10     N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                              11     N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                              12     N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                              13     N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                     14     N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                     15     N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                     16     N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                     17     N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                     18     N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                     19     Pyrrolyl-2                                                              20     NCH.sub.3 -Pyrrolyl-2                                                   21     NC.sub.6 H.sub.5 -Pyrrolyl-2                                            22     N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                              23     N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                              24     N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                              25     N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                             26     N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                             27     N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                             28     N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                              29     N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                              30     N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                              31     N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                     32     N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                     33     N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                     34     N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                     35     N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                     36     N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                     37     Furyl-2                                                                 38     5-CH.sub.3 -Furyl-2                                                     39     5-C.sub.6 H.sub.5 -Furyl-2                                              40     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 41     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 42     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 43     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                44     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                45     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                46     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 47     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 48     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 49     5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                        50     5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                        51     5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                        52     5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                        53     5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                        54     5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                        55     4-CH.sub.3 -Furyl-2                                                     56     4-C.sub.6 H.sub.5 -Furyl-2                                              57     4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 58     4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 59     4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                                 60     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                61     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                62     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                                63     4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 64     4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 65     4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                                 66     4-(4'-CN-C.sub.6 H.sub.4)-Furyl-2                                       67     4-(3'-CN-C.sub.6 H.sub.4)-Furyl-2                                       68     4-(2'-CN-C.sub.6 H.sub.4)-Furyl-2                                       69     4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                        70     4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                        71     4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                        72     Thienyl-2                                                               73     5-CH.sub.3 -Thienyl-2                                                   74     5-C.sub.6 H.sub.5 -Thienyl-2                                            75     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               76     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               77     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               78     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              79     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              80     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              81     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                               82     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                               83     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                               84     5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                      85     5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                      86     5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                      87     5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                      88     5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                      89     5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                      90     4-CH.sub.3 -Thienyl-2                                                   91     4-C.sub.6 H.sub.5 -Thienyl-2                                            92     4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               93     4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               94     4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                               95     4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              96     4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              97     4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                              98     4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                               99     4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                              100     4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                              101     4-(4'-CN-C.sub.6 H.sub.4)-Thienyl-2                                    102     4-(3'-CN-C.sub.6 H.sub.4)-Thienyl-2                                    103     4-(2'-CN-C.sub.6 H.sub.4)-Thienyl-2                                    104     4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                     105     4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                     106     4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                     107     Thienyl-3                                                              108     5-CH.sub.3 -Thienyl-3                                                  109     5-C.sub.6 H.sub.5 -Thienyl-3                                           110     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                              111     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                              112     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                              113     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                             114     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                             115     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                             116     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                              117     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                              118     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                              119     5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                     120     5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                     121     5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                     122     5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                     123     5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                     124     5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                     125     Pyrazolyl-4                                                            126     NCH.sub.3 -Pyrazolyl-4                                                 127     NC.sub.6 H.sub.5 -Pyrazolyl-4                                          128     N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                            129     N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                            130     N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                            131     N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                           132     N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                           133     N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                           134     N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                            135     N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                            136     N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                            137     N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                   138     N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                   139     N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                   140     N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                   141     N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                   142     N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                   143     3-CH.sub.3 N-Methylpyrazolyl-4                                         144     3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                                  145     3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                     146     3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                     147     3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                     148     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                    149     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                    150     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                    151     3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                     152     3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                     153     3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                     154     3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                            155     3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                            156     3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                            157     3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                            158     3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                            159     3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                            160     Isoxazolyl-5                                                           161     3-CH.sub.3 -Isoxazolyl-5                                               162     3-C.sub.6 H.sub.5 -Isoxazolyl-5                                        163     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                           164     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                           165     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                           166     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                          167     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                          168     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                          169     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                           170     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                           171     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                           172     3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                  173     3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                  174     3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                  175     3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                  176     3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                  177     3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                  178     4-Chloroisoxazolyl-5                                                   179     3-CH.sub.3 -Chloroisoxazolyl-5                                         180     3-C.sub.6 H.sub.5 -Chloroisoxazolyl-5                                  181     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Chloroisoxazolyl-5                     182     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Chloroisoxazolyl-5                     183     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Chloroisoxazolyl-5                     184     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Chloroisoxazolyl-5                    185     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Chloroisoxazolyl-5                    186     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Chloroisoxazolyl-5                    187     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Chloroisoxazolyl-5                     188     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Chloroisoxazolyl-5                     189     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Chloroisoxazolyl-5                     190     3-(4'-CN-C.sub.6 H.sub.4)-Chloroisoxazolyl-5                           191     3-(3'-CN-C.sub.6 H.sub.4)-Chloroisoxazolyl-5                           192     3-(2'-CN-C.sub.6 H.sub.4)-Chloroisoxazolyl-5                           193     3-(4'-ClC.sub.6 H.sub.4)-Chloroisoxazolyl-5                            194     3-(3'-ClC.sub.6 H.sub.4)-Chloroisoxazolyl-5                            195     3-(2'-ClC.sub.6 H.sub.4)-Chloroisoxazolyl-5                            196     Isoxazolyl-3                                                           197     5-CH.sub.3 -Isoxazolyl-3                                               198     5-C.sub.6 H.sub.5 -Isoxazolyl-3                                        199     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                           200     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                           201     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                           202     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                          203     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                          204     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                          205     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                           206     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                           207     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                           208     5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                  209     5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                  210     5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                  211     5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                  212     5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                  213     5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                  214     Isothiazolyl-5                                                         215     3-CH.sub.3 -Isothiazolyl-5                                             216     3-C.sub.6 H.sub.5 -Isothiazolyl-5                                      217     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                         218     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                         219     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                         220     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                        221     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                        222     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                        223     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                         224     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                         225     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                         226     3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                                227     3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                                228     3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                                229     3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                                230     3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                                231     3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                                232     Oxazolyl-4                                                             233     3-CH.sub.3 -Oxazolyl-5                                                 234     3-C.sub.6 H.sub.5 -Oxazolyl-5                                          235     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-5                             236     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-5                             237     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-5                             238     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-5                            239     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-5                            240     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-5                            241     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-5                             242     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-5                             243     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-5                             244     3-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-5                                    245     3-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-5                                    246     3-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-5                                    247     3-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-5                                    248     3-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-5                                    249     3-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-5                                    250     Thiazolyl-4                                                            251     2-CH.sub.3 -Thiazolyl-4                                                252     2-C.sub.6 H.sub.5 -Thiazolyl-4                                         253     2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                            254     2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                            255     2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                            256     2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                           257     2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                           258     2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                           259     2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                            260     2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                            261     2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                            262     2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                   263     2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                   264     2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                   265     2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                   266     2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                   267     2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                   268     NCH.sub.3 -1,2,4-Triazolyl-5                                           269     3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                                270     3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                         271     3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            272     3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            273     3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            274     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5           275     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5           276     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5           277     3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            278     3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            279     3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5            280     3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   281     3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   282     3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   283     3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   284     3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   285     3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                   286     1,3,4-Oxadiazolyl-2                                                    287     5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                        288     5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                                 289     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    290     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    291     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    292     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   293     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   294     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                   295     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    296     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    297     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                    298     5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           299     5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           300     5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           301     5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           302     5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           303     5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                           304     1,2,4-Oxadiazolyl-3                                                    305     5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                        306     5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                                 307     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    308     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    309     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    310     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   311     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   312     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                   313     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    314     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    315     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                    316     5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           317     5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           318     5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           319     5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           320     5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           321     5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                           322     1,2,4-Oxadiazolyl-5                                                    323     3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                        324     3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                                 325     3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    326     3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    327     3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    328     3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   329     3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   330     3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                   331     3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    332     3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    333     3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                    334     3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           335     3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           336     3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           337     3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           338     3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           339     3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                           340     1,2,4-Thiadiazolyl-3                                                   341     5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                       342     5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                                343     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   344     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   345     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   346     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  347     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  248     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                  249     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   350     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   351     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                   352     5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          353     5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          354     5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          355     5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          356     5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          357     5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                          358     1,3,4-Thiadiazolyl-2                                                   359     5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                       360     5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                                361     5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   362     5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   363     5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   364     5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  365     5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  366     5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                  367     5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   368     5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   369     5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                   370     5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          371     5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          372     5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          373     5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          374     5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          375     5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                          376     Pyridinyl-2                                                            377     Pyridinyl-4                                                            378     Pyridazinyl-3                                                          379     Pyridazinyl-4                                                          380     Pyridazinyl-2                                                          381     Pyrimidinyl-4                                                          382     Pyrimidinyl-5                                                          383     Pyrimidinyl-2                                                          384     1-Naphthyl                                                             385     2-Naphthyl                                                             ______________________________________                                    

                  TABLE 45                                                         ______________________________________                                          ##STR278##                                                                    I: R.sup.1 = H, X = CH.sub.3                                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3                                 VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = Cl                                     XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       No.      T.sub.m                                                               ______________________________________                                         1        H                                                                     2        2-F                                                                   3        3-F                                                                   4        4-F                                                                   5        2,4-F.sub.2                                                           6        2,4,6-F.sub.3                                                         7        2,3,4,5,6,-F.sub.5                                                    8        2,3-F.sub.2                                                           9        2-Cl                                                                  10       3-Cl                                                                  11       4-Cl                                                                  12       2,3,-Cl.sub.2                                                         13       2,4-Cl.sub.2                                                          14       2,5-Cl.sub.2                                                          15       2,6-Cl.sub.2                                                          16       3,4-Cl.sub.2                                                          17       3,5-Cl.sub.2                                                          18       2,3,4-Cl.sub.3                                                        19       2,3,5-Cl.sub.3                                                        20       2,3,6-Cl.sub.3                                                        21       2,4,5-Cl.sub.3                                                        22       2,4,6-Cl.sub.3                                                        23       3,4,5-Cl.sub.3                                                        24       2,3,4,6-Cl.sub.4                                                      25       2,3,5,6-Cl.sub.4                                                      26       2,3,4,5,6-Cl.sub.5                                                    27       2-Br                                                                  28       3-Br                                                                  29       4-Br                                                                  30       2,4-Br.sub.2                                                          31       2,5-Br.sub.2                                                          32       2,6-Br.sub.2                                                          33       2,4,6-Br.sub.3                                                        34       2,3,4,5,6-Br.sub.5                                                    35       2-I                                                                   36       3-I                                                                   37       4-I                                                                   38       2,4-I.sub.2                                                           39       2-Cl, 3-F                                                             40       2-Cl, 4-F                                                             41       2-Cl, 5-F                                                             42       2-Cl, 6-F                                                             43       2-Cl, 3-Br                                                            44       2-Cl, 4-Br                                                            45       2-Cl, 5-Br                                                            46       2-Cl, 6-Br                                                            47       2-Br, 3-Cl                                                            48       2-Br, 4-Cl                                                            49       2-Br, 5-Cl                                                            50       2-Br, 3-F                                                             51       2-Br, 4-F                                                             52       2-Br, 5-F                                                             53       2-Br, 6-F                                                             54       2-F, 3-Cl                                                             55       2-F, 4-Cl                                                             56       2-F, 5-Cl                                                             57       3-Cl, 4-F                                                             58       3-Cl, 5-F                                                             59       3-Cl, 4-Br                                                            60       3-Cl, 5-Br                                                            61       3-F, 4-Cl                                                             62       3-F, 4-Br                                                             63       3-Br, 4-Cl                                                            64       3-Br, 4-F                                                             65       2,6-Cl.sub.2, 4-Br                                                    66       2-CH.sub.3                                                            67       3-CH.sub.3                                                            68       4-CH.sub.3                                                            69       2,3-(CH.sub.3).sub.2                                                  70       2,4-(CH.sub.3).sub.2                                                  71       2,5-(CH.sub.3).sub.2                                                  72       2,6-(CH.sub.3).sub.2                                                  73       3,4-(CH.sub.3).sub.2                                                  74       3,5-(CH.sub.3).sub.2                                                  75       2,3,5-(CH.sub.3).sub.3                                                76       2,3,4-(CH.sub.3).sub.3                                                77       2,3,6-(CH.sub.3).sub.3                                                78       2,4,5-(CH.sub.3).sub.3                                                79       2,4,6-(CH.sub.3).sub.3                                                80       3,4,5-(CH.sub.3).sub.3                                                81       2,3,4,6-(CH.sub.3).sub.4                                              82       2,3,5,6-(CH.sub.3).sub.4                                              83       2,3,4,5,6-(CH.sub.3).sub.5                                            84       2-C.sub.2 H.sub.5                                                     85       3-C.sub.2 H.sub.5                                                     86       4-C.sub.2 H.sub.5                                                     87       2,4-(C.sub.2 H.sub.5).sub.2                                           88       2,6-(C.sub.2 H.sub.5).sub.2                                           89       3,5-(C.sub.2 H.sub.5).sub.2                                           90       2,4,6-(C.sub.2 H.sub.5).sub.3                                         91       2-n-C.sub.3 H.sub.7                                                   92       3-n-C.sub.3 H.sub.7                                                   93       4-n-C.sub.3 H.sub.7                                                   94       2-i-C.sub.3 H.sub.7                                                   95       3-i-C.sub.3 H.sub.7                                                   96       4-i-C.sub.3 H.sub.7                                                   97       2,4-(i-C.sub.3 H.sub.7).sub.2                                         98       2,6-(i-C.sub.3 H.sub.7).sub.2                                         99       3,5-(i-C.sub.3 H.sub.7).sub.2                                         100      2,4,6-(i-C.sub.3 H.sub.7).sub.3                                       101      2-s-C.sub.4 H.sub.9                                                   102      3-s-C.sub.4 H.sub.9                                                   103      4-s-C.sub.4 H.sub.9                                                   104      2-t-C.sub.4 H.sub.9                                                   105      3-t-C.sub.4 H.sub.9                                                   106      4-t-C.sub.4 H.sub.9                                                   107      2,3-(t-C.sub.4 H.sub.9).sub.2                                         108      2,4-(t-C.sub.4 H.sub.9).sub.2                                         109      2,5-(t-C.sub.4 H.sub.9).sub.2                                         110      2,6-(t-C.sub.4 H.sub.9).sub.2                                         111      3,4-(t-C.sub.4 H.sub.9).sub.2                                         112      2,4,6-(t-C.sub.4 H.sub.9).sub.3                                       113      4-n-C.sub.9 H.sub.19                                                  114      4-n-C.sub.12 H.sub.25                                                 115      4-n-C.sub.15 H.sub.31                                                 116      4-(1,1,3,3-Tetramethylbutyl)                                          117      4-(2,4,4-Trimethylpropyl)                                             118      2-t-C.sub.4 H.sub.9, 4-CH.sub.3                                       119      2-t-C.sub.4 H.sub.9, 5-CH.sub.3                                       120      2,6-(t-C.sub.4 H.sub.9).sub.2, 4-CH.sub.3                             121      2-CH.sub.3, 4-t-C.sub.4 H.sub.9                                       122      2-CH.sub.3, 6-t-C.sub.4 H.sub.9                                       123      2-CH.sub.3, 4-i-C.sub.3 H.sub.7                                       124      2-CH.sub.3, 5-i-C.sub.3 H.sub.7                                       125      3-CH.sub.3, 4-i-C.sub.3 H.sub.7                                       126      2-i-C.sub.3 H.sub.7, 5-CH.sub.3                                       127      2,4-(t-C.sub.4 H.sub.9).sub.2, 6-i-C.sub.3 H.sub.7                    128      2-Allyl                                                               129      3-Allyl                                                               130      4-Allyl                                                               131      2-Allyl, 6-CH.sub.3                                                   132      2-cyclo-C.sub.6 H.sub.11                                              133      3-cyclo-C.sub.6 H.sub.11                                              134      4-cyclo-C.sub.6 H.sub.11                                              135      2,4-(cyclo-C.sub.6 H.sub.11).sub.2, 6-CH.sub.3                        136      2-CH.sub.3, 4-cyclo-C.sub.6 H.sub.11                                  137      2-CH.sub.2 C.sub.6 H.sub.5                                            138      3-CH.sub.2 C.sub.6 H.sub.5                                            139      4-CH.sub.2 C.sub.6 H.sub.5                                            140      2-CH.sub.2 C.sub.6 H.sub.5, 4-CH.sub.3                                141      2-CH.sub.3, 4-CH.sub.2 C.sub.6 H.sub.5                                142      2-C.sub.6 H.sub.5                                                     143      3-C.sub.6 H.sub.5                                                     144      4-C.sub.6 H.sub.5                                                     145      4-(2-i-C.sub.3 H.sub.7 C.sub.6 H.sub.4)                               146      4-C.sub.6 H.sub.5, 2,6-(CH.sub.3).sub.2                               147      2-Cl, 4-C.sub.6 H.sub.5                                               148      2-Br, 4-C.sub.6 H.sub.5                                               149      2-C.sub.6 H.sub.5, 4-Cl                                               150      2-C.sub.6 H.sub.5, 4-Br                                               151      2-CH.sub.2 C.sub.6 H.sub.5, 4-Cl                                      152      2-CH.sub.2 C.sub.6 H.sub.5, 4-Br                                      153      2-Cl, 4-CH.sub.2 C.sub.6 H.sub.5                                      154      2-Br, 4-CH.sub.2 C.sub.6 H.sub.5                                      155      2-cyclo-C.sub.6 H.sub.11, 4-Cl                                        156      2-cyclo-C.sub.6 H.sub.11, 4-Br                                        157      2-Cl, 4-cyclo-C.sub.6 H.sub.11                                        158      2-Br, 4-cyclo-C.sub.6 H.sub.11                                        159      2-OCH.sub.3                                                           160      3-OCH.sub.3                                                           161      4-OCH.sub.3                                                           162      2-OC.sub.2 H.sub.5                                                    163      3-OC.sub.2 H.sub.5                                                    164      4-OC.sub.2 H.sub.5                                                    165      2-O-n-C.sub.3 H.sub.7                                                 166      3-O-n-C.sub.3 H.sub.7                                                 167      4-O-n-C.sub.3 H.sub.7                                                 168      2-O-i-C.sub.3 H.sub.7                                                 169      3-O-i-C.sub.3 H.sub.7                                                 170      4-O-i-C.sub.3 H.sub.7                                                 171      2-O-n-C.sub.6 H.sub.13                                                172      3-O-n-C.sub.6 H.sub.13                                                173      4-O-n-C.sub.6 H.sub.13                                                174      2-O-n-C.sub.8 H.sub.17                                                175      3-O-n-C.sub.8 H.sub.17                                                176      4-O-n-C.sub.8 H.sub.17                                                177      2-OCH.sub.2 C.sub.6 H.sub.5                                           178      3-OCH.sub.2 C.sub.6 H.sub.5                                           179      4-OCH.sub.2 C.sub.6 H.sub.5                                           180      2-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   181      3-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   182      4-O(CH.sub.2).sub.3 C.sub.6 H.sub.5                                   183      2,4-(OCH.sub.3).sub.2                                                 184      2-CF.sub.3                                                            185      3-CF.sub.3                                                            186      4-CF.sub.3                                                            187      2-OCF.sub.3                                                           188      3-OCF.sub.3                                                           189      4-OCF.sub.3                                                           190      3-OCH.sub.2 CHF.sub.2                                                 191      2-CO.sub.2                                                            192      3-NO.sub.2                                                            193      4-NO.sub.2                                                            194      2-CN                                                                  195      3-CN                                                                  196      4-CN                                                                  197      2-CH.sub.3, 3-Cl                                                      198      2-CH.sub.3, 4-Cl                                                      199      2-CH.sub.3, 5-Cl                                                      200      2-CH.sub.3, 6-Cl                                                      201      2-CH.sub.3, 3-F                                                       202      2-CH.sub.3, 4-F                                                       203      2-CH.sub.3, 5-F                                                       204      2-CH.sub.3, 6-F                                                       205      2-CH.sub.3, 3-Br                                                      206      2-CH.sub.3, 4-Br                                                      207      2-CH.sub.3, 5-Br                                                      208      2-CH.sub.3, 6-Br                                                      209      2-Cl, 3-CH.sub.3                                                      210      2-Cl, 4-CH.sub.3                                                      211      2-Cl, 5-CH.sub.3                                                      212      2-F, 3-CH.sub.3                                                       213      2-F, 4-CH.sub.3                                                       214      2-F, 5-CH.sub.3                                                       215      2-Br, 3-CH.sub.3                                                      216      2-Br, 4-CH.sub.3                                                      217      2-Br, 5-CH.sub.3                                                      218      3-CH.sub.3, 4-Cl                                                      219      3-CH.sub.3, 5-Cl                                                      220      3-CH.sub.3, 4-F                                                       221      3-CH.sub.3, 5-F                                                       222      3-CH.sub.3, 4-Br                                                      223      3-CH.sub.3, 5-Br                                                      224      3-F, 4-CH.sub.3                                                       225      3-Cl, 4-CH.sub.3                                                      226      3-Br, 4-CH.sub.3                                                      227      2-Cl, 4,5-(CH.sub.3).sub.2                                            228      2-Br, 4,5-(CH.sub.3).sub.2                                            229      2-Cl, 3,5-(CH.sub.3).sub.2                                            230      2-Br, 3,5-(CH.sub.3).sub.2                                            231      2,6-Cl.sub.2, 4-CH.sub.3                                              232      2,6-F.sub.2, 4-CH.sub.3                                               233      2,6-Br.sub.2, 4-CH.sub.3                                              234      2,4-Br.sub.2, 6-CH.sub.3                                              235      2,4-F.sub.2, 6-CH.sub.3                                               236      2,4-Br.sub.2, 6-CH.sub.3                                              237      2,6-(CH.sub.3).sub.2, 4-F                                             238      2,6-(CH.sub.3).sub.2, 4-Cl                                            239      2,6-(CH.sub.3).sub.2, 4-Br                                            240      3,5-(CH.sub.3).sub.2, 4-F                                             241      3,5-(CH.sub.3).sub.2, 4-Cl                                            242      3,5-(CH.sub.3).sub.2, 4-Br                                            243      2,3,6-(CH.sub.3).sub.3, 4-F                                           244      2,3,6-(CH.sub.3).sub.3, 4-Cl                                          245      2,3,6-(CH.sub.3).sub.3, 4-Br                                          246      2,4-(CH.sub.3).sub.2, 6-F                                             247      2,4-(CH.sub.3).sub.2, 6-Cl                                            248      2,4-(CH.sub.3).sub.2, 6-Br                                            249      2-i-C.sub.3 H.sub.7, 4-Cl, 5-CH.sub.3                                 250      2-Cl, 4-NO.sub.2                                                      251      2-NO.sub.2, 4-Cl                                                      252      2-OCH.sub.3, 5-NO.sub.2                                               253      2,4-Cl.sub.2, 5-NO.sub.2                                              254      2,4-Cl.sub.2, 6-NO.sub.2                                              255      2,6-Cl.sub.2, 4-NO.sub.2                                              256      2,6-Br.sub.2, 4-NO.sub.2                                              257      2,6-I.sub.2, 4-NO.sub.2                                               258      2-CH.sub.3, 5-i-C.sub.3 H.sub.7, 4-Cl                                 259      2-CO.sub.2 CH.sub.3                                                   260      3-CO.sub.2 CH.sub.3                                                   261      4-CO.sub.2 CH.sub.3                                                   262      2-CO.sub.2 (C.sub.2 H.sub.5)                                          263      3-CO.sub.2 (C.sub.2 H.sub.5)                                          264      4-CO.sub.2 (C.sub.2 H.sub.5)                                          265      2-CO.sub.2 (n-C.sub.3 H.sub.7)                                        266      3-CO.sub.2 (n-C.sub.3 H.sub.7)                                        267      4-CO.sub.2 (n-C.sub.3 H.sub.7)                                        268      2-CO.sub.2 (i-C.sub.3 H.sub.7)                                        269      3-CO.sub.2 (i-C.sub.3 H.sub.7)                                        270      4-CO.sub.2 (i-C.sub.3 H.sub.7)                                        271      2-CO.sub.2 (n-C.sub.6 H.sub.13)                                       272      3-CO.sub.2 (n-C.sub.6 H.sub.13)                                       273      4-CO.sub.2 (n-C.sub.6 H.sub.13)                                       274      2-CH.sub.2 OCH.sub.3                                                  275      3-CH.sub.2 OCH.sub.3                                                  276      4-CH.sub.2 OCH.sub.3                                                  277      2-CH.sub.2 O(C.sub.2 H.sub.5)                                         278      3-CH.sub.2 O(C.sub.2 H.sub.5)                                         279      4-CH.sub.2 O(C.sub.2 H.sub.5)                                         280      2-CH.sub.2 O(n-C.sub.3 H.sub.7)                                       281      3-CH.sub.2 O(n-C.sub.3 H.sub.7)                                       282      4-CH.sub.2 O(n-C.sub.3 H.sub.7)                                       283      2-CH.sub.2 O(i-C.sub.3 H.sub.7)                                       284      3-CH.sub.2 O(i-C.sub.3 H.sub.7)                                       285      4-CH.sub.2 O(i-C.sub.3 H.sub.7)                                       286      2-CHO                                                                 287      3-CHO                                                                 288      4-CHO                                                                 289      2-COCH.sub.3                                                          290      3-COCH.sub.3                                                          291      4-COCH.sub.3                                                          292      2-COCH.sub.2 CH.sub.3                                                 293      3-COCH.sub.2 CH.sub.3                                                 294      4-COCH.sub.2 CH.sub.3                                                 295      2-COCH.sub.2 CH.sub.2 CH.sub.3                                        296      3-COCH.sub.2 CH.sub.2 CH.sub.3                                        297      4-COCH.sub.2 CH.sub.2 CH.sub.3                                        298      2-COCH(CH.sub.3)CH.sub.3                                              299      3-COCH(CH.sub.3)CH.sub.3                                              300      4-COCH(CH.sub.3)CH.sub.3                                              301      2-Me-4-CHO                                                            302      2-Me-4-CH.sub.3 CO                                                    303      2-Me-4-CH.sub.3 CH.sub.2 CO                                           304      2-Me-4-CH.sub.3 CH.sub.2 CH.sub.2 CO                                  305      2-Me-4-CH.sub.3 CH(CH.sub.3)CO                                        306      2,5-Me.sub.2 -4-CHO                                                   307      2,5-Me.sub.2 -4-CH.sub.3 CO                                           308      2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CO                                  309      2,5-Me.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                         310      2,5-Me.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                               311      2-Cl-4-CHO                                                            312      2-Cl-4-CH.sub.3 CO                                                    313      2-Cl-4-CH.sub.3 CH.sub.2 CO                                           314      2-Cl-4-CH.sub.3 CH(CH.sub.3)CO                                        315      2,5-Cl.sub.2 -4-CHO                                                   316      2,5-Cl.sub.2 -4-CH.sub.3 CO                                           317      2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CO                                  318      2,5-Cl.sub.2 -4-CH.sub.3 CH.sub.2 CH.sub.2 CO                         319      2,5-Cl.sub.2 -4-CH.sub.3 CH(CH.sub.3)CO                               320      2-C(NOCH.sub.3)CH.sub.3                                               321      3-C(NOCH.sub.3)CH.sub.3                                               322      4-C(NOCH.sub.3)CH.sub.3                                               323      2-C(NOC.sub.2 H.sub.5)CH.sub.3                                        324      3-C(NOC.sub.2 H.sub.5)CH.sub.3                                        325      4-C(NOC.sub.2 H.sub.5)CH.sub.3                                        326      2-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     327      3-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     328      4-C(NO-n-C.sub.3 H.sub.7)CH.sub.3                                     329      2-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     330      3-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     331      4-C(NO-i-C.sub.3 H.sub.7)CH.sub.3                                     332      2-C(NO-Allyl)-CH.sub.3                                                333      3-C(NO-Allyl)-CH.sub.3                                                334      4-C(NO-Allyl)-CH.sub.3                                                335      2-C(NO-trans-Chloroallyl)-CH.sub.3                                    336      3-C(NO-trans-Chloroallyl)-CH.sub.3                                    337      4-C(NO-trans-Chloroallyl)-CH.sub.3                                    338      2-C(NO-Propargyl)-CH.sub.3                                            339      3-C(NO-Propargyl)-CH.sub.3                                            340      4-C(NO-Propargyl)-CH.sub.3                                            341      2-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     342      3-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     343      4-C(NO-n-C.sub.4 H.sub.9)CH.sub.3                                     344      2-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               345      3-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               346      4-C(NOCH.sub.2 C.sub.6 H.sub.5)CH.sub.3                               347      2-CH.sub.3 -4-CHNOCH.sub.3                                            348      2-CH.sub.3 -4-CHNOC.sub.2 H.sub.5                                     349      2-CH.sub.3 -4-CHNO-n-C.sub.3 H.sub.7                                  350      2-CH.sub.3 -4-CHNO-i-C.sub.3 H.sub.7                                  351      2-CH.sub.3 -4-CHNO-Allyl                                              352      2-CH.sub.3 -4-CHNO-(trans-Chloroallyl)                                353      2-CH.sub.3 -4-CHNO-Propargyl                                          354      2-CH.sub.3 -4-CHNO-n-C.sub.4 H.sub.9                                  355      2-CH.sub.3 -4-CHNOCH.sub.2 C.sub.6 H.sub.5                            356      2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.3)                                  357      2-CH.sub.3 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                           358      2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)                        359      2-CH.sub.3 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)                        360      2-CH.sub.3 -4-(CH.sub.3 CNO-Allyl)                                    361      2-CH.sub.3 -4-(CH.sub.3 CNO-trans-Chloroallyl)                        362      2-CH.sub.3 -4-(CH.sub.3 CNO-Propargyl)                                363      2-CH.sub.3 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)                        364      2-CH.sub.3 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)                  365      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.3)                           366      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOC.sub.2 H.sub.5)                    367      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.3 H.sub.7)                 368      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-i-C.sub.3 H.sub.7                  369      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Allyl)                             370      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-trans-Chloroallyl)                 371      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-Propargyl)                         372      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNO-n-C.sub.4 H.sub.9)                 373      2-CH.sub.3 -4-(C.sub.2 H.sub.5 CNOCH.sub.2 C.sub.6 H.sub.5)           374      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.3)                        375      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOC.sub.2 H.sub.5)                 376      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.3 H.sub.7)              377      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-i-C.sub.3 H.sub.7)              378      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Allyl)                          379      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-trans-Chloroallyl)              380      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-Proparyl)                       381      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNO-n-C.sub.4 H.sub.9)              382      2,5-(CH.sub.3).sub.2 -4-(CH.sub.3 CNOCH.sub.2 C.sub.6 H.sub.5)        383      2-C.sub.6 H.sub.5                                                     384      3-C.sub.6 H.sub.5                                                     385      4-C.sub.6 H.sub.5                                                     386      2-(2'-FC.sub.6 H.sub.4)                                               387      2-(3'-FC.sub.6 H.sub.4)                                               388      2-(4'-FC.sub.6 H.sub.4)                                               389      3-(2'-FC.sub.6 H.sub.4)                                               390      3-(3'-FC.sub.6 H.sub.4)                                               391      3-(4'-FC.sub.6 H.sub.4)                                               392      4-(2'-FC.sub.6 H.sub.4)                                               393      4-(3'-FC.sub.6 H.sub.4)                                               394      4-(4'-FC.sub.6 H.sub.4)                                               395      2-(2'-ClC.sub.6 H.sub.4)                                              396      2-(3'-ClC.sub.6 H.sub.4)                                              397      2-(4'-ClC.sub.6 H.sub.4)                                              398      3-(2'-ClC.sub.6 H.sub.4)                                              399      3-(3'-ClC.sub.6 H.sub.4)                                              400      3-(4'-ClC.sub.6 H.sub.4)                                              401      4-(2'-ClC.sub.6 H.sub.4)                                              402      4-(3'-ClC.sub.6 H.sub.4)                                              403      4-(4'-ClC.sub.6 H.sub.4)                                              405      2-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       406      2-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       407      2-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       408      3-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       409      3-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       410      3-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       411      4-(2'-CH.sub.3 C.sub.6 H.sub.4)                                       412      4-(3'-CH.sub.3 C.sub.6 H.sub.4)                                       413      4-(4'-CH.sub.3 C.sub.6 H.sub.4)                                       414      2-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     415      2-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     416      2-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     417      3-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     418      3-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     419      3-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     420      4-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                     421      4-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                     422      4-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                     423      2-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          424      2-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          425      2-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          426      3-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          427      3-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          428      3-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          429      4-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          430      4-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          431      4-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                          432      2-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              433      2-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              434      2-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              435      3-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              436      3-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              437      3-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              438      4-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              439      4-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              440      4-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                              441      2-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      442      2-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      443      2-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      444      3-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      445      3-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      446      3-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      447      4-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                      448      4-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                      449      4-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                      450      2-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       451      2-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       452      2-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       453      3-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       454      3-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       455      3-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       456      4-(2'-O.sub.2 NC.sub.6 H.sub.4)                                       457      4-(3'-O.sub.2 NC.sub.6 H.sub.4)                                       458      4-(4'-O.sub.2 NC.sub.6 H.sub.4)                                       459      2-(2'-NCC.sub.6 H.sub.4)                                              460      2-(3'-NCC.sub.6 H.sub.4)                                              461      2-(4'-NCC.sub.6 H.sub.4)                                              462      3-(2'-NCC.sub.6 H.sub.4)                                              463      3-(3'-NCC.sub.6 H.sub.4)                                              464      3-(4'-NCC.sub.6 H.sub.4)                                              465      4-(2'-NCC.sub.6 H.sub.4)                                              466      4-(3'-NCC.sub.6 H.sub.4)                                              467      4-(4'-NCC.sub.6 H.sub.4)                                              468      2-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       469      2-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       470      2-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       471      3-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       472      3-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       473      3-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       474      4-(2'-CF.sub.3 C.sub.6 H.sub.4)                                       475      4-(3'-CF.sub.3 C.sub.6 H.sub.4)                                       476      4-(4'-CF.sub.3 C.sub.6 H.sub.4)                                       477      2-OC.sub.6 H.sub.5                                                    475      3-OC.sub.6 H.sub.5                                                    476      4-OC.sub.6 H.sub.5                                                    478      2-O-(2'-FC.sub.6 H.sub.4)                                             479      2-O-(3'-FC.sub.6 H.sub.4)                                             480      2-O-(4'-FC.sub.6 H.sub.4)                                             481      3-O-(2'-FC.sub.6 H.sub.4)                                             482      3-O-(3'-FC.sub.6 H.sub.4)                                             483      3-O-(4'-FC.sub.6 H.sub.4)                                             484      4-O-(2'-FC.sub.6 H.sub.4)                                             485      4-O-(3'-FC.sub.6 H.sub.4)                                             486      4-O-(4'-FC.sub.6 H.sub.4)                                             487      2-O-(2'-ClC.sub.6 H.sub.4)                                            488      2-O-(3'-ClC.sub.6 H.sub.4)                                            489      2-O-(4'-ClC.sub.6 H.sub.4)                                            490      3-O-(2'-ClC.sub.6 H.sub.4)                                            491      3-O-(3'-ClC.sub.6 H.sub.4)                                            492      3-O-(4'-ClC.sub.6 H.sub.4)                                            493      3-O-(4'-ClC.sub.6 H.sub.4)                                            494      4-O-(2'-ClC.sub.6 H.sub.4)                                            495      4-O-(3'-ClC.sub.6 H.sub.4)                                            496      4-O-(4'-ClC.sub.6 H.sub.4)                                            497      2-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     498      2-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     499      2-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     500      3-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     501      3-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     502      3-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     503      4-O-(2'-CH.sub.3 C.sub.6 H.sub.4)                                     504      4-O-(3'-CH.sub.3 C.sub.6 H.sub.4)                                     505      4-O-(4'-CH.sub.3 C.sub.6 H.sub.4)                                     506      2-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   507      2-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   508      2-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   509      3-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   510      3-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   511      3-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   512      4-O-(2'-CH.sub.3 COC.sub.6 H.sub.4)                                   513      4-O-(3'-CH.sub.3 COC.sub.6 H.sub.4)                                   514      4-O-(4'-CH.sub.3 COC.sub.6 H.sub.4)                                   515      2-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        516      2-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        517      2-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        518      3-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        519      3-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        520      3-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        521      4-O-(2'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        522      4-O-(3'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        523      4-O-(4'-(CH.sub.3 C(NOAllyl))-C.sub.6 H.sub.4)                        524      2-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            525      2-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            526      2-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            527      3-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            528      3-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            529      3-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            530      4-O-(2'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            531      4-O-(3'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            532      4-O-(4'-CH.sub.3 O.sub.2 CC.sub.6 H.sub.4)                            533      2-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    534      2-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    535      2-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    536      3-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    537      3-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    538      3-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    539      4-O-(2'-CH.sub.3 OC.sub.6 H.sub.4)                                    540      4-O-(3'-CH.sub.3 OC.sub.6 H.sub.4)                                    541      4-O-(4'-CH.sub.3 OC.sub.6 H.sub.4)                                    542      2-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     543      2-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     544      2-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     545      3-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     546      3-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     547      3-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     548      4-O-(2'-O.sub.2 NC.sub.6 H.sub.4)                                     549      4-O-(3'-O.sub.2 NC.sub.6 H.sub.4)                                     550      4-O-(4'-O.sub.2 NC.sub.6 H.sub.4)                                     551      2-O-(2'-NCC.sub.6 H.sub.4)                                            552      2-O-(3'-NCC.sub.6 H.sub.4)                                            553      2-O-(4'-NCC.sub.6 H.sub.4)                                            554      3-O-(2'-NCC.sub.6 H.sub.4)                                            555      3-O-(3'-NCC.sub.6 H.sub.4)                                            556      3-O-(4'-NCC.sub.6 H.sub.4)                                            557      4-O-(2'-NCC.sub.6 H.sub.4)                                            558      4-O-(3'-NCC.sub.6 H.sub.4)                                            559      4-O-(4'-NCC.sub.6 H.sub.4)                                            560      2-O-(2'-CF.sub.3 C.sub.6 H.sub.5)                                     561      2-O-(3'-CF.sub.3 C.sub.6 H.sub.5)                                     562      2-O-(4'-CF.sub.3 C.sub.6 H.sub.5)                                     563      3-O-(2'-CF.sub.3 C.sub.6 H.sub.5)                                     564      3-O-(3'-CF.sub.3 C.sub.6 H.sub.5)                                     565      3-O-(4'-CF.sub.3 C.sub.6 H.sub.5)                                     566      4-O-(2'-CF.sub.3 C.sub.6 H.sub.5)                                     567      4-O-(3'-CF.sub.3 C.sub.6 H.sub.5)                                     568      4-O-(4'-CF.sub.3 C.sub.6 H.sub.5)                                     569      2-Pyridinyl-2'                                                        570      2-Pyridinyl-3'                                                        571      2-Pyridinyl-4'                                                        572      3-Pyridinyl-2'                                                        573      3-Pyridinyl-3'                                                        574      3-Pyridinyl-4'                                                        575      4-Pyridinyl-2'                                                        576      4-Pyridinyl-3'                                                        577      4-Pyridinyl-4'                                                        578      2-Pyrimidinyl-2'                                                      579      2-Pyrimidinyl-3'                                                      580      2-Pyrimidinyl-4'                                                      581      3-Pyrimidinyl-2'                                                      582      3-Pyrimidinyl-3'                                                      583      3-Pyrimidinyl-4'                                                      584      4-Pyrimidinyl-2'                                                      585      4-Pyrimidinyl-3'                                                      586      4-Pyrimidinyl-4'                                                      587      2-Pyrazolyl-1'                                                        588      2-Pyrazolyl-3'                                                        589      2-Pyrazolyl-4'                                                        590      3-Pyrazolyl-1'                                                        591      3-Pyrazolyl-3'                                                        592      3-Pyrazolyl-4'                                                        593      4-Pyrazolyl-1'                                                        594      4-Pyrazolyl-3'                                                        595      4-Pyrazolyl-4'                                                        596      2-Isoxazolyl-3'                                                       597      2-Isoxazolyl-4'                                                       598      2-Isoxazolyl-5'                                                       599      3-Isoxazolyl-3'                                                       600      3-Isoxazolyl-4'                                                       601      3-Isoxazolyl-5'                                                       602      4-Isoxazolyl-3'                                                       603      4-Isoxazolyl-4'                                                       604      4-Isoxazolyl-5'                                                       605      2-Isothiazolyl-3'                                                     606      2-Isothiazolyl-4'                                                     607      2-Isothiazolyl-5'                                                     608      3-Isothiazolyl-3'                                                     609      3-Isothiazolyl-4'                                                     610      3-Isothiazolyl-5'                                                     611      4-Isothiazolyl-3'                                                     612      4-Isothiazolyl-4'                                                     613      4-Isothiazolyl-5'                                                     614      2-Imidazolyl-1'                                                       615      2-Imidazolyl-2'                                                       616      2-Imidazolyl-4'                                                       617      3-Imidazolyl-1'                                                       618      3-Imidazolyl-2'                                                       619      3-Imidazolyl-4'                                                       620      4-Imidazolyl-1'                                                       621      4-Imidazolyl-2'                                                       622      4-Imidazolyl-4'                                                       623      2-Oxazolyl-2'                                                         624      2-Oxazolyl-4'                                                         625      2-Oxazolyl-5'                                                         626      3-Oxazolyl-2'                                                         627      3-Oxazolyl-4'                                                         628      3-Oxazolyl-5'                                                         629      4-Oxazolyl-2'                                                         630      4-Oxazolyl-4'                                                         631      4-Oxazolyl-5'                                                         632      2-Thiazolyl-2'                                                        633      2-Thiazolyl-4'                                                        634      2-Thiazolyl-5'                                                        635      3-Thiazolyl-2'                                                        636      3-Thiazolyl-4'                                                        637      3-Thiazolyl-5'                                                        638      4-Thiazolyl-2'                                                        639      4-Thiazolyl-4'                                                        640      4-Thiazolyl-5'                                                        ______________________________________                                    

                  TABLE 46                                                         ______________________________________                                          ##STR279##                                                                    I: R.sup.1 = H, X = CH.sub.3                                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3                                 VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = Cl                                     XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       V: R.sup.1 =                                                                   No.       B                                                                    ______________________________________                                         1         Pyrrolyl-3                                                           2         NCH.sub.3 -Pyrrolyl-3                                                3         NC.sub.6 H.sub.5 -Pyrrolyl-3                                         4         N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           5         N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           6         N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-3                           7         N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          8         N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          9         N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-3                          10        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           11        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           12        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-3                           13        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  14        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  15        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-3                                  16        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  17        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  18        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-3                                  19        Pyrrolyl-2                                                           20        NCH.sub.3 -Pyrrolyl-2                                                21        NC.sub.6 H.sub.5 -Pyrrolyl-2                                         22        N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           23        N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           24        N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrrolyl-2                           25        N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          26        N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          27        N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrrolyl-2                          28        N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           29        N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           30        N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrrolyl-2                           31        N-(4'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  32        N-(3'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  33        N-(2'-CNC.sub.6 H.sub.4)-Pyrrolyl-2                                  34        N-(4'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  35        N-(3'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  36        N-(2'-ClC.sub.6 H.sub.4)-Pyrrolyl-2                                  37        Furyl-2                                                              38        5-CH.sub.3 -Furyl-2                                                  39        5-C.sub.6 H.sub.5 -Furyl-2                                           40        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              41        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              42        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              43        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             44        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             45        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             46        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              47        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              48        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              49        5-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     50        5-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     51        5-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     52        5-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     53        5-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     54        5-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     55        4-CH.sub.3 -Furyl-2                                                  56        4-C.sub.6 H.sub.5 -Furyl-2                                           57        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              58        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              59        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Furyl-2                              60        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             61        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             62        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Furyl-2                             63        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              64        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              65        4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Furyl-2                              66        4-(4'-CNC.sub.6 H.sub.4)-Furyl-2                                     67        4-(3'-CNC.sub.6 H.sub.4)-Furyl-2                                     68        4-(2'-CNC.sub.6 H.sub.4)-Furyl-2                                     69        4-(4'-ClC.sub.6 H.sub.4)-Furyl-2                                     70        4-(3'-ClC.sub.6 H.sub.4)-Furyl-2                                     71        4-(2'-ClC.sub.6 H.sub.4)-Furyl-2                                     72        Thienyl-2                                                            73        5-CH.sub.3 -Thienyl-2                                                74        5-C.sub.6 H.sub.5 -Thienyl-2                                         75        5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            76        5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            77        5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            78        5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           79        5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           80        5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           81        5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            82        5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            83        5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            84        5-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   85        5-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   86        5-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   87        5-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   88        5-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   89        5-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   90        4-CH.sub.3 -Thienyl-2                                                91        4-C.sub.6 H.sub.5 -Thienyl-2                                         92        4-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            93        4-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            94        4-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-2                            95        4-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           96        4-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           97        4-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-2                           98        4-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            99        4-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            100       4-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-2                            101       4-(4'-CNC.sub.6 H.sub.4)-Thienyl-2                                   102       4-(3'-CNC.sub.6 H.sub.4)-Thienyl-2                                   103       4-(2'-CNC.sub.6 H.sub.4)-Thienyl-2                                   104       4-(4'-ClC.sub.6 H.sub.4)-Thienyl-2                                   105       4-(3'-ClC.sub.6 H.sub.4)-Thienyl-2                                   106       4-(2'-ClC.sub.6 H.sub.4)-Thienyl-2                                   107       Thienyl-3                                                            108       5-CH.sub.3 -Thienyl-3                                                109       5-C.sub.6 H.sub.5 -Thienyl-3                                         110       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            111       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            112       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thienyl-3                            113       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           114       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           115       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thienyl-3                           116       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            117       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            118       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thienyl-3                            119       5-(4'-CNC.sub.6 H.sub.4)-Thienyl-3                                   120       5-(3'-CNC.sub.6 H.sub.4)-Thienyl-3                                   121       5-(2'-CNC.sub.6 H.sub.4)-Thienyl-3                                   122       5-(4'-ClC.sub.6 H.sub.4)-Thienyl-3                                   123       5-(3'-ClC.sub.6 H.sub.4)-Thienyl-3                                   124       5-(2'-ClC.sub.6 H.sub.4)-Thienyl-3                                   125       Pyrazolyl-4                                                          126       NCH.sub.3 -Pyrazolyl-4                                               127       NC.sub.6 H.sub.5 -Pyrazolyl-4                                        128       N-(4'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          129       N-(3'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          130       N-(2'-CH.sub.3 C.sub.6 H.sub.4)-Pyrazolyl-4                          131       N-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         132       N-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         133       N-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Pyrazolyl-4                         134       N-(4'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          135       N-(3'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          136       N-(2'-NO.sub.2 C.sub.6 H.sub.4)-Pyrazolyl-4                          137       N-(4'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 138       N-(3'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 139       N-(2'-CNC.sub.6 H.sub.4)-Pyrazolyl-4                                 140       N-(4'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 141       N-(3'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 142       N-(2'-ClC.sub.6 H.sub.4)-Pyrazolyl-4                                 143       3-CH.sub.3 N-Methylpyrazolyl-4                                       144       3-C.sub.6 H.sub.5 N-Methylpyrazolyl-4                                145       3-(4'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   146       3-(3'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   147       3-(2'-CH.sub.3 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   148       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  149       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  150       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)N-Methylpyrazolyl-4                  151       3-(4'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   152       3-(3'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   153       3-(2'-NO.sub.2 C.sub.6 H.sub.4)N-Methylpyrazolyl-4                   154       3-(4'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          155       3-(3'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          156       3-(2'-CNC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          157       3-(4'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          158       3-(3'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          159       3-(2'-ClC.sub.6 H.sub.4)N-Methylpyrazolyl-4                          160       Isoxazolyl-5                                                         161       3-CH.sub.3 -Isoxazolyl-5                                             162       3-C.sub.6 H.sub.5 -Isoxazolyl-5                                      163       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         164       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         165       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-5                         166       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        167       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        168       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-5                        169       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         170       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         171       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-5                         172       3-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                173       3-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                174       3-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-5                                175       3-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                176       3-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                177       3-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-5                                178       4-Chloroisoxazolyl-5                                                 179       3-CH.sub.3 -4-Chloroisoxazolyl-5                                     180       3-C.sub.6 H.sub.5 -4-Chloroisoxazolyl-5                              181       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 182       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 183       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 184       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                185       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                186       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                187       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 188       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 189       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                 190       3-(4'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        191       3-(3'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        192       3-(2'-CNC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        193       3-(4'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        194       3-(3'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        195       3-(2'-ClC.sub.6 H.sub.4)-4-Chloroisoxazolyl-5                        196       Isoxazolyl-3                                                         197       5-CH.sub.3 -Isoxazolyl-3                                             198       5-C.sub.6 H.sub.5 -Isoxazolyl-3                                      199       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         200       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         201       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isoxazolyl-3                         202       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        203       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        204       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isoxazolyl-3                        205       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         206       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         207       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isoxazolyl-3                         208       5-(4'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                209       5-(3'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                210       5-(2'-CNC.sub.6 H.sub.4)-Isoxazolyl-3                                211       5-(4'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                212       5-(3'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                213       5-(2'-ClC.sub.6 H.sub.4)-Isoxazolyl-3                                214       Isothiazolyl-5                                                       215       3-CH.sub.3 -Isothiazolyl-5                                           216       3-C.sub.6 H.sub.5 -Isothiazolyl-5                                    217       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       218       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       219       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-Isothiazolyl-5                       220       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      221       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      222       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Isothiazolyl-5                      223       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       224       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       225       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-Isothiazolyl-5                       226       3-(4'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              227       3-(3'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              228       3-(2'-CNC.sub.6 H.sub.4)-Isothiazolyl-5                              229       3-(4'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              230       3-(3'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              231       3-(2'-ClC.sub.6 H.sub.4)-Isothiazolyl-5                              232       Oxazolyl-4                                                           233       2-CH.sub.3 -Oxazolyl-4                                               234       2-C.sub.6 H.sub.5 -Oxazolyl-4                                        235       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           236       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           237       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Oxazolyl-4                           238       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          239       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          240       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Oxazolyl-4                          241       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           242       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           243       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Oxazolyl-4                           244       2-(4'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  245       2-(3'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  246       2-(2'-CNC.sub.6 H.sub.4)-Oxazolyl-4                                  247       2-(4'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  248       2-(3'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  249       2-(2'-ClC.sub.6 H.sub.4)-Oxazolyl-4                                  250       Thiazolyl-4                                                          251       2-CH.sub.3 -Thiazolyl-4                                              252       2-C.sub.6 H.sub.5 -Thiazolyl-4                                       253       2-(4'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          254       2-(3'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          255       2-(2'-CH.sub.3 C.sub.6 H.sub.4)-Thiazolyl-4                          256       2-(4'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         267       2-(3'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         258       2-(2'-CH.sub.3 OC.sub.6 H.sub.4)-Thiazolyl-4                         259       2-(4'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          260       2-(3'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          261       2-(2'-NO.sub.2 C.sub.6 H.sub.4)-Thiazolyl-4                          262       2-(4'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 263       2-(3'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 264       2-(2'-CNC.sub.6 H.sub.4)-Thiazolyl-4                                 265       2-(4'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 266       2-(3'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 267       2-(2'-ClC.sub.6 H.sub.4)-Thiazolyl-4                                 268       NCH.sub.3 -1,2,4-Triazolyl-5                                         269       3-CH.sub.3 NCH.sub.3 -1,2,4-Triazolyl-5                              270       3-C.sub.6 H.sub.5 NCH.sub.3 -1,2,4-Triazolyl-5                       271       3-(4'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          272       3-(3'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          273       3-(2'-CH.sub.3 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          274       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         275       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         276       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5         277       3-(4'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          278       3-(3'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          279       3-(2'-NO.sub.2 C.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5          280       3-(4'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 281       3-(3'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 282       3-(2'-CNC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 283       3-(4'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 284       3-(3'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 285       3-(2'-ClC.sub.6 H.sub.4)NCH.sub.3 -1,2,4-Triazolyl-5                 286       1,3,4-Oxadiazolyl-2                                                  287       5-CH.sub.3 -1,3,4-Oxadiazolyl-2                                      288       5-C.sub.6 H.sub.5 -1,3,4-Oxadiazolyl-2                               289       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  290       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  291       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  292       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 293       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 294       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                 295       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  296       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  297       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                  298       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         299       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         300       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         301       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         302       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         303       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Oxadiazolyl-2                         304       1,2,4-Oxadiazolyl-3                                                  305       5-CH.sub.3 -1,2,4-Oxadiazolyl-3                                      306       5-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-3                               307       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  308       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  309       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  310       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 311       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 312       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                 313       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  314       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  315       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                  316       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         317       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         318       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         319       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         320       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         321       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-3                         322       1,2,4-Oxadiazolyl-5                                                  323       3-CH.sub.3 -1,2,4-Oxadiazolyl-5                                      324       3-C.sub.6 H.sub.5 -1,2,4-Oxadiazolyl-5                               325       3-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  326       3-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  327       3-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  328       3-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 329       3-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 330       3-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                 331       3-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  332       3-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  333       3-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                  334       3-(4'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         335       3-(3'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         336       3-(2'-CNC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         337       3-(4'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         338       3-(3'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         339       3-(2'-ClC.sub.6 H.sub.4)-1,2,4-Oxadiazolyl-5                         340       1,2,4-Thiadiazolyl-3                                                 341       5-CH.sub.3 -1,2,4-Thiadiazolyl-3                                     342       5-C.sub.6 H.sub.5 -1,2,4-Thiadiazolyl-3                              343       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 344       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 345       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 346       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                347       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                348       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                349       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 350       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 351       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                 352       5-(4'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        353       5-(3'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        354       5-(2'-CNC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        355       5-(4'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        356       5-(3'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        357       5-(2'-ClC.sub.6 H.sub.4)-1,2,4-Thiadiazolyl-3                        358       1,3,4-Thiadiazolyl-2                                                 359       5-CH.sub.3 -1,3,4-Thiadiazolyl-2                                     360       5-C.sub.6 H.sub.5 -1,3,4-Thiadiazolyl-2                              361       5-(4'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 362       5-(3'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 363       5-(2'-CH.sub.3 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 364       5-(4'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                365       5-(3'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                366       5-(2'-CH.sub.3 OC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                367       5-(4'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 368       5-(3'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 369       5-(2'-NO.sub.2 C.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                 370       5-(4'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        371       5-(3'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        372       5-(2'-CNC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        373       5-(4'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        374       5-(3'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        375       5-(2'-ClC.sub.6 H.sub.4)-1,3,4-Thiadiazolyl-2                        376       Pyridinyl-2                                                          377       Pyridinyl-4                                                          378       Pyridazinyl-3                                                        379       Pyridazinyl-4                                                        380       Pyridazinyl-2                                                        381       Pyrimidinyl-4                                                        382       Pyrimidinyl-5                                                        383       Pyrimidinyl-2                                                        ______________________________________                                    

                  TABLE 47                                                         ______________________________________                                         Selected physical data of some compounds                                        ##STR280##                                                                                              IR (cm.sup.-1) or                                    No.  X.sub.m   R.sup.1    .sup.1 h-NMR (ppm)                                                                           mp                                     ______________________________________                                         1    4-Cl      H                        133                                    2    3,4-Cl.sub.2                                                                             H                        109                                    3    4-t-C.sub.4 H.sub.9                                                                      H                         86                                    4    4-CH.sub.3                                                                               H                        117                                    5    4-CF.sub.3                                                                               H                        103                                    6    3-Br      H                         99                                    7    3-Cl      H                         93                                    8    3-CF.sub.3                                                                               H                         88                                    9    3,5-Cl.sub.2                                                                             H                        100                                    10   3,4-(CH.sub.3).sub.2                                                                     H                        127                                    11   3,4-Cl.sub.2                                                                             CH.sub.3                  74                                    12   3,4-Cl.sub.2                                                                             Allyl      3.65(S, 3H); 2.2(S, 6H)                              13   3,4-Cl.sub.2                                                                             Propargyl  3.65(S, 3H); 2.3(S, 3H);                                                       2.2(S, 3H)                                           14   3,4-Cl.sub.2                                                                             CH.sub.2 OCH.sub.3                                                                        3.65(S, 3H); 2.3(S, 3H);                                                       2.2(S, 3H)                                           15   3,4-Cl.sub.2                                                                             COOCH.sub.3              137                                    16   4-t-C.sub.4 H.sub.9                                                                      CH.sub.3   3.65(S, 3H); 2.25(S, 3H);                                                      2.2(S, 3H)                                           17   4-t-C.sub.4 H.sub.9                                                                      Allyl                     69                                    18   4-t-C.sub.4 H.sub.9                                                                      Propargyl                117                                    19   4-t-C.sub.4 H.sub.9                                                                      CH.sub.2 OCH.sub.3                                                                        3.65(S, 3H); 2.25(S, 3H);                                                                    117                                                              2.2(S, 3H)                                           20   4-t-C.sub.4 H.sub.9                                                                      COOCH.sub.3                                                                               3.65, 2.1     119                                    21   4-CH.sub.3                                                                               CH.sub.3                  69                                    22   4-CH.sub.3                                                                               Allyl      3.65(S, 3H); 2.25(S, 3H);                                                      2.2(S, 3H)                                           23   4-CH.sub.3                                                                               Propargyl  3.65(S, 3H); 2.3(S, 3H);                                                       2.2(S, 3H)                                           24   4-CH.sub.3                                                                               CH.sub.2 OCH.sub.3                                                                        3.65(S, 3H); 2.3(S, 3H);                                                       2.2(S, 3H)                                           25   4-CH.sub.3                                                                               COOCH.sub.3               97                                    26   4-CF.sub.3                                                                               CH.sub.3                  76                                    27   4-CF.sub.3                                                                               Allyl      3.65(S, 3H); 2.3(S, 3H);                                                       2.25(S, 3H)                                          28   4-CF.sub.3                                                                               Propargyl  3.65(S, 3H); 2.3(S, 3H);                                                       2.25(S, 3H)                                          29   4-CF.sub.3                                                                               CH.sub.2 OCH.sub.3                                                                        3.65(S, 3H); 2.25(S, 3H);                            30   4-CF.sub.3                                                                               COOCH.sub.3              103                                    31   4-Cl      CH.sub.3                 106                                    32   4-Cl      Allyl      3.65(S, 3H); 2.2(2S,                                                           each 3H)                                             33   4-Cl      Propargyl  3.65(S, 3H); 2.3(S, 3H);                                                       2.2(S, 3H)                                           34   4-Cl      CH.sub.2 OCH.sub.3                                                                        3.65(S, 3H); 2.25(S, 3H);                                                      2.2(S, 3H)                                           35   4-Cl      COOCH.sub.3              109                                    36   3-Br      CH.sub.3                  75                                    37   3-Br      Allyl      3.65(S, 3H); 2.2(2S,                                                           each 3H                                              38   3-Br      Propargyl  3.65(S, 3H); 2.3(S, 3H);                                                       2.2(S, 3H)                                           39   3-Br      CH.sub.2 OCH.sub.3        72                                    40   3-Br      COOCH.sub.3              131                                    41   3-Cl      CH.sub.3                  84                                    42   3-Cl      Allyl      3.65(S, 3H); 2.25(S, 3H);                                                      2.2(S, 3H)                                           43   3-Cl      Propargyl  3.65(S, 3H); 2.3(S, 3H);                                                       2.2(S, 3H)                                           44   3-Cl      CH.sub.2 OCH.sub.3        66                                    45   3-Cl      COOCH.sub.3              123                                    46   3-CF.sub.3                                                                               CH.sub.3                  63                                    47   3-CF.sub.3                                                                               Allyl                     64                                    48   3-CF.sub.3                                                                               Propargyl  3.65(S, 3H); 2.3(S, 3H);                                                       2.25(S, 3H)                                          49   3-CF.sub.3                                                                               CH.sub.2 OCH.sub.3        89                                    50   3-CF.sub.3                                                                               COOCH.sub.3              136                                    51   4-Br      COOCH.sub.3              103                                    52   4-Br      H                        108                                    53   4-Br      Propargyl  1710,1486,1469,1447,1376,                                                      1299,1252,1026,1008,774                              54   4-Br      CH.sub.2 OCH.sub.3                                                                        1715,1468,1445,1370,1301,                                                      1274,1090,1059,1008,775                              55   3,4-(CH.sub.3).sub.2                                                                     CH.sub.3                 oil                                    56   3,4-(CH.sub.3).sub.2                                                                     Allyl                    oil                                    57   3,4-(CH.sub.3).sub.2                                                                     Propargyl                oil                                    58   3,4-(CH.sub.3).sub.2                                                                     CH.sub.2 OCH.sub.3       oil                                    59   3,4-(CH.sub.3).sub.2                                                                     COOCH.sub.3              135                                    60   3,5-Cl.sub.2                                                                             CH.sub.3                  95                                    61   3,5-Cl.sub.2                                                                             Allyl                     97                                    62   3,5-Cl.sub.2                                                                             Propargyl                100                                    63   3,5-Cl.sub.2                                                                             CH.sub.2 OCH.sub.3       112                                    64   3,5-Cl.sub.2                                                                             COOCH.sub.3              160                                    ______________________________________                                    

                                      TABLE 48                                     __________________________________________________________________________     Selected physical data of some compounds                                        ##STR281##                                                                                              IR (cm.sup.-1) or                                    No.                                                                               X.sub.m         R.sup.1                                                                               .sup.1 h-NMR (ppm)                                                                           mp                                     __________________________________________________________________________     1  2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                            H                     82                                    2  2,4-(CH.sub.3).sub.2                                                                           H                    131                                    3  2,5-(CH.sub.3).sub.2                                                                           H                    124                                    4  2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                                     H                    102                                    5  2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                           H                    116                                    6  2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                            H                    122                                    7  2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                            CH.sub.3                                                                              4.0(S, 3H); 3.65(S, 3H)                              8  2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                            Allyl                101                                    9  2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                            Propargyl                                                                             4.0(S, 3H); 3.65(S, 3H)                              10 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                            CH.sub.2 OCH.sub.3                                                                    4.0(S, 3H); 3.65(S, 3H)                              11 2-CH.sub.3 -4-C(CH.sub.3)NOCH.sub.3                                                            COOCH.sub.3          122                                    12 2,4-(CH.sub.3).sub.2                                                                           CH.sub.3                                                                              3.65(S, 3H); 2.25(2s, each 3H)                       13 2,4-(CH.sub.3).sub.2                                                                           Allyl                 59                                    14 2,4-(CH.sub.3).sub.2                                                                           Propargyl                                                                             3.65(S, 3H); 2.25(3s, each 3H)                       15 2,4-(CH.sub.3).sub.2                                                                           CH.sub.2 OCH.sub.3    76                                    16 2,4-(CH.sub.3).sub.2                                                                           COOCH.sub.3          133                                    17 2,5-(CH.sub.3).sub.2                                                                           CH.sub.3                                                                              3.65(S, 3H); 2.3(S, 3H)                              18 2,5-(CH.sub.3).sub.2                                                                           Allyl                 56                                    19 2,5-(CH.sub.3).sub.2                                                                           Propargyl             80                                    20 2,5-(CH.sub.3).sub.2                                                                           CH.sub.2 OCH.sub.3                                                                    3.65(S, 3H); 2.3(S, 3H)                                                                       80                                    21 2,5-(CH.sub.3).sub.2                                                                           CH.sub.2 OCH.sub.3   140                                    22 2-CH.sub.3      H                    107                                    23 2-CH.sub.3      Propargyl            oil                                    24 2-CH.sub.3      COOCH.sub.3          135                                    25 2-CH.sub.3      CH.sub.2 OCH.sub.3   oil                                    26 2-CH.sub.3 -4-C(CH.sub.3)NO-Allyl                                                              H                     97                                    27 2-CH.sub.3 -4-C(CH.sub.3)NO-Allyl                                                              Propargyl            oil                                    28 2-CH.sub.3 -4-C(CH.sub.3)NO-Allyl                                                              COOCH.sub.3          130                                    29 2-CH.sub.3 -4-C(CH.sub.3)NO-Allyl                                                              HC.sub.2 OCH.sub.3   oil                                    30 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                                     CH.sub.3             oil                                    31 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                                     Allyl                 75                                    32 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                                     Propargyl             77                                    33 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                                     CH.sub.2 OCH.sub.3   oil                                    34 2-CH.sub.3 -4-C(CH.sub.3)NOC.sub.2 H.sub.5                                                     COOCH.sub.3          oil                                    35 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3                                                           CH.sub.3             oil                                    36 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3                                                           Allyl                104                                    37 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3                                                           Propargyl            oil                                    38 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3                                                           CH.sub.2 OCH.sub.3   oil                                    39 2-CH.sub.3 -4-C(CH.sub.3)NOOCH.sub.3                                                           COOCH.sub.3          158                                    40 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5                                                    CH.sub.3             oil                                    41 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5                                                    Allyl                 71                                    42 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5                                                    Propargyl            oil                                    43 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5                                                    CH.sub.2 OCH.sub.3   oil                                    44 2-CH.sub.3 -4-C(CH.sub.3)NOOC.sub.2 H.sub.5                                                    COOCH.sub.3          128                                    __________________________________________________________________________

                  TABLE 49                                                         ______________________________________                                          ##STR282##                                                                    I: R.sup.1 = H, X = CH.sub.3                                                   II: R.sup.1 = CH.sub.3, X = CH.sub.3                                           III: R.sup.1 = C.sub.2 H.sub.5, X = CH.sub.3                                   IV: R.sup.1 = Allyl, X = CH.sub.3                                              V: R.sup.1 = Propargyl, X = CH.sub.3                                           VI: R.sup.1 = CH.sub.2 OCH.sub.3, X = CH.sub.3                                 VII: R.sup.1 = CO.sub.2 CH.sub.3, X = CH.sub.3                                 VIII: R.sup.1 = H, X = Cl                                                      IX: R.sup.1 = CH.sub.3, X = Cl                                                 X: R.sup.1 = C.sub.2 H.sub.5, X = Cl                                           XI: R.sup.1 = Allyl, X = Cl                                                    XII: R.sup.1 = Propargyl, X = Cl                                               XIII: R.sup.1 = CH.sub.2 OCH.sub.3, X = Cl                                     XIV: R.sup.1 = CO.sub.2 CH.sub.3, X = Cl                                       No.     B                                                                      ______________________________________                                         1       2-Pyridyl                                                              2       3-Trifluoromethyl-2-pyridyl                                            3       5-Trifluoromethyl-2-pyridyl                                            4       3,5-Bis-(trifluoromethyl-2-pyridyl                                     5       3,5-Dichloro-2-pyridyl                                                 6       3-Chloro-5-trifluoromethyl-2-pyridyl                                   7       3,5-Dichloro-2-pyridyl                                                 8       2-Chloro-4-trifluoromethylphenyl                                       9       2-Benzothiazolyl                                                       10      5-Chloro-1-methyl-2-benzimidazolyl                                     11      2-Benzoxazolyl                                                         12      1-Methyl-5-trifluoromethylimide-azo 5,4-a!-pyridin-2-yl                13      5-Chloro-2-pyrimidinyl                                                 14      4-Methyl-5-phenyl-2-thiazolin-2-yl                                     15      4-Methyl-5-phenyl-2-oxazolin-2-yl                                      16      7-Trifluoromethyl-4-quinolinyl                                         ______________________________________                                    

                  TABLE 50                                                         ______________________________________                                         Selected physical data of some compounds                                        ##STR283##                                                                    No.    X.sub.m     IR (cm.sup.-1) or .sup.1 H-NMR (ppm)                                                            mp                                         ______________________________________                                         1      4-NO.sub.2                   112                                        2      3,4-Cl.sub.2                                                                               3.8(s, 3H); 3.75(s, 3H)                                     3      2,4-(CH.sub.3).sub.2                                                                       3.75(s, 3H); 3.7(s, 3H)                                     4      H           3.75(2s, each 3H)                                           5      4-i-C.sub.3 H.sub.7                                                                        3.8(s, 3H); 3.75(s, 3H)                                     6      3,4-(CH.sub.3).sub.2                                                                       3.8(s, 3H); 3.75(s, 3H)                                     7      3-CH.sub.3 -4-OCH.sub.3                                                                    3.85(s, 3H); 3.8(s, 3H);                                                       3.75(s, 3H)                                                 8      3-CH.sub.3 -4-O-                                                                           3.8(2s, each 3H)                                                   I-C.sub.3 H.sub.7                                                       9      4-CF.sub.3  3.8(s, 3H); 3.75(s, 3H)                                     10     3-CH.sub.3  3.8(2s, each 3H)                                            11     3-CF.sub.3  3.8(s, 3H); 3.75(s, 3H)                                     12     4-F         3.8(s, 3H); 3.75(s, 3H)                                     13     4-Br        3.8(s, 3H); 3.75(s, 3H)                                     14     3-Br        3.8(s, 3H); 3.75(s, 3H)                                     15     4-t-Bu      3.8(s, 3H); 3.75(s, 3H)                                     16     4-OCH.sub.3 3.85(s, 3H); 3.8(s, 3H);                                                       3.75(s, 3H)                                                 17     2-CH.sub.3  3.8(s, 3H); 3.75(s, 3H)                                     18     3-Cl        3.8(s, 3H); 3.75(s, 3H)                                     19     4-CN        3.8(s, 3H); 3.75(s, 3H)                                     20     4-C.sub.2 H.sub.5                                                                          3.8(s, 3H); 3.75(s, 3H)                                     ______________________________________                                    

                  TABLE 51                                                         ______________________________________                                         Selected physical data of some comounds                                         ##STR284##                                                                    No.   X.sub.m         IR (cm.sup.-1) or .sup.1 H-NMR (ppm)                                                           mp                                       ______________________________________                                         1     4-Cl            3.8(s, 3H); 3.75(s, 3H)                                  2     2-Cl            3.8(s, 3H); 3.75(s, 3H)                                  3     2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)                                                     3.8(s, 3H); 3.75(s, 3H)                                        N-Allyl                                                                  4     2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)                                                     3.9(s, 3H); 3.8(s, 3H);                                        NOCH.sub.3      3.75(s, 3H)                                              5     2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NO-                                                            3.8(s, 3H); 3.75(s, 3H)                                        trans-Cl-Allyl                                                           6     2-CH.sub.3 -4-C(C.sub.2 H.sub.5)NO-                                                            3.8(s, 3H); 3.75(s, 3H)                                        Allyl                                                                    7     2-CH.sub.3 -4-Cl                                                                               3.8(s, 3H); 3.75(s, 3H)                                  8     2-Cl-4-CH.sub.3 3.8(s, 3H); 3.75(s, 3H)                                  9     2-Cl-5-CH.sub.3 3.8(s, 3H); 3.75(s, 3H)                                  10    2-CH.sub.3 -4-C(C.sub.2 H.sub.5)N                                                              4.2(z, 2H); 3.8(s, 3H);                                        OC.sub.2 H.sub.5                                                                               3.75(s, 3H)                                              11    2-CH.sub.3 -4-C(C.sub.2 H.sub.5)N                                                              3.95(s, 3H); 3.8(s, 3H);                                       OCH.sub.3       3.75(s, 3H)                                              12    2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)                                                            3.8(s, 3H); 3.75(s, 3H)                                        NO-trans-Cl-Allyl                                                        13    2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)                                                            4.2(t, 2H); 3.8(s, 3H);                                        NOC.sub.2 H.sub.5                                                                              3.75(s, 3H)                                              14    2,5-(CH.sub.3).sub.2 -4-C(CH.sub.3)                                                            3.95(s, 3H); 3.8(s, 3H);                                       NOCH.sub.3      3.75(s, 3H)                                              15    2-CH.sub.3 -4-C(CH.sub.3)NO-                                                                   3.8(s, 3H); 3.75(s, 3H)                                        trans-Cl-Allyl                                                           16    2-CH.sub.3 -4-C(CH.sub.3)N-                                                                    4.2(t, 2H); 3.8(s, 3H);                                        OC.sub.2 H.sub.5                                                                               3.75(s, 3H)                                              17    2,5-(CH.sub.3).sub.2 -4-C(C.sub.2 H.sub.5)                                                     4.2(t, 2H); 3.8(s, 3H);                                        NOC.sub.2 H.sub.5                                                                              3.75(s, 3H)                                              ______________________________________                                    

                  TABLE 60                                                         ______________________________________                                          ##STR285##                                                                    No.         B                                                                  ______________________________________                                         1           Phenyl                                                             2           3-Phenoxyphenyl                                                    3           3-(2-Cyanophenoxy)-phenyl                                          4           4-Chlorophenyl                                                     5           3-Trifluoromethylphenyl                                            6           3-tert.-Butoxyphenyl                                               7           3,5-Dichlorophenyl                                                 8           3,5-Diethylphenyl                                                  9           2-Pyridyl                                                          10          4-Pyrimidinyl                                                      11          6-Phenoxy-pyrimidin-4-yl                                           12          6-Chloropyrimidin-4-yl                                             13          6-(2-Fluorophenoxy)-pyrimidin-4-yl                                 14          6-(2-Methylphenoxy)-pyrimidin-4-yl                                 15          6-(2-Cyanophenoxy)-pyrimdin-4-yl                                   16          6-(2,6-Difluorophenoxy)-pyrimidin-4-yl                             ______________________________________                                    

The novel compounds are suitable as fungicides.

The fungicidal compounds according to the invention, or agents containing them, may be applied for instance in the form of directly sprayable solutions, powders, suspensions (including high-percentage aqueous, oily or other suspen- sions), dispersions, emulsions, oil dispersions, pastes, dusts, broadcasting agents, or granules by spraying, atomizing, d usting, broadcasting or watering. The forms of application depend entirely on the purpose for which the agents are being used, but they must ensure as fine a distribution of the active ingredients according to the invention as possible. Normally, the plants are sprayed or dusted with the active ingredients, or the seeds of the plants are treated with the active ingredients.

The formulations are produced in known manner, for example by extending the active ingredient with solvents and/or carriers, with or without the use of emulsifiers and dispersants; if water is used as solvent, it is also possible to employ other organic solvents as auxiliary solvents. Suitable auxiliaries for this purpose are solvents such as aromatics (e.g., xylene), chlorinated aromatics (e.g., chlorobenzenes), paraffins (e.g., crude oil fractions), alcohols (e.g., methanol, butanol), ketones (e.g., cyclohexanone), amines (e.g., ethanolamine, dimethylformamide), and water; carriers such as ground natural minerals (e.g., kaolins, aluminas, talc and chalk) and ground synthetic minerals (e.g., highly disperse silica and silicates); emulsifiers such as nonionic and anionic emulsifiers (e.g., polyoxyethylene fatty alcohol ethers, alkyl sulfonates and aryl sulfonates); and dispersants such as lignin-sulfite waste liquors and methylcellulose.

Examples of surfactants are: alkali metal, alkaline earth metal and ammonium salts of aromatic sulfonic acids, e.g., ligninsulfonic acid, phenolsulfonic acid, naphthalenesulfonic acid and dibutylnaphthalenesulfonic acid, and of fatty acids, alkyl and alkylaryl sulfonates, and alkyl, lauryl ether and fatty alcohol sulfates, and salts of sulfated hexadecanols, heptadecanols, and octadecanols, salts of fatty alcohol glycol ethers, condensation products of sulfonated naphthalene and naphthalene derivatives with formaldehyde, condensation products of naphthalene or naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ethers, ethoxylated isooctylphenol, ethoxylated octylphenol and ethoxylated nonylphenol, alkylphenol polyglycol ethers, tributylphenyl polyglycol ethers, alkylaryl polyether alcohols, isotridecyl alcohol, fatty alcohol ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers, ethoxylated polyoxypropylene, lauryl alcohol polyglycol ether acetal, sorbitol esters, lignin-sulfite waste liquors and methyl cellulose.

Powders, dusts and broadcasting agents may be prepared by mixing or grinding the active ingredients with a solid carrier.

Granules, e.g., coated, impregnated or homogeneous granules, may be prepared by bonding the active ingredients to solid carriers. Examples of solid carriers are mineral earths such as silicic acids, silica gels, silicates, talc, kaolin, attapulgus clay, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground plastics, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate, and ureas, and vegetable products such as grain meals, bark meal, wood meal, and nutshell meal, cellulosic powders, etc.

Examples of formulations are given below.

I. A solution of 90 parts by weight of the compound from Table 7, No. 1 (7/1) and 10 parts by weight of N-methyl-α-pyrrolidone, which is suitable for application in the form of very fine drops.

II. A mixture of 20 parts by weight of compound 7/2, 80 parts by weight of xylene, 10 parts by weight of the adduct of 8 to 10 moles of ethylene oxide and 1 mole of oleic acid-N-monoethanolamide, 5 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, and 5 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil. By finely dispersing the mixture in water, a dispersion is obtained.

III. An aqueous dispersion of 20 parts by weight of compound 7/3, 40 parts by weight of cyclohexanone, 30 parts by weight of isobutanol, 20 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil.

IV. An aqueous dispersion of 20 parts by weight of compound 7/4, 25 parts by weight of cyclohexanol, 65 parts by weight of a mineral oil fraction having a boiling point between 210° and 280° C., and 10 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil.

V. A hammer-milled mixture of 80 parts by weight of compound 7/5, 3 parts by weight of the sodium salt of diisobutylnaphthalene-α-sulfonic acid, 10 parts by weight of the sodium salt of a lignin-sulfonic acid obtained from a sulfite waste liquor, and 7 parts by weight of powdered silica gel. By finely dispersing the mixture in water, a spray liquor is obtained.

VI. An intimate mixture of 3 parts by weight of compound 7/6 and 97 parts by weight of particulate kaolin. The dust contains 3wt % of the active ingredient.

VII. An intimate mixture of 30 parts by weight of compound 7/7, 92 parts by weight of powdered silica gel and 8 parts by weight of paraffin oil sprayed onto the surface of this silica gel. This formulation of the active ingredient exhibits good adherence.

VIII. A stable aqueous dispersion of 40 parts by weight of compound 7/8, 10 parts of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate, 2 parts of silica gel and 48 parts of water, which dispersion can be further diluted.

IX. A stable oily dispersion of 20 parts by weight of compound 7/9, 2 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, 8 parts by weight of a fatty alcohol polyglycol ether, 2 parts by weight of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate and 68 parts by weight of a paraffinic mineral oil.

The novel compounds are extremely effective on a broad spectrum of phytopathogenic fungi, in particular those from the class consisting of the Ascomycetes and Basidiomycetes. Some of them have a systemic action and can be used as foliar and soil fungicides.

The fungicidal compounds are of particular interest for controlling a large number of fungi in various crops or their seeds, especially wheat, rye, barley, oats, rice, Indian corn, lawns, cotton, soybeans, coffee, sugar cane, fruit and ornamentals in horticulture and viticulture, and in vegetables such as cucumbers, beans and cucurbits.

The compounds are applied by treating the fungi, or the seeds, plants, materials or soil to be protected against fungus attack with a fungicidally effective amount of the active ingredients.

The agents may be applied before or after infection of the materials, plants or seed by the fungi.

The compounds I are particularly useful for controlling the following plant diseases:

Erysiphe graminis in cereals,

Erysiphe cichoracearum and Sphaerotheca fuliginea in cucurbits,

Podosphaera leucotricha in apples,

Uncinula necator in vines,

Puccinia species in cereals,

Rhizoctonia solani in cotton,

Ustilago species in cereals and sugar cane,

Venturia inaequalis (scab) in apples,

Helminthosporium species in cereals,

Septoria nodorum in wheat,

Botrytis cinerea (gray mold) in strawberries and grapes,

Cercospora arachidicola in groundnuts,

Pseudocercosporella herpotrichoides in wheat and barley,

Pyricularia oryzae in rice,

Phytophthora infestans in potatoes and tomatoes,

Fusarium and Verticillium species in various plants,

Plasmopara viticola in grapes,

Alternaria species in fruit and vegetables.

The novel compounds may also be used for protecting materials (timber), for instance against Paecilomyces variotii.

The fungicidal agents generally contain from 0.1 to 95, an preferably from 0.5 to 90, wt % of active ingredient.

The application rates depend on the effect desired, and are from 0.02 to 3 kg of active ingredient per hectare.

When the active ingredients are used for treating seed, amounts of from 0.001 to 50, and preferably from 0.01 to 10, g per kg of seed are generally needed.

When the agents according to the invention are used as fungicides, they may be present together with other active ingredients, e.g., herbicides, insecticides, growth regulators, other fungicides, and fertilizers.

When they are mixed with other fungicides, the spectrum of fungicidal action is in many cases increased.

USE EXAMPLES

The active ingredients used for comparison purposes were isopropyl N-phenylcarbamate (A)--known from GB 574 995--, isopropyl N-3-chlorophenylcarbamate (B)--known from GB 574 995 --and methyl N-3,4-dichlorophenylcarbamate (C)--known from BE 612 550.

Example 1

Action on wheat mildew

Leaves of pot-grown wheat seedlings of the "Fruhgold" variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20° to 22° C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredients nos. 1, 2, 3, 4, 8, 9, 20, 23, 31, 33, 34, 35, 36, 42, 43, 44, 47, 48, 52, 53, 54, 55, 56, 57, 60, 61, 62, 63, 64, 67, 69, 70, 71, 72, 74, 78, 79, 85, 87, 89, 90, 91, 92, 93, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art comparative agents A (45%), B (45%) and C (45%).

Example 2

Action on Pyricularia oryzae (protective)

Leaves of pot-grown rice seedlings of the "Bahia" variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22° to 24° C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredients nos. 1, 2, 12, 18, 19, 22, 29, 39, 40, 42, 47, 49, 50, 52, 53, 54, 60, 61, 62, 63, 69, 70, 71, 72, 73, 74, 81, 83, 85, 87, 89, 90, 91, 92, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art comparative agents A (30%), B (30%) and C (30%).

Example 3

Action on wheat mildew

Leaves of pot-grown wheat seedlings of the "Fruhgold" variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20° to 22° C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredient no. 3 from Table 14, nos. 3 and 4 from Table 21, nos. 1, 3, 4, 5, 6, 7, 8, 9, 10, 11, 15, 17, 18, 19, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40 41, 42, 43 and 44 from Table 48, nos. 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20 and 23 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18 and 19 from Table 52, and nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (15%).

Example 4

Action on Pyricularia oryzae (protective)

Leaves of pot-grown rice seedlings of the "Bahia" variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22° to 24° C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredient nos. 3, 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20, 21, 22 and 24 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 19 and 20 from Table 52, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53, nos. 3 and 4 from Table 21, nos. 4 and 5 from Table 38, nos. 4, 7, 10, 16, 20, 21, 22, 23, 24, 25, 41, 42, 55, 56, 57, 58 and 59 from Table 47, and nos. 1, 4, 5, 6, 7, 8, 11, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40, 41, 42, 43 and 44 from Table 48 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (0%).

Use Example 5

Action on Botrytis cinerea

Paprika seedlings of the "Neusiedler Ideal Elite" variety were sprayed, after 4 to 5 leaves were well developed, to runoff with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. After the sprayed-on layer had dried, the plants were sprinkled with a conidial suspension of the fungus Botrytis cinerea, and placed at 22° to 24° C. in a chamber of high humidity. After 5 days, the disease had spread to such a great extent on the untreated plants that the necroses covered the major portion of the leaves.

    ______________________________________                                                         Percentage leaf attack after                                                   spraying with aqueous formu-                                                   lations containing 500 ppm                                     Active ingredient                                                                              of active ingredient                                           ______________________________________                                         Table 30, active ingr. no. 2                                                                    5                                                             Comparative substance A                                                                        100                                                            Comparative substance B                                                                        100                                                            Comparative substance C                                                                        100                                                            Untreated       100                                                            ______________________________________                                    

Use Example 6 Action on Plasmopara viticola

Leaves of potted vines of the Muller-Thurgau variety were sprayed with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. To assess the duration of action, the plants were set up, after the sprayed-on layer had dried, for 8 days in the greenhouse. Then the leaves were infected with a zoospore suspension of Plasmopara viticola. The plants were first placed for 48 hours in a water vapor-saturated chamber at 24° C. and then in a greenhouse for 5 days at from 20° to 30° C. To accelerate and intensify the sporangiophore discharge, the plants were then again placed in the moist chamber for 16 hours. The extent of fungus attack was then assessed on the undersides of the leaves.

    ______________________________________                                                         Percentage leaf attack after                                                   applying aqueous formu-                                                        lations containing 500 ppm                                     Active ingredient                                                                              of active ingredient                                           ______________________________________                                         Table 21, active ingr. no. 3                                                                    5                                                             Table 21, active ingr. no. 4                                                                    0                                                             Table 30, active ingr. no. 1                                                                   15                                                             Comparative substance A                                                                        65                                                             ______________________________________                                    

    ______________________________________                                                         Percentage leaf attack after                                                   applying aqueous formula-                                                      tions containing 500 ppm of                                    Active ingredient                                                                              active ingredient                                              ______________________________________                                         Comparative substance B                                                                        40                                                             Comparative substance C                                                                        25                                                             Untreated       65                                                             ______________________________________                                     

We claim:
 1. A compound of the formula I ##STR286## where Z is a trifluoromethyl, trichloromethyl, methoxy, amino, methylamino or dimethylamino;X,Y are hydrogen, fluoro, chloro, bromo, trifluoromethyl, cyano, nitro, alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, or X,Y together form a substituted aromatic, alicyclic, partially or completely hydrogenated ring; R¹ is alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, cycloalkenyloxy, or alkoxycarbonyloxy; A is a single bond, O, S, CR² ═CR³, CHR² O, CHR² S, CHR² --ON═CR⁴, CR² ═NO, ON═CR⁴, C.tbd.C, CHR² --CHR³, CHR² O--CO, or OCHR² ; B is hydrogen, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, arylalkyl, cycloalkylalkyl, or cycloalkenylalkyl; R²,R³ are hydrogen, alkyl, alkenyl, alkynyl, or cycloalkyl; R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, alkoxy, or cycloalkyl;provided that B is not hydrogen when A denotes a single bond.
 2. The compound of claim 1, wherein X and/or Y denote hydrogen.
 3. The compound of claim 1, whereX,Y are hydrogen, fluoro, chloro, bromo, trifluoromethyl, cyano, nitro, C₁ -C₆ -alkylalkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₆ -alkoxy, C₂ -C₆ -alkenyloxy, C₂ -C₆ -alkynyloxy, or X,Y together form a substituted aromatic or alicyclic partially or completely hydrogenated ring.
 4. The compound of claim 1, whereR² -R³ are hydrogen, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, or C₃ -C₁₀ -cycloalkyl; and R⁴ is hydrogen, cyano, C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₂ -C₆ -alkynyl, C₁ -C₆ -alkoxy, or C₃ -C₁₀ -cycloalkyl.
 5. The compound of claim 1, whereR¹ is C₁ -C₆ -alkoxy, C₂ -C₆ -alkenyloxy, C₂ -C₆ -alkynyloxy, C₃ -C₁₀ -cycloalkoxy, C₃ -C₁₀ -cycloalkenyloxy, or C₁ -C₆ -alkoxycarbonyloxy.
 6. A compound of formula ##STR287## where Z is methoxy;X,Y are hydrogen, fluoro, bromo, trifluoromethyl, cyano, nitro, alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, or X,Y together form a substituted aromatic, alicyclic, partially or completely hydrogenated ring; R¹ is alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, cycloalkenyloxy, or alkoxycarbonyloxy; A is a single bond, O, S, CR² ═CR³, CHR² O, CHR² S, CHR² --ON═CR⁴, CR² ═NO, ON═CR⁴, C.tbd.C, CHR² -CHR³, CHR² --O--CO, or OCHR² ; B is hydrogen, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, arylalkyl, cycloalkylalkyl, or cycloalkenylalkyl; R²,R³ are hydrogen, alkyl, alkenyl, alkynyl, or cycloalkyl; R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, alkoxy, or cycloalkyl; provided that B is not hydrogen when A denotes a single bond.
 7. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 1, or a plant tolerated acid or base adduct thereof.
 8. A process for combating fungi comprising the step of treating fungi, plants, seeds, soil or material threatened by fungal attack with a fungicidally effective amount of a compound of the compound of claim 1, or a plant-tolerated acid or base adduct thereof.
 9. The compound of claim 1, whereinB denotes hydrogen, or optional substituted C₁ -C₆ -alkyl, C₂ -C₆ -alkenyl, C₃ -C₁₀ -cycloalkyl, C₃ -C₁₀ -cycloalkenyl, C₃ -C₁₀ -cycloalkynyl, aryl, aryl C₁ -C₆ -alkyl, C₃ -C₁₀ -cycloalkyl-C₁ -C₆ -alkyl, or C₃ -C₁₀ -cycloalkenyl-C₁ -C₆ -alkyl .
 10. The compound of claim 1, where R¹ is C₁ - or C₂ -alkoxy.
 11. The compound of claim 1, where Z is methoxy.
 12. The compound of claim 1, where A is O, CH═CH, CH₂ --O, CH₂ --ON═CR⁴, or O--CH₂, and R⁴ is hydrogen, cyano, C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, or C₃ -C₆ -cycloalkyl.
 13. The compound of claim 1, where B is unsubstituted or substituted aryl.
 14. The compound of claim 1, whereR¹ is C₁₋ or C₂ -alkoxy, Z is methoxy, A is O, CH═CH, CH₂ --O, CH₂ --ON═CR4, or O--CH₂, and R⁴ is hydrogen, cyano, C₁ -C₄ -alkyl, C₁ -C₄ -alkoxy, or C₃ -C₆ -cycloalkyl, and B is unsubstituted or substituted aryl.
 15. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 10 or a plant tolerated acid or base adduct thereof.
 16. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 11 or a plant tolerated acid or base adduct thereof.
 17. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 12 or a plant tolerated acid or base adduct thereof.
 18. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 13 or a plant tolerated acid or base adduct thereof.
 19. A fungicide comprising an inert carrier and a fungicidally effective amount of the compound of claim 14 or a plant tolerated acid or base adduct thereof. 